Encyclopedia of Traditional Chinese Medicines Vol. 2

Encyclopedia of Traditional Chinese Medicines
Molecular Structures, Pharmacological Activities,

Natural Sources and Applications
Jiaju Zhou Guirong Xie Xinjian Yan
Encyclopedia of
Traditional Chinese Medicines
Molecular Structures, Pharmacological
Activities, Natural Sources and Applications
Vol. 2: Isolated Compounds D-G
Jiaju Zhou
1303, Buld. 10,
31 ZhongGuanCun NanDaJie,
HaiDian District,
100081, Beijing,
China
jjzhou@mail.ipe.ac.cn
Guirong Xie
Apt-2-1-302,
43 NongDa NanLu,
BoYaXiYuan,
HaiDian District,
100193, Beijing,
China
zhouxuexi@yahoo.cn
Xinjian Yan
523 Redland Blvd,
Rockville,
MD 20850,
USA
yunyan316@yahoo.com
ISBN 978-3-642-16737-9
e-ISBN 978-3-642-16738-6
DOI 10.1007/978-3-642-16738-6
Springer Heidelberg Dordrecht London New York
Library of Congress Control Number: 2011922128
# Springer-Verlag Berlin Heidelberg 2011
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Encyclopedia of Traditional Chinese Medicines

Molecular Structures, Pharmacological Activities, Natural Sources and Applications
Contents
Preface ........................................................................................................................... vii
Introduction .................................................................................................................. ix
How to Use This Book ............................................................................................... xix
Abbreviations and Symbols ....................................................................................... xxv
Cancer Cell Codes ..................................................................................................... xxix
Volume 1 Isolated Compounds (A-C)
A (entries 1~2071) ........................................................................................................... 3
B (entries 2072~2835) ................................................................................................ 241
C (entries 2836~4594) ................................................................................................ 327
Volume 2 Isolated Compounds (D-G)
D (entries 4595~6656) ..................................................................................................... 3
E (entries 6657~7700) ................................................................................................ 225
F (entries 7701~8043) ................................................................................................ 343
G (entries 8044~9185) ................................................................................................ 383
Volume 3 Isolated Compounds (H-M)
H (entries 9186~10927) ................................................................................................... 3
I (entries 10928~11806) ............................................................................................. 187
J (entries 11807~11990) ............................................................................................. 283
K (entries 11991~12399) ............................................................................................ 308
L (entries 12400~13280) ............................................................................................ 356
M (entries 13281~15227) ........................................................................................... 459
Volume 4 Isolated Compounds (N-S)
N (entries 15228~15880) ................................................................................................ 3
O (entries 15881~16484) ............................................................................................ 73
P (entries 16485~18281) ............................................................................................. 142
Q (entries 18282~18455) ............................................................................................ 350
R (entries 18456~19091) ............................................................................................ 375
S (entries 19092~20574) ............................................................................................. 453
vi
Volume 5 Isolated Compounds (T-Z)

T (entries 20575~22170) ................................................................................................. 3
U (entries 22171~22301) ............................................................................................ 184
V (entries 22302~22625) ............................................................................................ 201
W (entries 22626~22742) ........................................................................................... 238
X (entries 22743~22856) ............................................................................................ 254
Y (entries 22857~22960) ............................................................................................ 270
Z (entries 22961~23033) ............................................................................................ 284
References for Isolated Compounds ........................................................................... 293
TCM Plants and Congeners (entries T0001 ~ T6926) .................................................. 347
Volume 6 Indexes
Compound Pharmacological Activity Index .................................................................. 3
Compound Molecular Formula Index ........................................................................ 65
Compound Name Synonym Index .............................................................................. 285
TCM Plant English Name Index ................................................................................ 347
TCM Plant PIN-YIN/Chinese Name Index ................................................................ 458
TCM Plant Traditional Effect Index ........................................................................... 580
TCM Plant Traditional Indication Index .................................................................... 624
Preface
A significant preoccupation of modern traditional Chinese medicine (TCM)
research has been the characterization of TCM components, such as pertain to their
isolation, purification, structural determination, and pharmacological activity. As a
reference tool, this Encyclopedia of Traditional Chinese Medicines presents a
comprehensive and integrative work on surveying TCM plant sources, chemistry,
pharmacology and medicinal effects and indications in a systematic manner.
This encyclopedia is an integrated achievement of a long-term TCM research
project by the authors at the Chinese Academy of Sciences [14], involving three parts
and now organized in six volumes:
Part I (Volumes 1 to 4 and part of Volume 5) provides structural, physical,
pharmacological and natural source information on 23,033 isolated chemicals captured
from 5,535 references, basically up to year 2005. A great deal of effort has been paid on
overlapping or contradictory data in order to provide readers with an accurate and
reliable resource.
Part II (last part of Volume 5) describes 6,926 TCM plants and congeners, together
with their medicinal effects and indications. The contents of Part I and Part II are all
organized in alphabetical order.
Part III (Volume 6) includes seven indexes produced by a computer program.
Based on the indexes, users can readily find concerned contents in multiple ways.
With this encyclopedia, the authors attempt to provide a bridge for the
communication between the TCM system and Western medicinal systems, and a
platform with multiple-subjects in support of research and development of the health
sciences.
---------------------------
JJ Zhou, GR Xie and XJ Yan

Institute of Process Engineering, Chinese Academy of Sciences
Sep, 2010, Beijing
[1] Xinjian Yan, Jiaju Zhou and Guirong Xie, Traditional Chinese Medicines: Molecular structures, natural sources,
and applications, 1st edition, Ashgate Publishing house, 1999
[2] Jiaju Zhou, Guirong Xie and Xinjian Yan, Traditional Chinese Medicines: Molecular structures, natural sources,
and applications, 2nd edition, Ashgate Publishing house, 2002
[3] Jiaju Zhou, Guirong Xie and Xinjian Yan, Handbook of Chemical Components in Plant Origins of Traditional
Chinese Medicines, Chemical Industry Press, Beijing, 2004 (in Chinese)
[4] Jiaju Zhou, Guirong Xie and Xinjian Yan, Data Collection of Chemical Components in Plant Origins of
Traditional Chinese Medicines, Vol 13, Science Press, Beijing, 2009 (in Chinese)
vii
Introduction
This encyclopedia mainly consists two parts - compound and plant. Its core
content is the structural and pharmacological information of 23,033 phytochemicals, as
well as medical effects and indications of 6,926 plant species from which the
phytochemicals were isolated. The compounds, i.e. phytochemicals, are ordered
alphabetically, and their ordinal numbers are used as compound unique codes. The
plant species are coded from T0001 to T6926. With this code system, the complicated
many to many relationship between compounds and plants can be clearly expressed,
and any individual compound or plant could be located easily in this 6 volumes book.
1. Compound Entry
Format of Compound Entry. A compound entry starts with a title line, in which there
are two items: the compounds unique code and main name. Following the title line is
the compound physical, pharmacological and source information, which may include 8
items:
Title line (code number, main name)
A. Synonyms of the compound (if any);
B. CASRN number (if any);
C. Formula (relative molecular mass);
D. Physicochemical properties;
E. Pharmacological data (if any);
F. Source(s);
G. Reference(s);
H. Graphic structure.
Chemical Names and Synonyms. Generally, a compound may have one scientific
name and several trivial names. In the encyclopedia, based on original articles, we
select one name as the main name (appeared at the title line of each compound entry),
and use it to alphabetically order the 23,033 compounds in the first 5 volumes. The
main name is either a scientific name or a trivial name. All of other names of each
compound, if any, are presented after the title line.
Stereochemistry of Chemical Structure. We protracted all compound structures down
to atom-bond level including complicated glycosides, with stereo-chemical information
based on the data in the original papers. For example, the structure with full
stereochemistry of compound 22,834 (isolated from CHUAN XU DUAN Dipsacus
asperoides) is:
ix
hederagenin
H
O
28
OH
6
OO
OH 1
HO
OO
HO
OO
Glu OH 1
2
OH 1 Glu
OH
OO
OH
OH
1
Rham
OH
OH
3
Ara
HO
O O OH
O 1 Glu
HO
OO 3
OH
Glu 4 OH
1
OO
OH
Xyl OH 1 OH O
OH
1
OH
Rham
OH OH
3-O-[-D-Xylopyranosyl(14)--D-glucopyranosyl(14)]
[-L-rhamnopyranosyl(13)]--D-glucopyranosyl(13)-L-rhamnopyranosyl(12)--L-arabinopyranosyl hederagenin28-O--D-glucopyranosyl(16)--D-glucopyranoside
Normalization of Pharmacological Data. More than 8,000 TCM components in this

encyclopedia have a variety of pharmacological data, which are valuable not only for
the study of TCM, but also for the development of Western medicine. Because different
expressions are used for the same kind of data in different articles, we have to define
and normalize thousands pharmacological terms, so that the data could be expressed by
a unified way, and be easily understood by readers.
The pharmacological terms in the encyclopedia are presented by a multi-layered
structure. In the top layer, there are around 20 types of pharmacological activity terms,
they are cytotoxic (in vitro anticancer), antineoplastic (in vivo anticancer), antibacterial,
antifungal, antiviral, anti-HIV, anti-inflammatory, antioxidant, antimalarial, enzyme
inhibitors, NO production inhibitors, cardiovascular activity, smooth muscle relaxant
and stimulant, toxin and medium lethal dose LD50, and so forth. For each term there is
a regulation about how to describe related pharmacological data. The following is an
example:
Term name (in vitro/in vivo,
target cell 1, quantitative data,
control Compound, controls data;
terse description of related mechanism if any).
xi
Under the subtitle Pharm: of compound entry 248 (17-Acetoxylabda-7,12(E),14triene), a set of bio-data is presented as follows:
Pharm: Cytotoxic (in vitro,
BT474 human galactophore cancer cell, IC50 = 4.7g/mL,
control Doxorubicin hydrochloride, IC50 = 0.08g/mL;
CHAGO human undifferentiated lung cancer cell, IC50 = 5.7g/mL,
HepG2 human liver cancer cell, IC50 = 6.5g/mL,
Kato3 human gastric cancer cell, IC50 = 5.3g/mL,
SW620 human colorectal adenocarcinoma cell, IC50 = 5.6g/mL,
control Doxorubicin hydrochloride, IC50 = 1.1g/mL).
In order to standardize abbreviations of cancer cells, such as BT474, CHAGO,

etc., we defined and used 270 cancer cell codes (CCC) in the encyclopedia. For
explanations of these codes, please see Cancer Cell Codes in the Pharmacological
Models in Volume 1 of the encyclopedia.
By means of the formatted and structuralized methods, we normalized expressions
of most pharmacological data appeared in the encyclopedia. For complete information
of all 3367 normalized pharmacological activity terms, please see Compound
Pharmacological Activities Index in Volume 6.
2. Plant Entry
One Species One Entry. Conventionally, a TCM name may include more than one
plant species that have the same medical functions; therefore, a plant may not have an
independent TCM entry and may be described under a TCM name. In this book,
modern botany classification regulation is adopted and each plant species has an
independent entry.
For example, traditional Chinese medicine DAN SHEN includes three species.
They are equivalent in both effects and indications in TCM practice. In this
encyclopedia, we defined three plant entries for each one of them.
T5680 Salvia miltiorrhiza (Lamiaceae); DAN SHEN; Danshen;
T5681 Salvia miltiorrhiza f. alba (Lamiaceae); BAI HUA DAN SHEN; Whiteflower Danshen;
T5688 Salvia przewalskii (Lamiaceae); GAN XI SHU WEI CAO; Przewalsk Sage.
With this method, we are able to smoothly link TCM information with that of
modern botany.
Simplified Latin Name. For each TCM plant or TCM congener, four names are used
in the encyclopedia. They are Latin name, English name, PIN-YIN name and Chinese
xii
name, while the Chinese name only appears in TCM Plants PIN-YIN/Chinese Names
Index not in the main part of the book. For plant Latin name (e.g. scientific name), we
use a simplified nomenclature, in which the nomenclator(s) information is not included.
For example the Latin name of Chinese Angelica (DANG GUI) in the encyclopedia is
Angelica sinensis, not Angelica sinensis (Oliv.) Diels.
Family Name. According to the International Code of Botanical Nomenclature
(2007), the following eight authoritative family names are used in the encyclopedia.
The family names of long usage, which are not used in are the encyclopedia, indicated
in parentheses:
Apiaceae (Umbelliferae);
Arecaceae (Palmae);
Asteraceae (Compositae);
Brassicaceae (Cruciferae);
Clusiaceae (Guttiferae);
Fabaceae (Leguminosae);
Lamiaceae (Labiatae) and
Poaceae (Gramineae).
PIN-YIN Name and Chinese Name. A simplified PIN-YIN name system is used in
the encyclopedia. That is not to include the four-tone mark. However, there are
exceptions. Among the thousand PIN-YIN names in the book, there are seven
confusing cases. For each mistakable name, a superscript is attached to the name for
indicating its four-tone in order to distinguish it from other plant species. For example:
BAI MAO GEN(1) and BAI MAO GEN(4) are two different TCM plants:
T3416 Imperata cylindrica var. major (Poaceae); BAI MAO GEN(1); Lalang Grass Rhizome.
T3309 Hydrastis canadensis (Ranunculaceae); BAI MAO GEN(4); Golden-seal.
Other six cases are:

T1449 Cirsium japonicum (Asteraceae); DA JI(4); Japanese Thistle.
T2608 Euphorbia pekinensis (Euphorbiaceae); DA JI(3); Peking Euphorbia.
T4124 Matricaria chamomilla [Syn. Matricaria recutita] (Asteraceae); MU(3) JU; Mayweed.
T0197 Aegle marmelos (Rutaceae); MU(4) JU; Sepiaria.
T1039 Bruguiera gymnorrhiza (Rhizophoraceae); MU LAN(3); Common Bruguiera.
T3423 Indigofera tinctoria (Fabaceae); MU LAN(2); True Indigo.
T6798 Vitis vinifera (Vitaceae); PU(2) TAO; European Grape.
T6267 Syzygium jambos (Myrtaceae); PU(3) TAO; Roseapple.
T2107 Dendrobium nobile (Orchidaceae); SHI HU(4); Noble Dendrobium.
T2646 Evodia rutaecarpa var. officinalis (Rutaceae); SHI HU(3); Officinal Evodia.
T1221 Caryopteris divaricata (Verbenaceae); YOU(2); Divaricate Bluebeard.
T1478 Citrus grandis (Rutaceae); YOU(4); Pummelo.
xiii
Translation of TCM Effects Terms. In the Volume 5 of the encyclopedia, 6,926

TCM Plant entries list in alphabetical order of Latin names, including 2,923 original
TCM plants (including few of animals)[R01-R04] and 4,003 congeners (including a few of
non-TCM medicinal plants). For each TCM plant, two most important features are
traditional TCM effects and indications.
For preparing this encyclopedia, one of the greatest challenges is how to correctly
translate each TCM term into correspondent English, so that Western readers are able to
understand the true meaning of the content in the book. After comparing several
translation systems, we decided to use Wisemans terminological system[R05-R07] for this
book.
Wisemans system obeys two most important principles: (1). The Englishlanguage terms should be faithful to the original concepts in traditional Chinese
medicine. (2). The English-language TCM terminology should be flexible enough to
allow modifications and extensions so that derivative effects can be described by a
structuralized manner. For instance, the term quicken blood describes a general effect
meaning activating blood flow or promoting blood circulation. Elaboration of this
term produces quicken blood and transform stasis, quicken blood and relieve pain,
quicken blood and regulate menstruation, and so on. The following illustrations an
example of the structuralized expressions related to the term quicken blood:
quicken blood and disinhibit water
quicken blood and dispel stasis
quicken blood and dispel wind
quicken blood and disperse swelling
quicken blood and disperse welling abscess
quicken blood and dissipate binds
quicken blood and dissipate stasis
quicken blood and free menstruation
quicken blood and free network vessels
quicken blood and free vessels
quicken blood and joint bones
quicken blood and move qi
quicken blood and move stasis
quicken blood and nourish heart
quicken blood and promote milk
quicken blood and quiet spirit
quicken blood and regulate menstruation
quicken blood and relieve pain
quicken blood and resolve toxin
quicken blood and settle pain
quicken blood and soothe sinews
quicken blood and stanch bleeding
quicken blood and strengthen sinews
quicken blood and transform stasis
quicken blood and vessels
xiv
Translation of TCM Indications Terms. Based on Wisemans terminological system,

Chinese-English Dictionary of Traditional Chinese Medicine compiled by
Guangzhen Gao et al. [R08], An English-Chinese Medical Dictionary, Second Edition
compiled by Weiyi Chen et al.[R09], and other reference dictionaries, we defined over
3,800 standard indication terms for translating TCM indications terms from Chinese to
English. Among the 3,800 terms, 2,526 terms are actually used in the encyclopedia, in
which 85% terms are traditional TCM terms and the rest 15% are common modern
medicinal terms. Some typical examples of traditional TCM indication terms are as
follows:
yin vacuity internal heat
yin vacuity lung dryness
yin vacuity tidal fever
chest impediment
chest impediment and heart pain
chest impediment and heart pain over back
chest oppression and pain
chest oppression with breathe hard
distention pain in rib-side
distention pain in stomach duct
distention pain in stomach duct and abdomen
externally contracted summer heat-damp
externally contracted wind evil
externally contracted wind-cold
externally contracted wind-heat
knocks and falls
sores
sores clove boil
swelling of sores and boils
sore scab and lichen
toxin swelling of sores
In summary, this encyclopedia provides a collection of more than 23,000 TCM

chemical components isolated from natural resources and a large number of
pharmacological activity data of these components. It may be used not only as a
handbook to look for structures and pharmacological activities of TCM chemical
components and source plant information, but also a fundamental platform for studying
TCM with a systematic and integrative approach.
xv
Acknowledgements
We, the authors, would like to express our gratitude to Dr. Georga W.A. Milne,
former chief editor of JCICS of American Chemical Society. Dr. Milne originally urged
us to open a long-term project on TCM information study in 1993. From that time on,
he has been supporting and helping us in many aspects.
We would like to thank a number of Chinese scientists who are working on TCM
related fields for their support, help and information. Among them, special thanks are
given to Prof. Peigen Xiao (member of Chinese Engineering Academy, Institute of
Medicinal Plant Development, Chinese Academy of Medical Sciences & Peking Union
Medical College), Pref. Guanhua Du (Institute of Materia Medica, Chinese Academy of
Medical Sciences & Peking Union Medical College), Prof. Weiliang Wong (China
Academy of Chinese Medical Sciences), and Prof. Luhua Lai (Peking University).
We would like to thank the leaders and colleagues of the Institute of Process
Engineering (IPE), Chinese Academy of Sciences (CAS) for their understanding,
support, and help. Particularly, thanks go to Prof. Mooson Kwauk (member of the CAS),
Prof. Jinghai Li (member of the CAS, Vice president of CAS), Prof. Zhihong Xu, Prof.
Zhiguo Su, Prof. Suojiang Zhang (Director of IPE), Prof. Yunfa Chen (Vice director of
IPE), Prof. Huizhou Liu, Prof. Zhangyuan Yang, Prof. Hao Wen, and Prof. Xiaoxia Li.
We would like to thank our colleagues and students in the Molecule Design Group
in the Lab of Computer Chemistry (LCC) for their indispensable contributions
including information search, data collection, software development and technical
support, etc. Among them, special thanks are given to Mr. Wucheng Tang, Ms.
Hongping Xu, Ms. Qi Li, Asso. Prof. Dianfang Cao, Dr. Xianfeng He, Dr. Min He, Dr.
Jianfeng Pei, Dr. Tao Peng, Dr. Jing Lei, Dr. Aihua Xie, Dr. Chengzhong Liao, Dr.
Aijun Lu, Dr. Bing Liu, Dr. Haibo Liu, and Master Yingxin Qiao.
Cordial thanks are also given to Asso. Prof. Lanying Zhao, Asso. Prof. Peiwu
Wang and Asso. Prof. Yuanzhang Luo for their toilsome work on information collection
in the early stage of the project.
Finally, we would like to give heartfelt thanks to our family members. Without
their complete and never-ending support, this book would never have been completed.
xvi
Core References
(Comprehensive data sources of TCM plants)
R01
Jiangsu New Medical College Ed., Chinese Medicine Dictionary, Shanghai

Science and technology Press, Shanghai, 1979
R02 Huiyuan Zhang, Zhiying Zhang, Zunsun Yue, Rongling Guo, et al., Brief Flora of
Chinese medicine, Science Press, Beijing, 1994
R03 Chinese Materia Medica Editing Committee of the National Chinese Medicine
and Pharmacology Bureau, Chinese Materia Medica (ZHONG HUA BEN CAO),
Vol. 1Vol. 30, Shanghai Science and technology Press, Shanghai, 1999
R04 J. Buckingham (Executive Editor), Dictionary of Natural Products, Chapman &
Hall, London, Vol. 1Vol. 7 1994; Vol. 8, 1995; Vol. 9, 1996; Vol. 10, 1997; Vol.
11, 1998
(English translation tools)
R05
Nigel Wiseman, English-Chinese, Chinese-English Dictionary of Chinese

Medicine, Hunan Science and Technology Press, Chang Sha, 1996
R06 Nigel Wiseman, English-Chinese, Chinese-English Dictionary of Chinese Medicine,
Second Edition, Hunan Science and Technology Press, Chang Sha, 2007
R07 Nigel Wiseman and Ye Feng, A Practical Dictionary of Chinese Medicine, Second
Edition, Paradigm Publications, Brookline, Massachusetts, 1998
R08 Guangzhen Gao, Yixiang Yuan, Jixue Ren and Long Huang, Chinese-English
Dictionary of Traditional Chinese Medicine, Peoples Medical Publishing House,
Beijing, 1996
R09 Weiyi Chen et al., An English-Chinese Medical Dictionary, Second Edition,
Shanghai Science and technology Press, Shanghai, 1997
(Names of plant, bacteria, fungus)
R10 Yutang Zhao and Jinxiang Ji, Dictionarium Latino-Sinicum Nominum Scientificorum Plantarum, Jilin Science and Technology Press, Ji Lin, 1988
R11 Zongxun Wang et al. (Institute of Botany, Chinese academy of Sciences), New
Edited Plant Names in Latin-Chinese-English, Aerial Industry Press, Beijing, 1996
R12 M. Wrobel and G. Creber, Elseviers Dictionary of Plant Names in Latin, English,
French, German and Italian, Elsevier Science B.V., Amsterdam, 1996
R13 Jiaran Zhu et al., Dictionary of Seed-plant Names Latin-Chinese-English, Second
Edition, Science Press, Beijing, 2001
R14 Jiwu Wang, et al., Dictionary of Medicinal Plants, Tianjin Science and technology
Press, Tianjin, 2005
R15 Miaoying Cai, et al., Names of Bacteria, Second Edition, Science Press, Beijing, 1996
R16 C. J. Alexopoulos, M. Blackwell and C. W. Mims, (Yijian Yao and Yu Li
translated), Introductory Mycology, Fourth Edition, John Wiley & Sons, Inc.,
1996, Chinese Agricultural Press, Beijing, 2002
xvii
(Comprehensive data sources of compounds)

R17
Tatsuo Karikome, Wenben Yang translated, Phytochemistry, Science Press,

Beijing, 1985
R18 Jiwu Wang, et al., Handbook of Effective Components in Vegetal Medicines,
People Health Press, Beijing, 1986
R19 Zhenyu Song, et al., Modern Studies of Chinese Herbal Medicine, Vol. 1 to Vol. 3,
Union Press of Beijing Medical University and Peking Union Medical College,
Beijing, 1995, 1996, 1997
R20 Wenji Sun, et al., Brief Handbook of Natural Active Compounds, Medicinal
Science and Technology Press of China, Beijing, 1998
R21 Kee Chang Huang, The Pharmacology of Chinese Herbs, Second Edition, CRC
Press, Boka Raton, London, NewYork, Washington D.C., 1999
R22 Huifang Chen, et al., Lexicon of Active Components in Plants, Vol. 1 to Vol. 3,
Medicinal Science and Technology Press of China, Beijing, 2001
R23 Hangdong Sun, et al., Diterpenoids from Isodon Species, Science Press, Beijing, 2001
R24 M. Ou, et al., Brief Handbook of Components of Traditional Chinese Medicines,
The People's Medical Publishing House, Beijing, 2003
R25 Xiaotian Liang, et al., Fundamental Research on Common Traditional Chinese
Medicines. Vol. 1, Vol. 2, Science Press, Beijing, 2003, 2007
R26 Fakui Chen, Xiaoqiu Liu, et al., Determination of Effective Components in
Traditional Chinese Medicines, Peoples Medical Publishing House, Beijing, 2009
(Other dictionaries)
R27 Jisheng Chen, et al., English-Chinese Dictionary of Life Science, Scientific and
technological Literature Press, Beijing, 1992
R28 Scientific Terms Laboratory of Science Press, English-Chinese Biological
Dictionary, Second Edition, Science Press, Beijing, 1997
R29 Scientific Terms Laboratory of Science Press, Chinese-English Biological
Dictionary, Science Press, Beijing, 1998
R30 J. G. Harris and M. W. Harris, (Yufei Wang, et al., translated) Plant
Identification Terminology: An Illustrated Glossary, Spring Lake Publishing,
Payson UT, 2001, Science Press, Beijing, 2001
R31 Rensheng Xu, et al., Chemistry of Natural Products, Second Edition, Science
Press, Beijing, 2004
R32 Jingying Tan, English-Chinese Biological Dictionary of Biochemistry and
Molecular Biology, Second Edition, Science Press, Beijing, 2007
R33 Wenbao Chang, et al., Dictionary of Chemistry, Science Press, Beijing, 2008
How to Use the Books

1. Three Kinds of Many to Many Relationships
To help readers effectively search and use of the books, authors strongly suggest
readers being familiar with the structure of the encyclopedia and certain important
linkers or pointers between different data sets.
Firstly, in order to avoid confusing cases, please keep in mind the following three
features of the book:
(a) In the encyclopedia, all of pharmacological data belong to compounds, not to
plants. In other words, the encyclopedia doesnt include plants pharmacological data.
(b) All effect and indication terms belong to TCM plants, not to compounds. And
almost all of effect terms as well as 85% indication terms are pure Chinese traditional
concepts.
(c) In the encyclopedia, there are three kinds of many to many relationships: (i),
compounds to plants, which is the most important relationship. (ii), pharmacological
data to compounds in the molecular level only. (iii), plants to effects/indications in the
species level.
Pharm. data Compound 1
..
(Molecular level)
Plant T0001 effects, indications

.
(Species level)
Sketch Map of Three Important Many to Many Relationships
2. Seven Useful Indexes

In Volume 6, there are seven indexes for data searching.
The indexes 1-3 are tools to search compounds from different starting-points:
Index 1 (Compound Pharmacological Activity Index) links pharmacological terms
xix
xx
with related compound codes. For example, if there is a question as:

Which compounds have in vitro cytotoxic activity against human breast cancer
cells?
From the index 1, the answer can easily be obtained as follows:
Cytotoxic, BC hmn breast cancer cells 24, 349, 526, 2244, 3416, 3429, 3708, 4775, 5095,
6759, 6759, 6759, 12453, 12454, 15494, 15495, 18515, 20671.
Cytotoxic, BC-1 hmn breast cancer cells 1277, 2260, 5064, 5327, 6759, 6759, 8220, 8221,
8222, 8235, 10250, 10297, 10511, 11353, 13489, 13490, 13491, 13492, 13493, 13494,
13495, 15919, 17008, 18866, 20809.
Cytotoxic, BCA-1 hmn breast cancer cells 6759, 13468, 13469, 13470, 15739.
Cytotoxic, Bcap37 hmn breast cancer cells 843, 11392, 13123, 16183, 17717, 18499.
Then, from compounds code numbers, one can get detailed data for each
compound.
Index 2 (Compound Molecular Formula Index) connects a molecular formula to
its all isomers. For example, there are five isomers with formula C45H76O18:
C45H76O18
Abutiloside F, 40
Asp-IV, 1905
Asp-V, 1906
Trigoneoside IIIa, 21669
Trigoneoside IIIb, 21670
Index 3 (Compound Synonym Index) is useful for searching a compound from a

known name. A strong suggestion to readers is that when searching a compound from a
known name, to search twice probably is necessary: firstly from entry title in the
encyclopedia text and then from the index 3.
The indexes 47 are tools to search TCM plants:
Index 4 (TCM Plant English Name Index) links a Plant English Name to other
names of the plant, for example:
Chinese Angelica = T0495 Angelica sinensis = DANG GUI
Siberian Phlojodicarpus = T4804 Phlojodicarpus sibiricus = ZHANG GUO QIN
Dahurian Angelica = T0478 Angelica dahurica [Syn. Angelica porphyrocaulis] = BAI ZHI
Gigantic Angelica = T0483 Angelica gigas = CHAO XIAN DANG GUI
Narrowleaf Angelica = T0476 Angelica anomala = XIA YE DANG GUI
Index 5 (TCM Plant PIN-YIN and Chinese Name Index) links PIN-YIN name to
Latin name and/or English name, for example:
BAI HUA QIAN HU = T4768 Peucedanum praeruptorum = Whiteflower Hogfennel
BAI HUA SHE GAN = T3457 Iris dichotoma = Vesper Iris
BAI HUA SHE SHE CAO = T4485 Oldenlandia diffusa [Syn. Hedyotis diffusa] = Spreading Hedyitis
Index 6 (TCM Plant Traditional Effects Index) and Index 7 (TCM Plant
Traditional Indications Index) connect specific effect and/or indication to related plants.
xxi
For example, to search all plants with effect nourish heart and quiet spirit, the result
is:
nourish heart and quiet spirit:
T0944 Biota orientalis [Syn. Thuja orientalis; Platycladus orientalis],
T1292 Celastrus orbiculatus [Syn. Celastrus articulatus],
T1381 Choerospondias axillaris,
T4194 Menyanthes trifoliata,
T4400 Nelumbo nucifera,
T4902 Pimpinella thelungiana,
T5108 Polygonum multiflorum,
T5497 Rhodiola kirilowii,
T5701 Salvia yunnanensis.
If searching all plants with indication angina pectoris (a modern medicinal term),
externally contracted wind-cold (a TCM term), and externally contracted wind-heat
(a TCM term), you will obtain the following results:
angina pectoris: T1215 Carthamus tinctorius, T1395 Chrysanthemum morifolium [Syn. Dendranthema
morifolium], T1775 Crataegus pinnatifida, T1778 Crataegus pinnatifida var. major, T2274 Dryobalanops
aromatica, T2389 Epimedium acuminatum, T2390 Epimedium brevicornum, T2392 Epimedium davidii, T2394
Epimedium elongatum, T2398 Epimedium koreanum, T2401 Epimedium pubescens, T2402 Epimedium
sagittatum, T2404 Epimedium sutchuenense, T2406 Epimedium wushanense, T2846 Ganoderma japonicum
[Syn. Ganoderma sinense], T2848 Ganoderma lucidum, T2964 Ginkgo biloba, T3388 Ilex chinensis [Syn. Ilex
purpurea], T3396 Ilex pubescens, T3397 Ilex pubescens var. glaber, T3875 Liriope spicata var. prolifera,
T3925 Loranthus parasiticus [Syn. Loranthus chinenis; Taxillus chinensis], T3926 Loropetalum chinense,
T4303 Moschus moschiferus; Moschus berezovskii; Moschus sifanicus, T4507 Ophiopogon japonicus, T4608
Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng], T4953 Piper longum, T5312 Pueraria
edulis, T5313 Pueraria lobata [Syn. Pueraria thunbergiana; Pueraria pseudohirsuta], T5316 Pueraria
omeiensis, T5318 Pueraria phaseoloides, T5320 Pueraria thomsonii, T5680 Salvia miltiorrhiza, T5681 Salvia
miltiorrhiza f. alba, T5688 Salvia przewalskii, T6510 Trichosanthes kirilowii, T6513 Trichosanthes rosthornii
[Syn. Trichosanthes uniflora], T6584 Typha angustata, T6585 Typha angustifolia, T6587 Typha latifolia.
externally contracted wind-cold: T4039 Magnolia grandiflora, T4445 Notopterygium forbesii [Syn.
Notopterygium franchetii], T4446 Notopterygium incisum, T4956 Piper mullesua, T5727 Saposhnikovia
divaricata [Syn. Ledebouriella seseloides].
externally contracted wind-heat: T0480 Angelica decursiva [Syn. Peucedanum decursivum], T1395
Chrysanthemum morifolium [Syn. Dendranthema morifolium], T1933 Cyclea sutchuenensis, T2798 Fritillaria
verticillata var. thunbergii [Syn. Fritillaria thunbergii], T3819 Ligusticum brachylobum, T4413 Nepeta
cataria, T4761 Peucedanum longshengens, T4768 Peucedanum praeruptorum, T4769 Peucedanum rubricaule,
T6791 Vitex rotundifolia [Syn. Vitex trifollia var. simplicifolia], T6793 Vitex trifolia.
3. Data Survey Example of Compound Entry

At last, we would like to take Ursolic acid (compound code 22270 in the books) as
a data survey example. Under this compound there are a quite number of data as
follows:
xxii
22270 Ursolic acid

-Ursolic acid [77-52-1] C30H48O3 (456.72).
White solid powder (chloroformmethanol), mp 298~294C, 265~267C.
OH
H
H
HO
Pharm: (27 items)

Cytotoxic (KB, ED50 > 25g/mL, control Doxorubicin, ED50 = 0.12g/mL; Hep3B, ED50 >
25g/mL, control Doxorubicin, ED50 = 0.14g/mL; Colon205, ED50 > 25g/mL,
control Doxorubicin, ED50 = 0.10g/mL; HeLa, ED50 > 25g/mL, control Doxorubicin,
ED50 = 0.11g/mL)[4369];
cytotoxic (in vitro, HONE-1 cell, IC50 = (8.81.5)mol/L, control Etoposide, IC50 =
(0.50.2)mol/L, cis-Platin, IC50 = (3.20.5)mol/L; KB cell, IC50 = (8.22.7)mol/L,
Etoposide, IC50 = (0.90.3)mol/L, cis-Platin, IC50 = (4.40.9)mol/L; HT29 cell, IC50
= (4.71.5)mol/L, Etoposide, IC50 = (2.40.5)mol/L, cis-Platin, IC50 =
(5.71.1)mol/L)[5254];
antineoplastic (liver cancer cells in vitro, mus ascites carcinoma in vivo, life was
prolonged);
antibacterial (Escherichia coli, IZD = 13~15mm, control Chloramphenicol, IZD =
16~20mm, control DMSO (4%), IZD < 10mm; Staphylococcus aureus, IZD =
10~12mm, control Chloramphenicol, IZD = 16~20mm, control DMSO (4%), IZD <
10mm; Bacillus subtilis, IZD = 13~15mm; control Chloramphenicol, IZD = 16~20mm,
control DMSO (4%), IZD < 10mm)[5315];
antibacterial (Staphylococcus spp. in vitro, MIC = 300g/mL, gram-positive bacteria in
vitro, MIC = 50~400g/mL, gram-negative bacteria in vitro, MIC = 200~800g/mL,
microzyme in vitro, MIC = 100~700g/mL);
antitubercular (Mycobacterium tuberculosis, MIC = 41.9g/mL, cytotoxic, Vero cells, IC50
= 46.5g/mL, SI (IC50/MIC) = 1.11, positive control Rifampin, MIC = 0.03g/mL,
IC50 = 98.3g/mL, SI = 3277)[4986];
anticonvulsant (induced by corazol);
anti-inflammatory (rat, induced by embedding woolball, 12.5mg/(kgd) ip, 7 days,
effective);
anti-inflammatory (in vitro, murine macrophage RAW264.7 Cells, inhibits LPS-induced
NO and PGE2 release)[5016];
COX-2 enzyme selective inhibitor (mean IC50 of isomers = 130mol/L)[4415];
COX-2 enzyme inhibitor (PMA-treated hmn mammary and oral epithelial cells,
molecular mechanisms is mediated by a cAMP response element in the COX-2
promoter, associated with inhibition of protein kinases)[4415];
antipyretic (clearly reduces normal body temperature of rat);
reduces serum transaminase (animal, 100mg/kg);
antitrypanosomal (epimastigotes of Trypanosoma cruzi, MLC = 6.2mol/L, control
Gentian violet, MLC = 6.2mol/L)[2579];
mucin release stimulator (acts directly on airway mucin-secreting cells, increased mucin
release (40~50)% above control at the highest concentrations 0.00001~0.001mol/L,
possible use to treatment of chronic airway diseases)[4084];
platelet aggregation inhibitor (2~5mg/mL collagen-induced, IC50 = (5114)mol/L,
control ASA, IC50 = (4203)mol/L; 1~4mol/L epinephrine-induced with
0.8~1.0mg/mL collagen, IC50 = (82.62.8)mol/L, ASA, IC50 = (53.04.5)mol/L;
10~40mol/L Sodium arachidonate-induced with 0.8~1.0mg/mL collagen, IC50 =
xxiii
(66912)mol/L, ASA, IC 50 = (66.02.1)mol/L; 1~5mol/L PGH2/TXA2

receptor agonist U46619-induced with 0.8~1.0mg/mL collagen, IC 50 > 1000mol/L,
ASA, IC50 = (34012)mol/L) [4994];
tissue factor inhibitor inactive[5387];
antirheumatic[5341];
anti-diabetic[5341];
antiulcer[5341];
hypolipidemic[5341];
anti-atherosclerotic[5341];
anti-HIV[5341];
TGF-1 antagonist (inhibits the binding of 125I-TGF-1 to its receptor in Balb/c 3T3 cell,
IC50 = (6.90.8)mol/L, suggests TGF-1 antagonistic activity is responsible, at
least in part, for therapeutic efficacy of Clerodendranthus spicatus to treat humans
with renal disease)[5496];
glucocorticoid (enhances glycogen in liver, reduces glycogen in heart and striated muscles);
LD50 (mus, ip) = 680mg/kg.
Sources: (52 species)
BAI HUA SHE SHE CAO Oldenlandia diffusa [Syn. Hedyotis diffusa] (whole herb: mean
content of 16 origins = 0.211%)[5508],
BI LU GOU TENG Uncaria tomentosa,
CHE QIAN Plantago asiatica (whole herb: content scope = 0.28%~2.32%, mean content =
0.97%)[5508],
CHI NAN Syzygium buxifolium,
CHONG YA YAO Isodon ternifolius,
CI WU JIA YE Acanthopanax senticosus [Syn. Eleutherococcus senticosus],
DA CHE QIAN Plantago major,
DA ZAO Ziziphus jujuba (ripe fruit: mean content = 0.016%)[5508],
DAN SHEN Salvia miltiorrhiza,
DIAN NAN HONG HOU KE Calophyllum polyanthum (seed: yield = 0.0064%dw),
DONG LING CAO Rabdosia rubescens (whole herb: mean content = 0.414%[5508]; leaf:
mean content = 0.573%)[5508],
DU ZHONG Eucommia ulmoides,
DUAN TING SHAN MAI DONG Liriope muscari (tuber),
GOU GU YE Ilex cornuta (leaf: mean content = 0.96%)[5508],
GUANG JING QIAN CAO Rubia wallichiana (stem),
HONG HUA LU TI CAO Pyrola incarnata(whole herb: content = 2.06%)[5508],
HU BEI SHAN ZHA Crataegus hupehensis (dried ripe fruit: mean content = 0.455%),
JIAN YE TOU WU GEN Ligularia sagitta,
LIAN QIAN CAO Glechoma lungituba,
LIAN QIAO Forsythia suspensa,
LIU QIU SHE GEN CAO Ophiorrhiza liukiuensis (whole herb),
MA BIAN CAO Verbena officinalis (whole herb: mean content of 5 batch samples =
0.227%)[5508],
MAO CAO LONG Ludwigia octovalvis (whole herb: yield = 0.00012%dw),
MAO PAO TONG Paulownia tomentosa,
MAO XU CAO Clerodendranthus spicatus,
MU GUA Chaenomeles sinensis,
NV ZHEN ZI Ligustrum lucidum,
PI PA YE Eriobotrya japonica (dried leaf: mean content = 0.677%)[5508],
PI PA YE Eriobotrya japonica (stem and leaf),
PING CHE QIAN Plantago depressa (whole herb: mean content = 0.276%)[5508],
RI BEN LU TI CAO Pyrola japonica,
xxiv
RONG SHU Ficus microcarpa (aerial root),

SHAN DI XIANG CHA CAI Isodon oresbia,
SHAN LI HONG Crataegus pinnatifida var. major,
SHAN ZHA Crataegus pinnatifida (fruit: content scope = 0.31%~0.56%)[5501],
SHAN ZHU YU Cornus officinalis [Syn. Macrocarpium officinale] (dried ripe fruit: content
scope = 0.24%~0.32%[5501], mean content = 0.263%)[5508],
SHI NAN Photinia serrulata (leaf: mean content = 1.50%)[5508],
SHI SHENG BIAN LEI Gentianopsis paludosa,
SHI YE Diospyros kaki (dried leaf: mean content = 0.784%)[5508],
SHU HUA JIE CAO Valeriana laxiflora (aerial parts and root),
SUAN ZAO Ziziphus jujuba var. spinosa (ripe fruit: content = 0.030%)[5508],
SUO YANG Cynomorium songaricum (fleshy stem: content = 0.78%)[5508],
WEI LING CAI Potentilla chinensis,
WU GENG WU JIA PI Acanthopanax sessiliflorus (fruit),
XIA KU CAO Prunella vulgaris (dried spike: content = 0.780%)[5508],
YANG MEI SHU PI Myrica rubra (bark: content = 0.027%),
YE SHAN ZHA Crataegus cuneata (dried ripe fruit: mean content of 3 origins =
0.399%) [5508],
YI LANG QING LAN Dracocephalum kotschyi,
ZHI ZI Gardenia jasminoides [Syn. Gardenia florida] (dried ripe fruit: mean content =
0.041%) [5508],
ZHOU YE LU TI CAO Pyrola rugosa (whole herb: content = 3.00%)[5508],
Cussonia bancoensis,
Occurs in many plants.
Ref: 4, 367, 428, 454, 501, 592, 595, 600, 658, 660, 2579, 3005, 3061, 4084, 4163, 4369,
4415, 4527, 4767, 4772, 4986, 4994, 5016, 5254, 5315, 5382, 5387, 5341, 5496, 5501,
5508.
Abbreviations and Symbols

12(S)-HETE
12(S)-Hydroxy-5,8,10,14-EicosaTatraEnoic acid
cAMP-PDE
125
125
CAPE
I-TGF-1
5-FU
I-Transforming Growth Factor-1
5-FluoroUracil
5-HT
5-HydroxyTryptamine (serotonin)
95%FL (=CI95)
AA
AAPH
2,2'-Azo-bis-(2-AmidinoPropane)-diHydrochloride
ABTS+
ACAT
2,2'-Azino-Bis-(3-ethylbenzThiazoline 6-Sulphonic acid), radical

Acyl-CoA Cholesterol acyltransferase
ACE
Angiotensin Converting Enzyme
Ach
Acetylcholine
AChE
Acetylcholinesterase
ACTH
AdrenoCorticoTropic Hormone
AD
Alzheimers disease
ADM
ADP
AG
CB
cytochalasin B
CC
macrophage inflammatory protein (MIP-1), monocyte chemotactic
95% Fiducial Limits (=95% Confidence Interval)
Arachidonic Acid
protein (MCP-2), and C lymphotactin (ltn) (a chemokine family)

CC0
Minimum cytotoxic concentration
CC50
IC50 of cytotoxicity (concentration of the 50% cytotoxic effect)
CCR1
chemokine receptor 1
CD
concentration required to double enzyme (induction) activity
CD
Concentration required to double quinone reductase (induction)

activity
CD 50
medium Convulsive Dose
cGMP
cyclic guanosine monophosphate
cGMP-PDE
adriamycin
CGN
adenosine diphosphate
CGRP
aminoguanidine
cAMP-phosphodiesterase
Caffeic Acid Phenethyl Ester
cGMP-phosphodiesterase
cis-Golgi networt
Calcitonin gene-related peptide
CHO
Chinese hamster ovarian
AggRt
aggregation rate
CI
AIDS
acquired immunodeficiency syndrome
CI95 (=95%FL)
Chemopreventive index (=IC50/CD)
ALS
amyotrophic lateral sclerosis
CIC
ALT
alanine aminotransferase
CIMC
complete inhibiting minimum concentration
AMP
adenosine monophosphate
CINC-1
AMV
avian myeloblastosis virus
CMV
AP
angina pectoris
AP-1
6-Cyano-7-nitroquinoxaline-2,3-dione (non-NMDA receptor
antagonist)
APN
Aminopeptidase N
CNS
APV
dl-2-Amino-5-phosphonovaleric acid (a competitive antagonist of the
ConA
aq.
central nervous system

concanavalin A
NMDA receptor)
COX
cyclooxygenase
aqueous solution
COX-1
ASA
AcetylSalicylic Acid
COX-2
AST
aspartate transaminase; aspartate aminotransferase
CPT
AT-III
Antithrombase-III
ATPase
AZT
Adenosine triphosphatase
3'-azido-3'-deoxythymidine
BACE1
BChE
-Secretase
cyclooxygenase-2
CRF
corticotrophin releasing factor
CRH-1
CRP
corticotrophin releasing hormone-1

C-reactive protein
CV-3988
Butyrylcholinesterase
basic Fibroblast Growth Factor
CVS
Butylated HydroxyAnisole; 3-tert-Butyl-4-HydroxyAnisole
CXC
Butylated HydroxyToluene
CYP1A
BHT
bid
BLM
Cytochrome P450 2D6
bleomycin
CYP3A4
Cytochrome P450 3A4
Brine Shrimp lethality bioassay = Brine Shrimp Test
cAMP
Cytochrome P450 1A
CYP2D6
concentration
C5a
cardiac vascular system

Stromal cell-derived factor (SDF)-1 and IL-8 (a chemokine)
bis in die (Latin)

boiling point
BST
rac-3-(N-n-octadecylcarbamoyloxy)-2-methoxypropyl
2-thiazoliethyl phosphate
BHA
cyclooxygenase-1
camptothecin
bFGF
bp
cytokine-induced neutrophil chemoattractant 1

Cytomegalovirus
CNQX
activator protein-1
95% Confidence Interval (=95% Fiducial Limits)
complete inhibiting concentration
complement 5a
cyclic adenosine monophosphate
day
DCFH
2,7-dichlorodihydrofluorescein dye
DDDP
dec
DNA-dependent DNA polymerase

decompoposition
D-GalN
D-galactosamine
xxv
xxvi
DGAT
dil.
Diacylglycerol acyltransferase
dilute
DIZ
Diameter of Inhibitory Zone
GSH
Glutathione; N-(N-L--Glutamyl-L-cysteinyl)glycine
GTP
Guanosine TriPhosphate
GVHR
Graft-Versus-HostReaction
DMBA
9,10-dimethyl-1,2-benzanthracene (carcinogen); 7,12-dimethyl-
hour
benz[a]anthracene (carcinogen)
HAD
DMDP
(2R,3R,4R,5R)-2,5-DihydroxyMethyl-3,4-Dihydroxy-Pyrrolidine
HBeAg
hmn type B Hepatitis, e Antigen
DMSO
DiMethyl SulphOxide
HBsAg
hmn type B Hepatitis, Surface Antigen
hmn immunodeficiency virus associated dementia
DNA
deoxyribonucleic acid
HBV
DNJ
1-Deoxynojirimucin (one kind of polyhydroxy alkaloid, glucosidase
HC 50
inhibitor)
HCoV-229E
doxorubicin
HD
DOX
DPI
Diphenyleneiodonium
DPPH
1,1-DiPhenyl-2-PicrylHydrazyl free radical
DS8000
Dextran sulphate, prepared from average Mr 8000
DSCG
dw
DiSodium ChromoGlycate (anti-allergic agent)

dried weight
E.A.
Enzyme Activity
EBV-EA
EC
Epstein-Barr Virus Early Antigen
Effective Concentration
EC50
medium Effective Concentration
ED
Effective Dose
ED 25
ED 50
HER rat
HIV
HIV-1
HIV-RT
hmn
ia
IAA
(-)-Epigallocatechin gallate
Endothelial-Leukocyte Adhesion Molecule-1
Extracellular signal-Regulated Kinase

experimental times
Inhibiting Concentration
IC 50
median Inhibiting Concentration
IC 100
Absolute Inhibiting Concentration
ICAM-1
intradermal injection
Inhibiting Dose
ID 50
Median Inhibiting Dose
IFN
Freund's complete adjuvant
IFN-
IgG
N-formyl-L-Methionyl-L-Leucyl-L-Phenylalanine
IL
freezing point
interferon
Interferon-
IgE
influenza virus type A
Intercellular Cell Adhesion Molecule-1
Imprinting Control Region mouse
ID
fMLP
fw
indole-3-acetic acid
IC
Flu-A
Immunoglobulin E
Immunoglobulin G
interleukin
IL-1
Interleukin-1
Feeding ratio when the consumed area of control disc (CCD) is 50%
IL-1
interleukin-1
[FR = CTD(consumed area of treated disc)/CCD]
IL-1
interleukin-1
IL-2
Interleukin-2
G6PD
Glucose-6-Phosphate Dehydrogenase
IL-4
Interleukin-4
GABA
-aminobutyric acid
IL-6
Interleukin-6
IL-8
Interleukin-8
GaIN
GI
GI50
Glu
GOT
fresh weight
galactosamine
growth inhibition
IL-10
IL-12
the control
im
glutamate
in vitro
in vitro
in vivo
in vivo
Glutamate-Oxaloacetate Transaminase
Gastro protective effect
Indo
gpg
guinea pig
iNOS
GRO
Interleukin-10
the concentration of sample necessary to inhibit the growth to 50% of
Gp
GPT
OH
intra-arterial injection
Fagomine (one kind of polyhydroxy alkaloid, glucosidase inhibitor)

Feeding Index (= ((C-T)/(C+T)100)
FR50
herpes simplex virus 2

homovanillic acid
medium Effective Dose (in some cases for the medium
id
fp
herpes simplex virus 1
HVA
eosinophilous cytotaxin
FI
human
HSV-2
eotaxin
FCA
hmn immunodeficiency virus type 1 reverse transcriptase

hmn immunodeficiency virus reverse transcriptase
HSV-1
ICR
FAG
hmn immunodeficiency virus type 1 integrase
HIV-1 RT
Enzyme-Linked ImmunoSorbent Assay
ET
hmn immunodeficiency virus type 1
HIV-1 IN
ELISA
ERK
Hypertensive Essential Rat

hmn immunodeficiency virus
Effective Concentration)
Epidermal Growth Factor Receptor
ELAM-1
hmn coronavirus strain 229E
Huntingtons disease
hydroxyl radical
Epidermal Growth Factor (it protects MPP+-induced cell death)
EGFR
medium Hemolytic Concentration
Effective Dose for 25%
EGCG (EGCg)
EGF
Hepatitis B Virus
GlutamicPyruvic Transaminase
Growth-Related Oncogene
InRt
ip
Interleukin-12
intramuscular injection
indomethacin
inducible Nitric Oxide Synthase
inhibitive rate
intraperitoneal injection
xxvii
i.t.
intrathecal injection
MMP
iv
intravenous injection
MMP-2
Matrix MetalloProteinases
IZA
Inhibition Zone Area (mm2)
mp
IZD
Inhibition Zone Diameter (mm)
mPGES
J774.A1
JNK
murine monocyte/macrophage cell J774.A1
c-Jun NH2-terminal kinase
Matrix MetalloProteinase-2
melting point
microsomal ProstaGlandin E Synthase
MPP+
1-methyl-4-phenylpyridinium ion (neurotoxin)
MRSA
Methicillin-Resistant Staphylococcus aureus

Methicillin-Sensitive Staphylococcus aureus
KD50
Dose required to Knock down 50% of the population of insects
MSSA
LC50
concentration at which only 50% of the cell are viable
MTC
Minimal Toxic Concentration
LC50
concentration of inhibiting luminous intensity 50%
MTT
A Cytotoxicity measurement method (tetrazolium-based colorimetric
LCIC
LD
Lowest Complete Inhibition Concentration
assay used for cytotoxicity bioassay, see Rubinstein L. V., et al., Nat.
Lethal Dose
LD 100
100% Lethal Dose
LD 50
medium Lethal Dose
Cancer Inst., 82, 1113-1118, 1990)

mus
n
mouse
number of parallel experiments
LDH
lactate dehydrogenase
nAChR
neuronal nicotinic AcetylCholine Receptor
LDL
Low Density Lipoprotein
NADH
reduced nicotinamide adenine dinucleotide
L-NA
N-L-nitroarginine
NADPH
NG-monomethyl-L-arginine
L-NMMA
cytochrome C reductase
NCCLS
A standard antibecterial activity test method (see Wayne P. A.,
LOX
Lipoxygenase
National Committee for Clinical Laboratory Standards Performance
LPO
lipid peroxidation
Standards for Antimicrobial Disk Susceptibility Tests,6th ed.,
LPS
lipopolysaccharide
LTB4
Leukotriene B4
NDGA
LTC4
Leukotriene C4
NEP
LTD4
Leukotriene D4
NF
MA
maytenfolic acid
NF-B
MA
maslinic acid
NFAT
MA
minimal amount
NGF
Approved standards M2-A6. NCCLS, 1997)

Nordihydroguaiaretic acid
Neutral EndoPeptidase
Nuclear Factor
Nuclear Factor B
Nuclear Factor of Activated T cell
Nerve Growth Factor
MABA
Microplate Alamar Blue Assay
NMDA
MAC-1
integrin MAC-1
NO
N-methyl-D-aspartate
nitric oxide
MAO-A
Monoamine oxidase A
non-orl
MAO-B
Monoamine oxidase B
NOR1
MAPK
Mitogen-Activated Protein Kinase
hexenamid
MCC
Minimum Cytocidal Concentration
NOS-2
MCP
Monocyte Chemotactic Protein
OCIF
MCTHBE
Minimum Concentration for Total Haemolysis of Bovine

Erythrocytes (g/mL)
paraoral
(+/-)-(E)-4-methyl-2-[(E)-hydroxyimino]-5-nitro-6-methoxy-3-
orl
Nitric oxide synthase type-2

OsteoClastogenesis-Inhibitory Factor
oral
OVA
ovalbumin
MDA
Methylene Dihydroxy Amphetamine
oxazolone
MDA
Malondialdehyde
OZ
MDR
MultiDrug Resistance
MED
Minimal Effective Dose
P450
Platelet Activating Factor

Platelet Aggregation Factor
Minimal Fungicidal Concentration
PAF
MIA
Minimal Inhibitory Amounts (g/disc)
PAI-1
Minimum Inhibitory Concentration
Cytochrome P450
PAF
MFC
MIC
oxazolone
opsonized zymosan
Plasminogen Activator Inhibitor type 1
Para-3 (=PIV3)
MIC80
Minimal Inhibitive Concentration for 80%
PBMC
MIC90
Minimal Inhibitive Concentration for 90%
PCA reaction
min
minute
MIP-1/
MIQ
MK-801
macrophage inflammatory protein
Minimum inhibitory quantity (g)
Parkinsons Disease
PD
a cytotoxic model
pD2 (=pEC50)
PDE
phosphodiesterase
Minimum Lethal Concentration
PDTC
MLD
Minimum Lethal Dose
PEBP2A
Minimal Morphological Deformation Concentration
MMOC
Mouse Mammary Organ Culture model
negative logarithm (logM) of the concentration required to

produce 50% of the maximum response (EC50)
MLC
MMDC
Passive Cutaneous Anaphylaxis reaction
PD
dizocipline maleate (a non-competitive antagonist of the NMDA

receptor)
Parainfluenza type 3 virus
hmn Peripheral Blood Mononuclear Cell
pEC50
pyrrolidine dithiocarbamate
polyoma enhancer binding protein 2A
negative logarithm (logM) of the concentration required to
produce 50% of the maximum response (EC50)
xxviii
PEG
PolyEthylene Glycol
Singlet oxygen
PEP
Prolyl endopeptidase (a serine protease)
SIZ
sulfisoxazole
SNP
sodium nitroprusside
pet. ether
petroleum ether
PFTase
O2
farnesylprenyltransferase
SOD
PGD 2
prostaglandin D 2
sp.
PGE 2
prostaglandin E 2
SP-A
pulmonary surfactant Protein A
spp.
species (plural)
PGF 2
prostaglandin F 2
Superoxide dismutase
species
PGH2
prostaglandin H2
SRSA
PGI 2
prostacyclin (prostaglandin I2)
StRt
Stimulatory Rate
STZ
streptozotocin
PHA
phytohemagglutinin
Phe
Phenylephrine
pIC50
PK
negative logarithm (-logM) of IC 50

protein kinase
SuRt
survival rate
Syn.(= )
protein kinase C
T/C
PLA2
phospholipase A2
TACE
PMNs
Phorbol-12-Myristate-13-Acetate
polymorphonuclear cell
pNPPase
POA
p-nitrophenylphosphate enzyme
pentacyclic oxindole alkaloids
PPase1
Protein serine/threonine Phosphatase
PRA
Plaque Reduction Assay
PTH
parathyroid hormone
PTN
parthenolide
PTP1B
Protein Tyrosine Phosphatase 1B
Synonym
survival ratio
-Secretase (a serine protease)
TBARS
TC50
ThioBarbituric Acid Reactive Substance assay

50% cytoToxic Concentration
TCM
Traditional Chinese Medicines
TFP
Trifluoperazine (calmodulin antagonist)
TGF-1
TGI
Transforming Growth Factor-1

Total Growth Inhibition, concentration at which no growth was
observed
TI
Therapeutic Index (=IC50/EC50)
TNF-
QR
quinone reductase
TOA
RA
rheumatoid arthritis
topo II
Raji
EBV-transformed B cell line
TP
Tumor Necrosis Factor-

tetracyclic oxindole alkaloids
DNA topoisomerase II
Thymidine phosphorylase
rat
white rat
tPA
rbt
rabbit
TPA (=PMA)
RDDP
RNA-dependent DNA polymerase
RDS
Respiratory Distress Syndrome
rel-InRt
RM
relative inhibitive rate (taking the control compound as 100%)

Relative Mobility
RNA
ribonucleic acid
RNase H
ROS
RSV
RT
sAST
TrkA
TXA2
thromboxane A2
TXB2
thromboxane B2
UDP-MurNac
VCAM-1
VCR
UDP-N-acetylmuramic acid
Vascular Cell Adhesion Molecule-1
vincristine
various cancers, arteriosclerosis, rheumatism and ageing)
Veraguensin
Respiratory Syncytial Virus
VHR DS-PTPase
reverse-transcribed polymerase chain reaction
Vascular Endothelial Growth Factor
VHR protein
VP-16
veraguensin
VHR Dual-Specificity Protein Tyrosine Phosphatase
Vaccina open reading-frame H1-Related protein phosphatase
A positive control for cytotoxic assay (Sigma product)
serum alanine transaminase
VRE
Vancomycin-Resistant Enterococci sp
serum aspartate transaminase
VSE
Vancomycin-Sensitive Enterococci sp
subcutaneous injection
VSV
SC50
Half-maximal radical Scavenging Concentration
ww
SC50
50% Scavenging Concentration
XTT
ScRt
scavenging rate
SDF
Stromal cell-Derived Factor
Vesicular Stomatitis Virus

wet weight
sodium 3'-[1-(phenylaminocarbonyl)-3,4-tetrazolium]
bis(4-methoxy-6-nitrobenzene)sulfonic acid
homonym mark
SGOT
serum Glutamic OxalaceticTransaminase
(=Syn.)
SGPT
serum Glutamic Pyruvic Transaminase
SHR rat
12-O-tetradecanoyl phorbol 13-acetate
proto-oncogene TrkA
VEGF
Reverse Transcriptase
sALT
tissue Plasminogen Activator
reactive oxygen species (they are involved in the genesis of
RT-PCR
sc
inherent ribonuclease H
O2
superoxide anion
PKC
PMA (=TPA)
Slow-Reacting Substance of Anaphylaxis
Spontaneously Hypertensive Rats
SI
Selective index = cytotoxic CC50/target EC50
SI
Selective index = cytotoxic IC50/target IC50
SI
Selective index = cytotoxic IC50/target MIC
synonym mark
the name is given by the authors of the books
Cancer Cell Codes
This set of codes for 270 cancer cells, named as CCC code, are defined and tried out in the books for the first time
by the authors.
1A9
hmn ovarian cancer (cell).
CaEs-17
212
inducible Ha-ras oncogene transformed from the NIH/3T3 cell line.
CAKI
308
cultured mouse epidermal cells.
CAKI-1
3LL
mus Lewis lung cancer (cell).
Calu1
3PS
mouse leukemia (cell).
Capan1
renal cancer (cell).
Capan2
780-6
9KB
9L
hmn epidermatoid nasopharyngeal carcinoma (cell).

rat glioma (cell).
9PS
mouse lymphocytic leukemia (cell).
A2780
hmn esophageal cancer (cell).

hmn renal cancer (cell).
hmn lung cancer (cell).
pancreas cancer (cell).
CaSki
hmn cervical carcinoma (cell).
CEM
leukemia (cell).
CHAGO
hmn undifferentiated lung cancer (cell).
CNE
hmn nasopharyngeal carcinoma (cell).
A375
hmn melanoma (cell).
Col1
hmn colorectal cancer (cell).
A431
hmn epidermic cancer (cell).
Col2
A498
COLO320DM
A549
hmn non-small cell lung cancer (cell).
Colon205
ACHN
AGS
gastric adenocarcinoma (cell).
APM1840
B16
hmn leukemia (cell).
mouse melanoma (cell).
B16(F-10)
BAEC
BC
bovine aortic endothelial cells.

hmn breast cancer (cell).
BC-1
colorectal cancer (cell).
Colon26-L5
mus colorectal cancer (cell).
COS-7
monkey kidney cells.
CPAE
calf pulmonary arterial endothelial cells.
CT-26
mus colorectal cancer (cell).
CTV1
CXF94L
DLD
hmn tumor (cell).
hmn colorectal adenocarcinoma (cell).
DLD-1
BCA-1
DMS114
Bcap37
DMS273
Bel7402
hmn liver cancer (cell).
DU145
Bel7405
EAC
Ehrlich ascites cancer (cell).
BGC823
hmn gastric cancer (cell).
EJ-1
hmn bladder cancer (cell).
BIU87
bladder cancer (cell).
BL6
Bowes

prostatic cancer (cell).
FM3A
mus breast cancer (cell).
H.Ep.-2
hmn cutis cancer cells in throat.
skin cancer cells.
H116
Bre04
H9
BSY1
breast cancer (cell).
HBC4

lymphocytes.
BT474
hmn galactophore cancer (cell).
HBC5
BT549
hmn galactophore cancer (cell).
HCC2998
BXPC3
HCT
C6
rat glioma (cell).
HCT116
CA
HCT15

xxix
xxx
HCT8
HEK-293
HEL
hmn epithelial kidney cell.
hmn embryonic lung fibrocytes.
HeLa
culture cervical epithelial cancer (cell) from Henrietta Lack.
HeLa ATCC-17
HeLa-S3
hmn cervical epithelial cancer (cell).
hmn cervical epithelial cancer (cell).

normal hmn embryo lung fibroblasts.
HELF
Hep2
Hep2,2,15
Hep3B
hmn liver cancer (cell) transfected with hepatitis B virus.

Hepa
Hepa1c1c7
mus liver cancer (cell).
Hepa59T/VGH
HepG2
HEPZ
hmn epithelial cancer (cell).
KU-1
L1210
Lymphocytic leukemia (cell).
L5178Y
lymphosarcoma (cell).
L-6
rat skeletal myoblasts.
L615
mouse spleen leukemia (cell).
L7212
mouse leukemia (cell).
L-929
fibrosarcoma (cell).
LLC
mouse Lewis lung cancer (cell).
LMTK
mouse fiber cells.
LNCaP
hmn prostatic cancer (cell).
LNCaP-FGC
LO2
hmn liver cell.
LoVo
LoVo/Doxo
LOX
hmn colorectal cancer cell, drug-resistant subclone.
melanoma (cell).
HFF
hmn foreskin fibroblasts.
LOX-IMVI
HGF
normal hmn gingival fibroblast cells.
LS174T
HL-60
hmn acute promyelocytic leukemia (cell).
Lu04
HM02
Lu1
melanoma (cell).

HMC-1
hmn leukemic mast cells.
LXFL529L
HMEC
hmn microvascular endothelial cells.
M1
hmn large cell lung cancer (cell).
mus myelocytic leukemia (cell).
HO-8910
M14
HOG.R5
green fluorescent protein (GFP)-based reporter cell.
M4BEU
HONE-1
M5076
HOP-62
non-small cell lung cancer (cell).
Ma7373
Hs578T
MALME-3M
Hs740T
MBT-2
mus bladder cancer (cell).
Hs742T
MCF7
Hs756T
MCF7/6
HSC-2
hmn oral squamous cell carcinoma cells.
HSG
HT
hmn salivary gland tumor (cell).

sarcoma (cell).
HT1080
HT29
HT3
MCF7-ras
MDA231
hmn telomerase reverse transcriptase-retinal pigment
hmn umbilical vein endothelial cell.

hmn T-cell leukemia (cell).

hmn leukemia (cell) of adriamycin-resistent.

MDCK
Madin-Darby Canine.
MEL-28
hmn melanoma cell.
Meth-A
Meth-A sarcoma (cell).
MGc803
MI4
mus leukemia (cell).

melanoma (cell).
MIA-PaCa-2
MK1
MKN45
MKN7
MDR nasopharyngeal carcinoma (cell).
KB-VIN
vincristine-resistant nasopharyngeal carcinoma (cell).
MKN28

MKN74
MM1

highly invasive clone isolated from parental rat ascites hepatoma
AH130 cells.
Ketr3
Molt4
KG-1
Mono-Mac-6
KM12
KM20L2

hmn pancreas cancer (cell).
MKN1
KB16
hmn gastric adenocarcinoma (cell).
MH-60
KB15
KBV200

K562/ADM
KB3
Jurkat-T
KB
MCF7/ADR-RES
MDA-MB-435
hmn hepatoma (cell).
Kato3
melanoma (cell).
MDA-MB-231
epithelial cells.
K562
hmn fibrosarcoma (cell).
hTERT-RPE1
HUVEC

ovarian sarcoma (cell).

Huh7
melanoma (cell).
MQc80-3
MRC-5
hmn lymphoma (cell).

mononuclear cells.
gastric adenocarcinoma (cell).

hmn diploid embryonic cells.
xxxi
MS301
SF268
hmn brain tumor (cell).
MS310
SF295
N04
hmn neuroma (cell).
NCI-H1417
hmn small cell lung cancer (cell).
SF539
SGC
NCI-H187
hmn small cell lung cancer (cell).
SGC7901
NCI-H226
SiHa
NCI-H23
SKBR3
NCI-H460
SKCO1
NCI-H522
SK-MEL
NK/LY
ascites cancer (cell).
NSCLC-N6
NUGC
hmn caucasian melanoma (cell).
SK-MEL-2
SK-MES-1
NUGC-4
SK-OV-3
ovarian adenocarcinoma (cell).
SK-MEL-5
NUGC-3
OVCAR-2780
SK-MEL-28

bronchogenic carcinoma cell.
SMMC-7721
OVCAR-3
SNB75
OVCAR-4
SNB78
OVCAR-5
SNU638
OVCAR-8
SR
leukemia (cell).
St4
gastric cancer (cell).
P1534
P388
mus, transplanted leukemia (cell).

mouse lymphocytic leukemia (cell).
P388/ADM
mouse lymphocytic leukemia (cell) of adriamycin-resistent.
PACA-2
hmn pancreas cancer (cell) .
SVR
mouse endothelial cells.
SW620
T24

PANC1
T24S
PBMC
peripheral blood mononuclear cells.
T47D
T98G
hmn caucasian gioblastoma (cell).
TK10
PC12
PC3

PC-6
PLC/PRF/5
PSN1
hmn pancreas cancer (cell).
PTX10
ovarian cancer cells with -tubulin mutation.
QGY-7703
RAW264.7
RBL-2H3
RL33
RXF-393
RXF-631L

mouse cervical carcinoma (cell).
U251
brain tumor (cell).
U373
caucasian gioblastoma (cell).
U4
mouse macrophages.
U-87-MG
rbt lung cancer (cell).
RPMI-8226
U14

rat basophilic cells.
RPMI-7951
Tmolt3
mouse cervical carcinoma (cell).
U937
caucasian gioblastoma (cell).
hmn monocytic leukemia (cell).
UACC62
melanoma (cell).
melanoma (cell).
UO-31
leukemia (cell).
Vero
green monkey kidney tumour (cell).
W256
rat Walker sarcoma (cell).
WEHI-164
mus fibrosarcoma (cell).
S180
mouse sarcoma (cell).
WHCO1
S37
mouse sarcoma (cell).
WI-38
hmn lung fibrocyte (normal hmn diploid fibrocyte).
WiDr
colorectal adenocarcinoma (cell).
Wish
transformed epithelial tumour (cell).
Sca7901
SCL
SCL-37'6
SCL-6
SCL-9
XF-498
ZR-75-1
hmn esophageal cancer (cell).
hmn tumor (cell).

Volume 2
Isolated Compounds (D-G)
J. Zhou et al., Encyclopedia of Traditional Chinese Medicines Molecular Structures, Pharmacological Activities, Natural Sources
and Applications: Vol. 2: Isolated Compounds D-G, DOI 10.1007/978-3-642-16738-6, Springer-Verlag Berlin Heidelberg 2011
4600 Dahuribirin D
C32H28O10 (572.57). Colorless viscous oil, []D24 = 0.22 (c = 0.65,

dioxane). Source: BAI ZHI Angelica dahurica [Syn. Angelica
4595 Dactylyne
C14H17Br2ClO (396.55). mp 62~63C, []D25 = 38.2 (c = 0.19, CHCl3).
porphyrocaulis]. Ref: 4118.

O
Source: Laurencia sp., Aplysia dactylomela. Ref: 2306.

Br
Cl
Br
O
O
O
O
O
O
4596 Daechu alkaloid A
C10H13NO2 (179.22). Source: WU CI ZAO Ziziphus jujuba var. inermis.

Ref: 660.
4601 Dahuribirin E
C32H30O11 (590.59). Colorless viscous oil, []D24 = +4.6 (c = 0.62,
OH
HO
4597 Dahuribirin A
O
O
O
O
O
O
O
4602 Dahuribirin F

4598 Dahuribirin B
O
O
O
O
OH
O
O
O
O
OH
HO
4603 Dahuribirin G
C34H34O13 (650.64). Colorless viscous oil, []D24 = +5.2 (c = 0.54,
4599 Dahuribirin C
31
C33H30O11 (602.60). Colorless viscous oil, []D = +20.0 (c = 0.48,
O
O
O
O
O
O
O
O
O
H
O
OH
O
OH
O
4604 Daidzein
4606 Daidzin
4',7-Dihydroxyisoflavone [486-66-8] C15H10O4 (254.24). Pharm:
Daidzoside [552-66-9] C21H20O9 (416.39). Source: DA DOU Glycine max
Antifungal; antispasmodic (mus small intestine); CVS activity (enhances
(Soybean phytochemical concentrate: yield = 0.0074%dw)[4630], E MEI
collateral circulation and oxygen consumption upon lack of blood in
GE Pueraria omeiensis (root: content = 1.0 5%) [5508], FEN GE Pueraria
myocardium); estrogenic activity ; increases coronary flow (narcosis dog);
lobata var. thomsonii (root: content = 1.51%)[5508], GAN GE TENG GEN
lipase inhibitor; anti-inflammatory (NO production inhibitor)
[4415]
Pueraria thomsonii (root: content = 0.158%[5508]), GE GEN Pueraria
cytotoxic (KB, IC50 > 75mol/L, Helenalin, IC 50 =
lobata [Syn. Pueraria thunbergiana; Pueraria pseudohirsuta] (root:
(0.640.08)mol/L, Melphalan, IC50 = (6.00.5)mol/L; Mono-Mac-6,
content = 0.78%[5508]), SAN LIE YE GE Pueraria phaseoloides (root:
IC50 > 75mol/L, Helenalin, IC50 = (3.10.3)mol/L; Jurkat-T, IC 50 >
content = 0.72%)[5508], SHI YONG GE Pueraria edulis (root: content =
75mol/L, Helenalin, IC 50 = (1.140.08)mol/L, Melphalan,
0.44%)[5508]. Ref: 2, 660, 4630, 5508.
IC50 = (9.10.8)mol/L)
[5077]
; antibacterial (Staphylococcus aureus,
MIA = 1.00g, Chloramphenicol, MIA = 0.0001g; Bacillus subtilis,

O
MIA = 5.00g, Chloramphenicol, MIA = 0.0001g)[5247]; antifungal
OH
(Candida mycoderma, MIA = 0.05g, control Miconazole, MIA =

0.0001g)[5247]; antioxidant (DPPH scavenger, TLC, MIA = 0.1g, IC50 =
380g/mL; control Quercetin, MIA < 0.05g, IC50 = 7g/mL, Gallic acid,
MIA < 0.05g, IC50 = 4g/mL; Ascorbic acid, MIA < 0.10g, IC50 =
18g/mL)[5247]. Source: DA DOU Glycine max (Soybean phytochemical
concentrate: yield = 0.0058%dw)[4630], E MEI GE Pueraria omeiensis
(root: content = 0.055%)[5508], FEN GE Pueraria lobata var. thomsonii
(root: mean content of 2 origins = 0.035%)[5508], GE GEN Pueraria lobata
[Syn. Pueraria thunbergiana; Pueraria pseudohirsuta] (root: mean
content of 10 origins = 0.137%
[5508]
), HEI DA DOU Glycine max, HONG
CHE ZHOU CAO Trifolium pratense, HUANG HUA MU Piptanthus

nepalensis, HUANG MAO GE Pueraria calycina (root: content =
HO
OH
OH
OH
4607 Dalbergenone
[2543-95-5] C16H14O3 (254.29). mp 114~116C. Source: JIANG ZHEN
XIANG Dalbergia odorifera. Ref: 6.
O
0.030%)[5508], JI KUAN CI TONG Erythrina latissima (stem wood), MU

XU Medicago sativa, SAN LIE YE GE Pueraria phaseoloides (root:
content = 0.090%)[5508], SAN XIAO CAO Trifolium repens, SHAN DOU
GEN Sophora subprostrata [Syn. Sophora tonkinensis], SHI YONG GE
Pueraria edulis (root: content = 0.063%)[5508], SI TE WEN HUANG TAN
4608 Dalbergichromene
Dalbergia stevensonii, YUN NAN GE TENG Pueraria peduncularis
7-Methoxy-4-phenyl-2H-1-benzopyran-6-ol [32066-31-2] C16H14O3
(root: content = 0.053%)[5508], Bituminaria morisiana (leaf). Ref: 2, 4,
(254.29). mp 99~100C. Source: JIANG ZHEN XIANG Dalbergia
658, 660, 4415, 4630, 5077, 5247, 5508.
odorifera. Ref: 6.
O
HO
HO
4609 Dalbergin
OH
6-Hydroxy-7-Methoxy-4-phenylcoumarin [482-83-7] C16H12O4 (268.27).

mp 210C. Pharm: CVS activity (increases coronary flow and slows heart
4605 Daidzein 4',7-diglucoside
rate, perfused heart of rbt in vitro). Source: FEI ZHOU HUANG TAN
C27H30O14 (578.53). Source: GE GEN Pueraria lobata [Syn. Pueraria
Dalbergia melanoxylon, HE AN HUANG TAN Dalbergia riparia,
thunbergiana; Pueraria pseudohirsuta] (root: mean content of 7 origins =
JIANG ZHEN XIANG Dalbergia odorifera, JIAO ZHI HUANG TAN
0.453%[5508]), GAN GE TENG GEN Pueraria thomsonii. Ref: 2, 660,
Dalbergia cochinchinensis (stem: yield = 0.0024%dw)[4716], SI TE WEN
5508.
HUANG TAN Dalbergia stevensonii, XI A LA HUANG TAN Dalbergia

cearensis, XIAO DAO XING HUANG TAN Dalbergia cultrata, YIN DU
HO
OO
OH
HUANG TAN Dalbergia sissoo. Ref: 6, 658, 4716.
OH
OH
HO
OH
OH
OH
HO
4610 Dalbergiphenol
4614 Damascenine
C17H18O3 (270.33). Pharm: Testosterone 5-reductase inhibitor (25g/mL,
[483-64-7] C10H13NO3 (195.22). Pharm: Anti-inflammatory (rat, swollen
InRt = 8.2%, 50g/mL, InRt = 18.9%, 100g/mL, InRt = 51.8%; control
foot model); antipyretic. Source: YE HEI ZHONG CAO Nigella arvensis,
Glycyrrhetinic acid, 25g/mL, InRt = 31.7%, 50g/mL, InRt = 64.7%,
HEI ZHONG CAO Nigella damascena. Ref: 658.
100g/mL, InRt = 87.1%). Source: JIAO ZHI HUANG TAN Dalbergia

cochinchinensis (stem: yield = 0.0074%dw). Ref: 4716.
O
H
N
O
HO
4615 Dambonitol
[532-94-4] C8H16O6 (208.21). mp 210C. Source: JIA ZHU TAO Nerium
indicum, LUO SHI TENG Trachelospermum jasminoides. Ref: 6.
4611 Daldinin C
C22H26O9 (434.45). Pharm: Antioxidant (DPPH scavenger, IC50 =

412.0mol/L, control Ascorbic acid, IC50 = 16.5mol/L). Source: AN
ZONG TAN TUAN JUN Hypoxylon fuscum. Ref: 3771.
OH
OH
OH
4616 Dammara-20,24-dien-3-ol
[20460-34-8] C30H50O (426.73). mp 136~138C. Source: WU YUE CHA
HO
Antidesma bunius. Ref: 6.
O
O
O
OH
O
OH
H
4612 Daldinin E
H
HO
(2E,4E)-Hexa-2,4-dienoic
acid,2-methyl-7S-(acetyloxy)-3',4,4',5',6,6',7,8-octahydro-3'-hydroxy-6',7dimethyl-6,8-dioxospiro[3H-2-benzopyran-3,2'-[2H]pyran]-4-yl ester
4617 Dammar-20(21),24-diene-3,6,12-triol
C24H28O9 (460.49). Oil, []D20 = +87.7 (c = 0.3, CHCl3). Pharm:
C30H50O3 (458.73). Colorless fascicular crystals (MeOH), mp 145~148C.
Antioxidant (DPPH scavenger, IC50 = 178.9mol/L, control Ascorbic acid,
Source: XI YANG SHEN JING YE Panax quinquefolium. Ref: 4874.
IC50 = 16.5mol/L). Source: AN ZONG TAN TUAN JUN Hypoxylon

fuscum. Ref: 3771.
OH
HO
HO
O
O
OH
O
OH
4618 Dammar-24-ene-3,20-diol I
[19132-83-3] C30H52O2 (444.75). mp 142~144C. Source: MANG GUO
SHU PI Mangifera indica. Ref: 6.
4613 Daldinin F
HO
(2E,4E)-Hexa-2,4-dienoic
acid,4-methyl-7S-(acetyloxy)-3',4,4',5',6,6',7,8-octahydro-3'-hydroxy-6',7dimethyl-6,8-dioxospiro[3H-2-benzopyran-3,2'-[2H]pyran]-4-yl ester
C24H28O9 (460.49). Oil, []D20 = +28.9 (c = 0.4, CHCl3). Pharm:
Antioxidant (DPPH scavenger, IC50 = 212.3mol/L, control Ascorbic acid,
H
HO
IC50 = 16.5mol/L). Source: AN ZONG TAN TUAN JUN Hypoxylon
4619 20(S)-Dammar-23-ene-25-hydroperoxyl-3,6,12,20-tetrol
fuscum. Ref: 3771.
C30H52O6 (508.75). White crystalline powder, mp 142~145C. Source: XI

YANG SHEN JING YE Panax quinquefolium. Ref: 4874.
HO
OH
HO
O
O
O
O
O
OH
HO
OH
OH
4620 20(S),24(S)-Dammar-25(26)-ene-3,6,12,20,24-pentanol
4626 Danmelittoside
C30H52O5 (492.75). White crystalline powder, mp 142~144C. Source: XI
Monomelittoside C15H22O10 (362.34). Source: GAN DI HUANG
YANG SHEN JING YE Panax quinquefolium. Ref: 4874.
Rehmannia glutinosa [Syn. Rehmannia glutinosa f. huechingensis], OU
OH
ZHOU MI FENG HUA Melittis melissophyllum. Ref: 2, 1521.
HO
OH
OH
OH
HO
O
HO
HO
OH
H
OO
OH
OH
4621 20(S)-Dammar-25(26)-ene-3,6,12,20-tetrol
OH
C30H52O4 (476.75). Colorless fascicular crystals (MeOH), mp 259~260C.
4627 Danshenol A
Source: XI YANG SHEN JING YE Panax quinquefolium. Ref: 4874.
[189308-08-5] C21H20O4 (336.39). Taupe acicular crystals, mp 182C

(methanol), []D25 = 136.4 (c = 0.07, chloroform). Pharm: Aldose
reductase inhibitor (rat eye lens, IC50 = 0.1mol/L). Source: DAN SHEN
HO
OH
Salvia miltiorrhiza. Ref: 993.

O
O
HO
HO
O
OH
4622 Damnacanthal
[477-84-9] C16H10O5 (282.26). mp 208C. Source: HU CI Damnacanthus
indicus, TU LIAN QIAO Hymenodictyon excelsum. Ref: 6.
O
4628 Danshenol B
[189308-09-6] C22H26O4 (354.45). Yellow acicular crystals, mp 176C
O
O
OH
(methanol), []D25 = 131.6 (c = 0.10, chloroform). Pharm: Aldose

reductase inhibitor (rat eye lens, IC50 = 1.75mol/L). Source: DAN SHEN
Salvia miltiorrhiza. Ref: 993.
O
O
4623 Damnacanthol
[477-83-8] C16H12O5 (284.27). mp 288C. Source: HU CI Damnacanthus
HO
indicus. Ref: 6.
O
O
OH
OH
4629 Danshenspiroketallactone
[100414-80-0] C17H16O3 (268.32). White acicular crystals, mp 203~205C.
Source: DAN SHEN Salvia miltiorrhiza, GAN XI SHU WEI CAO Salvia
4624 Damsin
przewalskii. Ref: 38, 4538.
2,3-Dihydroambrosin [1216-42-8] C15H20O3 (248.32). mp 109~111C;

124~125C. Pharm: Schistosomacide; cytotoxic (KB, ED50 > 100g/mL);
molluscacide. Source: PU TONG TUN CAO Ambrosia ambrosioids,

TUN CAO Ambrosia artemisiifolia. Ref: 4, 658.
O
O
4630 Danshensu
[76822-21-4] C9H10O5 (198.18). White, long acicular crystals, mp
84~86C; sodium salt: white acicular crystals, mp 255~258C, []D20.5 =
+35 (water); []D27.5 = +14.8 (1N HCl). Pharm: Coronary vasodilator

O
(pig isolated coronary artery, 1.0g/mL, also against coronary contraction
4625 Damsinic acid
induced by morphine or propranolol)[5501]; increases tolerance to anoxia
[22844-19-5] C15H22O4 (266.34). mp 112~113C. Source: TUN CAO
(mouse ip300mg/kg or 50mg/kg, clearly extends survival time)[5501];
Ambrosia artemisiifolia. Ref: 1521.
anti-ischemia myocardial (rat im 20mg/kg, ischemia myocardial induced

by hypophysin)[5501]; anti-myocardial infarction (dog im 8mg/kg, rbt im
HO
10mg/kg)[5501]; antioxidant (strong O2 superoxide anion scavenger,

O
OH
protects myocardial ischemia-reperfusion injury in rat myocardium

mitochondrial membrane)[5501]; improves barrier of microcirculation (rbt
iv in ear 4~6mg/kg, induced by macromolecular dextran; mouse drop iv
1mg/0.1mL, induced by arterenol in mesentery)[5501]; platelet aggregation
4635 Danshenxinkun D
inhibitor (rbt iv in ear 20mg/kg; rat iv 100mg/kg; in vitro 5~600g/mL,
C21H20O4 (336.39). Pink acicular crystals, mp 178~180C. Source: DAN
[5501]
distinctly inhibits platelet aggregation induced by ADP or thrombin)
SHEN Salvia miltiorrhiza. Ref: 34.
Source: DAN SHEN Salvia miltiorrhiza (dried root: mean content =
0.664%)[5508] Ref: 661, 5501, 5508.
H OH
OH
OH
O
HO
HO
4636 Dantaxusin A
4631 Danshensuan B
5-Cinnamoyloxy-2,7,13-triacetoxy-2(320)abeo-taxa-4(20),11-dien
Salvianolic acid B [115939-25-8] C36H30O16 (718.63). Amorphous
e-9,10-dione C35H40O10 (620.7). Colorless amorphous powder, mp
yellowish powder, []D18 = +92 (c = 0.07, ethanol). Pharm: Free radical
114~116C, []D27 = +12 (c = 0.33, MeOH). Source: YUN NAN HONG
scavenger; fibrinolytic function; increases coronary flow; antioxidant
DOU SHAN Taxus yunnanensis (aerial parts). Ref: 3079.
(inhibits lipid peroxidization strongly, induced by vitamin Cnicotinamide ADP and Fe2+-cysteine in microsome of murine cerebral,
O
O
hepatic and renal cells); main component of phenol character acid in

Salvia miltiorrhiza. Source: DAN SHEN Salvia miltiorrhiza. Ref: 2, 900.
OH
HO
OH
O
O
H
HO
OH
O
O
O
HO
HO
O
O
OH
4637 Dantaxusin B
OH
C33H42O7 (550.7). Colorless amorphous powder, mp 245~246C, []D27 =
5-Cinnamoyloxy-9-hydroxy-10,13-diacetoxytaxa-4(20),11-diene
4632 Danshenxinkun A
8 (c = 0.33, MeOH). Source: YUN NAN HONG DOU SHAN Taxus

yunnanensis (aerial parts). Ref: 3079.
Neotanshinone A; Tanshiquinone A C18H16O4 (296.33). Pharm:
Antibacterial (Mycobacterium tuberculosis H37Rv, MIC = 0.78g/mL).
OH
Source: DAN SHEN Salvia miltiorrhiza. Ref: 658, 1285.

OH
OH
O
O
4638 Dantaxusin C
C37H44O12 (680.76). Colorless amorphous powder, mp 122~123C, []D24
= +1.25 (c = 0.33, MeOH). Source: YUN NAN HONG DOU SHAN
4633 Danshenxinkun B
Taxus yunnanensis (aerial parts). Ref: 4611.
Neotanshinone B; Tanshiquinone B C18H16O3 (280.33). Pharm:

O
O
O O
OH
O
H
H O
O
4639 Dantaxusin D
C37H46O11 (666.77). Colorless amorphous powder, mp 111~112 C, []D24
4634 Danshenxinkun C
= +6.88 (c = 0.33, MeOH). Source: YUN NAN HONG DOU SHAN
Neotanshinone C; Tanshiquinone C C16H12O3 (252.27). Pharm:
Taxus yunnanensis (aerial parts). Ref: 4611.

O
OH
O
O OH
O
O
O
H
H O
O
4640 Daphcalycinosidine C
4645 Daphnetin
C38H49NO12 (711.81). Colorless amorphous solid, []D22 = 15 (c = 0.6,
7,8-Dihydroxycoumarin [486-35-1] C9H6O4 (178.15). mp 257~258C;
MeOH). Source: NIU ER FENG ZI Daphniphyllum calycinum (fruit:
263~264C. Pharm: Analgesic; antibacterial (Staphylococcus aureus,
yield = 0.00042%). Ref: 4754.
Bacillus coli, Shigella flexneri and Bacillus pyocyaneus);

O
OH
anti-inflammatory; anti-ischemia, myocardial; immunomodulator (inhibits

immune response of specific cells and that of body fluid, but enhances
phagocytotic function of enterocelia Mphi macrophage); improves

O
O
HO
O
HO
H HO
H
O
myocardium metabolism and promotes restoration of myocardial function;

increases coronary flow; reduces consumption of oxygen in myocardium;
OH
sedative; LD50 (mus, ip) = 429mg/kg, (mus, iv) = 375mg/kg, (mus, orl) =
5.37g/kg. Source: HUI HUI DOU Cicer arietinum, LANG DU Stellera
chamaejasme, QIAN JIN ZI Euphorbia lathyris, RUI XIANG HUA

N
Daphne odora. Ref: 4, 6, 556, 658, 5501, 5507.

H
4641 Daphneligin
C21H26O6 (374.44). Amorphous powder, mp 136~138C, []D = +11.5 (c

= 0.10, CHCl3) Source: YOU RUI XIANG Daphne oleoides. Ref: 1883.
HO
OH
O
O
4642 Daphneolone
O
HO
OH
4646 Daphnetin-8-glucoside
[20853-56-9] C15H16O9 (340.29). mp 223~224C. Source: RUI XIANG
HUA Daphne odora. Ref: 6.
HO
[54835-64-2] C17H18O3 (270.33). Source: RUI XIANG GEN Daphne
HO
OO
OH
odora. Ref: 6.
OH
OH
4647 Daphnetin-7-methyl ether
OH
[19492-03-6] C10H8O4 (192.17). mp 175.5C. Source: BA XIAN HUA

Hydrangea macrophylla. Ref: 6.
OH
O
O
4643 Daphneticin
[83327-22-4] C20H18O8 (386.36). Pharm: Cytotoxic (W256). Source:
SHAN GAN RUI XIANG Daphne tangutica, AO YE RUI XIANG
Daphne retusa. Ref: 658.
OH
4648 Daphnetin-8-methyl ether

Hydrangetin [485-90-5] C10H8O4 (192.17). Needles (C6H6), mp 152C,
mp 157~157.5C, mp 185C. Pharm: Cytotoxic inactive (in vitro,
HONE-1 and NUGC cancer cell lines, no significant activity)[3069]. Source:
BA XIAN HUA Hydrangea macrophylla, QING HAO Artemisia apiacea

[Syn. Artemisia carvifolia; Artemisia caruifolia], QUAN YUAN YE HUA
JIAO Zanthoxylum integrifoliolum, ZHONG GUO XIU QIU Hydrangea

HO
OH
O
chinensis (root)[3069]. Ref: 6, 2176, 3069.

O
4644 Daphneticin-4''-O--D-glucopyranoside
C26H28O13 (548.51). mp 254~255C, []D = +23.5 (c = 0.10, DMSO).

Source: YOU RUI XIANG Daphne oleoides. Ref: 2279.
HO
HO
4649 Daphnetoxin
OH
OH
HO
[28164-88-7] C27H30O8 (482.54). Pharm: LD50 (mus, orl) = 0.25mg/kg.
Source: OU YA RUI XIANG Daphne mezereum. Ref: 658.
OH
O
O
HO
O
O
HO
OH
4650 Daphnin
4655 Daphnodorin H 3-methyl ether
Daphnetin-7-glucoside [486-55-5] C15H16O9 (340.29). mp 215C (dec).
C31H24O11 (572.53). Yellow amorphous powder. Source: YUAN HUA
Source: RUI XIANG HUA Daphne odora, SU MI Setaria italica. Ref: 6.
GEN Daphne genkwa. Ref: 4868.

HO
HO
OO
OH
OH
OH
OH
O
O
OH
HO
OH
OH
O
4651 Daphnodorin B
[95733-02-1] C30H22O10 (542.50). Source: LIAO GE WANG GEN
OH
Wikstroemia indica, RUI XIANG GEN Daphne odora. Ref: 2268, 1521.
4656 Daphnodorin H 3''-methyl ether
OH
C31H24O11 (572.53). Pale yellowish powder. Source: YUAN HUA GEN

Daphne genkwa. Ref: 4868.
HO
OH
OH
HO
OH
OH
O
O
OH
HO
OH
OH
4652 Daphnodorin G
OH
C30H22O11 (558.50). Source: YUAN HUA GEN Daphne genkwa. Ref:
OH
4868.
4657 Daphnoretin
HO
[2034-69-7] C19H12O7 (352.30). Yellow flossy, tiny acicular crystals

OH
HO
(ethanol) or yellow short, thick acicular crystals (acetonepyridine), mp

250~252C, 244~247C; yellow acicular crystals (tetrahydrofuran
O
OH
OH
O
methanol). Pharm: Antineoplastic. Source: LIAO GE WANG GEN

Wikstroemia indica, JING YA MA YE RUI XIANG Daphne gnidium. Ref:
661.
OH
OH
HO
4653 Daphnodorin G-3''-methyl ether

C31H24O11 (572.33). Yellow amorphous powder. Source: YUAN HUA
O
O
GEN Daphne genkwa. Ref: 4868.

4658 Daphnoretin methyl ether
HO
7-Methoxydaphnoritin C20H14O7 (366.33). Fine acicular crystals, mp

238~240C, soluble in methanol, ethanol, and insoluble in chloroform,
OH
O
HO
ether, and acetone. Source: LANG DU Stellera chamaejasme. Ref: 488.
OH
OH
OH
[14260-99-2] C19H26O12 (446.41). Source: JI SHI TENG Paederia
C30H22O11 (558.50). Source: YUAN HUA GEN Daphne genkwa. Ref:

4868.
scandens, JIAO RANG MU Daphniphyllum macropodum, XIE JI CU YE

MU Lasianthus wallichii (leaf). Ref: 1521, 2561, 4238.
O
HO
HO
OH
HO
O
OH
HO
OH
OH
OH
OH
O
4659 Daphylloside
4654 Daphnodorin H
OH
OH
10
4660 Darlinine
4666 Daturametelin A
[73069-56-4] C15H21NO (231.34). Straw-coloured crystals (EtOH), mp
C34H48O9 (600.76). Source: MAN TUO LUO YE Datura metel. Ref: 2,
59~61C, []D19 = +75 (CHCl3). Source: Darlingia darlingiana. Ref:
660.
1521.
O
H
N
OH
OH
C20H34O3 (322.49). Source: XI XIAN Siegesbeckia orientalis (aerial
O
O
OH
4661 Darutigenol
O
HO
OH
parts). Ref: 4438.

HO H
4667 Daturametelin B
OH

660.
H
HO
4662 Darutoside
HO
Darutin C26H44O8 (484.64). Source: XI XIAN Siegesbeckia orientalis
(aerial parts). Ref: 4438.

HO
O
H HO
OH
O
O
OH
OH
OH
4668 Daturametelin C
H
OO
HO
OH
OH
[123297-25-6] C29H40O5 (468.64). Source: MAN TUO LUO YE Datura

metel. Ref: 2, 660.
OH
4663 Dasycarpamine
HO
C17H21NO4 (303.36). mp 149C. Source: BAI XIAN PI Dictamnus
dasycarpus. Ref: 6.
OH
4669 Daturametelin E
C29H42O9S (566.72). Source: MAN TUO LUO YE Datura metel. Ref: 2,

660.
4664 Datumetelin
metel. Ref: 2.
HO
O
O
H
O
OH
O S O
4670 Daturametelin F
4665 Datumetine
C28H38O8S (534.67). Source: MAN TUO LUO YE Datura metel. Ref: 2,
[67078-20-0] C16H21NO3 (275.35). Source: MAN TUO LUO YE Datura
660.
metel. Ref: 2.
O
N
O
O
O
OH
O S O
O
H
H
11
4671 Daturametelin G-AC
4676 Daucic acid
[34098-52-7] C7H8O7 (204.14). Source: HE SHI FENG Daucus carota.
660.
Ref: 6.
OH
HO
O
O
O
O
OH
OH
4677 Daucoidin A
C19H20O6 (344.37). Yellowish glasses, []D20 = +46 (c = 0.30, MeOH).
Source: QIAN HU Angelica decursiva [Syn. Peucedanum decursivum].
O
O
O
Ref: 9.
4672 Daturic acid

O
DANG SHEN Codonopsis pilosula, LU HUI Aloe vera [Syn. Aloe

barbadensis], GAN DI HUANG Rehmannia glutinosa [Syn. Rehmannia
Margaric acid [506-12-7] C17H34O2 (270.46). mp 60~61C. Source:
OH
glutinosa f. huechingensis], XI YANG SHEN Panax quinquefolium, SHU

MI Panicum miliaceum. Ref: 2, 6.
4678 Daucoidin B
C19H20O6 (344.37). Colorless massive crystals, mp 140~141C, [] D20 =
+48.2 (c = 0.15, CHCl3). Source: QIAN HU Angelica decursiva [Syn.

Peucedanum decursivum]. Ref: 9.
HO
4673 Daturilin
Withametelin [113430-43-6] C28H36O4 (436.60). Source: MAN TUO
H
O
OH
4679 Daucol
[887-08-1] C15H26O2 (238.37). mp 113~115C, bp 124~132C/2mmHg.
LUO YE Datura metel. Ref: 2, 660, 1521.
Source: HU LUO BO ZI Daucus carota var. sativa, NAN HE SHI
Daucus carota, HE SHI FENG Daucus carota. Ref: 6, 660.
OH
O
4674 Daturilinol
4680 Daucosterol
metel. Ref: 2, 660.
-Daucosterol [474-58-8] C35H60O6 (576.86). White powder, mp 295C.

OH
O
O
O
H
H
H
Pharm: Platelet aggregation inhibitor (2~5mg/mL collagen-induced, IC50

= (1143)mol/L, control ASA, IC 50 = (4203)mol/L; 1~4mol/L
epinephrine-induced with 0.8~1.0mg/mL collagen, IC50 =
(53.22.3)mol/L, ASA, IC50 = (53.04.5)mol/L; 10~40mol/L
Sodium arachidonate-induced with 0.8~1.0mg/mL collagen, IC50 =
(66.54.0)mol/L, ASA, IC 50 = (66.02.1)mol/L; 1~5mol/L
PGH2/TXA2 receptor agonist U46619-induced with 0.8~1.0mg/mL
collagen, IC50 = (56.14.3)mol/L, ASA, IC 50 =
(34012)mol/L) [4994]; cytotoxic (P388, marginal activity); cytotoxic
4675 Daucene
inactive (in vitro, LNCaP, IC50 > 100mol/L)[4607]. Source: BAI MU
4,8-Daucadiene [16661-00-0] C15H24 (204.36). bp 96C/4mmHg. Source:
TONG GEN Akebia trifoliata var. australis, BAI TOU WENG Pulsatilla
NAN HE SHI Daucus carota. Ref: 6, 660.
chinensis, BAN XIA Pinellia ternata, BEI MA DOU LING GEN

Aristolochia contorta, BU GU ZHI Psoralea corylifolia, CAO CONG
RONG Boschniakia rossica, CHI SHAO Paeonia lactiflora wild,
CHUAN XIN LIAN Andrographis paniculata [Syn. Justicia paniculata],
CHUAN XU DUAN Dipsacus asperoides, CI WU JIA Acanthopanax
senticosus [Syn. Eleutherococcus senticosus], DAN SHEN Salvia
12
miltiorrhiza, DIAN NAN HONG HOU KE Calophyllum polyanthum
4682 Daurichromene B
(seed: yield = 0.0027%dw)[4767], DONG BEI CI REN SHEN Oplopanax
2R-(3'-Hydroxy-8'-methyl-4'-methyliden-7'-nonaenyl)-5-hydroxy-2,7-dim
elatus, FANG FENG Saposhnikovia divaricata [Syn. Ledebouriella
ethyl-2H-chromene C22H30O3 (342.48). Light yellow oil, []D26 = 27.7
seseloides], FANG XIANG JIANG Zingiber aromaticum (rhizome), GAN
(c = 0.13, CH3OH). Pharm: Antihistamine (inhibits histamine release, rat
DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa f.
peritoneal mast cells, compound 48/80-induced)[4755]. Source: MAN
huechingensis], GE GEN Pueraria lobata [Syn. Pueraria thunbergiana;
SHAN HONG Rhododendron dauricum (twig and leaf: yield = 0.0001%)
Pueraria pseudohirsuta], HAI JIN BI XIE Dioscorea spongiosa (rhizome:
Ref: 4755.
yield = 0.00012%)[4692], HUA DONG LAN CI TOU Echinops grijsii,

HUANG HUA BAI JIANG Patrinia scabiosaefolia, HUO XIANG
OH
Agastache rugosus, HUO YAN HUA Phlogacanthus curviflorus (root:

yield = 0.0385%dw)[4799], JIN QUE GEN Caragana sinica, JU YUAN
O
Citrus medica, LANG DANG ZI Hyoscyamus niger (seed: yield =

0.0004%dw)
[4607]
OH
, LIU QIU SHE GEN CAO Ophiorrhiza liukiuensis
(whole herb), MA TI YE Caltha palustris, MAO LIAN HAO Artemisia
4683 Daurichromene C
vestita, MU TONG Akebia quinata, MU TONG GEN Akebia quinata,
2R-(8'-Hydroxy-4',8'-dimethyl-3'E,6'Z-nonadienyl)-5-hydroxy-2,7-dimeth
REN SHEN Panax ginseng [Syn. Panax schinseng], ROU CONG RONG
yl-2H-chromene C22H30O3 (342.48). Light yellow oil, []D26 = 32.0 (c =
Cistanche deserticola, SAN QI Panax pseudo-ginseng var. notoginseng
0.10, CH3OH). Pharm: Antihistamine (inhibits histamine release, rat
[Syn. Panax notoginseng], SAN YE MU TONG GEN Akebia trifoliata,
SHAN FAN GEN Symplocos caudata, SHENG DI HONG JING TIAN
Rhodiola sacra, SHI LIU ZHONG ZI Punica granatum (seed: yield =
Ref: 4755.
0.0051%)[4792], SI CHI SI LENG CAO Schnabelia tetradonta (aerial parts:

OH
yield = 0.00058%dw)[4665], SUAN ZAO REN Ziziphus jujuba var. spinosa,

TIAN MA Gastrodia elata, TUN XING GUO Pygeum topengii, WU
GENG WU JIA PI Acanthopanax sessiliflorus (fruit), XIA KU CAO
Prunella vulgaris, XIAN GENG XI XIAN Siegesbeckia orientalis var.

pubescens [Syn. Siegesbeckia pubescens], XIANG TANG SONG CAO
OH
Thalictrum foetidum, XIAO QIAO MU ZI JIN NIU Ardisia arborescens
4684 Daurichromene D
(whole herb)[4769], XIN JIANG LAN CI TOU Echinops ritro, YA DAN ZI
2R-(9'-Hydroxy-4',8'-dimethyl-3'E,7'E-nonadienyl)-5-hydroxy-2,7-dimeth
Brucea javanica [Syn. Brucea sumatrana; Rhus javanica], YAO YONG
yl-2H-chromene C22H30O3 (342.48). Light yellow oil, []D26 = 26.0 (c =
PU GONG YING Taraxacum officinale, YI ZHU QIAN MA Urtica
dioica, ZHONG GUO XUAN FU HUA Inula britannica var. chinensis,
occurs in many plants. Ref: 2, 440, 447, 450, 454, 455, 471, 474, 502, 556,
580, 582, 585, 594, 596, 614, 622, 660, 1521, 2508, 2535, 4449, 4527,
Ref: 4755.
4607, 4665, 4692, 4767, 4769, 4792, 4799, 4994, 5501.

OH
4685 Dauricine
OO
HO
OH
[524-17-4] C38H44N2O6 (624.78). mp 115C. Pharm: Analgesic;
OH
antiarrhythmic; anti-inflammatory; antihypertensive; platelet aggregation
OH
OH
inhibitor (caused by ADP, adrenalin, collagen and arachidonic acid, in

vitro and in vivo); inhibits small intestinal contraction (rbt, in vitro) and
4681 Daurichromene A
reduces alvine tension (in vivo); antihypercholesterolemic (reduces the
2R-(7'-Hydroxy-4',8'-dimethyl-3'E,8'-nonadienyl)-5-hydroxy-2,7-dimethy
level of cholesterol in serum); LD (cat, iv) = 30mg/kg; LD50 (mus, ip) =
l-2H-chromene C22H30O3 (342.48). Light yellow oil, []D26 = 30.4 (c =
6mg/kg. Source: BIAN FU GE GEN Menispermum dauricum, MEI GUO
BIAN FU GE Menispermum canadense. Ref: 4, 6, 658, 5501.

Ref: 4755.
OH
O
OH
OH
N
H
13
4686 Dauricinoline
[30984-80-6] C37H42N2O6 (610.76). Source: BIAN FU GE GEN
Menispermum dauricum. Ref: 6.
H2N
N
H
OH
O
N
4691 Daurioxoisoporphine C
6-Methylamino-5,9-dimethoxyoxoisoaporphine C19H16N2O3 (320.35).
OH
Yellow amorphous powder. Source: BIAN FU GE GEN Menispermum

dauricum. Ref: 3071.
4687 Dauricoline
OH
N
H
HO
N
N
H
O
4692 Daurioxoisoporphine D
OH
5,6-Dimethoxyl-9-hydroxyoxoisoaporphine C18H13NO4 (307.31). Yellow
4688 Daurinoline
amorphous powder. Source: BIAN FU GE GEN Menispermum dauricum.
Ref: 3071.
N
H
HO
O
N
H
O
O
OH
OH
4693 Daurisoline
4689 Daurioxoisoporphine A
[70553-76-3] C37H42N2O6 (610.76). Cream powder (cyclohexane), mp
4-Demethoxytyraminoporphine C26H22N2O4 (426.48). Yellow crystals
96~102C, []D20 = 129 (c = 0.65, methanol). Pharm: Muscle relaxant;
(CHCl3), mp 234~235C. Pharm: Cytotoxic (in vitro, A549, IC50 =
LD50 (mus, iv) = (1.250.16)mg/kg. Source: BIAN FU GE GEN
8.8mol/L, HL-60, IC50 > 50mol/L, MCF7, IC50 = 3mol/L, P388, IC50 =
Menispermum dauricum (rhizome: mean content of 8 origins =
30.5mol/L; control VP-16: A549, IC50 = 0.5mol/L, HL-60, IC50 =
0.594%[5508]) Ref: 661, 5501, 5508.
5.4mol/L, MCF7, IC50 = 12.33mol/L, P388, IC50 = 0.1mol/L). Source:

BIAN FU GE GEN Menispermum dauricum. Ref: 3071.
HO
O
N
N
H
OH
N
H
O
OH
4694 Davidigenin
O
4690 Daurioxoisoporphine B
C15H14O4 (258.28). Source: BO TE LAN DA JI Euphorbia portlandica

(whole herb). Ref: 5019.
6-Amino-4,5,9-trimethoxyoxoisoaporphine C19H16N2O4 (336.35). Yellow

OH
amorphous powder. Pharm: Cytotoxic (in vitro, A549, IC50 > 50mol/L,
HL-60, IC50 > 50mol/L, MCF7, IC50 = 6.2mol/L, P388, IC50 = 9.6mol/L;
control VP-16: A549, IC50 = 0.5mol/L, HL-60, IC50 = 5.4mol/L, MCF7,
IC50 = 12.33mol/L, P388, IC50 = 0.1mol/L). Source: BIAN FU GE GEN
HO
OH
14
4699 Davuricoside D
4695 Davidiol A
C42H32O9 (680.72). Colorless powder, []D29 = 272 (c = 0.18, MeOH).
3,16,29-Trihydroxy-13,28-epoxy-oleanane-3-O--D-glucopyranosyl-(1
Source: BAI CI HUA GEN Sophora viciifolia. Ref: 3935.
2)-(6-methyl ester)--D-glucuronopyranoside C43H70O15 (827.03).

White amorphous powder, mp 184~186C (MeOH), []D20 = 16.00 (c =
OH
0.01, pyridine). Source: HUANG LIAN HUA Lysimachia davurica

HO
H
HO
OH
H
H
HO
O
OH
HO
OH
O
OH
OH
OO
OH
OH
4696 Davidiol B
29
C42H34O10 (698.73). Brown solid, []D = 82 (c = 0.04, MeOH). Source:
OO
HO
OH
BAI CI HUA GEN Sophora viciifolia. Ref: 3935.
OH
OH
OH
4700 Davuricoside J
HO
O
H
HO
OH
-glucuronopyranosyl]-28-O--D-glucuronopyranoside C48H78O19 (959.15).

White amorphous powder, mp 229~232C (MeOH:H2O = 9:1), []D20 =
H OH
OH
3,16,28-Trihydroxy-olean-12-en-3-O-[-D-glucopyranosyl-(12)--D
20.79 (c = 0.04, pyridine). Source: HUANG LIAN HUA Lysimachia

davurica (whole herb). Ref: 4834.
HO
OH
OH
4697 Davidiol C
C56H40O12 (904.94). Brown powder, []D29 = 124 (c = 0.11, MeOH).
HO
Source: BAI CI HUA GEN Sophora viciifolia. Ref: 3935.
OH
OO
HO
HO
OH
HO
OH
OO
OH
OH
O H
HO
OH
OH
OH
OO
HO
OH
O
H
H H
H
H
O
OH
OH
OH
4701 Dawoensin A
C26H36O8 (476.57). mp 240~242C, []D26 = 34.3 (c = 1.40, MeOH);
[]D25.6 = 37.8 (c = 0.332, MeOH). Pharm: Cytotoxic (in vitro, BGC823

hmn tumor cells, IC50 = 3.54g/mL, control VCR, IC50 =
H
OH
0.066g/mL)[4760]; cytotoxic (hmn tumor K562 cells, IC50 = 2.0g/mL,

control cis-Platin IC50 = 1.1g/mL)[4955]. Source: BAO YE XIANG CHA
HO
CAI Isodon melissoides (aerial parts: yield = 0.00031%dw), DAO FU
4698 Davisioside
XIANG CHA CAI Isodon dawoensis, DONG LING CAO Rabdosia
C22H28O10 (452.46). White amorphous powder, []D = 69 (c = 0.48,
rubescens (leaf). Ref: 4067, 4299, 4760, 4955.
MeOH). Source: Globularia davisiana (aerial parts). Ref: 4194.

HO
HO
H
O
O
H
O
HO
OO
OH
OH
OH
H
O
O
O
15
4702 2'-Deacetoxyaustrospicatine
4707 2-Deacetoxytaxinine B
[119777-80-9] C39H53NO10 (695.86). Source: AO DA LI YA HONG DOU
C35H42O9 (606.72). Source: XI MA LA YA HONG DOU SHAN Taxus
SHAN Austrotaxus spicata, XI MA LA YA HONG DOU SHAN Taxus
wallichiana. Ref: 662.

O O

O
O O
O O
O
O
O
O
4708 2-Deacetoxytaxinine J
[119347-14-7] C37H46O10 (650.77). Colorless crystals, mp 171~172C

(ethanol), []D14 = +50 (c = 1.2, acetone). Pharm: Cytotoxic (P388 in vitro,
4703 2'-Deacetoxyaustrotaxine
IC50 = 15.2g/mL, L1210 in vitro, IC50 = 4.9g/mL, 10g/mL InRt = 79.5%,
SHAN Austrotaxus spicata. Ref: 662.
KB in vitro, 10g/mL InRt = 27.6%). Source: MEI LI HONG DOU SHAN
Taxus mairei, YUN NAN HONG DOU SHAN Taxus yunnanensis (aerial
O O
parts)[3079, 4611], ZI SHAN Taxus cuspidata. Ref: 662, 900, 3079, 4611.
O O
O
O
O
O O
O
O
O
4704 2-Deacetoxy-5-decinnamoyl taxinine J
H
O
C28H40O9 (520.63). White massive crystals, mp 178~180C, []D12 =

+112.93 (c = 0.058, chloroform). Source: JIANG GUO ZI SHAN Taxus
4709 Deacetoxyvinblastine
baccata, XI MA LA YA HONG DOU SHAN Taxus wallichiana, YUN
C44H56N4O7 (752.96). Source: CHANG CHUN HUA Catharanthus
NAN HONG DOU SHAN Taxus yunnanensis. Ref: 296, 662.
roseus [Syn. Vinca rosea; Lochera rosea]. Ref: 2.
O O
O O
OH
O
O
N
H
O H
O
O
O
OH
N
O
4611.
OH
O
C33H42O8 (566.70). Source: HONG DOU SHAN Taxus chinensis, YUN

NAN HONG DOU SHAN Taxus yunnanensis (aerial parts)[4611]. Ref: 662,
H
H
4705 2-Deacetoxy-7,9-dideacetyltaxinine J
4710 4-Deacetyl-11(151)-abeo-baccatin VI
C35H44O13 (672.73). mp 222C, []D = 73.1 (CHCl3). Source: ZA JIAO
JIE ZHI HONG DOU SHAN Taxus x media. Ref: 662.
O
O OH
OH
O
O
O
HO
4706 13-Deacetoxy-13,15-epoxy-11(151)-abeo-13-epi-baccatin VI
O HO
C35H42O12 (654.72). []D = +23.9 (CHCl3), mp 150C. Source: ZA JIAO

O
4711 2-Deacetyl-9-acetoxytaxine B
C33H45NO7 (567.73). Source: JIANG GUO ZI SHAN Taxus baccata. Ref: 662.
O
OH O
H
O
O
O
O
O
H
H OH
16
4712 3-O-Deacetyl-9-O-acetylsalograviolide A
4716 Deacetyl asperulosidic acid
C17H20O6 (320.35). Colorless solid, []D22 = +29.80 (c = 0.0436,
Citroside A [14259-55-3] C16H22O11 (390.35). Colorless acicular crystals,
MeOH). Pharm: Antifungal (Aspergillus niger, MIC = 6.25g/mL;
mp 146C, []D34 = +11.1 (c = 0.36, water). Pharm: TNF- release
Aspergillus ochraceus, MIC = 3.13g/mL; Penicillium ochrocloron,
inhibitor (cultured mouse peritoneal macrophages, IC50 = 1g/mL)[1605];
MIC = 25g/mL; Cladosporium cladosporioides, MIC = 3.13g/mL;
Laxative. Source: CHANG WEI CU YE MU Lasianthus acuminatissimus
Fusarium tricinctum, MIC = 12.5g/mL; Phomopsis helianthi, MIC =
(root: yield = 0.0046%dw)[1605], HAI BA JI Morinda citrifolia (fruit),
1.56g/mL, Trichoderma viride, inactive). Source: NI GU LA SHI
JIAO RANG MU Daphniphyllum macropodum, XIE JI CU YE MU
CHE JU Centaurea nicolai. Ref: 2361.
Lasianthus wallichii (leaf), ZHI ZI Gardenia jasminoides [Syn. Gardenia

florida]. Ref: 661, 1605, 4238, 4542.
O
O
HO
HO
OH
H
OH
H
O
HO
HO
O
OH
OH
OH
4713 2-Deacetyl-10-acetyltaxine B
C33H45NO7 (567.73). Source: JIANG GUO ZI SHAN Taxus baccata.
Ref: 662.
4717 Deacetyl asperulosidic acid methyl ester

Methyldeacetylasperulosidate C17H24O11 (404.37). Pharm: Laxative (mus,
ED50 = 0.53g/kg). Source: SHUI ZHI Gardenia jasminoides var.
grandiflora, ZHI ZI Gardenia jasminoides [Syn. Gardenia florida]. Ref: 2,

6, 626, 658.
O OH
HO
O
O
H
O
O
H
H OH
O
H
HO
HO
OH
4714 7-Deacetyl-7-angeloyl-6-hydroxyazadiradione
OH
C31H38O6 (506.64). Pale yellow solid, mp 91~94C, []D = +69 (c = 0.658,
OH
CHCl3). Source: Quivisia papinae (seed). Ref: 3759.
4718 2'-Deacetylaustrospicatine
O

O
O
H
O
O
O O
O
O
OH
O
OH
4715 9-O-Deacetylanthemolide D
C17H22O7 (338.36). Pale yellow oil. Source: Anthemis carpatica (aerial
4719 7-Deacetylaustrospicatine
parts). Ref: 3974.

OH
OH
HO
O
O O
OH
N
O
O
H
O
O
O
O
17
4720 2'-Deacetylaustrotaxine
4724 4-Deacetylbaccatin IV
C30H42O13 (610.66). Source: ZA JIAO JIE ZHI HONG DOU SHAN
Taxus x media. Ref: 662.
O O
O O
O
O
O
O
O
O
OH
OH O
OH
O
4721 5-DeacetylbaccatinI
4725 7,9,10-Deacetylbaccatin VI
[30244-36-1] C30H42O12 (594.66). Source: JIANG GUO ZI SHAN Taxus
C31H40O11 (588.66). Source: JIA NA DA HONG DOU SHAN Taxus
baccata. Ref: 662.
canadensis. Ref: 662.
O O
O O
OH OH
H O
OH
OH O
OH
4722 10-Deacetyl baccatin III
4726 7,9-Deacetylbaccatin VI
C29H36O10 (544.62). Pharm: Cytotoxic (in vitro, 30g/mL: A498, InRt =
9-Dihydro-13-acetylbaccatin III C33H42O12 (630.70). mp 221C. Pharm:
27.0%; NCI-H226, InRt = 5.7%; A549, InRt = 12.2%; PC3, InRt = 1.6%;
NO production inhibitor (IC50 = 78.8mol/L, control L-NMMA, IC50 =
control Taxol, 30g/mL: A498, InRt = 98.2%; NCI-H226, InRt = 71.2%;
28.5mol/L) [5407]. Source: JIA NA DA HONG DOU SHAN Taxus
A549, InRt = 79.7%; PC3, InRt = 91.7%)[4800]. Source: DUAN YE
Canadensis, YUN NAN HONG DOU SHAN Taxus yunnanensis (wood).
HONG DOU SHAN Taxus brevifolia, JIANG GUO ZI SHAN Taxus
Ref: 662, 5407.
baccata, SU MEN DA LA HONG DOU SHAN Taxus sumatrana (twig

and leaf: yield = 0.0082%dw[4666]), YUN NAN HONG DOU SHAN
Taxus yunnanensis. Ref: 316, 563, 662, 4666, 4800.

O OH
HO
O OH
O
O
OH O
HO
OH O
H
O
O
O
O
OH
4727 10-Deacetylbaccatin VI
C35H44O13 (672.73). Source: YUN NAN HONG DOU SHAN Taxus
4723 7,9-Deacetylbaccatin IV
yunnanensis. Ref: 662.
C28H40O12 (568.62). Source: JIANG GUO ZI SHAN Taxus baccata,

DUAN YE HONG DOU SHAN Taxus brevifolia. Ref: 662.
O
OH O
O
O OH
OH
O
O
O
O
OH O
H
O
O
O
O
O
O
OH O
H
O
O
18
4728 9-Deacetylbaccatin VI
4733 7-Deacetyl-7-benzoyltaxchinin I
C45H48O13 (796.88). mp 255C. Source: DUAN YE HONG DOU SHAN
Taxus brevifolia. Ref: 662.
O
O OH
O
HO
O
O
OH O
O
O
HO
O
O
4729 9-Deacetyl-9-benzoyl-10-debenzoylbrevifoliol
C29H38O8 (514.62). mp 152C, []D = +18 (CHCl3). Source: DUAN YE
HONG DOU SHAN Taxus brevifolia. Ref: 662.
O
OH O
4734 7-Deacetylcanadensene
C28H40O11 (552.62). White amorphous solid, mp 95~96; []D25 = +5.33
(c = 0.003, CHCl3). Source: MEI LI HONG DOU SHAN Taxus mairei.
Ref: 662, 1914.
HO
OH
HO
O
O
4730 9-Deacetyl-9-benzoyl-10-debenzoyltaxchinin A
OH
C31H40O10 (572.66). []D = +19.4 (MeOH). Source: JIANG GUO ZI
OH
O
SHAN Taxus baccata. Ref: 662.
OH
O
O
HO
O
O
O
O
4735 13-Deacetylcanadensene
HO
HO
C28H40O11 (552.62). White amorphous solid, mp 98~99, []D24 = +4.52
OH
(c = 0.003, CHCl3) Source: MEI LI HONG DOU SHAN Taxus mairei.

O
Ref: 662, 1914.
4731 2-Deacetyl-2-benzoyl-5,13-diacetyltaxchinin A
O
C42H48O13 (760.84). mp 200~203C, []D = 21.5. Source: DUAN YE

O
OH
OH
O
O
O
HO
HO
O
O
4736 2-Deacetyl-5-decinnamoyltaxagifine
4732 7-Deacetyl-7-benzoyltaxayuntin C
C26H36O11 (524.57). Source: HONG DOU SHAN Taxus chinensis, SU
C47H50O14 (838.91). mp 234~236C. Source: DUAN YE HONG DOU
MEN DA LA HONG DOU SHAN Taxus sumatrana (twig and leaf)[4800].
SHAN Taxus brevifolia. Ref: 662.
Ref: 662, 4800.
O
O
O O
O
HO
O
O
O O
OH
O
O
H
H OH
O
O
OH
19
4737 2-Deacetyldecinnamoyltaxinine E
4742 Deacetylfruticolone
Deacetyldecinnamoyltaxinine E C26H38O8 (478.59). []D = +72 (CHCl3).
C20H28O5 (348.44). Colorless oil, [] D25 = +5.4 (c = 0.22, CHCl3).
Source: JIANG GUO ZI SHAN Taxus baccata, HONG DOU SHAN
Pharm: Insect antifeedant (fifth instar larvae of Spodoptera littoralis,
Taxus chinensis. Ref: 662.
dual-choice feeding assays, dose = 10g/cm2, FR50 = 1.030.07). Source:

GUAN CONG XIANG KE KE Teucrium fruticans. Ref: 3761.
O
O O
OH
H
O
O
OH
H
H OH
O
OH
4738 3-Deacetyleupalinin A
C20H26O7 (378.43). Source: CHENG GAN SHENG MA Eupatorium
4743 12-Deacetylganoderic acid H
lindleyanum (whole herb: yield = 0.0023%dw). Ref: 4762.
C30H42O8 (530.66). Source: LING ZHI Ganoderma lucidum (dried

sporocarp: yield = 0.0021%). Ref: 4603.
OH
O
HO
OH
OH
O
O
O
HO
Desacetyleupaserrin [38456-39-2] C20H26O6 (362.43). []D25 = +75.0 (c =

0.92, methanol). Pharm: Antineoplastic (P388, 18mg/kg); cytotoxic (KB,
ED50 = 0.29g/mL); larvacide (insect larva growth inhibitor). Source: AI
XIANG RI KUI Helianthus pumilus, BAN JU CHI ZHUANG ZE LAN
4739 Deacetyleupaserrin
4744 10-Deacetyl-10-glycolylbaccatin IV
C32H44O15 (668.70). Gum. Source: JIA NA DA HONG DOU SHAN
Taxus canadensis (needle leaf). Ref: 3958.
O
Eupatorium semiserratum, WEI GAN JU ZE LAN Eupatorium
HO
mikanioides, Helianthus sp. Ref: 658, 661.
O O
O
O
HO
O
OH
HO
O
O
O
4745 N-Deacetyllappaconitine
O
Puberanidine [11033-64-0] C30H42N2O7 (542.68). Pharm: Analgesic;

toxin. Source: GAN WAN WU TOU Aconitum finetianum. Ref: 658.
4740 14-Deacetyleurylene
C32H56O7 (552.80). Pharm: Cytotoxic (KB cells, IC50 = 0.52g/mL)
[4556]
Source: Eurycoma sp. Ref: 4556.
O
OH
N
H
OH
H
O OH
4741 N-Deacetylfinaconitine
[82872-81-9] C30H42N2O9 (574.68). Pharm: Analgesic; toxin. Source:
GAN WAN WU TOU Aconitum finetianum. Ref: 658.
OH
4746 Deacetyllaurenobiolide
C15H20O3 (248.32). Pharm: Anti-inflammatory (RAW264.7 cells,
LPS-induced: NF-B inhibitor, IC50 = (7.170.16)mol/L, control PTN,
IC50 = (3.420.08)mol/L; NO production inhibitor, IC50 =
(5.760.28)mol/L, PTN, IC50 = (2.410.06)mol/L, AG, IC50 =
O HO
O
N
OH
OH
NH2 OH
O H NH2
OH
(34.180.98)mol/L; TNF- production inhibitor, IC50 =

(27.761.76)mol/L, PTN, IC50 = (2.680.11)mol/L). Source: LIN DI
HAO Artemisia sylvatica (aerial parts). Ref: 3837.
O
O
OH
20
4747 8-Deacetylleopersin A
4752 15-O-Deacetyl-15-O-methylnimbolidin A
C20H30O5 (350.46). White powder. Source: BO SI YI MU CAO Leonurus
C39H48O11 (692.81). Colorless amorphous solid, []D21 = 5.8 (c = 1.26,
persicus. Ref: 2499.
CHCl3). Pharm: Cytotoxic (HeLa-S3, IC50 = 37.4mol/L, control 5-FU,

IC50 = 5.40mol/L, Cisplatin, IC50 = 2.46mol/L). Source: KU LIAN SHI
Melia azedarach (ripe fruit). Ref: 4528.
O
O
OH
O
O
4748 Deacetyllycoclavine
C16H27NO2 (265.40). Source: QIAN CENG TA Huperzia serrata [Syn.
Lycopodium serratum]. Ref: 4388.
OH
4753 15-O-Deacetyl-15-O-methylnimbolidin B
OH
N
O
O

4749 Deacetylmatricarin
C15H18O4 (262.31). mp 123~125C; 143~146C. Source: DAO LUAN YE
PU GONG YING GEN Taraxacum obovatum, YANG SHI CAO Achillea
millefolium, YI KUA Artemisia myriantha (aerial parts), YI ZHI HAO
Achillea alpina [Syn. Achillea sibirica]. Ref: 6, 4618, 5357.
O
O
OH
H
4754 15-O-Deacetylnimbolidin B
4750 Deacetylmatricarin 8-O--glucopyronoside
C21H28O9 (424.45). Colorless gum, [] D26 = 52.4 (c = 0.82, MeOH).
Source: DAO LUAN YE PU GONG YING GEN Taraxacum obovatum.
Ref: 5357.
O
O
HO
O
O
O
H
HO
O
OH
O
OH
OH
O
O
4751 Deacetylmetaplexigenin 3-O--D-oleandropyranosyl-(14)-D-oleandropyranoside

C35H56O12 (668.83). White powder, mp 118~121C, []D20 = +4.8 (c =
0.21, EtOH). Source: QING YANG SHEN Cynanchum otophyllum
(rhizome). Ref: 4574.
OH
O
OH
C35H42O9 (606.72). Amorphous powder, []D = 7 (c = 0.15). Source:

CHUAN LIAN PI Melia toosendan. Ref: 2374.
O
HO
OH
OH
O
OH
OH
O
OO
4755 1-Deacetylnimbolinin A
H
O
O
O
21
4756 1-Deacetylnimbolinin B
4760 3-O-Deacetylorthosiphol I
C33H44O9 (584.71). Amorphous powder. Source: CHUAN LIAN PI Melia
toosendan. Ref: 2374.
CHCl3). Pharm: NO production inhibitor (LPS-activated macrophage-like

J774.1 cells, IC50 = 66.3mol/L; control L-NMMA, IC50 = 26.0mol/L,
Polymixin B, IC50 = 27.8g/mL, Dexamethasone IC50 = 170mol/L).
HO
Source: XIONG RUI ZHUANG ZHI GUAN CAO Orthosiphon stamineus
OH
[Syn: Orthosiphon aristatus; Orthosiphon grandiflorus; Orthosiphon
spicatus] (aerial parts: yield = 0.000045%dw). Ref: 4322, 4741.
H
O
O
O
O
OH
4757 Deacetylnomilin
C26H32O8 (472.54). Source: YOU HE Citrus grandis. Ref: 6.
O
HO
OH
4761 2-O-Deacetylorthosiphol J

OH
J774.1 cells, IC50 = 24.1mol/L; control L-NMMA, IC50 = 26.0mol/L,

Source: XIONG RUI ZHUANG ZHI GUAN CAO Orthosiphon
stamineus [Syn: Orthosiphon aristatus; Orthosiphon grandiflorus;

Orthosiphon spicatus] (aerial parts). Ref: 4322.
O
4758 Deacetyloleandrin
C30H46O8 (534.70). mp 235~238C. Source: JIA ZHU TAO Nerium
HO
indicum. Ref: 6.
O
OH
H
O
4762 10-Deacetyl-13-oxobaccatin III

OH
H
H
OH
OO
OH

29.7%; NCI-H226, InRt = 49.2%; A549, InRt = 43.9%; PC3, InRt =
65.3%; control Taxol, 30g/mL: A498, InRt = 98.2%; NCI-H226, InRt =
71.2%; A549, InRt = 79.7%; PC3, InRt = 91.7%). Source: SU MEN DA
LA HONG DOU SHAN Taxus sumatrana (leaf and twig). Ref: 4800.
OH O
OH
4759 7-O-Deacetylorthosiphol B
OH O
H
O
O
J774.1 cells, IC50 = 102mol/L; control L-NMMA, IC50 = 26.0mol/L,

Orthosiphon spicatus] (aerial parts). Ref: 4322.
4763 10-Deacetyl-10-oxobaccatin III

79.1%; NCI-H226, InRt = 97.3%; A549, InRt = 54.7%; PC3, InRt =
100%; control Taxol, 30g/mL: A498, InRt = 98.2%; NCI-H226, InRt =
71.2%; A549, InRt = 79.7%; PC3, InRt = 91.7%). Source: SU MEN DA
LA HONG DOU SHAN Taxus sumatrana (leaf and twig). Ref: 4800.
O O
OH
O
HO
O
O
O
OH
H
OH
HO
OH O
H
O
O
22
4764 10-Deacetyl-10-oxobaccatin V
4769 Deacetylpseudolaric acid A
C29H34O10 (542.59). Source: HONG DOU SHAN Taxus chinensis. Ref:
C20H26O5 (346.43). Source: TU JING PI Pseudolarix amabilis [Syn. Larix
662.
amabilis; Pseudolarix kaempferi] (root cortex: yield = 0.00003%dw). Ref:

O O
4637.
OH
OH
HO
OH O
H
OH
4770 Deacetylpseudolaric acid C2
4765 10-Deacetyl-10-oxo-7-epitaxol
C45H47NO13 (809.88). []D25 = 60.4 (MeOH). Source: DUAN YE
HONG DOU SHAN Taxus brevifolia, SU MEN DA LA HONG DOU
SHAN Taxus sumatrana (twig and leaf: yield = 0.000026%dw)[4666]. Ref:
C20H24O7 (376.41). Source: TU JING PI Pseudolarix amabilis [Syn. Larix

amabilis; Pseudolarix kaempferi] (root cortex: yield = 0.00025%dw). Ref:
4637.
662, 4666.
OH
HO
O O
OH O
OH
4771 N-Deacetylranaconitine
[82872-80-8] C30H42N2O8 (558.68). Pharm: Analgesic; toxin. Source:
GAN WAN WU TOU Aconitum finetianum. Ref: 658.

H
4766 10-Deacetyl-10-oxo-7-epitaxuyunnanine A
25
C44H53NO13 (803.91). []D = 70.8 (CHCl3). Source: YUN NAN

HONG DOU SHAN Taxus yunnanensis. Ref: 662.
O O
O
OH
O
OH
O
O
OH
OH
O
OH
NH2 OH
O
O
OH O
OH
H
O
O
4772 Deacetylsecomahoganin
C27H34O8 (486.57). White amorphous powder. Source: TAO HUA XIN
MU Swietenia mahogany (leaf). Ref: 4420.
4767 O-Deacetylpachysandrine B
C29H50N2O2 (458.73). mp 184~185C. Source: XUE SHAN LIN
Pachysandra terminalis. Ref: 6.
N
O
H
OH
OH
4768 Deacetylpicraline-3,4,5-trimethoxybenzoat
4773 10-Deacetylspicatine
C31H34N2O8 (562.63). White acicular crystals, mp 222C, []D17 = 185
C33H42O9 (582.70). Source: AO DA LI YA HONG DOU SHAN
(c = 0.052, chloroform). Source: DIAN JI GU CHANG SHAN Alstonia
Austrotaxus spicata. Ref: 662.

O
O
O
O
OH OH
N
H H
O
N
O
O
H O
H
O
23
4774 8-Deacetylsungpanconitine
4779 7-Deacetyltaxayuntin D
C33H47NO9 (601.74). Source: ZHUA KUI GUA YE WU TOU Aconitum
C45H48O13 (796.88). mp 164~166C. Source: DUAN YE HONG DOU
hemsleyanum var. leueanthus (root: yield = 0.0027%dw). Ref: 4678.
SHAN Taxus brevifolia. Ref: 662.
H
H
HO
H
O
O
O
O
O
OH
OH
4775 Deacetyltanghinin
HO
C30H44O9 (548.68). Pharm: Cytotoxic (KB, ED50 = 0.05g/mL, BC, ED50
O
O
= 1.48g/mL, NCI-H187, ED50 = 0.1g/mL)[2594]. Source: NIU XIN QIE

ZI Cerbera manghas. Ref: 2594.
O
4780 2-Deacetyltaxine A
Taxine C C33H45NO9 (599.73). mp 220~221C, []D = 106 (CHCl3),
[]D = 73 (CHCl3). Source: JIANG GUO ZI SHAN Taxus baccata. Ref:
662, 1498.
O
OH
OO
OH
HO
OH
HO
C30H42O12 (594.66). mp 82~83C, []D = 51 (CHCl3). Source: HONG
OH
4776 2-Deacetyltaxachitriene A
OH
DOU SHAN Taxus chinensis. Ref: 662.

4781 2-Deacetyltaxine B
O
O
2-Deacetyl-7,10-diacetyl-5-deaminoacyl taxine A C26H36O9 (492.57). mp
O
O
O
178~179C, []D = 218.2 (CHCl3). Source: JIA NA DA HONG DOU

SHAN Taxus canadensis (needle leaf), YUN NAN HONG DOU SHAN
Taxus yunnanensis. Ref: 662, 3958.
OH
OH
4777 5-Deacetyltaxachitriene B
C28H40O11 (552.62). mp 96~98C, []D = +67.7 (MeOH). Source: HONG
OH

O
O
H
O
OH
O
OH
OH
O
O
4782 10-Deacetyl taxinine B

C35H42O10 (622.72). Colorless thin acicular crystals, mp 245~248C.
Source: ZI SHAN Taxus cuspidata. Ref: 291, 662.
OH
4778 4-Deacetyltaxagifine III
[135962-71-9] C22H32O10 (456.49). mp 221~223C, []D = +38.1
OH O
O
O
(MeOH). Source: HONG DOU SHAN Taxus chinensis. Ref: 662.

O
HO
OH O
HO
O
H
H OH OH
O
O
H O
O
24
4783 10-Deacetyltaxol
4787 10-Deacetyltaxuyunnanine A
C45H49NO13 (811.89). []D = 3 (pyridine). Source: XI MA LA YA
10-Deacetyltaxol C C44H55NO13 (805.93). []D = 50.9 (CHCl3). Source:
HONG DOU SHAN Taxus wallichiana, JIANG GUO ZI SHAN Taxus
SU MEN DA LA HONG DOU SHAN Taxus sumatrana (twig and leaf:
baccata. Ref: 662.
yield = 0.000026%dw)[4666], YUN NAN HONG DOU SHAN Taxus

yunnanensis. Ref: 662, 4666.
OH O
O
N
OH
HO
O
O
OH O
OH
OH
O
O
OH O
OH
H
O
O
4784 10-Deacetyltaxol B
4788 10-Deacetyltaxuyunnanine C
10-Deacetylcephalomannine C43H51NO13 (789.88). []D = 2 (pyridine).
C26H38O7 (462.59). Pharm: Cytotoxic (in vitro, Colon26-L5, EC50 =
Source: XI MA LA YA HONG DOU SHAN Taxus wallichiana, JIANG
76.1g/mL; HT1080, EC50 = 53.8g/mL; control 5-FU , 26-L5, EC50 =
GUO ZI SHAN Taxus baccata. Ref: 662.
0.29g/mL; HT1080, EC50 = 0.07g/mL)[4661]; NO production inhibitor

(IC50 = 28.5mol/L, control L-NMMA, IC 50 = 28.5mol/L)[5407].
OH O
O
N
OH
Source: YUN NAN HONG DOU SHAN Taxus yunnanensis (wood: yield
= 0.0031%dw). Ref: 4661, 5407.
H
O
O
OH O
OH
OH
H
O
O
O
H O
4785 13-O-Deacetyltaxumairol Z
C31H40O12 (604.66). Amorphous powder, []D25 = 42 (c = 0.5, CHCl3).
Source: MEI LI HONG DOU SHAN Taxus mairei (root). Ref: 4250.
4789 6-Deacetyl-teucrolivin A
C22H28O8 (420.46). Amorphous solid, []D25 = +39.60 (c = 1.0, CHCl3).
Source: DONG FANG XIANG KE KE Teucrium orientale. Ref: 2552.
HO
O
OH
OH
HO
O
HO
HO
OH
4790 12-O-Deacetyltrichilin H
4786 7-Deacetyltaxuspine L
C30H44O12 (596.68). Gum. Source: JIA NA DA HONG DOU SHAN
Taxus canadensis (needle leaf). Ref: 3958.

O
O
O
H
O
OH
OH
O
O H O
OH
O O
O
OH
O
O
O
O
H
H
O
OH
25
4791 Deacetylturraeanthin
4796 Deacylmetaplexigenin
C30H48O4 (472.71). mp 202~206C. Source: RI BEN KU LIAN Melia
C21H32O6 (380.48). Source: LUO MO Metaplexis japonica, BAI SHOU
azedarach var. japonica. Ref: 6, 660.
WU Cynanchum bungei, ROU HONG MA LI JIN Asclepias incarnata

(aerial parts). Ref: 6, 3925.
HO
O
OH
OH
H
HO
4797 Deacylmetaplexigenin 3-O--D-oleandropyranosyl-(14)--D-
4792 8-Deacetylyunaconitine
[93460-55-0] C33H47NO10 (617.74). White amorphous powder. Source:
GONG GA SHAN WU TOU Aconitum liljestrandii, GUA YE WU TOU
Aconitum hemsleyanum. Ref: 2191.
OH
O
pyranoside
C46H74O18 (915.09). Amorphous powder, []D27 = +18.6 (c = 1.17,
parts). Ref: 3925.
O
OH
O
H
digitoxopyranosyl-(14)--D-digitoxopyranosyl-(14)--D-digitoxo
MeOH). Source: ROU HONG MA LI JIN Asclepias incarnata (aerial

O
OH
HO
HO
OH
OH
OH
O
OH
OO
4793 10-Deacetylyunnanaxane
C29H44O8 (520.67). Source: JIE ZHI HONG DOU SHAN Taxus media.
OO
OH
Ref: 662.
OH
OO
OH
O
OH
OH
H O
OO
OH
OH
4798 Deaminoacyltaxine A
C24H34O8 (450.53). Source: JIANG GUO ZI SHAN Taxus baccata. Ref:
4794 Deacylbrownioside
C39H62O13 (738.92). Colorless needles (CHCl3-MeOH), mp 258~260C
662.
O
(dec), []D23.9 = 100 (c = 0.175, pyridine). Source: XIAO HUA DUN

YE SHU YU Dioscorea parviflora (fresh rhizome). Ref: 4858.
O
OH
OH
HO
O
OH
O
O
O
OO
HO
4799 Deapio platycodin D
OH
3-O--D-Glucopyranosyl-2,3,16,23,24-pentahydroxyolean-12-ene-28-
OH
OH O O
oic acid 28-O--D-xylopyranosyl-(14)--L-rhamnopyranosyl-(12)-L-arabinopyranoside C52H84O24 (1093.23). Source: JIE GENG

Platycodon grandiflorum. Ref: 4900.
OH OH
4795 Deacylcynaropicrin
C15H18O4 (262.31). mp 152C, []D20 = +120 (c = 0.5, methanol). Pharm:
Cytotoxic (HeLa, ID50 = 5g/mL). Source: YAN DI FENG MAO JU
HO
OH
OH O O
Saussurea salsa. Ref: 661.

OO
HO
H
OH
HO
HO
OH
OH
OH
OH
OO
OH
OO
OH
OH
O
OH OH OH
26
4800 Deapio platycodin D3
4804 N-Debenzoyl-N-butanoyl-10-deacetylpaclitaxel
3-O--D-Glucopyranosyl-(16)--D-glucopyranosyl 2,3,16,23,24-
C42H51NO13 (777.87). mp 244C. Source: JIANG GUO ZI SHAN Taxus
pentahydroxyolean-12-ene-28-oic acid 28-O--D-xylopyranosyl-(14)-
baccata. Ref: 662.
-L-rhamnopyranosyl-(12)--L-arabinopyranoside C58H94O29 (1255.38).

Source: JIE GENG Platycodon grandiflorum. Ref: 4900.
OH O
O
H
OH
H
O
O
HO
OH
OH
OH
OH
OH
OH
HO
OH
H
O
O
OH
OH
OO
OH
OO
OO
HO
OH O
OH
4805 N-Debenzoyl-N-cinnamoyltaxol
OO
OO
OH
OH
C49H53NO14 (879.97). mp 180C, []D = 16.6 (MeOH). Source: ZA

JIAO JIE ZHI HONG DOU SHAN Taxus x media. Ref: 662.
O
OH OH OH
O O
4801 10-Debenzoyl-2-acetoxy-brevifoliol
C26H38O10 (510.59). mp 180C, []D = +32.6 (MeOH). Source: XI MA
O
O
LA YA HONG DOU SHAN Taxus wallichiana. Ref: 662.
OH
OH O
OH
H
O
O
O
O
HO
O
O
4806 14-Debenzoylfranchetine
C24H37NO5 (419.57). White amorphous powder. Source: GONG GA
HO
HO
OH
SHAN WU TOU Aconitum liljestrandii. Ref: 2191.
OH
4802 19-Debenzoyl-19-acetyltaxinine M

O
4807 N-Debenzoyl-N-(2-methylbutyryl)taxol
O
O O
O O
HO
O
C45H55NO14 (833.94). mp 226C, []D = 48 (MeOH). Source: ZA JIAO
O
O

O
OH
H O H
O O
O
N
O
O
OH O
OH
4803 2-Debenzoyl-14-benzoyloxy-10-deacetylbaccatin III
OH
O
O
H
O

4808 7-Debenzoyloxy-10-deacetyl-brevifoliol
OH O
OH
C22H34O6 (394.51). mp 160~162C, []D = 24 (MeOH). Source: XI MA

LA YA HONG DOU SHAN Taxus wallichiana. Ref: 662.
HO
O
H
OH OH O
O
HO
HO
H
OH
OH
27
4814 Debilic acid
4809 8-O-Debenzoylpaeoniflorin
C16H24O10 (376.36). Colorless amorphous solid, [] D23 = 12.8 (c =
[475-85-4] C18H13NO7 (355.31). mp > 350C (dec). Source: JI SHI TENG
0.195, MeOH). Source: Ducrosia anethifolia (aerial parts). Ref: 5469.
GUO Paederia scandens, QING MU XIANG Aristolochia debilis [Syn.

Aristolochia longa]. Ref: 6, 660.
OO
HO
OH
OH
OH
OH
O
OH
O
O
OH
NO2
4810 N-Debenzoyl-N-propanoyl-10-deacetyl paclitaxel

C41H49NO13 (763.85). mp 245C. Source: JIANG GUO ZI SHAN Taxus
4815 Debilone
baccata. Ref: 662.
9-Hydroxy-1(10)-aristolen-2-one [26808-51-5] C15H22O2 (234.34). mp

OH O
O
N
135C. Source: GAN SONG Nardostachys chinensis. Ref: 6.
OH
HO
O
O
OH O
OH
H
O
O
4816 Debneyol
[99694-82-3] C15H26O2 (238.37). Pharm: Antifungal (in vitro,
4811 11-O-Debenzoyltashironin
C15H22O5 (282.34). Colorless solid, []D22 = 65 (c = 0.72, CHCl3).
Pharm: Neurotrophic activity (primary culture of rat cortical neurons,
Cladosporium cucumerinum, ED50 = 50~70g/mL) Source: YAN CAO

Nicotiana tabacum. Ref: 1087, 1114.
0.1-10mol/L). Source: Illicium merrillianum (pericarp: yield =
HO
OH
0.00019%dw). Ref: 3046.
4817 (E,E)-2,4-Decadienal
OH
HO
[25152-84-5] C10H16O (152.24). Source: XING REN Prunus armeniaca.
O
OH
Ref: 2.
4812 2-Debenzoyl-2-tigloyl-10-deacetylbaccatin III
662.
H
O
OH O
OH
4818 (2E,8E)-2,8-Decadiene-4,6-diyne-1,10-diol 1-O--D-glucopyranoside
HO
OH O
C16H20O7 (324.33). Amorphous powder, []D21 = 77 (c = 0.2, MeOH).
Source: CANG ZHU Atractylodes lancea. Ref: 4348.
O
HO
OO
HO
4813 2-Debenzoyl-2-tigloyltaxol
OH
Isocephalomannine C45H53NO14 (831.92). mp 232C, []D = 44
OH
OH
(MeOH). Source: ZA JIAO JIE ZHI HONG DOU SHAN Taxus x media.
4819 Decadienoic acid
Ref: 662.
[13159-49-4] C10H16O2 (168.24). Source: PI JIU HUA Humulus lupulus.

O
Ref: 1521.
O O
OH
O
OH
O
O
OH
OH O
H
O
O
28
4820 3-O-(2'E,4'E-Decadienoyl)-20-O-acetylingenol
4824 3-O-(2E,4Z-Decadienoyl)-20-deoxyingenol
Ingenol-3-(2,4-decadienoate)-20-acetate C32H44O7 (540.70). Colorless oil,
C30H42O5 (482.67). Colorless gum, []D23 = +42.1 (c = 0.28, MeOH).
[]D23 = +84.1 (c = 0.10, MeOH). Pharm: Cytotoxic (in vitro animal cap
Pharm: Induces cell cleavage arrest (Xenopus laevis embryo cells at the
assay to screen for inhibitors of cell division, treatment of cultured
blastular stage, at 0.5g/mL compound results in > 75% cell cleavage
individual Xenopus cells from the early Xenopus laevis embryo at the
arrest). Source: GAN SUI Euphorbia kansui. Ref: 4368.
blastular stage, 0.5g/mL, cleavage arrest > 75%)[4645]. Source: GAN SUI
Euphorbia kansui (root: yield = 0.00006%dw)[4645]. Ref: 660, 4645.
H
O
O
HO
HO
O
H
HO
H H
O
HO
4825 3-O-(2'E,4'E-Decadienoyl)ingenol
C30H42O6 (498.67). Colorless oil, []D23 = +89.09 (c = 0.10, MeOH).

Pharm: Cytotoxic (in vitro animal cap assay to screen for inhibitors of cell
4821 3-O-(2'E,4'Z-Decadienoyl)-5-O-acetylingenol
division, treatment of cultured individual Xenopus cells from the early
Xenopus laevis embryo at the blastular stage, 0.5g/mL, cleavage arrest >
75%). Source: GAN SUI Euphorbia kansui (root: yield = 0.00009%dw).
Ref: 4645.
Ref: 4645.
H H
HO
O
O
O
HO
HO
O
H
OH
4826 3-O-(2'E,4'Z-Decadienoyl)ingenol
OH
C30H42O6 (498.67). Pharm: Cytotoxic (in vitro animal cap assay to screen
for inhibitors of cell division, treatment of cultured individual Xenopus
4822 3-O-(2'E,4'Z-Decadienoyl)-20-O-acetylingenol
cells from the early Xenopus laevis embryo at the blastular stage,
C32H44O7 (540.70). Colorless oil. Pharm: Cytotoxic (in vitro animal cap
0.5g/mL, cleavage arrest > 75%). Source: GAN SUI Euphorbia kansui
assay to screen for inhibitors of cell division, treatment of cultured
(root: yield = 0.00011%dw). Ref: 4645.
individual Xenopus cells from the early Xenopus laevis embryo at the
blastular stage, 0.5g/mL, cleavage arrest > 75%). Source: GAN SUI
Euphorbia kansui (root: yield = 0.00007%dw). Ref: 4645.
H
H
HO
HO
O
HO
H
H
H H
OH
HO
C30H42O6 (498.67). Colorless oil, []D23 = 7.69 (c = 0.13, MeOH).

4823 3-O-(2E,4E-Decadienoyl)-20-deoxyingenol
C30H42O5 (482.67). Colorless gum, []D23 = +57.5 (c = 0.16, MeOH).
Pharm: Induces cell cleavage arrest (Xenopus laevis embryo cells at the
blastular stage, at 0.5g/mL compound results in > 75% cell cleavage
Ref: 4645.
arrest). Source: GAN SUI Euphorbia kansui. Ref: 4368.
O
O
HO
HO
O
H
H
O
HO
HO
OH
29
4832 Decamine
Weedone [17349-05-2] C26H31NO5 (437.54). mp 223~224C. Pharm:
Antibacterial (Bacillus diphtheriae in vitro, 4g/mL); antifungal (Candida
albicans in vitro, 8g/mL). Source: ZI WEI HUA Lagerstroemia indica,
DI KE DONG Decodon verticillatus, ZI WEI YE Lagerstroemia indica.
Ref: 6, 658.
Ref: 4645.
HO
H
H
OH
HO
HO
OH H
4833 Decanal
Capric aldehyde [112-31-2] C10H20O (156.27). Source: DONG LING

CAO Rabdosia rubescens, GAN JIANG Zingiber officinale, JU PI Citrus
4829 20-O-(2'E,4Z-Decadienoyl)ingenol
reticulata, YU XING CAO Houttuynia cordata. Ref: 2.

4834 Decane
Ref: 4645.
n-Decane [124-18-5] C10H22 (142.29). Source: SHAN ZHA Crataegus

pinnatifida. Ref: 2.
HO
HO
O H HH
HO
4835 -Decanolactone
[706-14-9] C10H18O2 (170.25). Source: XING REN Prunus armeniaca,

NAN HE SHI Daucus carota. Ref: 2, 660.
4830 Decaffeoylacteoside
Decaffeoylverbascoside C20H30O12 (462.45). Pharm: Antioxidant (ferric
thiocyanate method, 0.5mmol/L, peroxidation value = 6.6%, control BHA,
0.5mmol/L, peroxidation value = 4.5%, control Vitamin E, 0.5mmol/L,
peroxidation value = 14.7%)[4508]. Source: ROU CONG RONG Cistanche
deserticola, TIAN SHE CAO Lippia dulcis (aerial parts). Ref: 2448,
4508.
4836 2-(Decan-9-one)-N-methyl-4-quinolone
C20H27NO2 (313.44). Source: MENG DA NA YUN XIANG Ruta
Montana (whole herb). Ref: 3910.
O
HO
OH
OO
OH
OH
OH
N
O
OH
OH OH
4831 2,6-Decamethylene pyridine

C15H23N (217.36). Source: SHE XIANG Moschus moschiferus; Moschus
berezovskii; Moschus sifanicus. Ref: 2.
4837 Decanoylacetaldehyde
Houttuynin C12H22O2 (198.31). Pharm: Antibacterial (in vitro,
gram-positive bacteria, gram-negative bacteria; in vitro and in vivo,
houttuynin isoniazone inhibits Mycobacterium tuberculosis strongly, MIC
= 0.78~3.10mg/mL); immunoenhancer (chronic bronchitis patient, orl
90mg, 3 times daily, after seven days the level of properdin in blood has
ascending tendency). Source: YU XING CAO Houttuynia cordata (aerial
parts: content = 0.05%[5501]). Ref: 2, 4, 1974, 2056, 5501.
30
4843 cis-4-Decenoic acid
4838 20-O-(Decanoyl)ingenol
C30H46O6 (502.7). Pharm: Cytotoxic (in vitro animal cap assay to screen
Obtusilic acid [505-90-8] C10H18O2 (170.25). bp 148~150C/13mmHg.
for inhibitors of cell division, treatment of cultured individual Xenopus
Source: CHENG QIE ZI Litsea cubeba, SAN ZUAN FENG Lindera
cells from the early Xenopus laevis embryo at the blastular stage,
obtusiloba, ZHEN CAI Litsea pungens. Ref: 6, 1521, 2825, 2956.

O
0.5g/mL, cleavage arrest > 75%). Source: GAN SUI Euphorbia kansui
OH
(root: yield = 0.00007%dw). Ref: 4645.

H
H
H
HO
HO
4844 trans-4-Decenoic acid
[26303-90-2] C10H18O2 (170.25). bp 148~150C/13mmHg. Source: SAN
HO
ZUAN FENG Lindera obtusiloba. Ref: 6.
O
O
4839 12-O-Decanoylphorbol-13-(2-methylbutyrate)
OH
C35H54O8 (602.82). Oil, []D = +56 (c = 0.05, CHCl3). Pharm:

Anti-HIV-1 (MT-4 cells, HIV-1-induced cytopathic effect inhibitor, IC100
4845 Decentapicrin A
= 7.81g/mL, CC0 = 31.3g/mL, control DS8000, IC100 = 3.9g/mL, CC0
C23H26O11 (478.46). Source: GUANG LIANG JIA LONG DAN
> 1000g/mL); PKC activator inactive (10ng/mL, activity rate =
Gentianella nitida (whole herb). Ref: 3542.
0%)[3921]. Source: BA DOU Croton tiglium. Ref: 3921.
H
O
OO
HO
OH
HO
O
O HO
OH
OH
OH
4846 Dechloroacutumidine
4840 Decarbomethoxy naucl echine
C18H23NO6 (349.39). []D25 = 68 (c = 0.2, MeOH) Source: BIAN FU
C19H19N3O (305.38). Pharm: Antibacterial (in vitro: Staphylococcus aureus,
GE Menispermum dauricum. Ref: 1946.
Bacillus subtilis, Bacillus coli, Bacillus diphtheriae, Streptococcus sp.,
Streptobacillus sp., Salmonella sp., Bacillus proteus, Bacillus lactis,
OH
Klebsiella pneumoniae); antileishmanial; antifungal (Aspergillus niger).

Source: KUAN YE WU TAN Nauclea latifolia. Ref: 2178.
N
H H
NH
O
O
OH
4847 Dechlorodauricumine
C19H25NO6 (363.41). Amorphous powder, []D25 = +20.7 (c = 0.10,
MeOH). Source: BIAN FU GE GEN Menispermum dauricum. Ref: 5326.
4841 1-Decene
C10H20 (140.27). Source: KUAN DONG HUA Tussilago farfara. Ref:
OH
660.
O
N
O
O
O
4842 (2E)-2-Decene-4,6-diyne-1,8-diol 8-O--D-apiofuranosyl-
4848 Decinine
(16)--D-glucopyranoside
[10183-64-9] C26H31NO5 (437.54). mp 222~224C. Source: ZI WEI YE
Lagerstroemia indica. Ref: 6.
Source: CANG ZHU Atractylodes lancea (rhizome). Ref: 4384.
O
O
HO
OO
OH OH
OH
OH
OH
OH
OH
31
4849 Decinnamol taxinine J
4854 Decinnamoyltaxinine E
5-Hydroxy-2,7,9,10,13-Pentaacetoxy-4(20),11-taxadiene
C30H42O11 (578.66). Colorless prisms. Source: AO DA LI YA HONG
662.
DOU SHAN Austrotaxus spicata, DUAN YE HONG DOU SHAN Taxus

brevifolia, HONG DOU SHAN Taxus chinensis. Ref: 662, 2488.
O O
O O
O O
O O
O
O
H O
OH
H O H
OH
4855 Decinnamoyltaxinine B 11,12-oxide
4850 5-Decinnamoyl-11-acetyl-19-hydroxyl taxagifine
C30H40O14 (624.64). White massive crystals, mp 209~210C, []D14 =
12.1 (chloroform). Source: YUN NAN HONG DOU SHAN Taxus

O
yunnanensis. Ref: 296, 662.

O O
O
O
O O
OH
O
O O
O
O
O
O
H O
OH
OH
H O
O
4856 Decodine
4851 13-Decinnamoyl-9-deacetyltaxchinin B

O
O
O
OH O
HO
HO
OH
O
O
HO
O
4852 Decinnamoyl-1-hydroxy-taxinine J
4857 Decoside
C30H42O9 (546.66). Pharm: Toxin (vertebrate). Source: YANG JIAO AO
662.
ZI Strophanthus divaricatus. Ref: 658.

O O
O O
O
O
O
O
OH O
OH
O
H
OH
OH
OO
4853 5-Decinnamoyltaxagifine
662.
O O
HO
O O
4858 Decoyl vanillylamide
C16H25NO3 (279.38). Source: LA JIAO Capsicum frutescens. Ref: 6.
O
O
H O
O
OH
O
N
H
O
OH
32
4859 Decumbensol
4864 Decussine
C19H20O6 (344.37). Colorless massive crystals, mp 183~183.5C, [] D20 =
[75375-52-9] C20H19N3 (301.39). Yellow rhomboid crystals (methanol),
+202 (c = 0.53, CHCl3). Source: QIAN HU Angelica decursiva [Syn.
mp 203~205C. Pharm: Neuromuscular blocker. Source: DUI SHENG
Peucedanum decursivum]. Ref: 9.
MA QIAN Strychnos decussata. Ref: 661.
HO
O
O
4860 Decumbesterone A
C29H46O7 (506.69). Pharm: Antineoplastic (inhibits EBV-EA induction
strongly). Source: BAI MAO XIA KU CAO Ajuga decumbens. Ref: 693.
4865 n-Decyl acetate

[112-17-4] C12H24O2 (200.32). mp 15.05C, bp 244C. Source: HEI MA
OH
OH
YI Formica fusca. Ref: 6.
HO
H
HO
OH
HO
O
O
4861 Decumbic acid
4866 4a,N-Dedihydronoraugustamine
C9H12O4 (184.19). mp 125~127C, []D25 = +44.3 (c = 0.47, CHCl3).
C16H15NO4 (285.30). mp 127~130C, []D20 = 242.6 (c = 0.27, MeOH).
Source: Lasiodiplodia theobromae (fruit). Ref: 3867.
Pharm: Antiprotozoal inactive (Plasmodium falciparum, Leishmania

donovani, Trypanosoma brucei, Trypanosoma cruzi). Source: KEN NI
YA WEN SHU LAN Crinum kirkii (bulb). Ref: 3892.
HO
4862 Decursin
[5928-25-6] C19H20O5 (328.37). mp 110~111C. Pharm: AChE inhibitor
(in vitro, IC50 = 390mol/L)[3058]; reduces muscular twitching (cultured
O O
myocardial cells line). Source: QIAN HU Angelica decursiva [Syn.

Peucedanum decursivum], CHAO XIAN DANG GUI Angelica gigas
(underground part)[3058]. Ref: 6, 658, 3058.
4867 N-Deethyl-N-19-didehydrosachaconitine
C21H31NO4 (361.49). Amorphous solid, []D25 = +181.8 (c = 0.11,
CHCl3). Source: BAN HUA WU TOU Aconitum variegatum (aerial parts).
Ref: 5270.
O
O
H
O
4863 Decursinol
O
OH
OH
[23458-02-8] C14H14O4 (246.27). mp 176~177C. Pharm: AChE inhibitor

(in vitro, IC50 = 28mol/L)[3058]; reduces muscular twitching (cultured
myocardial cells line). Source: DA TIAO WEN XIE HAO Seseli
grandivittatum, MU(4) JU Aegle marmelos, QIAN HU Angelica decursiva
[Syn. Peucedanum decursivum], CHAO XIAN DANG GUI Angelica
gigas (underground part)[3058]. Ref: 6, 658, 3058.
4868 Deformylflustrabromine
C16H21BrN2 (321.26). Pharm: Affinity to nAChR (42* subtype, Ki =
(3400500)nmol/L, control ()-Nicotine, Ki = (0.8380.132)nmol/L; 7*
subtype, Ki > 50000nmol/L, ()-Nicotine, Ki = (1275)nmol/L). Source:
BEI HAI XIAN TAI CHONG Flustra foliacea. Ref: 5029.
N
H
O
HO
O
Br
NH
33
4869 Deformylflustrabromine B
4873 Dehydroabietic acid
C16H21BrN2 (321.26). Pharm: Affinity to nAChR (42* subtype, Ki >
8,11,13-Abietatrien-18-oic acid [1740-19-8] C20H28O2 (300.44). Colorless
50000nmol/L, control ()-Nicotine, Ki = (0.8380.132)nmol/L; 7*
acicular crystals, mp 174C, []D20 = +66 (c = 0.60, diethyl ether). Pharm:
subtype, Ki = (170002200)nmol/L, ()-Nicotine, Ki = (1275)nmol/L).
Activates nerve (stimulates release of neurotransmitter inhibitor
Source: BEI HAI XIAN TAI CHONG Flustra foliacea. Ref: 5029.
(-aminobutyric acid) and neurotransmitter stimulant); antifungal (in vitro,

Pyricularia oryzae, InRt = 100%); antiulcerative; used in treatment of
N
H
hypertension and tachycardia caused by smoking; vasodilator. Source:

XIAN MAI XIANG CHA CAI Rabdosia nervosa, LEI GONG TENG
Br
Tripterygium wilfordii. Ref: 900.
4870 Degalactotigonin
[39941-51-0] C50H82O22 (1035.20). Pharm: Antineoplastic (inhibits 32P
combines with phospholipid in HeLa cells, 50g/mL, InRt = 57.8%).
Source: ZHI MU Anemarrhena asphodeloides. Ref: 2, 1636.
O
O
H
H
HO
OO
OH
OH
OH
HO
OH
OH
4874 Dehydroabietic acid methyl ester

C21H30O2 (314.47). Pharm: Antineoplastic (EBV-EA induced by TPA,
mol ratio/TPA = 1000, relative percentage of EBV-EA = 0% (positive
control value 32pmol, 20ng TPA =100%), viability of Raji cells = 60%;
reference compound -Carotene, relative percentage = 8.6%). Source: FU
OO
OH
OH
HO
H
O
LING Poria cocos (sclerotium: yield = 0.0013%dw). Ref: 4616.
OH
OH
OH
4871 Deglucocheirotoxin
C29H42O10 (550.65). mp 188~191C. Source: LING LAN Convallaria
keiskei [Syn. Convallaria majalis]. Ref: 6.
O
H
O
4875 Dehydroagastol
19(43)-Abeo-11,14-dihydroxy-12-methoxy-abieta-8,11,13,15-tetraen-7
-one C21H26O4 (342.44). Yellow green acicular crystals, mp 159~161C,
O
H
H
OO
HO
soluble in hexane, chloroform and methanol. Source: GUANG HUO

XIANG Pogostemon cablin [Syn. Mentha cablin]. Ref: 210, 660.
OH
OH
O
HO
OH OH
4872 Deguelin
OH
Degueline [522-17-8] C23H22O6 (394.43). Yellow crystals, mp 180~182C

H
(methanol); 171C, []D20 = 107 (c = 0.2, benzene). Pharm: Ornithine

decarboxylase inhibitor (induced by ester phorbol, IC50 = 0.0003g/mL);
larvacide (larva of mosquito); nematocide (MLD = 1mol/L); anti-tumor
promotor (in vivo, mouse skin tumor, inhibits TPA-induced EBV-EA
activation, 100(mol ratio/32 pmol TPA), EBV-EA positive cells = 72.3%
viability, positive control -Carotene, EBV-EA positive cells = 82.7%
viability)[4982]. Source: MU LAN
(2)
Indigofera tinctoria, HUI YE GEN
Tephrosia purpurea, MAO YU TENG Derris elliptica, YU TENG Derris
4876 Dehydroandrographolide
C20H28O4 (332.44). Colorless acicular crystals (recrystalsliztion in 30 and
50% ethanol), mp 204C. Pharm: Anti-inflammatory; antipyretic; used in
treatment of infectious diseases of respiratory tract and intestinal tract.
Source: CHUAN XIN LIAN Andrographis paniculata [Syn. Justicia
paniculata] (dried aerial parts: content = 1.19%[5508]) Ref: 661, 5508.
trifoliata (stem), Tephrosia sp., Lonchocarpus sp. Ref: 6, 900, 4982.

O
O
H
O
O
HO
H
OH
34
4877 1,2-Dehydroapateline
4881 Dehydrobaimuxinol
C34H30N2O5 (546.63). Yellow amorphous powder, []D25 = +128 (c =
[105013-74-9] C15H24O2 (236.36). Colorless acicular crystals, mp
0.42, MeOH). Pharm: Exhibited in vitro anticholinesterase activities, IC50
136~138C, []D26 = +25 (c = 1.6, chloroform). Source: BAI MU
= (116.52.5)mol/L, control Galanthamine, IC50 = (0.50.0)mol/L).
XIANG Aquilaria sinensis. Ref: 13, 58.
Source: CHUI MU FANG JI Cocculus pendulus. Ref: 4051.

O
O
N
OH
4882 (3S,7R)-5,6-Dehydro-1,7-bis(4-hydroxyphenyl)-4-de-O-meth-
OH
4878 6,7-Dehydroartemisinic acid

C15H20O2 (232.33). Source: HUANG HUA HAO Artemisia annua. Ref: 2, 660.
ylcentrolobine
MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 71.2mol/L, control
5-FU, ED50 = 0.53mol/L; HT1080, ED50 = 45.3mol/L, 5-FU, ED50 =

8.0mol/L). Source: YUN NAN CAO KOU Alpinia blepharocalyx (seed:
yield = 0.000071%dw). Ref: 3048.
HO
OH
HO
4879 Dehydroascorbic acid

[490-83-5] C6H6O6 (174.11). mp 196C (dec). Source: HUI XIANG JING
YE Foeniculum vulgare, JIANG MANG Cassia sophera, MA BO
Lasiosphaera fenzlii. Ref: 6.
11,24-Dioxo-5,21-dien-cucuebit-3-O--D-xylopyranosyl-16-O--L-rha
OH
mnopyranoside C41H64O12 (748.96). White amorphous powder, []D28 = 0
OH
O
4883 Dehydrobryogenin glycoside
(c = 0.176, MeOH). Source: KU XUAN SHEN Picria felterrae (whole

herb). Ref: 4853.
O
O
4880 9(11)-Dehydroaxinysterol
C28H40O3 (424.63). White amorphous solid, []D25 = +78.9 (c = 0.89,
CHCl3). Pharm: Cytotoxic (Breast: HBC4 IC50 = 0.85g/mL; BSY1 IC50
OH
= 0.60g/mL; HBC5 IC50 = 0.96g/mL; MCF7 IC50 = 0.36g/mL;

MDA-MB-231 IC50 = 1.26g/mL; Lung: NCI-H23 IC50 = 0.54g/mL;
NCI-H226 IC50 = 0.63g/mL; NCI-H522 IC50 = 0.57g/mL; NCI-H460
IC50 = 0.81g/mL; A549 IC50 = 0.96g/mL; DMS273 IC50 = 0.54g/mL;
OO
OO
OH
OH
DMS114 IC50 = 0.48g/mL; Stomach: St4 IC50 = 0.69g/mL; MKN1 IC50
OH OH
OH
= 0.42g/mL; MKN7 IC50 = 0.48g/mL; MKN28 IC50 = 0.84g/mL;

MKN45 IC50 = 0.54g/mL; MKN74 IC50 = 0.54g/mL; Kidney:
4884 Dehydrobufotenine
RXF-631L IC50 = 0.72g/mL; ACHN IC50 = 0.51g/mL; Colon:
[17232-69-8] C12H14N2O (202.26). Source: CHAN SU Bufo bufo
HCC2998 IC50 = 0.57g/mL; KM12 IC50 = 0.60g/mL; HT29 IC50 =
gargarizans; Bufo melanostictus. Ref: 2.
0.57g/mL; HCT15 IC50 = 0.75g/mL; HCT116 IC50 = 0.48g/mL;

Ovary: OVCAR-3 IC50 = 0.19g/mL; OVCAR-4 IC50 = 0.60g/mL;
OVCAR-5 IC50 = 0.54g/mL; OVCAR-8 IC50 = 0.22g/mL; SK-OV-3
N
O
IC50 = 0.81g/mL; CNS: U251 IC50 = 0.63g/mL; SF268 IC50 =
NH
1.02g/mL; SF295 IC50 = 0.75g/mL; SF539 IC50 = 0.84g/mL; SNB75

IC50 = 2.16g/mL; SNB78 IC50 = 1.17g/mL; Prostate: DU145 IC50 =
0.54g/mL; PC3 IC50 = 0.57g/mL; Melanoma: LOX-IMVI IC50 =
0.60g/mL). Source: Sponge Axinyssa sp. Ref: 4231.
4885 7-Dehydrocholesterol
[434-16-2] C27H44O (384.65). mp 142~143C; 150C. Source: SHUI
LONG GU Polypodium niponicum. Ref: 6.
H
H
H
HO
H
HO
35
4886 Dehydrocoreximine (perchlorate)
4890 Dehydrocorydalmine
2,3,10,11-Substituted pseudoprotoberberine alkaloid C19H18NO4+
[6877-27-6] C20H20NO4+ (338.39). Source: CHANG JU YAN HU SUO
(324.36). Pale yellow crystalline solid, mp 243~247C. Source: XIAO
Corydalis longicalcarata (rhizome: content = 0.208%[5508]), HUI LV YAN
HUA MU BAN SHU Xylopia parviflora (bark and root). Ref: 3794.
HU SUO Corydalis adunca (rhizome: content = 0.122%[5508]), YAN HU

SUO Corydalis yanhusuo [Syn. Corydalis turtschaninovii f. yanhusuo].
Ref: 6, 5508.
O
N
HO
O
+
O
OH
OH
4887 11-Dehydrocorticosterone
4891 Dehydrocostuslactone
[72-23-1] C21H28O4 (344.45). mp 183.0~183.5C. Source: NIU SHEN
C15H18O2 (230.31). mp 60.5C. Pharm: Plant growth regulator;
Bos taurus domesticus; Bubalus bubalis, ZI HE CHE Homo sapiens.

Ref: 6.
antitrypanosomal (epimastigotes of Trypanosoma cruzi, MLC =

6.3mol/L); anti-inflammatory (NO production inhibitor)[4415]; cytotoxic
(in vitro, HepG2, CD50 = 3.5g/mL; HeLa, CD50 = 3.5g/mL; OVCAR-3,
CD50 = 2.5g/mL; control Cisplatin, HepG2, CD50 = 2.8g/mL; HeLa,
OH
CD50 = 5.2g/mL; OVCAR-3, CD50 = 3g/mL; without significant
antibacterial effect)[4720]. Source: CHUAN MU XIANG Vladimiria
H
H
souliei [Syn. Jurinea souliei] (root: content scope of 4 origins =
0.482%~1.620%, mean content of = 1.29%[5508]), MU XIANG Saussurea
lappa [Syn. Aucklandia lappa] (root: mean content of 10 origins =

1.83%[5508]; yield = 0.019%dw[4720]), YUE GUI YE Laurus nobilis, YUE
4888 Dehydrocorybulbine
C21H22NO4+ (352.41). Source: YAN HU SUO Corydalis yanhusuo [Syn.
Corydalis turtschaninovii f. yanhusuo]. Ref: 2.
XI MU XIANG Vladimiria denticulata. Ref: 2, 6, 658, 660, 4248, 4415,

4720, 5508.
H
H
O
OH
H
O
4892 cis-Dehydrocrotonin
C19H22O4 (314.38). Source: GE LUN BI YA BA DOU Croton

schiedeanus. Ref: 4552.
4889 Dehydrocorydaline
+
[30045-16-0] C22H24NO4 (366.44). Pharm: Antiulcerative (rat, sc, gastric

ulcer); coronary vasodilator; increases coronary flow; inhibits gastric
secretion; increases tolerance to anoxia (mus); used in treatment of

coronary heart disease (main effective component in Corydalis yanhusuo
YAN HU SUO). Source: CHANG JU YAN HU SUO Corydalis

longicalcarata (rhizome: content = 0.025%[5508]), DONG BEI YAN HU
SUO Corydalis ambigua var. amurensis [Syn. Corydalis ambigua], DUI

YE YUAN HU Corydalis ledebouriana (rhizome: content = 0.032%[5508]),
HUI LV YAN HU SUO Corydalis adunca (rhizome: content =
0.069%[5508]), XI SHEN SHAN ZI JIN Corydalis pallida var. tenuis, YAN
HU SUO Corydalis yanhusuo [Syn. Corydalis turtschaninovii f.
yanhusuo] (rhizome: mean content of 5 origins = 0.152%[5508]). Ref: 2,
658, 5508.
4893 trans-Dehydrocrotonin
C19H22O4 (314.38). Pharm: Antiulcerogenic[5351]; cytotoxic (HL-60 cells,
MTT assay, 24h, IC50 = 300mol/L, 96h, IC50 =180mol/L, control
Myricetin, 24h, IC50 = 192mol/L; protein quantification, 24h, IC50 =
500mol/L, 96h, IC50 =150mol/L, control Myricetin, 24h, IC50 =
300mol/L). Source: KA ZHU BA DOU Croton cajucara. Ref: 5351.
O
O
O
O
O
O
O
36
4894 Dehydro--curcumene
4899 Dehydrodeltatsine
[4999-58-0] C15H20 (200.33). Source: CE BAI ZHI JIE Thuja orientalis
C25H39NO7 (465.59). Amorphous solid, []D25 = +20 (c = 0.1, CHCl3).
[Syn. Platycladus orientalis; Biota orientalis]. Ref: 6.
Source: DONG FANG FEI YAN CAO Consolida orientalis (aerial parts).
Ref: 4283.
H
O
H
OH
H
4895 Dehydrocurdione
H
O
[38230-32-9] C15H22O2 (234.34). Pharm: NO production inhibitor
OH
inactive (mus peritoneal macrophages, induced by LPS, 100mol/L, InRt

= (12.83.1)%, control L-NMMA, 100mol/L, InRt = (79.20.9)%,
p<0.01)[4150]. Source: PING E SHU Curcuma zedoaria [Syn. Curcuma
aeruginosa], JIANG HUANG Curcuma longa. Ref: 6, 640, 4150.
4900 (3S,7S)-5,6-Dehydro-4-de-O-methylcentrolobine
C19H20O3 (286.37). Pharm: Cytotoxic (Colon26-L5, ED50 > 100mol/L,
control 5-FU, ED50 = 0.53mol/L; HT1080, ED50 = 79.4mol/L, 5-FU,
ED50 = 8.0mol/L). Source: YUN NAN CAO KOU Alpinia
blepharocalyx (seed: yield = 0.000014%dw). Ref: 3048.

OH
HO
4896 1,2-Dehydrocycloparvifloralone
22
C15H22O6 (298.34). Colorless amorphous powder, []D = +14 (c = 1.77,

CH3OH). Pharm: Neurotrophic bioassay inactive (primary culture of rat
cortical neurons, 0.1-10mol/L). Source: Illicium merrillianum (pericarp:
4901 3-Dehydrodeoxyandrographolide
yield = 0.00038%dw). Ref: 3046.
C20H28O4 (332.44). Colorless lamellar crystals (MeOH), mp 140~142C.

HO
paniculata] (leaf). Ref: 4913.
O
O OH
OH
OH
4897 Dehydrodeacetylheterophylloidine
C21H25NO3 (339.44). Amorphous, []D25 = 73.3 (c = 0.17, CHCl3).
Source: WU ZHU FEI YAN CAO Delphinium pentagynum (aerial parts).
Ref: 3831.
OH
4902 (7R,8S)Dehydrodiconifery alcohol-9'-O--D-glucoside
C26H32O11 (520.54). Source: GUAN HUA ROU CONG RONG Cistanche

tubulosa. Ref: 2448.
O
N
HO
O
HO
O
HO
4898 Dehydrodeguelin
6,12-Dehydrodeguelin [3466-23-7] C23H20O6 (392.41). Straw yellow
OH
OH
OH
solid, mp 215~225C. Pharm: cAMP phosphodiesterase inhibitor (rat

heart, IC50 = 6.2mol/L); larvacide (larva of mosquito); nematocide (in
vitro, 0.1g/mL, larva of Toxocara canis, after 6 hours cultivation, RM =
30, after 24 hours, RM = 0). Source: MU LAN
(2)
Indigofera tinctoria,
HUI YE GEN Tephrosia purpurea. Ref: 946, 1138, 1188.
4903 (7S,8R)Dehydrodiconifery alcohol-4-O--D-glucoside

[107870-88-2] C26H32O11 (520.54). White powder, []D21= 45.8 (c = 0.9,
MeOH). Source: GUAN HUA ROU CONG RONG Cistanche tubulosa,
MAO JIAN QIU LUO Lychnis coronaria Ref: 2189, 2448.
O
O
HO
OH
OO
OH
OH
OH
OH
O
O
37
4904 Dehydrodiconiferyl alcohol 4,'-di-O--D-glucopyranoside
4909 Dehydroeburicoic acid
[109792-90-7] C32H42O16 (682.68). Source: DU ZHONG Eucommia
3-Hydroxy-24-methylene-lanosta-7,9(11)-dien-21-oic acid [6879-05-6]
ulmoides. Ref: 2.
C31H48O3 (468.73). mp 286~288C. Source: A LI HONG Fomes

officinalis, FU LING Poria cocos. Ref: 6, 660.
HO
HO
OO
HO
OH
OH
O
OH
OH
OH
HO
OH
4905 (7S,8R) Dehydrodiconiferyl alcohol 9'--glucopyranoside
HO
C26H32O11 (520.54). Pale yellow amorphous powder, []D15 = 19.5 (c =

0.4, CHCl3). Source: SUO YANG Cynomorium songaricum (stem). Ref:
4114.
4910 Dehydroeburiconic acid

[18449-25-7] C31H46O3 (466.71). mp 240~242C. Source: A LI HONG
Fomes officinalis. Ref: 6.
HO
O
HO
O
HO
O
O
O
OH
OH
HO
OH
4906 Dehydrodieugenol
[4433-08-3] C20H22O4 (326.40). Pharm: Antifungal (using extract of bark

of Litsea turfosa). Source: NI ZHAO MU JIANG ZI Litsea turfosa. Ref:
658.
4911 8,9-Dehydro-10-epi-ryanodine
O
OH HO
C25H33NO9 (491.54). Crystals (CHCl3:Me2CO = 1:1), mp 165C, []D =
+20 (c = 0.1). Pharm: Cardiac contraction inhibitor (guinea-pig papillary

muscle, causes a prolongation of the latency time and decrease of
contraction force, EC50 = 17nmol/L)[5139]. Source: QU CHONG CAO
Spigelia anthelmia (aerial parts). Ref: 5139.
4907 (13S)-8,9-Dehydro-18,21-dihydroxy-10-epi-ryanodine
C25H33NO11 (523.54). Crystals (CHCl3:MeOH = 1:1), mp 162C, []D =
+7 (c = 0.2). Source: QU CHONG CAO Spigelia anthelmia (aerial parts).
Ref: 5139.
O
HO
OH
OH
HO
OH
OH
HO
OH
OH
H
HO
OH
OH
NH
H
OH
N
H
OH
4912 Dehydroevodiamine
C19H15N3O (301.35). Pharm: Uterine stimulant (rat, in vitro); slows heart
4908 8,9-Dehydro-20,21-dihydroxy-10-epi-ryanodine
rate (anesthetic rat); antihypertensive (anesthetic rat). Source: WU ZHU
C25H33NO11 (523.54). Crystals (CHCl3:MeOH = 1:1), mp 173C, []D =
YU Evodia rutaecarpa (dried unripe fruit). Ref: 5031, 5501.

Ref: 5139.
OH
HO
OH
N
H
O
O
OH
OH
OH
OH
OH
N
N
38
4913 3R,8R-Dehydrofalcarindiol
4918 Dehydroflourensic acid
C17H22O2 (258.36). Pale yellow oil, []D25 = +39.8 (c = 2.66, CHCl3).
C15H20O3 (248.32). Oil. Pharm: Phytotoxin (inhibits radicle growth,
Pharm: 12-Lipoxygenase inhibitor inactive (10g/mL, InRt = 0%;
Amaranthus hypochondriacus, IC50 = 196mol/L, control 2,4-D, IC50 =
30g/mL, InRt = 0%; control Baicalein, 10g/mL, InRt = 56.23%);
180mol/L; Echinochloa crusgalli, IC50 = 620mol/L, control 2,4-D, IC50
cytotoxic (in vitro, MTT assay: LS174T colorectal cancer, IC50 =
= 230mol/L); CaM interactor (cAMP phosphodiesterase inhibitor, IC50 =
(14.87.2)g/mL, control Doxorubicin, IC50 = (324100)ng/mL; SKCO1
23.2mol/L, control Chlorpromazine, IC50 = 10.2mol/L, interacted with
colorectal cancer, IC50 = (13.35.4)g/mL, Doxorubicin, IC50 =
bovine-brain calmodulin and inhibited the activation of the
(28.510)ng/mL; COLO320DM colorectal cancer, IC50 = 9.6g/mL,
calmodulin-dependent enzyme cAMP phosphodiesterase). Source: FU
Doxorubicin IC50 = (1163168)ng/mL; WIDr colorectal cancer, IC50 =
CHUI FE LAO JU Flourensia cernua. Ref: 3433.
10.9g/mL; MDA231 breast cancer, IC50 = 37.6g/mL; MCF7 breast
cancer, IC50 = 5.8g/mL). Source: DAN ZI HAO Artemisia monosperma.
Ref: 5249.
OH
OH
H
4919 Dehydrogeijerin
H
H
H
OH
[16850-91-2] C15H14O4 (258.28). mp 132C. Source: YAN JIAO CAO

Boenninghausenia albiflora. Ref: 2495.
H
O
4914 Dehydrofalcarinol
[36150-08-0] C17H22O (242.36). Source: YIN CHEN HAO Artemisia
capillaris. Ref: 2.
4920 12,13-Dehydrogeranylgeraniol
C20H32O (288.48). Clear oil. Pharm: Antioxidant (HL-60, PMA-induced
peroxide-catalyzed oxidation of 2,7-dichlorodihydrofluorescein dye
(DCFH) by reactive oxygen species (ROS), 5g/mL (17.4mol/L), InRt =
HO
28%)[3060]. Source: MEI ZHOU SAN BAI CAO Saururus cernuus (stem
4915 Dehydrofalcarinone
and leaf), SHUANG CHA ZAO Bifurcaria bifurcata. Ref: 3060, 5146.
[4117-05-9] C17H20O (240.35). Source: YIN CHEN HAO Artemisia
OH
capillaris. Ref: 2.
4921 6-Dehydrogingerdione
[76060-35-0] C17H22O4 (290.36). Pharm: Anti-inflammatory
(prostaglandin biosynthesis inhibitor, IC50 = 2.3mol/L); antidiarrheal

(mus, orl, 10mg/kg, inhibits 5-HT-induced diarrhea and loss of body
4916 6-Dehydroferruginol
temperature); antihepatotoxin (rat liver cells, in vitro, 1.0mg/mL, liver
C20H28O (284.45). Pharm: 12(S)-LOX inhibitor inactive (hmn Platelets,
toxicosis induced by CCl4, GPT = (702)% of that of control, p<0.001);
100g/mL, 12(S)-HETE Production inhibitor inactive)[4980]. Source: DU

SONG SHI Juniperus rigida, OU ZHOU CI BAI Juniperus communis
prostaglandin syntheatase inhibitor (IC50 = 1.0mol/L). Source: SHENG

JIANG Zingiber officinale. Ref: 2, 1815, 1816, 1817, 1820.
(wood). Ref: 6, 4980.

OH
OH
O
HO
4922 10-Dehydrogingerdione
H
[82206-04-0] C21H30O4 (346.47). Pharm: Anti-inflammatory
4917 3,4-Dehydrofloridanolide
C15H22O5 (282.34). Colorless amorphous, []D20 = +44 (c = 1.90, CHCl3).
Source: Illicium merrillianum (pericarp). Ref: 5113.
(prostaglandin biosynthesis inhibitor, IC50 = 1.0mol/L); antihepatotoxin

(rat liver cells, in vitro, 1.0mg/mL, liver toxicosis induced by CCl4, GPT =
(801)% of that of control, p<0.01). Source: SHENG JIANG Zingiber
officinale. Ref: 2, 1815, 1817.
O
HO
OH
OH
HO
HO
39
4923 Dehydroglaucine
4928 9(11)-Dehydrohecogenin
[22212-26-6] C21H23NO4 (353.42). Yellow lamellar crystals, mp
C27H40O4 (428.62). mp 230~232C. Source: FAN MA Agave americana,
121~122C. Pharm: Antibacterial (Staphylococcus aureus, Bacillus
WU CI FAN MA Agave americana var. marginata [Syn. Agave
subtilis, and Mycobacterium smegmatis, MIC = 25g/mL); antifungal
americana var. variegata], Agave deserti. Ref: 2503.
(Candida albicans, MIC = 25g/mL; Saccharomyces cerevisiae, MIC =

50g/mL). Source: BEI MEI E ZHANG QIU Liriodendron tulipifera,
O
O
HUANG HAI YING SU Glaucium flavum. Ref: 661.
O
H
H
H
HO
4929 6-Dehydrohinokiol
C21H30O (298.47). Source: TAI WAN SHAN Taiwania cryptomerioides.

Ref: 2526.
4924 Dehydroglyasperin C
C21H22O5 (354.41). Source: CU MAO GAN CAO Glycyrrhiza aspera.
OH
Ref: 2431.
O
HO
OH
4930 Dehydrohirsutanonol
OH
1,7-Di-(3',4'-dihydroxyphenyl)-4-hepten-3-one C19H20O5 (328.37).
4925 Dehydroguggulsterone M
Syrupy solid. Pharm: Antioxidant (superoxide radical scavenger, IC50 =
C22H28O3 (340.47). Amorphous powder, []D = +36.5 (c = 0.76, MeOH)
1.2mol/L; DPPH scavenger, IC50 = 2.4mol/L)[4535]; cytotoxic (TK10,
Source: A MAN SU DAN MO YAO Commiphora wightii. Ref: 2062.
GI50 = 6.8g/mL, control Etoposide, GI 50 = 8.1g/mL; MCF7, GI50 =

1.9g/mL, Etoposide, GI 50 = 0.33g/mL; UACC62, GI50 = 4.8g/mL,
Etoposide, GI 50 = 0.97g/mL)[5195]. Source: CHI YANG Alnus japonica
(leaf), SHI ZI XING HU JI SHENG Viscum cruciatum (aerial parts). Ref:
4535, 5195.
H
O
4926 5',6'-Dehydroguiachrysine
C40H42N4O3+2 (626.81). Orange-brown colored amorphous powder.
Pharm: Neuromuscular toxicity (neuromuscular transmission inhibitor,
IC50 = 21.5mol/L; Venezuelan calabash curare, IC50 = 6.5mol/L).
Source: Strychnos guianensis (stem cortex). Ref: 5202.
N
OH
OH
HO
OH
4931 (13S)-8,9-Dehydro-18-hydroxy-10-epi-ryanodine
contraction force, EC50 = 1500nmol/L). Source: QU CHONG CAO
H
N
HO
OH
HN
OH
OH
OH
HO OH
OH
O
N
H
4927 5',6'-Dehydroguiaflavine
+2
C40H40N4O2 (608.79). Orange-brown colored amorphous powder.
OH
O
4932 8,9-Dehydro-20-hydroxy-10-epi-ryanodine
Pharm: Neuromuscular toxicity (neuromuscular transmission inhibitor,
IC50 = 24mol/L; Venezuelan calabash curare, IC50 = 6.5mol/L). Source:
Strychnos guianensis (stem cortex). Ref: 5202.

contraction force, EC50 = 440nmol/L). Source: QU CHONG CAO

H
N
O
H
HO
HN
OH
OH
OH
N
H
O
O
OH
OH
OH
40
4933 8,9-Dehydro-21-hydroxy-10-epi-ryanodine
4938 11-Dehydroklaineanone
C20H26O6 (362.43). Pharm: Plant growth inhibitor (Cucumber seedling,
root growth, IC50 = (55.61.0)mol/L, shoot growth, IC50 =
(77.31.0)mol/L; Rice seedling, root growth, IC50 > 200mol/L, shoot
contraction force, EC50 = 1900nmol/L)[5139]. Source: QU CHONG CAO
growth, IC50 > 200mol/L). Source: CHANG YE KUAN MU Eurycoma
longifolia (leaf). Ref: 5215.

OH
OH
OH
O
OH
HO OH
OH
O
H
OH
N
H
OH
4939 11,13-Dehydrolanuginolide
C17H22O5 (306.36). Colorless acicular crystals (ether), mp 167C (dec),
4934 Dehydrojinkoheremol
[]D = 96.5 (c = 0.74, CHCl3). Pharm: Cytotoxic (KB, ED50 =
C15H24O (220.36). Source: CHEN XIANG Aquilaria agallocha. Ref: 13.
1.8g/mL). Source: NAN YA HAN XIAO Michelia doltsopa. Ref: 661.
O
O
OH
O
O
4935 Dehydrojuvabione
C16H24O3 (264.37). Pharm: Insect juvenile hormone. Source: XIANG ZHI
LENG SHAN Abies balsamea. Ref: 658.
4940 3,4-Dehydrolarreatricin
Dehydrolarreatricin C18H18O4 (298.34). Pharm: Antioxidant (Takamatsu
DCFH method, myelomonocytic HL-60 cells, IC50 > 62.5g/mL; control
NDGA, IC50 = (0.70.3)g/mL, Vitamin C, IC50 = (1.90.7)g/mL,
Trolox, IC50 = (1.40.5)g/mL)[3850]; cytotoxic (XTT assay, HL-60 cells,

O
IC50 = (27.60.4)g/mL; control NDGA, IC50 = (2.60.2)g/mL, Vitamin

C, IC50 > 10.0g/mL, Trolox, IC50 > 10.0g/mL)[3850]. Source: SAN CHI
LA RUI A Larrea tridentata (leaf). Ref: 1521, 3850.

4936 5,6-Dehydrokawain
[15345-89-8] C14H12O3 (228.25). Pharm: Anticonvulsant; local anesthetic;
OH
cytotoxic inactive (Colon26-L5, HT1080, 100mol/L)[3042]. Source: DA
OH
CAO KOU Alpinia speciosa, DIAO ZHANG GEN PI Lindera umbellata
HO
[Syn. Lindera erythrocarpa], KA WA HU JIAO Piper methysticum, YUN
4941 Dehydroleucodin
NAN CAO KOU Alpinia blepharocalyx (seed: yield = 0.00390%)[3042].
Mesatlantin E [36150-07-9] C15H16O3 (244.29). mp 131C (diethyl
Ref: 658, 3042.
ether petroleum ether), [] 589nm22 = +77; []578nm22 = +81; []546nm22 =

+92; []430nm22 = +155 (c = 2.5, chloroform). Pharm: Antiulcerative (rat
and mus, stomach/duodenum mucous membrane damage caused by
EtOH); cytotoxic (KB ATCC CCL17, IC50 = 1.3g/mL)[5399]. Source:

YAN XIANG JU Chrysanthemum lavandulifolium, YI KUA Artemisia
4937 Dehydrokerlin
myriantha (aerial parts)[4618], Warionia saharae. Ref: 900, 4618, 5399.

O
C20H24O4 (328.41). Source: DUO SUI SHU WEI CAO Salvia

polystachya (aerial parts). Ref: 3901.
O
H
H
4942 Dehydrolindestrenolide
O
[32810-35-8] C15H16O2 (228.29). mp 111~113C. Source: WU YAO

Lindera strychnifolia [Syn. Lindera aggregata]. Ref: 6.
O
O
41
4943 Dehydrologanin
4949 6,12-Dehydromillettone
Ketologanin [152-91-0] C17H24O10 (388.37). Source: CHANG CHUN HUA
C22H16O6 (376.37). Yellow crystals, mp>300C. Pharm: Antimalarial
Catharanthus roseus [Syn. Vinca rosea; Lochera rosea], MA QIAN ZI
(antiplasmodial, chloroquine-resistant W2 strain of Plasmodium
Strychnos nux-vomica, SHAN ZHU YU Cornus officinalis [Syn.
falciparum, IC50 = 33.3mol/L, control Chloroquine, IC50 = 0.094mol/L,
[9]
Macrocarpium officinale] (fruit: yield = 0.00022%dw) . Ref: 2, 9, 639, 660.
control Quinine, IC50 = 0.209mol/L; chloroquine-sensitive D6 strain of

Plasmodium falciparum, IC50 = 39.1mol/L, control Chloroquine, IC50 =
0.009mol/L, control Quinine, IC50 = 0.044mol/L). Source: Millettia
usaramensis ssp. usaramensis. Ref: 3454.
O
H
HO
O
OH
OH
OH
O
O
4944 3,4-Dehydrolycopen-16-al
C40H52O (548.86). Source: QIAN NIAN BU LAN XIN Solanum

4950 Dehydromiltirone
dulcamara. Ref: 6.
1-Dehydromiltirone C19H20O2 (280.37). Red acicular crystals, mp

45~46C; red oleaginous substance. Source: HONG GEN CAO Salvia
prionitis, DAN SHEN Salvia miltiorrhiza. Ref: 102, 116.
O
4945 9(11)-Dehydromanogenin
C27H40O5 (444.62). mp 240C. Source: FAN MA Agave americana, WU
CI FAN MA Agave americana var. marginata [Syn. Agave americana var.
variegata], Agave deserti. Ref: 2503.
4951 Dehydromorroniaglycone
O
O
C11H14O5 (226.23). White crystals, mp 119~120C, []D21 = 47.17 (c =

O
0.053, EtOH). Source: SHAN ZHU YU Cornus officinalis [Syn.
HO
Macrocarpium officinale] (fruit: yield = 0.00044%dw)[9]. Ref: 9, 479,

H
HO
5502.
O
4946 Dehydromatricaria ester

Methyl-cis-2-decen-4,6,8-triynate [2739-57-3] C11H8O2 (172.19). mp
H
O
114~115C. Source: AI YE Artemisia argyi, QI ZHOU YI ZHI HAO
Conyza canadensis [Syn. Erigeron canadensis]. Ref: 6.

4952 1,2-Dehydroneomajucin
C15H18O7 (310.31). Amorphous solid, []D20 = 7.8 (c = 0.16, EtOH).

H
Source: JIA DI FENG PI Illicium jiadifengpi (pericarp: yield =
0.00013%dw). Ref: 4621.
4947 trans-Dehydromatricaria ester

Methyl-trans-2-decene-4,6,8-triynoate [692-94-4] C11H8O2 (172.19). mp
O
HO
O
105C. Source: BI MA GEN Ricinus communis, DA YE BAI TOU
OH
O
WENG Anaphalis margaritacea. Ref: 6.

O
HO
O
O
H
4948 7,11-Dehydromatrine
[46862-63-9] C15H22N2O (246.36). Source: KU SHEN Sophora
flavescens [Syn. Sophora angustfolia]. Ref: 2.
4953 2,3-Dehydroneomajucin
C15H18O7 (310.31). Source: JIA DI FENG PI Illicium jiadifengpi
(pericarp). Ref: 4621.
O
HO
O
OH
O
N
H
H
HO
42
4954 Dehydroneotenone
4960 Dehydropinguisenol
C19H12O6 (336.30). Source: DI GUA ZI Pachyrhizus erosus. Ref: 4180.
C15H20O2 (232.33). Source: YE TAI Trocholejeunea sandvicensis. Ref:

3909.
OH
4961 Dehydropipernonaline
4955 Dehydroodorine
C18H22N2O2 (298.39). Source: DA YE SHU LAN Aglaia elliptifolia (leaf:
C21H25NO3 (339.44). Colorless crystals. Pharm: Protective gastric lesions
yield = 0.00104%dw). Ref: 3031.
(rat, ethanol-induced, 25mg/kg orl, length = (50.614.2)mm, control,

length = (118.616.2)mm, InRt = 57.3%; indomethacin-induced in rats,
dose, 25mg/kg orl, length = (34.111.0)mm, control, length =
H
N
(89.59.8)mm, InRt = 61.9%). Source: Piper chaba (fruit). Ref: 4935.

O
4956 (+)-2,3-Dehydro-10-oxo--isosparteine
C15H22N2O (246.36). Colorless needles, mp 98~103, []D26 = +132 (c =
0.6, EtOH). Source: FA GUO JIN QUE ER Cytisus monspessulanus. Ref:

4962 Dehydropodophyllotoxin
1943.
C22H18O8 (410.38). mp 275~276C. Source: GUI JIU Dysosma versipellis
O
H
N
[Syn. Podophyllum versipelle], LIU JIAO LIAN Dysosma pleiantha [Syn.
YE Diphylleia grayi, TAO ER QI Podophyllum emodii [Syn.
Podophyllum pleianthum] (rhizome: content = 0.019%)[5508], SHAN HE
4957 Dehydrooxoperezinone
Podophyllum emodii var. chinense; Podophyllum sikkimenosis;
C15H14O4 (258.28). Orange needles (CHCl3/CH3OH), mp > 280C. Pharm:
Sinopodophyllum emodii] (rhizome: mean content of 2 origins =
Anti-HIV (in vitro, acutely infected H-9 lymphocyte cells, IC50 =
0.037%)[5508], WO ER QI Diphylleia sinensis (rhizome: mean content of 4
25.1g/mL, EC50 = 17.5g/mL, TI = 1.43); cytotoxic inactive (in vitro,
origins = 0.072%[5508]). Ref: 6, 279, 5508.

OH
MCF7 and A549). Source: GUAN MU TONG Aristolochia

manshuriensis (stem: yield = 0.00069%). Ref: 4706.
O
O
O
O
HO
O
O
4958 3,4-Dehydropalicoside
C27H33N2O9+ (529.57). Amorphous powder, []D25 = 27 (c = 0.175,
MeOH). Source: Strychnos vanprukii (stem). Ref: 3471.
4963 7-Dehydroporiferasterol
Corbisterol [19432-13-4] C29H46O (410.69). Pharm: Anti-inflammatory
(inflammation caused by TPA in mus, 1mg/ear, InRt = 85%, ID50 =
0.5mg/ear). Source: YAN CAO Nicotiana tabacum. Ref: 900.
N
H
HO
H
O
O
O HO
O
OH
OH
OH
HO
4959 7,8-Dehydropenstemoside
4964 Dehydroprotostemonine
C17H24O11 (404.37). Colorless powder, mp 119~120C. Source: DU YI
C23H29NO6 (415.49). Amorphous, []D20 = +72 (c = 0.3, MeOH). Pharm:
WEI Lamiophlomis rotata [Syn. Phlomis rotata]. Ref: 381.
Insecticidal (neonate larvae of Spodoptera littoralis, LC50 = 6.1mg/L,
HO HO
EC50 = 0.8mg/L). Source: DI TANG BAI BU Stemona kerrii, Stemona

curtisii. Ref: 3409.
OO
HO
OH
O
OH
N H
H
OH
43
4965 6,7-Dehydroroyleanone
4971 7-Dehydrostigmasterol
C20H26O3 (314.43). Red crystals, mp 160~164C. Source: XIU QIU SHU
C29H50 O (414.72). Source: HUANG BAI Phellodendron amurense.
WEI CAO Salvia hydrangea (root). Ref: 5447.
Ref: 2.
H
OH
O
H
O
HO
4972 16-Dehydrostrophanthidin
4966 Dehydrosafynol
C23H30O6 (402.49). mp 226C; 253~262C, []D = +82.3. Source: HEI
C13H10O2 (198.22). Pharm: Plant antitoxin. Source: HONG HUA
GANG LIU Periploca nigrescens. Ref: 1521, 2498.
Carthamus tinctorius. Ref: 658.
O
H
OH
OH
H
OH
4967 Dehydro--sanshool
HO
OH
C18H25NO (271.41). Pharm: Anti-PAF. Source: Zanthoxylum sp. Ref:

2176.
4973 16-Dehydrostrophanthidol
C23H32O6 (404.51). mp 242~247C, []D = 68.9. Source: HEI GANG LIU
Periploca nigrescens. Ref: 1521, 2498.
H
N
HO
4968 Dehydroshikimic acid

C7H8O5 (172.14). mp 150~152C; 201~202C. Source: HE ZI Terminalia
chebula, HE ZI YE Terminalia chebula. Ref: 6.
OH
4974 1-Dehydrotanshinone
OH
OH
HO
C19H16O3 (292.34). Dark red acicular crystals, mp 147~148C. Source:

DAN SHEN Salvia miltiorrhiza. Ref: 116.
HO
OH
4969 7-Dehydrosophoramine
O
[67767-18-4] C15H18N2O (242.32). Source: HUANG BAI Phellodendron

amurense. Ref: 2.
O
4975 8,9-Dehydrothymol 3-O-tiglate
C15H18O2 (230.31). Source: PEI LAN Eupatorium fortunei (aerial parts).
H
H
Ref: 3077.
N
O
4970 Dehydrostephalagine
C19H17NO3 (307.35). Pharm: Cytotoxic inactive (yeast assay:

RS321NYCp50(gal), RS321NpRAD52(gal), RS321NpRAD52(glu)).
Source: DING KE LA QIAN JIN TENG Stephania dinklagei (stem). Ref:
(goldfish). Source: QIAN MA YE ZE LAN Eupatorium urticaefolium.
Ref: 658.
O
O
4976 Dehydrotremetone
[3015-20-1] C13H12O2 (200.24). Pharm: Antibacterial; fish toxin
5457.
O
O
44
4981 1-Dehydroxybaccatin VI
4977 4-O-8',5'-5''-Dehydrotriferulic acid

C30H26O12 (578.53). Source: YU MI FU Zea mays (bran). Ref: 3420.
C37H46O13 (698.77). Colorless crystals, mp 220~221C, []D = 21.2

(CHCl3). Source: JIE ZHI HONG DOU SHAN Taxus media, MEI LI
OH
HONG DOU SHAN Taxus mairei. Ref: 139, 662.

O
O O
OH
HO
O
O
O
OH
H O
OH
O
O
4978 Dehydrotumulosic acid
4982 4-Dehydroxycrinamabine
C31H48O4 (484.73). Pharm: Antineoplastic (EBV-EA induced by TPA,
C16H19NO4 (289.33). Pharm: Antitrypanosomal (Trypanosoma brucei rhodesiense
mol ratio/TPA = 1000, relative percentage of EBV-EA = 0% (positive
strain STIB-900, stage trypomastigotes, IC50 = 11.07g/mL); antimalarial
control value 32pmol, 20ng TPA =100%), viability of Raji cells = 70%;
inactive (Plasmodium falciparum strain NF-54, stage IEF). Source: GUAN
reference compound -Carotene, relative percentage = 8.6%). Source: FU
MU WEN SHU LAN Crinum macowanii (bulb). Ref: 4000.
LING Poria cocos (sclerotium: yield = 0.00084%dw). Ref: 4616.
OH
HO
O
H
HO
OH
4983 Dehydroxycubebin
C20H20O5 (340.38). Source: QIANG DAO YAO Hypoestes purpurea [Syn. Justicia
purpurea; Hypoestes sinica] (aerial parts: yield = 0.000034%dw). Ref: 4783.
HO
4979 1-Dehydroxybaccatin III

4984 1-Dehydroxy-4-deacetylbaccatin IV
C30H42O12 (594.66). Source: MEI LI HONG DOU SHAN Taxus mairei. Ref: 662.
O
O O
OH
O O
O
HO
H O
H
O
O
O
O
O
H
OH
4985 Dehydroxyhexaspermone C
rel-4',7-Dimethoxy-4-oxo-2,3-trans-isoflavanyl-(22'')-4'',5''-dihydroxy4980 1-Dehydroxybaccatin IV
7''-methoxy-2'',3''-trans-isoflavanone C33H28O9 (568.59). White or
C32H44O13 (636.70). Colorless prisms, []D = +5 (CHCl3), mp 286C, mp
colorless solid, mp 133~135C, [] D23.7 = 117.0 (c = 0.05, MeOH).
259~260C, []D = +99 (CHCl3). Pharm: NO production inhibitor (IC50

= 32.2mol/L, control L-NMMA, IC50 = 28.5mol/L)[5407]. Source:
Pharm: Antibacterial inactive (MDR Staphylococcus aureus: RN4220

strain, 64g/mL, control Erythromycin, MIC = 128g/mL; XU212
HONG DOU SHAN Taxus chinensis, JIE ZHI HONG DOU SHAN Taxus
strain, 64g/mL, control Tetracycline, MIC = 128g/mL; SA-1199-B
media, YUN NAN HONG DOU SHAN Taxus yunnanensis (wood). Ref:
strain, 64g/mL, control Norfloxacin, MIC = 32g/mL). Source:
662, 2488, 5407.
CHANG E JIN LIAN MU PI Ochna macrocalyx. Ref: 5372.
O
O O
HO
O
O
H O
H
O
O
OH
H
H
H
O
45
4986 6-Dehydroxylongilactone
4990 Delafrine
6-Dehydrolongilactone C19H26O6 (350.42). Pharm: Cytotoxic (P388, IC50 =
C27H45NO3 (431.66). Source: XI BEI MU Fritillaria imperialis (bulb).
0.66g/mL, A549 cells, remarkable activity, MCF7 cells, IC50 <
Ref: 4217.
2.5g/mL)[4556]; plant growth inhibitor (Cucumber seedling, root growth,

IC50 = (25.70.5)mol/L, shoot growth, IC50 = (48.60.5)mol/L; Rice
seedling, root growth, IC50 > 200mol/L, shoot growth, IC50 >
[5215]
200mol/L)
. Source: CHANG YE KUAN MU Eurycoma longifolia
HO
HO
OH
O
O
O
OH
OH
(leaf), Eurycoma sp. Ref: 4556, 5215.
OH
4991 Delajacine
C37H54N2O9 (670.85). White amorphous powder. Source: QIN LING CUI
QUE HUA Delphinium giraldii. Ref: 2506.
4987 2-Dehydroxy-5-O-methylembelin
C18H28O3 (292.42). Pharm: Cytotoxic inactive (in vitro, HL-60, IC50 >
O
100g/mL; Bel7402, IC50 > 100g/mL; HeLa, IC50 > 100g/mL; U937,
O
O
H
H
IC50 > 100g/mL; control Colchicine, HL-60, IC50 = 1.6g/mL; Bel7402,
IC50 = 0.4g/mL; HeLa, IC50 = 0.1g/mL; U937, IC50 = 0.1g/mL)[4746].
Source: LA ZHU GUO Aegiceras corniculatum (stem and twig: yield =
0.00005%). Ref: 4746.
NH
OH
OH
O
O
O
4992 Delamide
C13H16N2O4 (274.28). Source: FU ZI Aconitum carmichaeli. Ref: 16.
O
O
4988 Deidaclin
H
N
C12H17NO6 (198.22). Pharm: Toxin. Source: GE YANG XI FAN LIAN
NH2
O
Passiflora coriaceae. Ref: 658.
4993 Delavaconitine
[1356-52-1] C29H39NO6 (497.64). mp 59~64C, []D17 = 9.56; nitrate:
mp 154C; perchlorate: mp 241C; picrolonate: mp 241C; chloraurate:
OO
HO
OH
mp 215C. Pharm: Analgesic; local anesthetic; LD (rbt, iv) = 5~10mg/kg,

N
OH
(dog, iv) = 10~12mg/kg; LD50 (mus, sc) = 106mg/kg, (mus, iv) =
OH
28mg/kg. Source: MA ER SHAN WU TOU Aconitum delavayi. Ref: 661.
4989 Deisobutyryl bakkenolide H

O
93.0 (c = 0.365, MeOH). Pharm: Platelet aggregation inhibitor

(100mol/L AA-induced, 100g/mL, InRt = (91.76.8)%, p<0.001,
thrombin-induced, 100g/mL, InRt = (1.11.1)%). Source: TAI WAN

FENG DOU CAI Petasites formosanus. Ref: 2377.
OH
H
collagen-induced, 100g/mL, InRt = (85.513.0)%, p<0.001, Aspirin,

(21.01.7)%, p<0.001, Aspirin, 50g/mL, InRt = (9.61.2)%; 0.1g/mL
4994 Delavaine
[27989-72-6] C20H23NO5 (357.41). mp 140~150C. Source: DI BU
RONG Stephania delavayi [Syn. Stephania epigaea]. Ref: 1521.
O
O
O
O
O
O
control Aspirin, 50g/mL, InRt = (1000.0)%; 10g/mL

50g/mL, InRt = (12.21.7)%; 2nmol/L PAF-induced, 100g/mL, InRt =
HO
C19H28O5 (336.45). Colorless needles (MeOH), mp 178~180C, [] D =
OH
O
O
O
46
4995 Delavayine A
4999 Delbruline
C19H28NO2 (302.44). Yellow powder, []D22 = 5.1 (c = 0.90, C5H5N).
[106982-82-5] C26H41NO7 (479.62). Source: FU ZI Aconitum carmichaeli.
Pharm: Antinociceptive (acetic acid-induced, 50mg/kg, sc, inhibitive
Ref: 16.
percent = 45%; control Aminopyrine, 50mg/kg, orl, inhibitive percent =
87%, 50mg/kg, sc, inhibitive percent = 94%). Source: MA TONG HUA
Incarvillea arguta]. Ref: 3908.
O
H
OH
H
H
O
5000 Delbrunine
4996 Delavine
[98243-57-3] C27H45NO2 (415.67). Colorless needles (EtOH), mp
Ref: 16.
179~182C (dec), []D25 = 17.2 (c = 0.5, CHCl3). Pharm: cAMP
phosphodiesterase inhibitor (IC50 = 88mol/L); AChE inhibitor (IC50 =

(105.51.5)mol/L, control Eserine, IC 50 = (0.410.01)mol/L)
[4217]
OH
control Eserine, IC50 = (0.8570.008)mol/L)
OH
H
butyrylcholinesterase (BChE) inhibitor (IC50 = (1.710.11)mol/L,

[4217]
. Source: LENG SHA
O
H
BEI MU Fritillaria delavayi, XI BEI MU Fritillaria imperialis (bulb).
Ref: 2, 660, 1755, 4217.

5001 Delbrusine
N
H
H
HO
Ref: 16.
O
H
OH
O
H
4997 Delavinone
[96997-98-7] C27 H 43 NO 2 (413.65). Source: LENG SHA BEI MU
Fritillaria delavayi, GAN SU BEI MU Fritillaria przewalskii. Ref:

2, 660.
5002 Delcarduchol
C21H27NO3 (341.45). Source: Delphinium carduchorum. Ref: 2288.
N
H
OH
H
H
HO
5003 Delcorine
4998 Delbonine
[95066-33-4] C27H43NO8 (509.65). Amorphous solid, []D = +35.3 (c =
[52358-55-1] C26H41NO7 (479.62). Pharm: Inhibits intestinal contraction
0.8, CHCl3). Source: CHUAN QIAN CUI QUE HUA Delphinium
(rat and rbt, in vitro); inhibits respiration; uterine relaxant (gpg);
bonvalotii, DONG FANG FEI YAN CAO Consolida orientalis (aerial
antihypertensive. Source: GUANG FEI YAN CAO Delphinium
parts). Ref: 1521, 4283.
corumbosum. Ref: 658.
25
H
OH
O
H
H
N
H
OH
H
H
O
O
O
H
OH
47
5004 Delcosine
5009 Delphicrispuline
Delphamine [545-56-2] C24H39NO7 (453.58). mp 203~204C. Pharm:
Neofinaconitine C30H42N2O6 (526.68). []D20 = +23.8 (c = 0.8, CHCl3)
Antihypertensive (anesthetic, cat, 10mg/kg); toxin (poikilotherms).
Source: GAN WAN WU TOU Aconitum finetianum, TU ER QI CUI QUE
Source: FEI YAN CAO Consolida ajacis [Syn. Delphinium ajacis],
HUA Delphinium crispulum. Ref: 1913, 2690.
QIANG GU FEI YAN CAO Delphinium consolida, XIAO CAO WU

Delphinium yunnanense. Ref: 6, 16, 658.
H
H
OH
N
NH2
OH
OH
H
O
H
OH
H
OH
5005 Delectine
[58485-71-5] C31H44N2O8 (572.70). White amorphous powder. Source: E
5010 Delphin
MEI CUI QUE HUA Delphinium omeiense. Ref: 2190.
Delphinidin-3,5-diglucoside [17670-06-3] C27H31O17+ (627.54). Source:
H
O
O
OH
H
BAI FAN DOU Phaseolus vulgaris, FEI YAN CAO Consolida ajacis
[Syn. Delphinium ajacis], MU XU Medicago sativa, QIE ZI Solanum
melongena, YA ZHI CAO Commelina communis. Ref: 6.
OH
OH
HO
OH
NH2
OH
OH
OH
[58480-82-3] C24H39NO7 (453.58). White amorphous powder. Source: E
Delphinidol C15H11O7+ (303.25). Pharm: Pigment; leukocyte elastase
OH
H
MMP-2/9 inhibitor[4416]. Source: BU XUE CAO Limonium gmelinii,
N
H
HO
FENG XIAN HUA Impatiens balsamina, PU(3) TAO Syzygium jambos,
OH
OH
OH
5011 Delphinidin
OH
OH
MEI CUI QUE HUA Delphinium omeiense. Ref: 2190.

H
OH
OH
5006 Delectinine
OH
O
OH
TAO ER QI Podophyllum emodii [Syn. Podophyllum emodii var.

chinense; Podophyllum sikkimenosis; Sinopodophyllum emodii]. Ref: 6,
658, 4416.
5007 Delgrandine
C41H43NO12 (741.80). Source: FU ZI Aconitum carmichaeli. Ref: 16.
O
HO
+
OH
HO
O
O
OH
HO
O
O
OH
OH
5008 Delphatine
[25488-62-4] C26H43NO7 (481.64). Pharm: Anti-inflammatory (modified assay
5012 Delphinidin-3-arabinoside
of Berridge, 100g/mL, InRt = 17.39%)[5271]; tyrosinase inhibitor inactive
[28500-01-8] C20H19O11+ (435.37). Source: ZI WEI HUA Lagerstroemia
(control Kojic acid, IC50 = (16.670.52)mol/L, L-Mimosine, IC50 =
indica. Ref: 6.
(3.680.02)mol/L)[5271]; antioxidant (DPPH scavenger, 1mol/L, ScRt = 55.4%;

OH
control 3-t-Butyl-4-hydroxyanisole, 1mol/L, ScRt = 92.5%)[5271]. Source: FU
H
H
OH
N
H
OH
OH
ZI Aconitum carmichaeli, Aconitum leave (aerial parts). Ref: 16, 5271.
HO
OH
OH
O
OH
OH
OH
48
5013 Delphinidin-3-O-[2-O-(2-O-(trans-caffeoyl)--D-glucopyranos-
yl)--D-galactopyranoside]-7-O-[6-O-(trans-caffeoyl)--D-glucopyra-
yl)-6-O-(2-O-(tartaryl)malonyl)--D-galactopyranoside]-7-O-[6-O-(tra
noside]-3'-O-[-D-glucuronopyranoside]
ns-caffeoyl)--D-gluco-pyranoside]-3'-O-[-D-glucuronopyranoside]
C57H61O34+ (1290.10). Source: HUA GUAN YIN LIAN HUA Anemone
coronaria. Ref: 1956.

OH
OH
OH
OH
OO
OH
HO
O
OH
OH
HO
OH
HO
OH
OH
HO
OH
OO
O
OH
OH
HO
OH
OO
OH
OH
OH
OH
OH
OH
O
OH
O OH
HO
OH
OH
O
O
OH
O
OH
O
OH HO HO
O
O
O
OH
O
OH
OO
OH
O
OH
O
OH
OH
OH
5017 Delphinidin-3-O-[6-O-(p-coumaroyl)--D-glucopyranoside]5-O-[4-O-acetyl-6-O-malonyl--D-glucopyranoside]
C41H41O23+ (901.77). Source: Salvia uliginosa. Ref: 2367.

OH
OH
yl)-6-O-(malonyl)--D-galactopyranoside]-7-O-[6-O-(trans-caffeoyl)-
-D-glucopyranoside]-3'-O-[-D-glucuronopyranoside]
O
OH
OO
OH
HO
OH O
HO
O
HO
OH
OH
O OH
OH
HO
O
OH
OH
OH
OH
OH
OH
OH
OO
O
O
OH
O
OH
O
HO
HO
OH
O
OH
5018 Delphinidin-3-O--D-(6-(E)-p-coumaryl) galactopyranoside

C30H27O14+ (611.54). Source: CHA YE Camellia sinensis [Syn. Thea
OH
OH
OO
sinensis]. Ref: 759.

OH
OH
OH
OH
OH
HO
O
HO
OH
HO
OH
O
OH
yl)-6-O-(2-O-(tartaryl)malonyl)--D-galactopyranoside] -7-O-[6-O-
OH
(trans-caffeoyl)--D-glucopyranoside]
5019 Delphinidin-3,7-di-O--glucopyranoside-3',5'-di-O-(6-O-p-cou-
maroyl--glucopyranoside)
C57H63O31+ (1244.12). Source: TA SI MA NI YA JIE GENG LAN Dianella

tasmanica (berry), HEI JIE GENG LAN Dianella nigra (berry). Ref: 5214.
O
OH
OH
O
OO
HO
OH HO HO O
OH
O
OO
OH
OH
OH HO
OH
O
OH
OH
OH
OH
O
OH
O
OH
OH
OH
OH
OH
O
OH
O HO
HO
OO
OH
OH
O
OH
HO
OO
O
OH
HO
OH
OH
OH
OH
OH
OH
49
5020 Delphinidin-3-diglucoside
5025 Delphinidin-3-O-(-D-glucopyranoside)-5-O-(6-O-malonyl-(-
C27H31O17+ (627.54). Source: SHUI HU LU Eichhornia crassipes. Ref: 6.
D-glucopyranoside
C30H33O20+ (713.59). Source: HE LAN ZHONG ZHI FAN HONG HUA
OH
Crocus antalyensis cv. Ref: 1897.
HO
OH
OH
OH
HO
OO
OO
OH
OH
OH
HO
OH
OH
OH
HO
OH
OH
5026 Delphinidin-3-O--D-glucopyranoside-7,3',5'-tri-O-(6-O-p-couOH
OH
O
HO
OO
O
OH
OH
maroyl--glucopyranoside)
C66H69O33+ (1390.27). Source: TA SI MA NI YA JIE GENG LAN
Dianella tasmanica (berry), HEI JIE GENG LAN Dianella nigra (berry).
Ref: 5214.
OH
OH
OH
O
O
OH
HO
Empetrin [68852-84-6] C21H21O12+ (465.39). Source: CHA YE Camellia

sinensis [Syn. Thea sinensis]. Ref: 759.
OO
O
OH
OH
HO
OH
OH
OH
[6906-38-3] C21 H21O12+ (465.39). Source: BAI FAN DOU Phaseolus

vulgaris, HEI DA DOU PI Glycine max, QIE ZI Solanum melongena.
Ref: 6.
C30H27O17+ (659.54). Source: LAN SHUI LIAN Nymphaea caerulea. Ref: 1863.
OH
HO
HO
OH
OO
OH
OH
OH
HO
OH
O
O
OH
HO
OH
5027 Delphinidin-3-glucoside
5023 Delphinidin-3'-O-(2''-O-galloyl-6''-O-acetyl--galactopyranoside)
HO
OH
OH
5028 Delphinidin-3-O-(6-O-malonyl--D-glucoside)-5-O--D-gluco-
OH
OH
side
5024 Delphinidin-3'-O-(2''-O-galloyl--galactopyranoside)
C30H33O20+ (713.59). Source: JU QU Cichorium intybus. Ref: 1955.
C28H25O16+ (617.50). Source: LAN SHUI LIAN Nymphaea caerulea. Ref: 1863.
OH
HO
OH
OH
OH
OH
HO
OH
O
O
OH
HO
O
OH
OH
HO
OH HO
O
O
OH
OH
OH
OH
OH
OH
OH
O
O
OH
5022 Delphinidin-3-O--D-galactopyranoside
HO
OH
OH
C33H35O23 (799.63). Source: JU QU Cichorium intybus. Ref: 1955.
HO
O
OH
OH
OH
HO
OO
5021 Delphinidin-3,5-di-O-(6-O-malonyl--D-glucoside)
HO
OH
HO
OH
OH
HO
OH
OH
OH
HO
O
O
O
HO
OH
O
OH
HO
OO
HO
OH
OH
OH
HO
OH
O
OH
OH
OH
OH
OH
50
5029 Delphinidin-3-neohesperidoside
5033 Delsemine A
C24H23O15 (551.44). Dark red amorphous powder. Source: HU DIE HUA
C37H53N3O10 (699.85). []D30 = +368 (c = 0.7, CHCl3). Source: E MEI
DOU Clitoria ternatea (petal). Ref: 3480.
CUI QUE HUA Delphinium omeiense, FU ZI Aconitum carmichaeli.

Ref: 16, 2190.
OH
OH
HO
OH O
OH
OH
OH
OH
OH
OH
O
NH
OH
NH2
5030
Delphinidin-3-O-(2''-O--rhamnosyl-6''-O-malonyl)--glucoside
C30H33O19 (697.59). Dark red amorphous powder. Source: HU DIE HUA
5034 Delsemine B
DOU Clitoria ternatea (petal). Ref: 3480.
C37H53N3O10 (699.85). []D30 = +28.2 (c = 0.6, CHCl3). Source: E MEI CUI

QUE HUA Delphinium omeiense, FU ZI Aconitum carmichaeli. Ref: 16, 2190.
OH
OH
HO
OH
O
H
OH O
OH
OH O O
HO
OH
OH
OH
NH
NH2
O
OH OH
5031
5035 Delsoline
Delphinidin-3,7,3',5'-tetra-O-(6-O-p-coumaroyl--glucopyranoside)
[509-18-2] C25H41NO7 (467.61). mp 213.0~216.5C. Pharm: Causes
C75H75O35 (1536.41). Source: TA SI MA NI YA JIE GENG LAN Dianella
paroxysm convulsion and breath inhibition (mus, administration by
tasmanica (berry), HEI JIE GENG LAN Dianella nigra (berry). Ref:
non-intestinal tract); insecticidal; antihypertensive (anesthetic cat and dog,
5214.
5~15mg/kg); smooth muscle relaxant. Source: E MEI CUI QUE HUA

Delphinium omeiense, FEI YAN CAO Consolida ajacis [Syn. Delphinium
HO
ajacis], GAN WAN WU TOU Aconitum finetianum, QIANG GU FEI
OH
OO
YAN CAO Delphinium consolida, SHAN DI WU TOU Aconitum
OH
OH
OH
monticola. Ref: 6, 658, 2190.

H
OH
OH
O
OH
OH
OH O OH
O
OO
OH
OH
OH
H
O
OH
OH
O
H
OH
OH
OH
OH
5036 Deltaline
[6836-11-9] C27H41NO8 (507.63). Pharm: Antispasmodic;
HO
antihypertensive (rat, iv, 20mg/kg). Source: FU ZI Aconitum carmichaeli,
5032 Delphinine
[561-07-9] C33H45NO9 (599.73). Pharm: Inhibits respiration; similar
action with aconitine. Source: SI TA WEI CUI QUE HUA Delphinium
staphisagria. Ref: 658.
GAO FEI YAN CAO Delphinium elatum, WANG GUO CUI QUE HUA
Delphinium dictyocarpum, XI FANG CUI QUE Delphinium occidentale,
YI LI CUI QUE HUA Delphinium iliense. Ref: 16, 658.
H
OH
O
H
H
O
O
OH
O
O
H
O
O
H
O
O
51
5037 Deltamine
5041 Deltoside
C51H82O23 (1063.21). Pharm: Raw material for partial synthesis of
Ref: 16.
steroid hormone (its diosgenin is used). Source: SAN JIAO

YE SHU YU Dioscorea deltoidea, XIAO HUA DUN YE SHU YU
H
Dioscorea parviflora. Ref: 10.
O
OH
O
H
HO
O
H
OH
OH
OH
5038 Deltatsine
[92631-66-8] C25H41NO7 (467.61). Amorphous powder, +1H2O, []D20 =
+28.6 (c = 2.4, EtOH). Source: E MEI CUI QUE HUA Delphinium
HO
omeiense, KANG DING CUI QUE HUA Delphinium tatsienense. Ref:

1521, 2190.
OH
H
OO
O OOH
OO
OH
O
H
OH
HO
OH
O
OH
OH
OH
OH OH
H
N
O
H
5042 Demethoxybergenin
OH
C13H15O8 (298.25). Colorless needles, mp 305C (dec., MeOH), []D20 =

22.7 (c = 0.08, MeOH). Pharm: Cytotoxic inactive (murine breast
cancer cell line FM3A, 100mol/L). Source: YOU SE ZI JIN NIU
5039 Deltoin
Ardisia colorata (fruit). Ref: 4244.
[19662-71-6] C19H20O5 (328.37). Source: FANG FENG Saposhnikovia

divaricata [Syn. Ledebouriella seseloides], YUN QIAN HU Peucedanum
OH
rubricaule. Ref: 2, 177.
OH
OH O
H
O
O
HO
OH
5040 Deltonin
5043 6-Demethoxycapillarisin
Trilloside A [55659-75-1] C45H72O17 (885.07). mp 290~292C. Pharm:
C15H10 O6 (286.24). Source: YIN CHEN HAO Artemisia capillaris.
Raw material for partial synthesis of steroid hormone (its aglucon is
Ref: 2.
used); phosphatase inhibitor (HeLa cell stimulated by TPA and joined by

32
P)[2165]. Source: SAN JIAO YE SHU YU Dioscorea deltoidea, SHAN
HO
YAO Dioscorea batatas [Syn. Dioscorea opposita], XIAO HUA DUN YE
OH
SHU YU Dioscorea parviflora, YU ER QI Trillium camtschaticum, ZA
OH
JIAO BAI HE Lilium speciosum x L. nobilissimum. Ref: 6, 10, 658, 2165.
O
O
H
H
HO
5044 Demethoxy-cochinchinone D
C23H24O6 (396.44). Pharm: Antioxidant inactive (DPPH scavenger,
50mol/L, ScRt = 5.2%; control BHT, 50mol/L, ScRt = 51.7%, IC50 =
28.9mol/L)[4423]. Source: HUANG NIU MU Cratoxylum cochinchinense
(root). Ref: 4423.
OO
OH
HO
OH
OO
OH O O
O
O
OH
OH
OH
OH OH
O
OH
52
5045 Demethoxycurcumin
5051 6''-Demethoxyneocalycopterone
1-(4-Hydroxy-3-methoxyphenyl)-7-(4-hydroxyphenyl)-1,6-heptadiene-3,5-dio
C34H32O9 (584.63). Pale amorphous solid, mp 157~159C (Et2O petrol),
ne C20H18O5 (338.36). Yellow needles, mp 180~181C. Pharm:
[]D20 = 199.14 (c = 0.350). Source: E CHI TENG Calycopteris
Neuroprotective (in vitro protects PC12 cells from -Amyloid insult:
floribunda (green part). Ref: 3779.
anti-A(25-35), ED50 = (4.00.5)g/mL; anti-A(1-41), ED50 =

(5.00.5)g/mL; control Congo red: anti-A(25-35), ED50 = (37.55.4)g/mL;
anti-A(1-41), ED50 = (39.25.2)g/mL). Source: JIANG HUANG Curcuma
O
longa (turmeric powder: yield = 0.0012%dw). Ref: 4643.

O
HO
O
O
O
OH
HO
O
O
5046 (+)-5'-Demethoxyepiexcelsin
C21H20O7 (384.39). Colorless crystals (Me2CO), []D20 = +116.3 (c =
1.35, CHCl3) Source: DIE DA LAO Litsea verticillata. Ref: 1984.
O
Source: YE XIA ZHU Phyllanthus urinaria. Ref: 3410.
O
H
5052 5-Demethoxyniranthin
C23H30O6 (402.49). White amorphous solid, []D25 = +15.4 (c = 0.19).
O
O
5047 5-Demethoxyfumagillol
(3R,4R,6R)-4-[(2R,3R)-2-Methyl-3-(3-methyl-but-2-enyl)-oxiranyl]-1-oxa
O
-spiro[2,5]octan-6-ol C15H24O3 (252.36). Colorless oil. Pharm:
Anti-angiogenic (angiogenesis inhibitor, calf CPAE cell, IC50 =

7.06mol/L, control TNP-470, IC50 = 0.0011mol/L, mus L5178Y cell,
5053 18-Demethoxypubescenine
IC50 > 39.6mol/L, control TNP-470, IC50 > 24.5mol/L). Source: YAN
C25H39NO7 (465.59). Amorphous solid, []D25 = +1.1 (c = 0.4, CHCl3).
QU MEI Aspergillus fumigatus. Ref: 4061.
Source: DONG FANG FEI YAN CAO Consolida orientalis (aerial parts).
Ref: 4283.
H
H
OH
O
H
H
OH
N
O
5048 Demethoxymatteucinol
C17H16O4 (284.31). []D25 = 48.1 (c = 0.52, acetone). Source: YANG PU

TAO YE Syzygium samarangense. Ref: 4100.
OH
OH
5054 Demethoxypurpeline
C20H22N2O (306.41). Yellow amorphous solid Source: BA XI LUO FU
HO
MU Rauvolfia bahiensis. Ref: 1952.
O
OH
5049 6-Demethoxy-4'-methoxylcapillarisin
C16H12O6 (300.27). Source: YIN CHEN HAO Artemisia capillaris. Ref: 2.
5055 7-Demethoxytylophorine
Antofine C23H25NO3 (363.46). Yellow needles (MeOH CHCl 3), [] D26 =
HO
115.30 (c = 0.477, CHCl3); colorless gum, [] D21 = 58.3 (c = 0.11, CHCl3).
Pharm: Cytotoxic (inhibits growth of hmn cancer cells, hmn lung cancer cells
O
OH
A549, IC50 = (7.00.2)ng/mL, control Ellipticine, IC50 = (50025)ng/mL; hmn

colon cancer cells Col2, IC50 = (8.60.3)ng/mL, Ellipticine, IC50 =
5050 11-Demethoxymyrtoidine
(34035)ng/mL; action mechanism is to arrest in the G2/M phase of cell
C22H24N2O4 (380.45). Crystals (EtOAc n-hexane), mp 237~240C,
cycle)[5342]. Source: NIU XIN PIAO ZI Cynanchum komarovii, XU CHANG
20
[]D = 28.9 (c = 0.4, CH2Cl2). Source: Strychnos myrtoides. Ref: 2297.
QING Cynanchum paniculatum (root). Ref: 2206, 5342.

O
O
N H
N
O
H
H
O
O
O
53
5056 14-Demethyl-14-acetylanhweidelphinine
5062 DemethylaristofolinE
C36H44N2O11 (680.76). Amorphous, []D25 = +67.1 (c = 0.16, CHCl3).
3,4-Methylenedioxyphenanthrene-1-carboxylic acid C16H10O4 (266.26).
Source: WU ZHU FEI YAN CAO Delphinium pentagynum (aerial parts).
Yellow crystalline solid (CHCl3/(CH3)2CO), mp 256~258C. Pharm:
Ref: 3831.
Anti-HIV inactive (in vitro, acutely infected H-9 lymphocyte cells)[4706];

H
cytotoxic inactive (in vitro, MCF7 and A549). Source: GUAN MU

TONG Aristolochia manshuriensis (stem: yield = 0.00083%). Ref: 4706.
O
O
OH
N
O
OH
O
O O
OH
N
O
5057 N-Demethyl-acronycine
[13255-08-8] C19H17NO3 (307.35). Source: JIU LI XIANG Murraya
paniculata [Syn. Chalcas paniculata]. Ref: 11.
O
5063 Demethylauraptenol
(S)-()-7-Hydroxy-8-(2-hydroxy-3-methyl-3-butenyl)-2H-1-benzopyran2-one C14H14O4 (246.27). Pharm: Antineoplastic (Raji cells, antitumor
promotor, in vivo, inhibits TPA-induced EBV-EA activation, compound
N
H
concentration = 500(mol ratio/32 pmol TPA): EBV-EA-positive cells =
(15.31.6)% (viability > 80%), -Carotene, EBV-EA-positive cells =
5058 N(4)-Demethylalstonerinal
C20H22N2O2 (322.41). Source: XIA YE JI GU CHANG SHAN Alstonia
angustifolia (leaf). Ref: 3780.
H
(22.81.8)% (viability > 80%), compound IC50 = 207(mol ratio/32

pmol TPA), -Carotene, IC50 = 400(mol ratio/32 pmol TPA),
Curcumin, IC 50 = 341(mol ratio/32 pmol TPA))[5048]. Source: TAI WAN
HUANG BO Phellodendron amurense var. wilsonii (leaf: yield =
H
O
NH
(34.31.1)% (viability >80), Curcumin, EBV-EA-positive cells =
0.00016%dw), Citrus hassaku. Ref: 4722, 5048.
H
O
5059 N(4)-Demethylalstonerine
HO
C20H22N2O2 (322.41). Source: XIA YE JI GU CHANG SHAN Alstonia
HO
angustifolia (leaf). Ref: 3780.

H
H
O
NH
N
H
5064 Demethylcalabaxanthone
1,7-Dihydroxy-8-(3-methylbut-2-enyl)-6',6'-dimethylpyrano(2',3':3,2)-xan
thone C23H22O5 (378.43). Pharm: Cytotoxic (KB cancer cell lines, IC50 =
5060 N(4)-Demethylalstophyllal oxindole

C21H24N2O4 (368.44). Source: DA YE TANG JIAO SHU Alstonia
macrophylla (leaf: yield = 0.00001%). Ref: 3020.
H
H
NH
O
10.9g/mL, control Ellipticine, IC50 = 1.33g/mL; BC-1, IC50 =

2.85g/mL, Ellipticine, IC50 = 1.46g/mL; NCI-H187, IC50 = 3.13g/mL
Ellipticine, IC50 = 0.39g/mL)[1619]; antitubercular (Mycobacterium
tuberculosis, MIC = 12.5g/mL) [4358]. Source: DAO NIAN ZI Garcinia
mangostana (unripe fruit: yield = 0.0068%dw)[1619]. Ref: 1619, 4358.
O
H
OH
HO
5061 N(4)-Demethylalstophylline oxindole

O
H
C15H10O7 (302.24). Yellow needles, mp 272~274C. Source: HUANG

HAO Artemisia scoparia [Syn. Artemisia capillaris var. scoparia] (bud).
Ref: 4815.
NH
O
5065 6-Demethylcapillarisin
O
H
OH
OH
HO
O
OH
54
5066 Demethylcephalotaxinone
5071 Demethyldelavaine A
C17H17NO4 (299.33). Source: HAI NAN CU FEI Cephalotaxus
hainanensis [Syn. Cephalotaxus mannii], SAN JIAN SHAN

Cephalotaxus fortunei (drupe: yield = 0.00020%)[4675], ZHONG GUO CU
FEI ZHI YE Cephalotaxus sinensis [Syn. Cephalotaxus harringtonia var.
O
H
sinensis]. Ref: 2, 660, 4675.
O
H
OH
OH
NH
HO
OH
5067 Demethylcoclaurine
Higenamine [5843-65-2] C16H17NO3 (271.32). mp 260~262C. Pharm:
5072 Demethyldelavaine B
Enhances cardiac motility; raises heart rate; antiasthmatic (gpg, asthma
caused by histamine, bronchial smooth muscle relaxant); treatment of

H
chronic arrhythmia; coronary, cerebral and peripheral vasodilator. Source:

O
FU ZI Aconitum carmichaeli, LIAN ZI Nelumbo nucifera, XIAO YE
O
H
O
H
MAI MA TENG Gnetum parvifolium [Syn. Gnetum indicum], RI BEN
WU TOU Aconitum japonicum, WU TOU Aconitum carmichaeli. Ref: 2,
OH
O
H
4, 658, 1521, 5501.
OH
NH
HO
OH
NH
HO
5073 6-Demethyldelsoline
C24H39NO7 (453.58). Colorless massive crystals, mp 202~204C. Source:
HO
ZI HUA GAO WU TOU Aconitum excelsum. Ref: 689.

5068 Demethyl coniferin
C15H20O8 (328.32). White powder. Source: SHAN TONG ZI Idesia
H
OH
polycarpa. Ref: 2494.
OH
H
OO
OH
O
H
OH
HO
O
H
OH
OH
OH
OH
5074 4'-Demethyldeoxypodophyllotoxin
OH
4-Demethyl-deoxypodophyllotoxin C21H20O7 (384.39). Colorless lamellar

5069 ()-N-Demethylcrychine
crystals, mp 246~248C, []D20 = 127.3 (c = 0.11, CHCl3). Pharm:
C18H15NO4 (309.32). Yellow powder (acetone), []D = 74.3 (c = 0.02,
Antineoplastic (P388); antimitotic; cytotoxic (KB, ED50 = 0.0012g/mL);
MeOH). Source: HOU KE GUI Cryptocarya chinensis (wood). Ref:
cytotoxic (KB, IC50 = 17.7ng/mL, control Vinblastine, IC50 = 9.7ng/mL;
3092.
LNCaP, IC50 = 10.0ng/mL, Vinblastine, IC50 = 10.5ng/mL; Col2, IC50 =

23.1ng/mL, Vinblastine, IC50 = 8.1ng/mL)[5336]. Source: BAI BA JIAO
LIAN Dysosma majorensis [Syn. Podophyllum majorense; Dysosma
lichuanensis] (rhizome: content = 0.0089%)[5508], BI LIN BA JIAO LIAN
NH
O
Dysosma furfuracea (rhizome: mean content in different seasons =

5070 4'-Demethyldehydropodophyllotoxin
C21H16O8 (396.36). White needles, mp > 320C. Source: LIU JIAO LIAN
Dysosma pleiantha [Syn. Podophyllum pleianthum]. Ref: 4801.
OH
0.75%)[5508], CHONG MING BA JIAO LIAN Dysosma subrosea

(rhizome: content = 0.020%)[5508], CHUAN BA JIAO LIAN Dysosma
veitchii (rhizome: content = 0.0092%)[5508], DA XIAN YUAN ZHI
Polygala macradenia, GUANG XI BA JIAO LIAN Dysosma
guangxiensis (rhizome: content = 0.0042%)[5508], GUI JIU Dysosma
O
O
O
versipellis [Syn. Podophyllum versipelle] (rhizome: content = 0.15%)[5508],

LIU JIAO LIAN Dysosma pleiantha [Syn. Podophyllum pleianthum]
(rhizome: content = 0.076%)[5508], LUN SHENG SHAN XIANG Hyptis

verticillata, PEI NI YUAN ZHI Polygala paenea, TAO ER QI
O
OH
Podophyllum emodii [Syn. Podophyllum emodii var. chinense;

Podophyllum sikkimenosis; Sinopodophyllum emodii] (rhizome: mean
55
content of 3 origins = 0.46%[5508]), WO ER QI Diphylleia sinensis
5079 8-Demethylfarrerol
(rhizome: content = 0.56%)[5508], XI MA LA YA YUAN ZHI Polygala
C16H14O5 (286.29). mp 267~270C. Source: MAN SHAN HONG
emodi, XIAO BA JIAO LIAN Dysosma difformis (rhizome: content =
Rhododendron dauricum. Ref: 6, 507.
0.0031%)[5508], YUE NAN LIE LAN Bursera tonkinensis (root), ZU YE

CAO Polygala peltatum. Ref: 661, 3543, 5336, 5508.
OH
HO
H
O
O
OH
O
H
5080 Demethylfuropinnarin
C16H14O4 (270.29). Source: JU MAO LEI A WEI Ferulago capillaries

O
(aerial parts), QIANG HUO Notopterygium incisum, KUAN YE QIANG
O
OH
HUO Notopterygium forbesii [Syn. Notopterygium franchetii]. Ref: 2,
5075 4'-Demethyldesoxypodophyllotoxin-4-O--D-glucoside
325, 660, 3938.

OH
20
C27H30O12 (546.53). []D = +20.6 (c = 0.14, CHCl3). Pharm: Cytotoxic

inactive (100g/mL: KB, LNCaP, and Col2 cells). Source: YUE NAN
LIE LAN Bursera tonkinensis (root). Ref: 5336.
O
O
O
5081 9-Demethylhomolycorine
O
[6879-81-8] C17H19NO4 (301.35). mp 213~214C. Pharm: Cytotoxic (hmn

lymphoma Molt4, ED50 = 18.5g/mL, mouse fiber cell LMTK, ED50 =
0.8g/mL). Source: SHI SUAN Lycoris radiata [Syn. Amaryllis radiata].
OO
HO
Ref: 6, 1847.
OH
OH
OH
5076 ()-10-O-Demethyldiscretine
C19H21NO4 (327.38). Source: YOU GOU YING ZHAO Artabotrys
H
H
uncinatus (root). Ref: 3083.

HO
OH
O
O
HO
5082 ()-3'-O-Demethyl-5-hydroxymatairesinol
(8R,8'R)-3'-O-Demethyl-5-hydroxymatairesinol C19H20O7 (360.37). []D23
= 27.5 (c = 0.10, MeOH). Source: Macrococculus pomiferus (stem).
5077 N-Demethyldoryphornine
Ref: 3869.
7-Hydroxy-6-methoxy-1(2H)-isoquinolinone C10H9NO3 (191.19).

Colorless rods (MeOH), mp 257~259C. Source: BIAN FU GE GEN
HO

HO
O
N
HO
H
O
HO
5078 4-Demethylepipodophyllotoxin 7'-O--D-glucopyranoside

C27H30O13 (562.53). White needles, []D15 = 29.3 (c = 0.63, MeOH).
Source: TAO ER QI Podophyllum emodii [Syn. Podophyllum emodii var.
chinense; Podophyllum sikkimenosis; Sinopodophyllum emodii] (root and
rhizome). Ref: 4142.
OH
5083 14-Demethyl-14-isobutyrylanhweidelphinine
C38H48N2O11 (708.81). Amorphous substance, []D25 = +65.2 (c = 0.14,
CHCl3). Source: WU ZHU FEI YAN CAO Delphinium pentagynum
OH
O
O
O
O
HO
OH
OH
OH
N
O
OH
O
O O
N
O
OH
56
5084 Demethylligstroside
5089 N-Demethylnoracronycine
C24H30O12 (510.50). Colorless amorphous powder, [] D26 = 110 (c =
[13396-93-5] C18H15NO3 (293.33). Source: JIU LI XIANG Murraya
0.32, MeOH). Source: MEI GUO BAI CEN Fraxinus americana (leaf).

O
Ref: 5091.
HO
O
O
OH
N
H
5090 N-Demethylphyllocryptine
C19H21NO4 (327.38). Source: HOU KE GUI Cryptocarya chinensis
OO
HO
OH
OH
(wood). Ref: 3092.

OH
OH
OH
O
5085 ()-3'-O-Demethyl-5-methoxymatairesinol
(8R,8'R)-3'-O-Demethyl-5-methoxymatairesinol C20H22O7 (374.39).
[]D23 = 6.0 (c = 0.12, MeOH). Source: Macrococculus pomiferus
(stem). Ref: 3869.
5091 4-Demethyl-picropodophyllotoxin
HO
C21H20O8 (400.39). Source: TAO ER QI Podophyllum emodii [Syn.

O
HO

Sinopodophyllum emodii] (root and rhizome). Ref: 3543.
OH
O
OH
5086 Demethylmoracin I
Anticancer Benzofuran PMV70P691-006 C19H18O4 (310.35). Brown
powder, mp 82~83C. Pharm: Aromatase inhibitor (in vitro, IC50 =
O
O
31mol/L; control Aminoglutethimide, IC50 = 6.4mol/L)[3090, 5038].

Source: GOU SHU Broussonetia papyrifera. Ref: 3090, 5038.
OH
5092 4-Demethyl-picropodophyllotoxin 7'-O--D-glucopyranoside

C27H30O13 (562.53). White powder, []D29 = 5.18 (c = 0.6, MeOH).
Source: TAO ER QI Podophyllum emodii [Syn. Podophyllum emodii var.
HO
chinense; Podophyllum sikkimenosis; Sinopodophyllum emodii] (root and
OH
rhizome). Ref: 3543.

OH
OH
5087 N-Demethylnicaustrine
[126617-16-1] C42H52N2O11 (760.89). Source: AO DA LI YA HONG
O
O
DOU SHAN Austrotaxus spicata. Ref: 662.

O
O
O O
OH
O O
O
O
O
H O
HN
5093 4-Demethyl-podophyllotoxin
cancer; supertoxic agent. Source: BAI BA JIAO LIAN Dysosma
5-Hydroxy-6,7,8,3',4'-pentamethoxyflavone [2174-59-6] C20H20O8

(388.38). mp 144C. Source: A ER TAI ZI WAN Heteropappus altaicus,
JU PI Citrus reticulata. Ref: 2, 6.
majorensis [Syn. Podophyllum majorense; Dysosma lichuanensis]

(rhizome: content = 0.013%)[5508], BAI YA MA Linum album, BI LIN BA
JIAO LIAN Dysosma furfuracea (rhizome: mean content in different
seasons = 0.47%)[5508], CHONG MING BA JIAO LIAN Dysosma
subrosea (rhizome: content = 0.48%)[5508], CHUAN BA JIAO LIAN
O
O
O
OH
Antineoplastic; antimitotic; antiviral; laxative; used in treatment of skin
5088 Demethylnobiletin
OH
4'-Demethylpodophyllotoxin [40505-27-9] C21H20O8 (400.39). Pharm:
OO
HO
Dysosma veitchii (rhizome: content = 0.022%)[5508], GUANG XI BA

JIAO LIAN Dysosma guangxiensis (rhizome: content = 0.0071%)[5508],
GUI JIU Dysosma versipellis [Syn. Podophyllum versipelle] (rhizome:
content = 0.0053%)[5508], KU YUAN ZHI Polygala polygama, LIU JIAO

OH
57
LIAN Dysosma pleiantha [Syn. Podophyllum pleianthum] (rhizome:
5097 Demethylsecologanol
mean content = 0.11%)[5508], TAO ER QI Podophyllum emodii [Syn.
C16H24O10 (376.36). Amorphous, []D23 = 108.3 (c = 0.06, MeOH).
Source: LIU QIU SHE GEN CAO Ophiorrhiza liukiuensis (whole herb).
Sinopodophyllum emodii] (rhizome: mean content of 5 origins =
Ref: 4527.
0.63%[5508]), WO ER QI Diphylleia sinensis (rhizome: mean content of 4

origins = 0.78%[5508]), XIAO BA JIAO LIAN Dysosma difformis
[5508]
(rhizome: content = 0.22%)
HO
OH
. Ref: 658, 3543, 5508.
OH
H
HO
OO
OH
OH
O
O
O
OH
5098 7-Demethylsuberosin
[21422-04-8] C14H14O3 (230.27). Pharm: AChE inhibitor (in vitro, IC50 =
OH
2.4mmol/L)[3058]; antineoplastic (Raji cells, antitumor promotor, in vivo,

inhibits TPA-induced EBV-EA activation, compound concentration =
5094 4-Demethyl-podophyllotoxin 7'-O--D-glucopyranoside
500(mol ratio/32 pmol TPA), EBV-EA-positive cells = (15.41.7)%
C27H30O13 (562.53). Source: TAO ER QI Podophyllum emodii [Syn.
(viability = 60%), -Carotene, EBV-EA-positive cells = (34.31.1)%
(viability > 80), Curcumin, EBV-EA-positive cells = (22.81.8)%
Sinopodophyllum emodii] (root and rhizome). Ref: 3543.
(viability > 80%); IC50 = 172(mol ratio/32 pmol TPA), -Carotene,

IC50 = 400(mol ratio/32 pmol TPA), Curcumin IC50 = 341(mol ratio/32
HO
pmol TPA))[5048]. Source: BAI ZHI Angelica dahurica [Syn. Angelica
OH
OH
porphyrocaulis], CHAO XIAN DANG GUI Angelica gigas (underground

part)[3058], LI HUA JU Citrus tachibana, Citrus rugulosa, Citrus jambhiri,
OH
Citrus sulcata, Citrus tamurana. Ref: 2, 3058, 5048.
O
O
O
O
OH
HO
5095 Demethylracemosol
5099 De-O-methyltenuicausine
C20H22O4 (326.40). Pharm: Cytotoxic (KB, EC50 = 5.6g/mL, control
[221640-45-5] C40H44N4O3 (628.82). White amorphous powder, mp
Ellipticine, EC50 = 0.3g/mL; BC, EC50 = 3.6g/mL, Ellipticine, EC50 =
190C, []D13 = 198.5 (c= 0.047, CHCl3). Source: CHUAN SHAN
0.3g/mL)
[5092]
; antimalarial (Plasmodium falciparum, EC50= 2.0g/mL,
CHENG Melodinus hemsleyanus. Ref: 412.
control Chloroquine diphosphate, EC50= 0.16g/mL). Source: MA LA BA

YANG TI JIA Bauhinia malabarica (root). Ref: 5092.
N
N
H
HO
HO
OH
N
H
O
OH
5096 Demethylregelin
5100 N-Demethylthalistyline
C30H46O4 (470.70). Pharm: DPPH scavenger inactive (for 40mol/L
[62251-51-8] C40H48N2O8 (682.82). Yellow amorphous powder, []D25 =
DPPH radical, SC50 > 40mol/L). Source: SUO LA MU Salacia
+151 (c = 0.2, methanol). Pharm: Antibacterial (Mycobacterium
prinoides [Syn. Salacia chinensis] (stem). Ref: 4378.
smegmatis, MIC 100g/mL); antihypertensive (dog, rbt). Source:

CHANG ZHU TANG SONG CAO Thalictrum longistylum, BING GUO
OH
TANG SONG CAO Thalictrum podocarpum. Ref: 661.

O
OH
N
H
O
O
O
O
N
H
58
5101 Demethylwedelolactone
5105 (S)-Dencichine
Norwedelolactone [6468-55-9] C15H8O7 (300.23). Green needles (MeOH),
[5302-45-4] C5H8N2O5 (176.13). Pharm: Hemostatic (mouse, perfusion in
mp 360C. Pharm: Antihepatotoxin (rat, liver toxicosis induced by CCl4,
stomach, 1mg/kg, platelets increase = (24~30)%)[5501]; LD50 (mouse,
GaIN and phalloidin, 67.6g/mL for liver toxicosis induced by phalloidin,
perfusion in stomach) = (83617)mg/kg[5501]. Source: SAN QI Panax
InRt = 98%, CD50 = 22.3g/mL, promotes regeneration of liver cells
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (root: mean
obviously); hemostatic (ED50 = 0.3mg/kg, 0.5mg/kg reduces bleeding
content in different standards = 0.350%[5508]; 0.87%[5501]). Ref: 1521,
time by 4.2min); antifungal (Aspergillus niger, 100mg/L InRt = 50%).
5501, 5508.
Source: MO HAN LIAN Eclipta prostrata [Syn. Eclipta alba], PENG QI

JU Wedelia chinensis [Syn. Solidago chinensis; Wedelia calendulacea],
2758, 2759, 2760.
OH
NH2
N
H
OH
5106 Dendramine
OH
HO
O H
HO
OH
XIAO LIAN QIAO Hypericum erectum. Ref: 6, 2754, 2755, 2756, 2757,
[7668-75-9] C16H25NO3 (279.38). mp 186~188C. Source: SHI HU
Dendrobium nobile. Ref: 6.
5102 Demethylwedelolactone-7-glucoside
C21H18O12 (462.37). Source: MO HAN LIAN Eclipta prostrata [Syn.
Eclipta alba]. Ref: 6.
OH
O
OH
OH
5107 Dendrine
OH
HO
OO
(4)
OH
OH
(4)
OH
5103 4-Demethylxuulanin-4-ethyl ether
4-Ethoxy-5-methoxy-6'',6''-dimethyl-2H-pyrano-(2'',3'':7,6)-flavan
C23H26O4 (366.46). Yellow oil. Source: Lonchocarpus xuul (stem cortex).
Ref: 3973.
5108 Dendrobine
[2115-91-5] C16H25NO2 (263.38). mp 135~136C. Pharm: Antipyretic;
causes hyperspasmia in toxic doses; inhibits respiration; antihypertensive;
analgesic; uterine stimulant. Source: SHI HU
(4)
Dendrobium nobile (the
compound was isolated from the plant by Y.Inubushi, et al. in 1965)[5505],

5104 Demissine
FEN LAI SHI HU Dendrobium findleyanum. Ref: 6, 658, 5501, 5505.
[6077-69-6] C50H83NO20 (1018.21). Pharm: Antifungal; cardiotonic.

Source: CHA QIE Solanum chacoense, KE MO SEN QIE Solanum
commersonii, AI QIE Solanum demissum, SHI XIAN QIE Solanum
decemlineata, JU SHI QIE Solanum juzepczukii. Ref: 658, 661.
H
O
H
H
H
H
HO
OO
OH
HO
OO
5109 Dendrobiumane A
C15H26O3 (254.37). Colorless gum, []D24 = +2.3 (c = 0.35, EtOH).
Source: XI JING SHI HU Dendrobium moniliforme (fresh stem). Ref:
5490.
OH
HO
H
HO
O
HO
OH
OH
O
N
OH
OH
OH
OO
OH
OH
H
H
OH
59
5110 Dendrobiumane B
5116 Dendromoniliside A
C15H24O4 (268.36). Colorless gum, []D23 = 7.0 (c = 0.80, EtOH). Source: XI
2,12-Dihydroxycopacamphan-15-one 2-O--D-glucopyranoside
JING SHI HU Dendrobium moniliforme (fresh stem). Ref: 5490.
C21H34O8 (414.5). White amorphous powder, mp215~216C (dec), []D20

= 0.6 (c = 0.4, H2O). Pharm: Proliferation stimulator (B cells in vitro,
OH
0.00001mol/L, p<0.05); proliferation inhibitor (T cells in vitro,

0.0000001mol/L, p<0.05, without any obvious cytotoxic effects). Source:
HO
XI JING SHI HU Dendrobium moniliforme (stem: yield = 0.0007%dw).
H
O
Ref: 4717.
HO
5111 Dendrobiumane C
C15H22O4 (266.34). Colorless gum, []D24 = +122.7 (c = 0.05, EtOH). Source:
OO
HO
HO
O
OH
XI JING SHI HU Dendrobium moniliforme (fresh stem). Ref: 5490.
OH
HO
5117 Dendromoniliside B
HO
2,3,12-Trihydroxypicrotoxane-3(15)-olid-11-oic acid
H
O
2-O--D-glucopyranoside C21H32O11 (460.48). Colorless prism crystals
(MeOH:H2O = 1:1), mp 225~227C, []D20 = 18.3 (c = 0.5, MeOH).
5112 Dendrobiumane D
Source: XI JING SHI HU Dendrobium moniliforme (stem: yield =
C15H24O5 (284.36). Colorless gum, []D23 = +5.7 (c = 0.31, EtOH). Source: XI
0.0003%dw). Ref: 4717.

OH
OH
O
HO
HO
OH
O
OO
HO
HO
OH
O
O
OH
5113 Dendrobiumane E
C15H18O7 (310.31). Colorless gum, []D24 = +4.1 (c = 0.21, EtOH). Source: XI
5118 Dendromoniliside C
2,3,8-Trihydroxy-9-(11)-epoxypicrotoxan-3(15)-olide
8-O--D-glucopyranoside C21H32O10 (444.48). White amorphous powder,
OH
mp 170~172C, []D20 = 0.5 (c = 0.4, H2O). Pharm: Proliferation
O
O
stimulator (B cells in vitro, 0.00001mol/L, p<0.05); proliferation inhibitor

OH
O
(T cells in vitro, 0.0000001mol/L, p<0.05, without any obvious cytotoxic

effects). Source: XI JING SHI HU Dendrobium moniliforme (stem: yield
= 0.0007%dw). Ref: 4717.
5114 Dendrocyin
Isocucurbitacin; 24-Ethoxy-20-25-epoxy-3,16-dihydroxy-9-methyl-
OH
(methanol), mp 195~198C. Source: Dendrosicyos socotrana (stem). Ref:
OH
HO
H
3855.
O
OH
OH
19-norlanost-5(6) ene-2,11,22-trione C32H48O7 (544.74). White prisms
5119 Dendromoniliside D
O
H
2,3,11,12-Tetrahydroxypicrotoxan-3(15)-olide
OH
11-O--D-glucopyranoside C21H34O10 (446.5). White amorphous powder,

mp 205~207C, []D20 = 0.4 (c = 1.2, H2O). Source: XI JING SHI HU
HO
Dendrobium moniliforme (stem: yield = 0.0003%dw). Ref: 4717.
5115 Dendrolasin
HO
[23262-34-2] C15H22O (218.34). bp 148~150C/16mmHg. Source: TAN

XIANG Santalum album. Ref: 6.
HO
HO
OO
OH
HO
H
O
OH
60
5120 Dendronobiloside A
5125 Dendroside F
10,12-Dihydroxypicrotoxane 10,12-di-O--D-glucopyranoside C27H48O12

(564.68). White amorphous powder,
[]D20
= 62.9 (c = 0.6, MeOH). Pharm:
C21H34O9 (430.50). White amorphous powder, []D20 = 30.6 (c = 0.5,

(4)
MeOH). Source: SHI HU
Dendrobium nobile, XI JING SHI HU
Immunoenhancer (in vitro, stimulates significantly proliferation of mouse B
Dendrobium moniliforme (stem: yield = 0.00016%dw)[4717]. Ref: 1931,
lymphocytes, 1.0mol/L, p<0.01, control Astragaloside I, 1.0mol/L,
4717.
(4)
p<0.05). Source: SHI HU
Dendrobium nobile (stem). Ref: 3084.
HO
OO
OH
HO
HO
HO
HO
O O
HO
OH
OH
OH
OH
O
HO
HO
5121 Dendronobiloside B
6,10,12-Trihydroxypicrotoxane 10-O--D-glucopyranoside C21H38O8
(418.53). White amorphous powder, []D20 = 63.6 (c = 0.5, MeOH).
Pharm: Immunosuppressant (in vitro, inhibits proliferation of mouse T
lymphocytes, 0.1-10.0mol/L, p<0.05). Source: SHI HU
(4)
5126 Dendroside G
(4)
MeOH) Source: SHI HU
Dendrobium
nobile (stem). Ref: 3084.
HO
OO
OH
HO
HO
HO
OH
OH
OH
OH
OH
HO
HO
5122 Dendroside A
10,12,14-Trihydroxyalloaromadendrane 14-O--D-glucopyranoside
C21H36O8 (416.52). White amorphous powder; mp 145~147C, []D14 =
48.6 (c 0.1, MeOH). Pharm: Immunoenhancer (in vitro, stimulates
significantly proliferation of mouse T lymphocytes, 0.1mol/L, p<0.01,
5127 Dendroxine
(4)

control Astragaloside I, 10mol/L, p<0.05; stimulates significantly

proliferation of mouse B lymphocytes, 10mol/L, p<0.01, Astragaloside I,
(4)
1.0mol/L, p<0.05). Source: SHI HU
Dendrobium nobile (stem). Ref:
3084.
HO
HO
HO
O O
OH
H
O
HO
OH
5128 Dengibsin
C14H10O4 (242.23). Source: MI HUA SHI HU Dendrobium densiflorum
5123 Dendroside D
20
C27H44O14 (592.64). White amorphous powder, []D = 31.3 (c = 0.5,

(4)
(stem). Ref: 5171.

OH
OO
HO
OH
OH
OH
OH
H
OO
HO
OH
OH
5129 Deniagenin
3,11,12,14,17,20-Hexahydroxy pregn-5-ene C21H34O6 (382.50).
OH
White amorphous powder, mp 110C, []D = 66.7(c = 0.3, CHCl3).
5124 Dendroside E
HO
OO
OH
(4)
Source: ROU LEI NIU NAI CAI Marsdenia roylei (aerial parts). Ref:
3490.
OH
OH
H
HO
OH
OH
OH
OH
OH
HO
OH
OH
61
5130 Denicunine
EBV-EA-positive cells = (22.81.8)% (viability > 80%); IC50 =
Calogenin 3-O-3-O-methyl--D-fucopyranosyl-(14)-O--D-oleandro-
496(mol ratio/32 pmol TPA), -Carotene, IC50 = 400(mol ratio/32
pyranoside C35H58O10 (638.85). mp 148C, []D = +20 (c = 0.11, MeOH).
pmol TPA), Curcumin IC50 = 341(mol ratio/32 pmol TPA))[5048].
Source: YIN DU BA QIA Hemidesmus indicus (stem). Ref: 5081.
Source: CHENG ZI Citrus junos, SHAN HUANG PI Clausena excavata,

YE HUANG PI Clausena dentata, ZHI GEN PI Poncirus trifoliata. Ref:
OH
6, 1521, 5367, 5048.

O
OH
O
OO
OO
HO
O
5135 ()-Denudatin B
C21H24O5 (356.42). Colorless oleaginous substance, []D15 = 76.4 (c =
OH
0.11, CHCl3). Pharm: PAF antagonist (IC50 = 7.5mol/L); PAF receptor
5131 Denin
antagonist (5g/mL, InRt = 80.1%, 10g/mL, InRt = 100%); used in
Desacylkondurangogenin C-3-O--D-glucopyranosyl-(14)-O--L-fuco-
treatment of rheumatic arthritis and asthma; calcium antagonist
pyranoside C33H56O14 (676.81). White amorphous powder, mp 232C,
(28mol/L, activity = 100%); calcium antagonist (gpg, colon bands);
[]D = +12.5(c = 0.016, CHCl3). Source: ROU LEI NIU NAI CAI
vascular relaxant (inhibits inward flow of calcium, increase cGMP);
Marsdenia roylei (aerial parts). Ref: 3490.
anti-platelet (nonspecific). Source: WANG CHUN YU LAN Magnolia

biondii [Syn. Magnolia fargesii], HAI FENG TENG Piper kadsura [Syn.
OH
OH
Piper futokadsura]. Ref: 267, 658, 1578, 1609, 1610, 1611.
HO
OH
HO
OH
OH
O
O
HO
O
OH
OO
5136 Denudatine
OH
[26166-37-0] C22H33NO2 (343.51). Pharm: Antiarrhythmic (rat, aconitine

induced arrhythmia, inhibits rapid inward flow of sodium ion; CaCl 2 induced
5132 Densiflorol A
C16H16O4 (272.30). White amorphous powder. Source: MI HUA SHI HU
Dendrobium densiflorum (stem). Ref: 5171.
OH
arrhythmia, reduces heart rate); antihypertensive (rat, iv, 25~50mg/kg,

slightly blood pressure goes down); eclamptogenic (mus, iv, ED50 =
55.6mg/kg); Intestinal smooth muscle relaxant (dog intestine, reduces
tension and creep); antineoplastic (leukemia); cytotoxic; LD50 (mus, iv) =
128mg/kg, (mus, orl) = 290mg/kg. Source: LU CUI QUE Delphinium
denudatum, FU ZI Aconitum carmichaeli. Ref: 16, 1621, 1622, 1623,
1624.
HO
H
5133 Densiflorolorin
C14H10O5 (258.23). Red amorphous powder. Source: MI HUA SHI HU
OH
OH
Dendrobium densiflorum (stem). Ref: 5171.
5137 14-Deoxo-14-O-acetylorthosiphol Y
OH
OH
J774.1 cells, IC50 = 118.7mol/L; control L-NMMA, IC50 = 35.7mol/L).
5134 Dentatin
Poncitrin [22980-57-0] C20H22O4 (326.40). mp 95~96C; mp 93~94C.
Pharm: Antibacterial (Mycobacterium tuberculosis, MIC = 50g/mL,
control Isoniazide, MIC = 0.040~0.090g/mL, Kanamycin sulfate, MIC =

Orthosiphon spicatus] (aerial parts: yield = 0.00038%dw). Ref: 4741.
2.0~5.0g/mL)[5367]; antifungal inactive (Candida albicans, control

Amphotericin, IC50 = 0.01g/mL)
[5367]
HO
; antineoplastic (Raji cells,
antitumor promotor, in vivo, inhibits TPA-induced EBV-EA activation,

compound concentration = 500(mol ratio/32 pmol TPA),
EBV-EA-positive cells = (47.91.4)% (viability > 80%), -Carotene,
EBV-EA-positive cells = (34.31.1)% (viability > 80), Curcumin,
O
O
H
O
O
OH
O
O
O
62
5138 13-Deoxo-13-acetyloxy-1-deoxynortaxine B
5143 2-Deoxo-5-deoxy-8-O-acetyl-17,18-epoxy pumilin
2,9-Dihydroxy-10,13-diacetoxy-5-(3'-N-methylamino-3'-phenyl)-pr
C22H26O7 (402.45). Yellow oil, []D22 = 0.03 (c = 3.88, CH2Cl2). Source:
opionyloxytaxa-4(20),11-diene C34H47NO8 (597.76). Gum, []D22 = +47
Balsamorhiza sagittata (aerial parts), Balsamorhiza macrophylla (aerial
(c = 0.21, CHCl3). Source: JIA NA DA HONG DOU SHAN Taxus
parts). Ref: 991.
canadensis (needle leaf), JIANG GUO ZI SHAN Taxus baccata. Ref: 662,
3886.
O
O OH
O
O
H
H OH
H
H
5144 11-Deoxoglycyrrhetinic acid
5139 13-Deoxo-13-acetyloxy-1-deoxytaxine B
11-Deoxyglycyrrhetinic acid C30H48O3 (456.72). Source: GUANG GUO
C35H49NO8 (611.78). Source: JIANG GUO ZI SHAN Taxus baccata. Ref:
GAN CAO Glycyrrhiza glabra, LEI GONG TENG Tripterygium wilfordii,
662.
ZHANG GUO GAN CAO Glycyrrhiza inflata. Ref: 2, 660, 670.
OH
O OH
O
O
N
H
H
OH
H
HO
5140 13-Deoxo-3-acetyloxytaxine B
C35H49NO9 (627.78). Source: JIANG GUO ZI SHAN Taxus baccata. Ref:
5145 9-Deoxo-9-hydroxytaxol
662.
C47H53NO14 (855.94). mp 174~176C, []D = 13.1 (MeOH). Source:

YUN NAN HONG DOU SHAN Taxus yunnanensis. Ref: 662.
O
O OH
O
H
OH OH
O
O
OH
5141 2-Deoxo-8-O-acetyl pumilin
O OH
OH O
OH
C22H26O7 (402.45). Yellow oil, []D22 = 0.024 (c = 2.75, CH2Cl2). Source:
H
O
O
Balsamorhiza sagittata (aerial parts), Balsamorhiza macrophylla (aerial

parts). Ref: 991.
5146 5-Deoxyabyssinin II
4',7-Dihydroxy-3'-methoxy-5'-prenylflavanone C21H22O5 (354.41).
O
O
HO
Amorphous powder, []D = 0 (c = 0.01, MeOH). Pharm: Antimalarial

(Plasmodium falciparum D6, IC50 = (13.60.9)g/mL, control
Chloroquine, IC50 = (0.0090.002)g/mL, Quinine, IC50 =
(0.040.01)g/mL; Plasmodium falciparum W2, IC50 = (13.31.5)g/mL,
Chloroquine, IC50 = (0.080.003)g/mL, Quinine, IC50 =
5142 Deoxodehydrocyclopiloselloidone
(0.210.01)g/mL)[3879]. Source: A BI XI NI YA CI TONG Erythrina
Desoxodehydrocyclopiloselloidone C18H22O2 (270.37). Source: MAO DA
abyssinica (stem cortex). Ref: 3879.
DING CAO Gerbera piloselloides. Ref: 6.

O
OH
O
HO
63
5147 6-Deoxy-6-acetoxyatalantin acetate
5152 Deoxyandrographolide
Limonoid C31H38O11 (586.64). White lamellar prismatic crystals, mp
C20H30O4 (334.46). Pharm: Antibacterial; antispirochetic;
208~209C. Source: DONG FENG JU YE Atalantia buxifolia [Syn.
anti-inflammatory (rat, edema on ears caused by oleum crotonis); reduces
Severinia buxifolia]. Ref: 402.
effusion of Evans blue from blood capillary (caused by xylene or acetic

acid); stimulates function of adrenal cortex; LD50 (mus, orl) > 20mg/kg.

paniculata]. Ref: 2, 658, 1521, 5501.
O
O
O
O
O
5148 8-Deoxy-9-O-acetylanthemolide B
HO
C17H22O7 (338.36). Amorphous solid, []D25 = 54 (c = 0.32, MeOH).
OH
Source: Anthemis carpatica (aerial parts). Ref: 3974.

OH
5153 14-Deoxyandrographolide-3-O-sulfate
C20H30O7S (414.52). White amorphous powder. Source: REN NIAO
Homo sapiens. Ref: 4300.
HO O
O
O
5149 Deoxyaconitine
Ref: 16, 1521.
O
HO
H
H
N
H
O
O
O
H
OO
HO
O
S
H
OH
O
OH
5154 1-Deoxy-L-arabinitol
Source: YIN DU ZANG HUI XIANG Carum ajowan (fruit). Ref: 3547.
5150 27-Deoxyactein
C37H56O11 (676.85). Pharm: Cytotoxic (HSC-2 cells, IC50 = 211mol/L,
control Etoposide, IC50 = 24mol/L; HGF cells, IC50 = 276mol/L)[4158].
Source: ZONG ZHUANG SHENG MA Cimicifuga racemosa (rhizome).
Ref: 4158.
H
HO
HO
O
O
H
H
OH
5155 3-Deoxybidensyneoside B
(E)-8-Decene-4,6-diyne-1,10-diol 1-O--D-glucopyranoside C16H22O7
OH
(326.35). Colorless crystals, mp 164C, []D23 = 67.7 (c = 0.5, MeOH).
OO
Pharm: Antihistamine (mast cells, inhibits histamine release induced by
OH
OH
OH
antigen-antibody reaction, IC50 = 0.085mol/L, control Indumethacin,

IC50 = 0.625mol/L)[4105]; NO production inhibitor (mus macrophages
OH
5151 11-Deoxyalisol A
RAW264.7, activated by 100ng/mL LPS at 37C, for 18h, IC50 =
C30H50O4 (474.73). Colorless powder. Source: ZE XIE Alisma orientale
0.116mol/L, activated by 100ng/mL LPS + 10U/mL IFN- at 37C, for
[Syn. Alisma plantago-aquatica var. orientale]. Ref: 2213.
18h, IC50 = 0.078mol/L)[4105]. Source: XIAO HUA GUI ZHEN Bidens

parviflora (whole herb). Ref: 4105.
OH
OH
OH
HO
OO
HO
OH
H
O
OH
H
OH
64
5156 Deoxycalyxin A
5161 Deoxycholic acid
C35H34O8 (582.66). Light yellow amorphous solid, []D25 = +147.9 (c =
7-Deoxycholic acid [83-44-3] C24H40O4 (392.58). Pharm: Antispasmodic
0.035, MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 27.4mol/L;
(main antispasmodic component in Bos taurus domesticus; Bubalus
HT1080, ED50 = 26.5mol/L; control Curcumin, Colon26-L5, ED50 =
bubalis NIU HUANG)[5501]; choleretic (bile secretion promotor)[5501];
23.2mol/L; HT1080, ED50 = 23.4mol/L). Source: YUN NAN CAO
anti-inflammatory (mouse, acetic acid-induced, ip, inhibits increase of
KOU Alpinia blepharocalyx (seed: yield = 0.000056%). Ref: 3035.
vaso-permeability)[5501]; antibacterial (Vibrio cholerae, Bacillus coli,

Staphylococcus tetragenus, Staphylococcus aureus, Streptococcus
OH
sp.)[5501]; antiviral (mouse, encephalitis B virus)[5501]; LD50 (mouse,

perfusion in stomach) = 1.06g/kg, (mouse, iv) = 0.15g/kg[5501]. Source:
HO
NIU HUANG Bos taurus domesticus; Bubalus bubalis (gallstone: mean

content = 1.65%[5508]), XIONG DAN Selenarctos thibetanus; Ursus
H
OH
OH
arctos. Ref: 2, 658, 5501, 5508.
OH
OH
OH
OH
5157 Deoxycamptothecin
H
[34141-35-0] C20H16N2O3 (332.36). mp 171~172C. Source: XI SHU

HO
Camptotheca acuminata. Ref: 6, 1521.

O
5162 3-Deoxycimigenol
N
N
C30H48O4 (472.71). mp 202~203C. Source: RI BEN SHENG MA

O
Cimicifuga japonica. Ref: 2215.
5158 3'-Deoxycapsanthin
(3R,5'R)-3-Hydroxy-,-caroten-6'-one C40H56O2 (568.89). Source:

H
HONG HAI JIAO Capsicum annuum (fruit: yield = 0.00005%). Ref:
OH
O
OH
3007.
H
5163 Deoxycorticosterone
HO
21-Hydroxypregn-4-ene-3,20-dione [64-85-7] C21H30O3 (330.47). mp

141~142C. Source: NIU SHEN Bos taurus domesticus; Bubalus bubalis,
5159 6-Deoxycatalpol
ZI HE CHE Homo sapiens. Ref: 6.
C15H22O9 (346.34). Source: ROU CONG RONG Cistanche deserticola,

O
GUAN HUA ROU CONG RONG Cistanche tubulosa. Ref: 2448.

H
H
H
O
O
HO
HO
OH
H
OO
5164 14-Deoxy-12-(cysteine-S-yl)-andrographolide-3-O-sulfate
OH
C23H39NO9S2 (533.66). White amorphous powder. Source: REN NIAO
OH
OH
Homo sapiens. Ref: 4300.
5160 7-Deoxycephalofortuneine
[128508-20-3] C20H27NO4 (345.44). Source: SAN JIAN SHAN
Cephalotaxus fortunei. Ref: 2, 1521.
NH2
OH
O
N
O
HO
O
O
H
H
OH
HO
65
5165 12-Deoxydanshenxinkun B
5170 10-Deoxy-4,18-epoxy-12-methoxy-4,5-seco-pisiferan-19-ol
18,20-Dinor-1,3,5(10),6,8,12-abietahexaene-11,14-dione C18H16O2
[245110-74-1] C21H32O3 (332.49). Gum, []D25 = +25.8 (c = 0.03,
(264.33). Red needles (CHCl3 n-hexane), mp 187~197C. Source: JIAO
CHCl3). Source: HONG GUI Chamaecyparis formosensis. Ref: 2315.
ZHI SHU WEI CAO Salvia glutinosa (dried root). Ref: 2384.
O
O
OH
O
O
5171 1-Deoxy-L-erythritol
5166 8-Deoxy-14-dehydro-aconosine
C22H33NO3 (359.51). Source: FU ZI Aconitum carmichaeli. Ref: 16.
HO
HO
O
H
OH
5172 1-Deoxy-L-erythritol 3-O--D-glucopyranoside

Source: HUI QIN Pimpinella anisum (fruit). Ref: 3402.
5167 14-Deoxy-11,12-didehydroandrographolide
C20H28O4 (332.44). Source: CHUAN XIN LIAN Andrographis
HO
paniculata [Syn. Justicia paniculata]. Ref: 2, 1521.
OO
HO
OH
OH
OH
OH
5173 1-Deoxyeucommiol
H
HO
C9H16O3 (172.23). Source: DU ZHONG Eucommia ulmoides. Ref: 2.
HO
OH
5168 Deoxyelephantopin
HO
[29307-03-7] C19H20O6 (344.37). mp > 320C. Pharm: Antineoplastic

(mus, in vivo, Walker cancer); cytotoxic. Source: KU DI DAN
Elephantopus scaber, KA LUO LAI NA DI DAN CAO Elephantopus
carolinianus. Ref: 5, 6, 658.
O
5174 10-Deoxyeucommiol
C9H16O3 (172.23). Yellow oil, []D17 = 33.77 (c = 3.61, MeOH). Source:
DIAO DENG SHU Kigelia pinnata. Ref: 3418.
HO
OH
OH
OH
O
O
5175 Deoxygaudichaudione A
C33H40O6 (532.68). Pharm: Cytotoxic (hmn leukemia:

doxorubicin-resistant K562, IC50 = (3.040.18)g/mL, control
5169 6-Deoxy-6,9-epoxy-8-hydroxy-10-epi-ryanodine
Adriamycin, IC50 = (1.790.17)g/mL; drug-sensitive K562, IC50 =
(1.740.22)g/mL, Adriamycin, IC50 = (0.110.01)g/mL). Source:
8 (c = 0.2). Source: QU CHONG CAO Spigelia anthelmia (aerial parts).
TENG HUANG SHU Garcinia hanburyi (resin). Ref: 1583.
Ref: 5139.
OH
HO
OH
OH
N
H
O
O
HO
OH
OH
OH
66
5176 10-Deoxygeniposidic acid
5181 Deoxyharringtonine
[36804-95-2] C28H37NO8 (515.61). Pharm: Antineoplastic (mouse P388,
mouse spleen leukemic L615). Source: HAI NAN CU FEI Cephalotaxus

hainanensis [Syn. Cephalotaxus mannii], RI BEN CU FEI Cephalotaxus
HO
harringtonia, SAN JIAN SHAN Cephalotaxus fortunei (drupe: yield =
0.00060%)[4675], ZHONG GUO CU FEI ZHI YE Cephalotaxus sinensis

[Syn. Cephalotaxus harringtonia var. sinensis]. Ref: 2, 5, 660, 4675.
O
HO
H
O
O
OH
OH
OH
OH
5177 1-Deoxy-D-glucitol
H
C6H14O5 (166.18). Source: SHI LUO ZI Anethum graveolens (fruit). Ref:
4177.
H
OH
HO
5182 6-Deoxyisojacareubin
C18H14O5 (310.31). Yellow needles, mp 218~220C. Source: BIAN DI
OH
JIN Hypericum wightianum (whole herb). Ref: 4426.
OH
O
OH
OH
5178 Deoxygomisin A
Schizandrin B; Schisandrin B; Wuweizisu B; -Schisandrin [61281-37-6]
C23H28O6 (400.48). Rhombic crystals (methanol), mp 117~119C, []D17 =
O
OH
32 (ethanol). Pharm: Antihepatotoxin; antitussive. Source: HONG HUA

WU WEI ZI Schisandra rubriflora, REN SHEN Panax ginseng [Syn.
Panax schinseng], WU WEI ZI Schisandra chinensis (dried ripe fruit:
5183 14-Deoxy-15-isopropylidene-11,12-didehydroandrographolide
content scope of 6 origins = 0.80%~5.00%, mean content = 2.68%[5508]).
C23H32O4 (372.51). Colorless needles (MeOH), mp 207~209, []D28 =
Ref: 2, 4, 39, 658, 1521, 5501, 5508.
21.8 (c = 0.002, MeOH). Source: CHUAN XIN LIAN Andrographis

paniculata [Syn. Justicia paniculata]. Ref: 2036.
O
O
O
O
O
O
5179 (+)-9-Deoxygoniopypyrone
C13H14O4 (234.25). Pharm: Cytotoxic inactive (HepG2, Hep3B,
MDA-MB-231, MCF7)
[5056]
. Source: TAI WAN GE NA XIANG
HO
HO
Goniothalamus amuyon (stem: yield = 0.00067%fw), TAI WAN GE NA

XIANG Goniothalamus amuyon (leaf and stem). Ref: 4686, 5056.
5184 6-Deoxyjacareubin
1,5-Dihydroxy-6',6'-dimethylpyrano(2',3':3,2)xanthone C18H14O5 (310.31).
H O
O
O
Pharm: Cytotoxic (HSC-2 cells, CC50 = 0.48mmol/L; HGF, CC50 >

0.65mmol/L)[3025]; anti-hypotension (PAF-induced, ID50 =
(14.53.2)mol/kg, control Ginkgolide B, ID50 = (38.52.7)mol/kg,
HO H
CV-3988, ID50 = (2.41.2)mol/kg)[5050]. Source: GOU JI Cudrania

5180 Deoxygoniopypyrone A
C13H14O4 (234.25). Colorless needles, mp 170~172C, []D23 = 35.5 (c
= 0.07, MeOH). Pharm: Cytotoxic inactive (HepG2, Hep3B,
MDA-MB-231, MCF7). Source: TAI WAN GE NA XIANG
Goniothalamus amuyon (leaf and stem). Ref: 5056.
cochinchinensis (root: yield = 0.00013%dw)[3025], HAI TANG GUO

Calophyllum inophyllum (the compound was isolated from the plant by
F.S.AL-Jeboury, et al. in 1971)[5505], HAI TANG GUO Calophyllum
inophyllum (root)[5050], HEI XIAN TIAO TENG HUANG Garcinia
nigrolineata (stam bark)[3482]. Ref: 3025, 3482, 5050, 5505.
OH
O
O
H
HO
O
H
O
OH
67
5185 4'-Deoxykanokoside A
5190 C-8-(S)-7-Deoxyloganic acid
C21H32O12 (476.48). Amorphous, []D20 = 122 (c = 0.1, MeOH). Pharm:
C16H24O9 (360.36). Source: BI LU GOU TENG Uncaria tomentosa (inner
Cytostatic/cytotoxic (GI50 = 1~9g/mL). Source: CHANG HUA XIE
bark). Ref: 5161.
CAO Centranthus longiflorus ssp. longiflorus. Ref: 2035.

H
HO
O
O
HO
OH
O OH
HO
OH
OH
HO
OH
5186 4'-Deoxykanokoside C
Cytostatic/cytotoxic (GI50 = 1~9g/mL). Source: CHANG HUA XIE
CAO Centranthus longiflorus ssp. longiflorus. Ref: 2035.
O
OO
HO
OH
O
HO
OH
O
OH
OH
OH
5191 Deoxyloganin
[26660-57-1] C17H26O9 (374.39). Pharm: Laxative. Source: Strychnos sp.,
Vinca sp., Menyanthes sp. Ref: 658.
O
OH
5187 8-Deoxylactucin
OH
OH
OH
O
H
HO
OO
OH
OH
OH
C15H16O4 (260.29). Pharm: Antineoplastic; cytotoxic. Source: YE WO JU

Lactuca serriola, JU QU Cichorium intybus. Ref: 658.
5192 1-Deoxy-D-lyxitol
Source: BEI SHA SHEN Glehnia littoralis (fruit). Ref: 3525.
H
O
HO
HO
HO
OH
OH
5188 Deoxylapachol
[3568-90-9] C15H14O2 (226.28). Pharm: Anthelmintic (termites); irritant
(to skin). Source: ZI BAI PI Catalpa ovata, YOU MU Tectona grandis.
5193 8-Deoxymerrilliortholactone
C15H24O6 (300.35). Source: Illicium merrillianum (pericarp). Ref: 4257.
Ref: 658.
OH
O
O
HO
OH
OH
5189 7-Deoxy-8-epi-loganic acid

C16H24O9 (360.36). Yellow powder, []D23 = 22.5 (c = 0.50, C5H5N).
Pharm: Antinociceptive (acetic acid-induced, 50mg/kg, orl, inhibitive
percent = 5%, 100mg/kg, orl, inhibitive percent = 49%, 50mg/kg, sc,
5194 1-Deoxy-3-methacrylyl-11-methoxymeliacarpinin
[177795-23-2] C32H42O12 (618.68). Colorless powder, mp 274~276C
(chloroform), []D = 16.3 (c = 0.2, chloroform). Pharm: Cytotoxic (P388,
IC50 = 47.0g/mL). Source: KU LIAN PI Melia azedarach. Ref: 1104.
O
inhibitive percent = 0%, 100mg/kg, sc, inhibitive percent = 6%; control
O
H
Aminopyrine, 50mg/kg, orl, inhibitive percent = 87%, 50mg/kg, sc,

[3908]
inhibitive percent = 94%)
. Source: BO SI YI MU CAO Leonurus
OH
O
O
Cistanche deserticola. Ref: 2448, 2499, 3908.
H
OO
OH
OH
OH
5195 3'-Deoxy-4-O-methylsappanol
O
HO
O
HO
persicus, MA TONG HUA Incarvillea arguta], ROU CONG RONG

HO
C17H18O5 (302.33). Source: SU MU Caesalpinia sappan (heartwood). Ref:

4494.
HO
OH
OH
68
5196 Deoxymorellin
5201 Deoxypeganine
Desoxymorellin C33H38O6 (530.67). mp 126C. Pharm: Cytotoxic (HeLa
[495-59-0] C11H12N2 (172.23). mp 87~88C. Pharm: Cholinergic. Source:
and HEL, MIC = 0.39g/mL). Source: TENG HUANG Garcinia morella.
LUO TUO PENG Peganum harmala. Ref: 6, 658.
Ref: 1081, 1099, 1172.

N
N
O
O
5202 4-Deoxyphorbol 12,13-bis(isobutyrate)

OH
[250258-02-7] C28H40O7 (488.63). Oil, []D = +47 (c = 0.64, CHCl3).
5197 3,5-Deoxyneotigogenin
Source: DUN YE DA JI Euphorbia obtusifolia var. obtusifolia. Ref: 2365.
C27H40O2 (396.62). Source: CHA RUI SHU YU Dioscorea collettii, BI

XIE Dioscorea hypoglauca [Syn. Dioscorea collettii var. hypoglauca].
Ref: 10.
O
H
OH
O H
OH
5198 1-Deoxynojirimycin
Moranoline [19130-96-2] C6H13NO4 (163.17). Pharm: -Glucosidase
5203 3-Deoxypseudoanisatin
inhibitor (IC50 = 0.3mmol/L)[4155]. Source: SANG ZHI Morus alba. Ref:
C15H22O5 (282.34). []D18 = 40.2 (c = 0.44, MeOH). Source: Illicium
2170, 4155.
merrillianum (pericarp). Ref: 4257.
H
N
HO
OH
OH
O O
OH
OH
OH
5199 Deoxynupharidine
[1143-54-0] C15H23NO (233.36). Pharm: Anesthetic (rhizoma of source
plant RI BEN PING PENG CAO Nuphar japanicum); sedative (rhizoma
5204 6-Deoxypseudoanisatin
of source plant RI BEN PING PENG CAO Nuphar japanicum). Source:
7-Deoxypseudoanisatin C15H22O5 (282.34). White acicular crystals (acetic
RI BEN PING PENG CAO Nuphar japonicum, OU ZHOU PING PENG
ester), mp 235~237C, []D25 = +15.5 (c = 1.406, ethanol). Source: HONG
CAO Nuphar luteum. Ref: 658.
HUI XIANG Illicium henryi, MIN WAN BA JIAO Illicium minwanense

(pericarp: yield = 0.0054%dw)[4697]. Ref: 100, 315, 1521, 4697.
H
N
OH
HO
5200 14-Deoxy-11-oxoandrographolide
[42895-57-8] C20H28O5 (348.44). mp 98~100C. Source: CHUAN XIN
LIAN Andrographis paniculata [Syn. Justicia paniculata], JI XING ZI
Impatiens balsamina. Ref: 2, 6.
5205 (3R)-Deoxypumiloside
C26H28N2O8 (496.52). Source: LIU QIU SHE GEN CAO Ophiorrhiza
liukiuensis (whole herb). Ref: 4527.
O
O
H
HO
H
OH
N
N
H
H
HO
H
OO
OH
OH
OH
69
5206 Deoxyrhaponticin
5212 3-Deoxysappanone B
4'-O-Methyl piceid [36469-58-6] C21H24O8 (404.42). Pharm:
C16H14O5 (286.29). Pharm: Xanthine oxidase inhibitor (noncompetitive
-Glucosidase inhibitor (IC50 = 280g/mL). Source: TIAN SHAN DA
inhibitory activity in concentration-dependent manner, IC50 = 36.8mol/L,
HUANG Rheum wittrocki, ZHANG YE DA HUANG Rheum palmatum.
Ki = 27.4mol/L, control Allopurinol, competitive type, IC50 = 2.5mol/L,

Ki = 1.80mol/L). Source: SU MU Caesalpinia sappan (heartwood). Ref:
Ref: 2, 609, 660, 1438, 1780.
4494.
HO
O
HO
OH
O
OH
OO
HO
OH
OH
5213 Deoxyschizandrin
OH
Wuweizisu A; Schizandrin A [61281-38-7] C24H32O6 (416.52). []D23 =
5207 1-Deoxy-D-ribitol
C5H12O4 (136.15). Source: SHI LUO ZI Anethum graveolens (fruit). Ref: 4177.
+86.7 (c = 0.30, CHCl3). Pharm: Antihepatotoxin (mus, due to carbon

tetrachloride, promotes markedly glycogenic in liver); NFAT transcription
inhibitor (IC50 = (7.230.21)mol/L, control Cyclosporin A, IC50 =
OH
(1.200.29)nmol/L)[5343]. Source: HONG HUA WU WEI ZI Schisandra
OH
rubriflora, HUA ZHONG WU WEI ZI Schisandra sphenanthera (dried
OH
ripe fruit: content scope of 12 origins = 0.07%~5.65%, mean content =
1.65%[5508]), WU WEI ZI Schisandra chinensis (dried ripe fruit: content
OH
scope of 6 origins = 0.17%~1.10%, mean content = 0.52%[5508]). Ref: 2,

658, 5343, 5508.
5208 2-Deoxy-D-ribitol1
C5H12O4 (136.15). Colorless syrup, []D22 = 17. Source: BEI SHA
SHEN Glehnia littoralis (fruit). Ref: 3525.
OH
O
O
O
CH2
OH
OH
O
O
OH
5214 Deoxyshikonin
5209 2-Deoxy-D-ribono-1,4-lactone
[43043-74-9] C16H16O4 (272.30). Pharm: Antibacterial (Staphylococcus
Dihydro-4-hydroxy-5-hydroxymethyl-2(3H)-furanone C5H8O4 (132.12).
aureus 209P, MIC = 40g/kg; Staphylococcus aureus TPR27, MIC =
Colorless oil liquid. Source: SHI LUO ZI Anethum graveolens (fruit),
20g/kg; Staphylococcus epidermidis TPR25, MIC = 80g/kg; Sarcina
WEI LING XIAN Clematis chinensis. Ref: 871, 2079, 4177.
lutea NIHJ, MIC = 40g/kg; Bacillus subtilis, MIC = 40g/kg). Source:

JIA ZI CAO Arnebia guttata, XIN ZANG JIA ZI CAO Arnebia euchroma
HO
(root: mean content of 3 origins = 0.174%[5508]), ZI CAO Lithospermum
erythrorhizon. Ref: 2, 658, 660, 5501, 5508.
HO
OH
OH
5210 (6S,9R)-Deoxyroseoside
C19H30O7 (370.45). Source: LIU QIU SHE GEN CAO Ophiorrhiza
liukiuensis (whole herb). Ref: 4527.
5215 20-Deoxyspiganthine
C25H35NO8 (477.56). Crystals (CHCl3:Me2CO = 1:1), mp 144~147C,
O
HO
[]D = +12 (c = 0.1). Pharm: Cardiac contraction inhibitor (guinea-pig

papillary muscle, causes a prolongation of the latency time and decrease
OH
OH
of contraction force, EC50 = 54nmol/L). Source: QU CHONG CAO

OH
5211 3'-Deoxysappanol
HO
OH
OH
OH
OH
HO
C16H16O5 (288.30). Source: SU MU Caesalpinia sappan (heartwood). Ref: 4494.
O
N
H
OH
O
HO
OH
70
5216 3,5-Deoxytigogenin
5220 1-Deoxy-D-xylitol
C27H40O2 (396.62). Source: CHA RUI SHU YU Dioscorea collettii,
CHAI HUANG JIANG Dioscorea nipponica ssp. rosthornii, CHUAN
4177.
LONG SHU YU Dioscorea nipponica, DUN YE SHU YU Dioscorea

zingiberensis, BI XIE Dioscorea hypoglauca [Syn. Dioscorea collettii var.
hypoglauca], FU ZHOU SHU YU Dioscorea futschauensis, HUANG
SHAN YAO Dioscorea panthaica, MIAN BI XIE Dioscorea septemloba,
H
HO
H
OH
H
OH
OH
SHU KUI YE SHU YU Dioscorea althaeoides, XIAN XI SHU YU

Dioscorea gracillima, XIAO HUA DUN YE SHU YU Dioscorea
parviflora. Ref: 6, 10, 660.
5221 Derricidin
C20H20O3 (308.38). Source: HONG E JI XUE TENG Millettia
O
erythrocalyx (stem cortex: yield = 0.0013%dw). Ref: 4624.
OH
5222 Derriscandenoside A
5217 Deoxytrillenoside A
25
C47H70O23 (1003.07). Amorphous powder, []D = 113.2 (c = 0.8,
7,8-Dihydroxy-4'-methoxyisoflavone8-O--glucopyranoside C22H22O10
MeOH). Source: JI LIN YAN LING CAO Trillium kamtschaticum
(446.41). Colorless viscous gum, []D29 = 55.56 (c = 0.36, CHCl3).
(underground part). Ref: 4403.
Source: PAN YUAN YU TENG Derris scandens. Ref: 1976.

O
O
OH
OH
O OH
O
OH
OH
OH
OO
OH
HO
OH
HO
OO
OH
OH
OH
OH
O OH
5223 Derriscandenoside B
7,8-Dihydroxy-4'-methoxyisoflavone
OH OH
7-O-[-rhamnopyranosyl-(16)]--glucopyranoside C28H32O14 (592.56).
5218 Deoxytrillenoside B
Colorless viscous gum, []D29 = 51.47 (c = 1.36, CHCl3). Source: PAN
C42H62O19 (870.95). Source: JI LIN YAN LING CAO Trillium
YUAN YU TENG Derris scandens. Ref: 1976.
kamtschaticum (underground part). Ref: 4403.

OH
OH
O
OO
OH
O OH
OH
OH OH
OH
O
OH
OH
OH
OH
OO
O
OH O O
OH
OH
5224 Derriscandenoside C
8-Hydroxy-4',7-dimethoxyisoflavone
OH OH
8-O-[-rhamnopyranosyl-(16)]--glucopyranoside C29H34O14 (606.59).

Colorless viscous gum, []D29 = 40.54 (c = 0.74, CHCl3). Source: PAN
5219 Deoxyvasicinone
[530-53-0] C11H10N2O (186.22). mp 109~110C. Pharm: Cholinergic.
Source: LUO TUO HAO Peganum nigellastrum, LUO TUO PENG
Peganum harmala, LUO TUO PENG ZI Peganum harmala. Ref: 6, 658.
OH
OO
OH
OH
OH OH O
OH
N
O
71
5225 Derriscandenoside D
5230 Derrisisoflavone B
Afromosin 7-O-[-rhamnopyranosyl-(16)]--glucopyranoside
C25H26O6 (422.48). Pale brown amorphous, []D = +3.0 (c = 0.054,
C29H34O14 (606.59). Colorless viscous gum, []D29 = 68.18 (c = 0.44,
EtOH). Pharm: Antifungal (dermatophyte Trichophyton
CHCl3). Source: PAN YUAN YU TENG Derris scandens. Ref: 1976.
mentagrophytes, 500~1000g/mL). Source: PAN YUAN YU TENG

Derris scandens. Ref: 2347.
OH
OO
OO
HO
HO
OH
OH
OH OH
OH
OH
5226 Derriscandenoside E
OH
5231 Derrisisoflavone C
C29H34O15 (622.59). Colorless viscous gum, []D29 = 90.90 (c = 0.11,
C26H28O6 (436.51). Colorless amorphous, []D = 63.8 (c = 0.043, EtOH).
CHCl3). Source: PAN YUAN YU TENG Derris scandens. Ref: 1976.
Pharm: Antifungal (dermatophyte Trichophyton mentagrophytes,

250g/mL). Source: PAN YUAN YU TENG Derris scandens. Ref: 2347.
OH
OO
OO
HO
OH
OH
OH OH
OH
OH
5227 Derriscanoside A
O
C28H32O13 (576.56). Light yellow powder, mp 115~117C. Pharm:

Antioxidant (DPPH scavenger, 10mol/L, ScRt = 18%, control BHT,
10mol/L, ScRt = 43%)[5319]. Source: PAN YUAN YU TENG Derris
scandens, TIAN SHAN ZHU ZI Garcinia dulcis (fruit). Ref: 664, 5319.
OH
5232 Derrisisoflavone D
C26H28O6 (436.51). Colorless amorphous, []D = 10.8 (c = 0.088,
OH
OO
OO
OH
OH
OH
OH OH
HO
OH
5228 Derriscanoside B
C29H34O14 (606.59). Light yellow powder, mp 145~147C. Source: PAN
OO
C26H28O6 (436.51). Pale brown amorphous, []D = +2.0 (c = 0.089, EtOH).
OO
OH
5233 Derrisisoflavone E
O
OH
OH

500~1000g/mL). Source: PAN YUAN YU TENG Derris scandens. Ref: 2347.
OH
OH
OH OH
5229 Derrisisoflavone A
C26H28O5 (420.51). Pale yellow amorphous, with yellow fluorescence.
500~1000g/mL)
OH
O
HO
[2347]
; antioxidant (DPPH scavenger, ScRt = 81.58%,
control BHT, ScRt = 71.5%)[3810]; antibacterial (Staphylococcus aureus
ATCC 25923, MIC = 16g/mL, Vancomycin, MIC = 0.5g/mL; MRSA

SK1, MIC = 4g/mL, Vancomycin, MIC = 1.0g/mL)
[3810]
; increases
blood pressure (anesthetized rats, increases in mean arterial blood

pressure, 4.0mg/kg, 7.5mmHg)[3810]. Source: PAN YUAN YU TENG
Derris scandens. Ref: 2347, 3810.
OH
5234 Derrisisoflavone F
C25H26 O6 (422.48). Colorless amorphous, []D = +20.6 (c= 0.12,
O
HO
HO
OH
OH
OH
72
5235 Derrone
5239 Desacetylcinobufotalin
5-Hydroxy-3-(4-hydroxyphenyl)-8,8-dimethyl-4H,8H-benzo[1,2-b:3,4-b']
C24H32O6 (416.52). Pharm: Cytotoxic (in vitro, KB, IC50 = 10g/mL;
dipyran-4-one [76166-59-1] C20H16O5 (336.35). Pharm: Antibacterial
HL-60, IC50 = 4.3g/mL; MH-60, IC50 > 25g/mL)[3082]. Source: CHAN
(Escherichia coli, MIA = 100.0g, control Chloramphenicol, MIA =
SU Bufo bufo gargarizans; Bufo melanostictus. Ref: 2, 6, 3082.
0.001g; Bacillus subtilis, MIA = 20.0g, Chloramphenicol, MIA =

O
0.001g; Staphylococcus aureus, MIA = 0.1g, Chloramphenicol, MIA =

0.001g)
[3785]
; antifungal (Candida mycoderma, MIA = 1.00g,
Miconazole, MIA = 0.0001g) [3785]; hepatoprotective (mus primary

cultured hepatocytes, antihepatotoxin induced by D-galactosamine (GalN),
OH
100mol/L, InRt = (4.01.0)%, inactive, control Silybin, 100mol/L,
InRt = (77.05.5)%)[4095]. Source: CU ZHUANG YU TENG Derris

robusta (seed), GUANG BU DING GONG TENG Erycibe expansa,
OH
Bolusanthus speciosus (root wood). Ref: 3785, 4095.
OH
5240 Desacetyluvaricin
OH
H
HO
[98767-45-4] C37H66O6 (606.93). Colorless oil, []D25 = +30.3 (c = 0.26,

CHCl3). Pharm: Cytotoxic (hmn hepatoma cell lines HepG2, IC50 =
0.062ng/mL, control Adriamycin, IC50 = 0.241g/mL; hmn hepatoma
cells transfected with hepatitis B virus Hep2,2,15, IC 50 = 0.071ng/mL,

Adriamycin, IC50 = 0.450g/mL). Source: CI GUO FAN LI ZHI Annona
5236 Desacetoxymatricarin
[17946-87-1] C15H18O3 (246.31). Pharm: Antineoplastic; cytotoxic; plant
muricata. Ref: 5377.
growth inhibitor. Source: BAN GUAN MU MU JU Matricaria

OH
suffruticosa, Achillea sp., Artemisia sp. Ref: 658.
OH
O
O
O
5241 Desacyl-boninsaponin A
C54H88O25 (1137.29). Source: RI BEN HOU PI XIANG Ternstroemia
japonica (fresh fruit: yield = 0.00066%fw). Ref: 4730.
5237 Desacetylbufotalin
C24H34O5 (402.54). Pharm: Cytotoxic (in vitro, KB, IC50 = 0.79g/mL;
HL-60, IC50 = 0.025g/mL; MH-60, IC50 > 25g/mL)[3082]. Source:
CHAN SU Bufo bufo gargarizans; Bufo melanostictus. Ref: 2, 6, 3082.
OH
HO
HO
HO
H
H
HO
HO
OH
O
OH
OH
O
HO
OO
OH
OO
O HO
O
O
HO
HO
OH
OH
OH
OH
OH
5238 Desacetylcinobufagin
C24H32O5 (400.52). Pharm: Cytotoxic (in vitro, KB, IC50 = 0.44g/mL;
HL-60, IC50 = 1g/mL; MH-60, IC50 > 25g/mL)
[3082]
. Source: CHAN
SU Bufo bufo gargarizans; Bufo melanostictus. Ref: 2, 6, 3082.
5242 Desacylkondurangogenin C
C21H36O5 (368.52). White amorphous powder, mp 127C, []D =
+135.6(c = 0.14, CHCl3). Source: ROU LEI NIU NAI CAI Marsdenia
roylei (aerial parts). Ref: 3490.
O
O
OH
HO
OH
H
H
HO
OH
HO
OH
73
5243 Desacyl-theasaponin E
5248 Deserpidine
C52H82O25 (1107.22). Source: PU ER CHA Camellia sinensis var.
[131-01-1] C32H38 N2O8 (578.67). Three crystals types (methanol): -,
assamica (seed and leaf). Ref: 4537.
mp 228~232C; -, mp 230~232C; -, mp 138C and 226~232C

(two-melting points, 173 solidifying), []D20 = 163 (c = 0.5,
OH
pyridine). Pharm: CNS depressant; antihypertensive. Source: CUI TU

LUO FU MU Rauvolfia vomitoria, GU BA LUO FU MU Rauwolfia
OH
H
O
HO
OO
OH
OH
serpentina. Ref: 661.
OH
OH
cubana, HAI BIN LUO FU MU Rauwolfia littoralis, HUI BAI MAO

LUO FU MU Rauwolfia canescens, YIN DU LUO FU MU Rauwolfia
OH
HO
HO
OO
OH
OH
OO
OH
N
H
OH
OH
5244 Desaspidinol
O
O
[437-72-9] C11H14O4 (210.23). Source: GUAN ZHONG Dryopteris
O
O
crassirhizoma. Ref: 6, 1521.

O
HO
5249 5-Desgalloylstachyurin
C34H24O22 (784.56). Source: BAI SHAO Paeonia albiflora [Syn. Paeonia
lactiflora] (fresh fruit: yield = 0.015%fw). Ref: 4695.
OH
5245 Descurainin
5-Hydroxymethyl-6-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxa-bicyclo[3,2
OH
HO
,1]oct-3-en-2-one C16H18O6 (306.32). Colorless needles, mp 193~195C,

[]D20 = +1.7 (c = 0.23, MeOH). Source: BO NIANG HAO Descurainia
O
HO
O
Sophia (seeds). Ref: 2548.
O
O
OH
H
HO
OH
OH
O
HO
HO
OH HO
H
O
OH
OH HO
HO
OH
5246 Descurainolide A
4-(4-Hydroxy-3,5-dimethoxy-phenyl)-5-methyl-dihydro-furan-2-one
C13H16O5 (252.27). Colorless needles, mp 117~118C, []D20 = +0.3 (c =
0.19, Me2CO). Source: BO NIANG HAO Descurainia Sophia (seeds).
Ref: 2548.
[40043-49-0] C50H82O22 (1035.20). Amorphous powder, []D28 = 38.7

(c = 0.10, chloroform: methanol = 1:1). Pharm: cAMP phosphodiesterase
5250 Desglucolanatigonin II
inhibitor (IC50 = 123mol/L). Source: CI JI LI Tribulus terrestris. Ref:

706, 738, 951.
O
O
OH
O
H
5247 Descurainolide B
HO
trans-3-(4-Hydroxy-3,5-dimethoxy-benzylidene)-5-(4-hydroxy-3,5-dimet
HO
hoxy-phenyl)-dihydrofuran-2-one C21H22O8 (402.40). Colorless needles,

mp 201~203C, []D20 = +2.3 (c = 0.37, MeOH). Source: BO NIANG
HAO Descurainia Sophia (seeds). Ref: 2548.
O
O
OH
OH
H
OO
O O
OH
OH
HO
OH HO
OH
O
O
O
O
OH
O
HO
O
OH
OH
H
H
74
5251 Desglucomusennin
5256 N-Desmethyl-8-ethoxy pretazettine
C45H72O16 (869.07). Pharm: Anthelmintic. Source: QU CHONG HE
C19H23NO5 (345.40). Amorphous, []D28 = +34 (c = 0.14, CHCl3). Pharm:
HUAN Albizzia anthelmintica. Ref: 658.
AChE inhibitor (IC50 = (4198)mol/L, control Galanthamine, IC50 =

(1.90.2)mol/L) [4952]. Source: LIN JING ZHONG ZI WEN SHU LAN
Crinum bulbispermum. Ref: 2369, 4952.
O
H
H
OH O O
OH
OH
OH
H
N
O
O
OH O O
OH
5257 Des-O-methylicariin
OH OO
OH
Epimedoside A [39012-04-9] C32H38O15 (662.65). mp 235~237C. Source:

CU MAO YIN YANG HUO Epimedium acuminatum, CHUAN E YIN
OH
YANG HUO Epimedium fargesii, YIN YANG HUO Epimedium

brevicornum, YIN YANG HUO GEN Epimedium brevicornum. Ref: 2, 6,
5252 Desmanthin 2
[85541-03-3] C28H24O16 (616.49). Yellow powder, mp 196C. Source: YI
112, 514, 567, 624.
LI NUO HE HUAN CAO Desmanthus illinoensis. Ref: 1521.

OH
OH
HO
OO
OH
O
HO
O
HO
OH
OH
O
O
OO
OH
OH
OH OO
OHOH
5258 Des-O-methyllasiodiplodin
C16H22O4 (278.35). Pharm: Prostaglandin biosynthesis inhibitor (20g/mL,
OH OH
5253 N-Desmethoxyhumantenine
C20H24N2O2 (324.43). mp 238~240C, []D = 188.5. Source: GOU
InRt = 62.5%). Source: ZI CAO Lithospermum erythrorhizon, XIN

ZANG JIA ZI CAO Arnebia euchroma. Ref: 2193.
HO
OH
WEN Gelsemium elegans. Ref: 14.

O H
OH
HO
OH
OH
N
O
N
H
5259 4'-Desmethylpiplartine
5254 N-Desmethoxyrankinidine
[122590-02-7] C19H22N2O2 (310.40). mp 258~260C, []D = 169.2.
Source: GOU WEN Gelsemium elegans. Ref: 14.
O H
N-(4'-Hydroxy-3',5'-dimethoxycinnamoyl)-3-pyridin-2-one C16H17NO5
(303.32). Yellow oil. Source: Piper cenocladum (leaf). Ref: 3896.
O
O
N
O
HO
O
HN
O
N
H
5260 N-Desmethylthalidezine
5255 N-Desmethyl-8-ethoxy pretazettine

C19H23NO5 (345.40). Amorphous, []D28 = +160.63 (c = 0.09, CHCl3).
Pharm: AChE inhibitor (IC50 = (23413)mol/L, control Galanthamine,
IC50 = (1.90.2)mol/L)[4952]. Source: LIN JING ZHONG ZI WEN SHU
[65230-06-0] C37H40N2O7 (624.74). Colorless acicular crystals (methanol),

mp 173~174C, []D25 = +280 (c = 0.14, methanol). Pharm:
Antihypertensive (dog, rat). Source: BING GUO TANG SONG CAO
Thalictrum podocarpum. Ref: 661.
LAN Crinum bulbispermum. Ref: 2369, 4952.
OH
O
O
H
N
O
HN
H
O
O
H
O
O
O
75
5261 Desmethylxanthohumol
5266 Desmodilactone
C20H20O5 (340.38). Source: PI JIU HUA Humulus lupulus (strobile). Ref:
C8H13NO3 (171.20). Colorless massive crystals, mp 84~85C, []D18 =
4789.
16.4 (c = 0.11, MeOH). Source: GUANG JIN QIAN CAO Desmodium

styracifolium. Ref: 260.
OH
O
H
N
HO
OH
O
OH
5262 Desmethylxanthohumol B
()-{(2E)-1-(3,4-Dihydro-3,5,7-trihydroxy-2,2-dimethyl-2H-1-benzopyra
5267 Desmodimine
n-6-yl)-3-(4-hydroxyphenyl)-2-propen-1-one}; DMX-B C20H20O6
[150036-83-2] C12H15NO4 (237.26). Colorless gummy substance. Source:
(356.38). Yellow orange solid. Source: PI JIU HUA Humulus lupulus
GUANG JIN QIAN CAO Desmodium styracifolium. Ref: 260.
(strobile). Ref: 4789.

HO
OH
OH
O
OH
OH
5268 Desmosdumotin A
5263 Desmethylxanthohumol J
(2E)-1-[2,3-Dihydro-4,6-dihydroxy-2-(1-hydroxy-1-methylethyl)-7-benzo
furanyl]-3-(4-hydroxyphenyl)-2-propen-1-one; DMX-J C20H20O6
(356.38). Yellow orange solid. Source: PI JIU HUA Humulus lupulus
5-Hydroxy-7-methoxy-8-formyl-3-benzoyl-2,6-dimethyl-2S,3R-dihydroc
hromone C20H18O6 (354.36). Yellow massive crystals (CHCl3 MeOH),
mp 124~125C. Source: MAO YE JIA YING ZHAO GEN Desmos
dumosus. Ref: 685.
(strobile). Ref: 4789.
O
O
HO
OH
O
OH
OH
OH
5269 Desmosdumotin D
2-Methoxy-3-methyl-4,6-dihydroxy-5(3'-hydroxyl)cinnamoylbenzaldehy
5264 Desmodianone D
de C18H16O6 (328.32). Yellow acicular crystals (CHCl3 MeOH), mp
2,3-Dihydro-5,7-dihydroxy-6-methyl-3-(1a,2,3,3a,8b,8c-hexahydro-6-hyd
147~148C. Pharm: Anti-HIV (a lead candidate)[4881]. Source: MAO YE
roxy-1,1,3a-trimethyl-1H-4-oxabenzo[f]cyclobut[c,d]inden-7-yl)-4H-1-be
JIA YING ZHAO GEN Desmos dumosus. Ref: 685, 4881.
nzopyran-4-one C26H28O6 (436.51). Source: DAN HUI BAI SHAN MA

HUANG Desmodium canum. Ref: 3444.
O
O
OH
H
HO
OH
OH
O
HO
OH
5270 Desmosflavone
5265 Desmodianone E
5-Hydroxy-7-methoxy-6,8-dimethyflavone C17H14O5 (298.30). Orange
2,3-Dihydro-5,7-dihydroxy-6-methyl-3-(6a,7,8,10a-tetrahydro-3-hydroxy
sandy crystals (chloroform), mp 197~198C. Source: JIA YING ZHAO
-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-2-yl)-4H-1-benzopyran-4-one
Desmos cochinchinensis [Syn. Desmos chinensis]. Ref: 312.
C26H28O6 (436.51). Source: DAN HUI BAI SHAN MA HUANG

Desmodium canum. Ref: 3444.
OH
O
HO
OH
OH
O
HO
76
5271 16-Desoxybarringtogenol C
5275 8-Desoxy-3,4-epoxyrupiculin-B
C30H50O4 (474.73). mp 288.0~290.5C. Source: RI BEN QI YE SHU
C15H18O4 (262.31). Colorless gum, []D22 = +46 (c = 0.1, EtOH). Pharm:
Aesculus turbinata. Ref: 6.
Cytotoxic (in vitro, KB, IC50 = 2.0g/mL). Source: Warionia saharae

(leaf: yield = 0.0008%dw). Ref: 4620.
OH
HO
OH
OH
H
HO
O
O
5272 Desoxycordifoline
C28H30N2O11 (570.56). mp 144~146C. Pharm: Antibacterial (in vitro:
5276 8-Desoxygartanin
Staphylococcus aureus, Bacillus subtilis, Bacillus coli, Bacillus
C23H24O5 (380.44). Pharm: Antioxidant (DPPH scavenger, 10mol/L, ScRt
diphtheriae, Streptococcus sp., Streptobacillus sp., Salmonella sp.,
= 8%, control BHT, 10mol/L, ScRt = 43%)[5319], cytotoxic (KB cancer cell
Bacillus proteus, Bacillus lactis, Klebsiella pneumoniae); antileishmanial;
lines, inactive; BC-1, inactive; NCI-H187, IC50 = 16.88g/mL Ellipticine,
antifungal (Aspergillus niger). Source: DI SHI WU TAN Nauclea
IC50 = 0.39g/mL)[1619]; antibacterial (MRSA, MIC = 16g/mL; control
diderrichii. Ref: 2178.
Vancomycin, MIC = 2g/mL)[4735]. Source: DAO NIAN ZI Garcinia

mangostana (young fruit: yield = 0.0060%dw)[1619], DAO NIAN ZI
Garcinia mangostana (fruit hull), HEI XIAN TIAO TENG HUANG
OH
Garcinia nigrolineata (leaf: yield = 0.00047%dw)[4735], MEI LI TENG
N
H
HUANG Garcinia speciosa (trunk bark and stems), TIAN SHAN ZHU ZI
O
O
HO
Garcinia dulcis (fruit). Ref: 1619, 3066, 4735, 5319, 5491.
OH
OH
OH
OH
5273 Desoxycordifolinic acid
OH
OH
[88839-94-5] C27H28N2O11 (556.53). mp 206~208C, []D = 45.7 (c =

0.126, MeOH). Pharm: Antibacterial (in vitro: Staphylococcus aureus,
5277 Desrhamnosylacteoside
C23H26O11 (478.46). Source: CHANG YE CHE QIAN Plantago
Source: DI SHI WU TAN Nauclea diderrichii. Ref: 2178.
lanceolata. Ref: 5020.
OH
N
H
OH
OH
H
O H
OO
HO
OH
OH
HO
O
HO
O
O
OH
OH
HO
OH
OH
5278 Desrhamnosylisoacteoside
C23H26O11 (478.46). Source: CHANG YE CHE QIAN Plantago
5274 8-Desoxy-3,4-epoxyrupiculin-A
lanceolata. Ref: 5020.
C15H18O4 (262.31). Colorless gum, []D22 = 22 (c = 0.1, EtOH). Pharm:

Cytotoxic (in vitro, KB, IC50 = 1.7g/mL). Source: Warionia saharae
(leaf: yield = 0.0004%dw). Ref: 4620.
OO
HO
OH
HO
OH
O
H
O
OH
HO
HO
OH
O
77
5279 Detetrahydroconidendrin
5283 Dhurrin
C20H16O6 (352.35). Pharm: Antibacterial (18 methicillin-resistant
p-Hydroxymandelonitril-glucoside [21401-21-8] C14H17NO7 (311.29).
Staphylococcus aureus MRSA, MIC = 4, 8, 16, or >64g/mL)[3052];
Pharm: Toxin. Source: AO ZHOU JIAN GUO Macadamia ternifolia,
antioxidant (ferric thiocyanate method, 0.5mmol/L, stronger than control
GAO LIANG Sorghum vulgare, KUN LAN SHU Trochodendron
Vitamin E; DPPH radical scavenger, DPPH 0.1mmol/L, 0.02mmol/L,
aralioides, LIU LI JU Borago officinalis, YE YING SU Papaver
stronger than control L-Cysteine)[4791]. Source: DAN YE MAN JING Vitex
nudicaule, Platanus sp. Ref: 6, 658, 1521.
rotundifolia [Syn. Vitex trifollia var. simplicifolia] (underground part:

N
yield = 0.00017%dw)[3052], HUANG JING ZHONG ZI Vitex negundo

[4791]
(seed: yield = 0.0051%)
. Ref: 3052, 4791.
HO
OO
OH
O
O
OH
OH
OH
HO
5284 7,18-Diacetoxyabiet-8(14)-en-13-ol
O
C24H38O5 (406.57). Colorless oil, []D = +14.7 (c = 1.0, CHCl3). Pharm:
OH
Cytotoxic (A549, IC50 > 5g/mL; H116, IC50 > 5g/mL; PSN1, IC50 >
5g/mL; T98G, IC50 > 5g/mL; SKBR3, IC50 > 5g/mL). Source: BEI
5280 Detetrahydroconidendrin B
FEI XUE SONG Cedrus atlantica (cone). Ref: 5248.
C21H18O6 (366.37). Brown amorphous solid. Source: DAN YE MAN
OH
JING Vitex rotundifolia [Syn. Vitex trifollia var. simplicifolia]

(underground part: yield = 0.000057%dw). Ref: 3052.
O
O
O
OH
5285 1,2-Diacetoxy-6-benzoyloxy-9-cinnamoyloxy--dihydro-
agarofuran
O
C35H40O9 (604.70). Pharm: NO production inhibitor (mus, macrophage
RAW264.7 cells, activated by LPS, IC50 = 43.7mol/L, control

Aminoquanidine IC50 = 18.2mol/L). Source: NAN SHE TENG GUO
5281 Detetrahydroconidendrin C
Celastrus orbiculatus [Syn. Celastrus articulatus]. Ref: 2584.
C21H18O6 (366.37). Yellowish oil. Source: DAN YE MAN JING Vitex
rotundifolia [Syn. Vitex trifollia var. simplicifolia] (underground part:
yield = 0.000042%dw). Ref: 3052.
O
O
O
O
O
OH
5286 1,8-Diacetoxy-9-benzoyloxydihydro--agarofuran

MeOH). Pharm: Intestinal smooth muscle relaxant (in vitro, rat ileum,
5282 Dextrobursehernin
1g/mL, relaxant effect = (7.31.7)%, control Papaverine, relaxant
C21H22O6 (370.41). Colorless liquid, []D25 = +36.0 (c = 1.0). Source: YE
effect = (28.67.3)%). Source: DENG YOU TENG ZI Celastrus
XIA ZHU Phyllanthus urinaria. Ref: 3410.
paniculatus. Ref: 5002.
O
O
O
O
O
O
O
O
O
O
78
5287 (2R*,3S*,4R*,5R*,9S*,11S*,15R*)-5,15-Diacetoxy-3-benzoyloxy-
5292 1,6-Diacetoxy-8,9-dibenzoyloxy--dihydroagarofuran
14-oxolathyra-6(17),12E-diene
C33H38O9 (578.67). Pharm: NO production inhibitor (mus, macrophage
Euphorbia factor L3 C31H38O7 (522.64). Colorless oil. Source: HAI BO NA
RAW264.7 cells activated by LPS, very weak activity). Source: NAN SHE
DA JI Euphorbia hyberna. Ref: 1521, 2153.
TENG GUO Celastrus orbiculatus [Syn. Celastrus articulatus]. Ref: 2584.
O
O
O
O
O
O H
O
O
O
O
5288 (3S,5S)-3,5-Diacetoxy-1,7-bis(4-hydroxy-3-methoxyphenyl)heptane
C25H32O8 (460.53). Colorless oil, []D26 = +7.0 (c = 0.68, CHCl3). Source:
SHENG JIANG Zingiber officinale. Ref: 3803.
O
trihydroxy-11(151)-abeo-taxene
C38H44O12 (692.77). []D = 8 (CHCl3). Source: JIANG GUO ZI SHAN
5293 4,7-Diacetoxy-2,9-dibenzoyloxy-5,20-epoxy-10,13,15-
Taxus baccata. Ref: 662.
OH
HO
5289 9,10-Diacetoxy-5-cinnamoyloxytaxa-4(20),11-dien-13-ol
C 33 H 42 O 7 (550.70). Colorless gum, []D
24
O
HO
= 13 (c = 0.03, CHCl 3 ).
Source: YUN NAN HONG DOU SHAN Taxus yunnanensis (seed). Ref:
3991.
HO
HO
HO
O
O
O
O
5294 9,10-Diacetoxy-5,13-dihydroxy-4(20),11-taxadiene
Diacetoxydihydroxytaxadiene C24H36O6 (420.55). mp 235C, []D = +146
(from Taxus baccata), mp 234~236C, []D = +144.2 (CHCl3) (from Taxus
5290 1R,5R-Diacetoxycyclomyltaylan-10-one
C19H26O5 (334.42). Amorphous powder, []D20 = 23.2 (c = 0.9, MeOH).
mairei). Source: HONG DOU SHAN Taxus chinensis, JIANG GUO ZI

SHAN Taxus baccata, MEI LI HONG DOU SHAN Taxus mairei. Ref: 662.
O
Source: Bazzania madagassa. Ref: 4458.
O
O O
HO
neotecleanin
C30H36O10 (556.62). Colorless needle-like crystals (MeCNH 2O), mp
179~180C. Source: Turraea wakefieldii (root cortex). Ref: 3459.
O
O
C24H36O6 (420.55). Colorless oil, []D = +6.2 (c = 0.13, CHCl3). Pharm:

5g/mL; T98G, IC50 > 5g/mL; SKBR3, IC50 > 5g/mL). Source: BEI FEI
XUE SONG Cedrus atlantica (cone). Ref: 5248.
O
O
O
O
O
O
HO
H
O
H
OH
5295 7,18-Diacetoxy,9,13-epi-dioxiabiet-8(14)-ene
5291 11,12-Diacetoxy-1-deoxo-14,15-epoxy-3-hydroxy-2-oxo-
O
O
O
O
79
5296 (1R,2R,5Z,7R,8S,9R,10R,12R,14R,17S)-2,14-Diacetoxy-8,17-epoxy-
5300 1,2-Diacetoxy-8-(-furancarbonyloxy)-9-benzoyloxy-13-iso-
9,12-dihydroxybriara-5,11(20)-dien-19-one
butanoyloxy-4,6-dihydroxy--dihydroagarofuran
C24H32O9 (464.52). Colorless oil, []D25 = +113 (c = 0.1, CHCl3); []D25 =
C35H42O14 (686.72). Amorphous white powder, mp 248~249C, []D24 = +7.6
+115.1 (c = 0.08). Source: CUI DENG XIN LIU SHAN HU Junceella
(c = 0.66, CHCl3). Pharm: Insecticidal (Mythimna separata, KD50 = 73.3g/g).
fragilis, LEI DENG XIN LIU SHAN HU Junceella gemmacea. Ref: 2554.
Source: DIAO GAN MA Celastrus angulatus (root cortex). Ref: 5228.
O
O
O
O
O
HO
O
O
H
O O
OH
O
O
HO
OH
5297 rel-(2S,5R,6R,8S,9S,10R,18S,19R)-diacetoxy-18,19-epoxy-6-hy-
5301 11,12-Diacetoxyharrisonin
droxy-2-(2-methylbutanoyloxy)cleroda-3,13(16),14-triene
C31H36O14 (362.62). Colorless crystals (acetone), mp.249~250C. Source: A
C29H42O8 (518.65). Pharm: Cytotoxic (in vitro, PC3, IC50 = 1.8mol/L,
BI XI NI YA NIU JIN GUO Harrisonia abyssinica. Ref: 2351.
control Paclitaxel, IC50 = 0.016mol/L; Hep3B, IC50 = 2.4mol/L, Paclitaxel,
membranacea (leaf and twig: yield = 0.023%dw). Ref: 3010.

O
O
O
5298 7,12-Diacetoxy-14,15-epoxy-11-hydroxyneotecleanin
C30H38O9 (542.63). White amorphous solid, mp 180~182C. Source: Turraea
5302 3,5-Diacetoxy-1-(4-hydroxy-3,5-dimethoxyphenyl)-7-(4-hydroxy-3methoxyphenyl) heptane

C26H34O9 (490.56). Source: GAN JIANG Zingiber officinale, SHENG JIANG
Zingiber officinale. Ref: 2.
wakefieldii (root cortex). Ref: 3459.

O
O
O OH
OH
HO
H
O
OH
O
O
O
OH
HO
O
IC50 = 0.031mol/L). Source: MO ZHI JIAO GU CUI Casearia
5303 10,18-Diacetoxy-8-hydroxy-2,6-dolabelladiene
5299 11,12-Diacetoxy-14,15-epoxyneotecleanin
C24H38O5 (406.57). Colorless needles, mp 136~138C, []D25 = 115 (c =
C30H36O9 (540.62). White amorphous solid, mp 161~162C. Pharm:
0.0016, CHCl3). Pharm: Anti-HSV-1 (Vero cells infected by HSV-1, 50mol/L,
Larvicidal (mosquito late third or early fourth-instar larvae of Anopheles
(895)% of cytopathic effect inhibition of herpes virus); cytotoxic inactive
gambiae s.s., LD50 = 7.07mg/L). Source: Turraea wakefieldii (root cortex).
(200mol/L); HIV-1 RT inhibitor (40mol/L, InRt = 20%, positive control
Ref: 3459.
AZT, 0.01mol/L, InRt = 85%). Source: BA XI ZONG ZAO Dictyota pfaffii.

O
O
O O
Ref: 5023.
H
O
H
H
OH
80
5304 9,10-Diacetoxy-13-hydroxy-5-O-(-D-glucopyranosyl)taxa-
5309 ent-(16S)-1,14-Diacetoxy-7-hydroxy-17-methoxykauran-15-one
4(20),11-diene
C30H46O11 (582.69). Amorphous solid, []D22 = +33 (c = 0.3, CHCl3). Source:
CHCl3). Source: DONG JIN BA DOU Croton tonkinensis (leaf). Ref: 4444.
JIA NA DA HONG DOU SHAN Taxus canadensis (needle: yield =

0.000075%dw). Ref: 4734.
O
O
O
O
HO
O
O
OH
5310 2,5-Diacetoxy-14-(2'S,3'R)-3'-hydroxy-2'-methylbutanoate-
H
HO
HO HO
10-O-(-D-glucopyranosyl)taxa-4(20),11-diene
OO

canadensis (needle: yield = 0.00013%dw). Ref: 4734.
OH
5305 ent-1,7-Diacetoxy-14-hydroxykaur-16-en-15-one
C24H34O6 (418.53). White amorphous powder, []D15 = 22 (c = 0.10, MeOH).
HO
HO
Source: DONG JIN BA DOU Croton tonkinensis (leaf). Ref: 4057.
HO
HO
H
O H O
OH
H
O
HO
5311 7,12-Diacetoxy-11-hydroxyneotecleanin
C24H34O6 (418.53). White amorphous powder, []D = 16 (c = 0.10, MeOH).
C30H38O8 (526.63). White amorphous solid, mp 186~187C. Pharm:
Source: DONG JIN BA DOU Croton tonkinensis (leaf). Ref: 4057.
Larvicidal (mosquito late third or early fourth-instar larvae of Anopheles
15
gambiae s.s., LD50 = 7.05mg/L). Source: Turraea wakefieldii (root cortex).

Ref: 3459.
O
O
O
O
OH
O
O OH
H
O
CHCl3). Source: DONG JIN BA DOU Croton tonkinensis (leaf). Ref: 4444.
5312 1,2-Diacetoxy-8-isobutanoyloxy-9-benzoyloxy-13-(-methyl)
butanoyloxy-4,6-dihydroxy--dihydroagarofuran
H
O
C35H48O13 (676.77). Amorphous white powder, mp 95~96C, []D24 = 12.8
O
OH
(c = 0.60, CHCl3). Pharm: Insecticidal (Mythimna separata, KD50 =

135.3g/g). Source: DIAO GAN MA Celastrus angulatus (root cortex). Ref:
5228.
5308 6,7-Diacetoxy-13-hydroxy-labda-8,14-diene
[2413]
C24H38O5 (406.57). Pharm: Affinity to dopamine-D2-receptor
. Source:
SUI HUA MU JING Vitex agnuscastus. Ref: 2413.
O
O
H
OH
O
O
O
O
O
O
O
HO
O
OH
81
5313 7,18-Diacetoxy-13-methoxyabiet-8(14)-ene
5317 6,7-Diacetoxyroyleanone
C25H40O5 (420.59). Colorless oil, []D = +43.7 (c = 0.1, CHCl3). Source: BEI
C24H32O7 (432.52). Yellowish solid, []D23 = 56.7 (c = 0.3, CHCl3). Source:
FEI XUE SONG Cedrus atlantica (cone). Ref: 5248.
TAI WAN SHAN Taiwania cryptomerioides (bark). Ref: 4443.
OH
O
O
O
O
O
O
5314 8,10-Diacetoxy-2-methoxy-3,11(13)-guaiadiene-12,6-olide
C20H26O7 (378.43). []D25 = 32.4 (c = 0.75, CHCl3). Pharm: Cytotoxic (in
vitro, ACHN cell, IC50 = (3.260.28)g/mL, control Adriamycin, IC50 =
5318 Diacetoxytetrahydroxytaxadiene
(0.090.03)g/mL; LOX-IMVI, IC50 = (3.780.31)g/mL, Adriamycin, IC50 =
2,9-Diacetoxy-1,5,10,13-tetrahydroxytaxa-4(20),11-diene C24H36O8
(0.050.02)g/mL; SW620, IC50 = (4.750.18)g/mL, Adriamycin, IC50 =
(452.55). mp 154C, []D = 22 (CHCl3) Source: JIANG GUO ZI SHAN
(0.190.07)g/mL; PC3, IC50 = (3.820.26)g/mL, Adriamycin, IC50 =
Taxus baccata, HONG DOU SHAN Taxus chinensis. Ref: 662.
(0.760.12)g/mL; A549, IC50 = (3.670.29)g/mL, Adriamycin, IC50 =

(0.280.09)g/mL)[5455]; anti-apoptosis (etoposide-induced, IC50 =
(13.70.9)g/mL; control PDTC, IC50 = (8.00.5)g/mL). Source: BEI YE JU
OH O
Chrysanthemum boreale. Ref: 5455.

O
HO
OH
OH O H
O
O
5319 5,3'-Diacetoxy-3,6,7,4'-tetramethoxyflavone
5315 2,5-Diacetoxy-14-2'-methylbutanoate-10-O-(-D-glucopyra-
C23H22O10 (458.43). mp 140~142C. Pharm: Cytotoxic (in vitro, Col2, ED50 =
nosyl)taxa-4(20),11-diene
15.9g/mL; hTERT-RPE1, ED50 = 0.4g/mL; HUVEC, ED50 = 0.1g/mL; KB,
C35H54O12 (666.81). Amorphous solid, []D22 = +32 (c = 0.15, CHCl3).

Source: JIA NA DA HONG DOU SHAN Taxus canadensis (needle: yield =
ED50 = 0.2g/mL; HUVEC, ED50 = 0.1g/mL; Lu1, ED50 = 0.7g/mL).

Source: HUANG JING YE Vitex negundo. Ref: 4699.
0.00014%dw). Ref: 4734.

O
HO
HO
HO
HO
O
O
O
O H O
O
O
5320 2,7-Diacetoxy-5,10,13-trihydroxy-2(320)abeotaxane-9-one
5316 11,12-Diacetoxyneotecleanin
[260367-32-6] C24H34O8 (450.53). Source: MEI LI HONG DOU SHAN Taxus
C30H36O8 (524.62). White amorphous solid, mp 154~156C, []D20 = 34.0 (c
mairei. Ref: 2414.
= 1.59, CHCl3). Pharm: Larvicidal (mosquito late third or early fourth-instar
larvae of Anopheles gambiae s.s., LD50 = 7.83mg/L). Source: Turraea

wakefieldii (root cortex). Ref: 3459.
O
O
O O
H
O
OH
O
HO
H
H
O
HO
82
5321 7,13-Diacetoxy-2,5,10-trihydroxy-2(320)abeotaxane-9-one
5326 3,12-Diacetyl-7-benzoyl-8-nicotinoylingol
2,10-Dideacetyltaxin B' [219999-48-1] C24H34O8 (450.53). Colorless crystals,
C37H41NO10 (659.74). White powder, mp 90~92C, []D25 = 61 (c = 0.5,
mp 220~222C, []D25 = 11.2 (c = 0.002, CHCl3). Source: MEI LI HONG
CHCl3). Source: YIN DU DUO ZHI DA JI Euphorbia nivulia. Ref: 1985.
DOU SHAN Taxus mairei. Ref: 2414.
O
O
O
O
O
O
HO
O
O
OH
O
OH
5327 N,O-Diacetylcassine
5322 7,9-Diacetoxy-5,13,14-trihydroxy-10-oxotaxa-4(20),11-diene
C22H39NO4 (381.56). Pharm: Cytotoxic (P388 IC50 = 5.2g/mL, control 5-FU,
C24H34O8 (450.53). Source: AO DA LI YA HONG DOU SHAN Austrotaxus
IC50 = 0.99g/mL; KB, IC50 = 5.2g/mL, Doxorubicin, IC50 = 0.57g/mL;
spicata. Ref: 662.
BC-1, IC50 = 7.1g/mL, Doxorubicin, IC50 = 0.21g/mL); cytotoxic (brine
O O
shrimp lethality, IC50 = 17.0g/mL, control Monocrotophos, IC50 = 0.24g/mL).

Source: ZHUANG GUAN FAN XIE Senna spectabilis (flower). Ref: 5480.
HO
OH
H
OH
5323 (3E,7E)-2,10-Diacetoxy-5,13,20-trihydroxy-3,8-secotaxa3,7,11-trien-9-one
C24H34O8 (450.53). []D = 15.5 (CHCl3). Source: HONG DOU SHAN
Taxus chinensis. Ref: 662.
5328 2,10-Diacetyl-5-cinnamoyl-7-hydroxy phototaxicin II

O
O
O
O OH
OH
O
OH
HO
O
H O
OH
5324 7,16-Diacetoxy withanolide D

7,16-Diacetoxy-4,20R-dihydroxy-5,6-epoxy-1-oxowitha-2,24-dienolide
C33H42O10 (586.69). mp 163~166 (EtOAc) Source: BA XI YE YAN Acnistus
5329 2,9-Diacetyl-5-cinnamoylphototaxicin II
O
arborescens. Ref: 2003.
OH O
O
OH
H
O
O
H O
H
H
H
H
O
OH
5330 2,10-Diacetyl-5-cinnamoylphototaxicin II
5325 3,12-Diacetyl-8-benzoylingol
C31H38O9 (554.64). White powder, mp 95~97, []D25 = 27 (c = 0.5, CHCl3).
O OH
Source: YIN DU DUO ZHI DA JI Euphorbia nivulia. Ref: 1985.

O
O
O
O
O
O
O
O
OH
O
H O
O
83
5331 Diacetyldecinnamoyltaxicin I
5335 3,15-Di-O-acetyl-9-hydroxyamphoricarpolide
2,10-Di-O-acetyl-5-decinnamoyl-taxicin I C24H34O8 (450.53). mp 165C, []D
C19H24O7 (364.40). Colorless gum, [] D25 = +3.4 (c = 0.25, CHCl3). Source:
= +30 (CHCl3). Source: JIANG GUO ZI SHAN Taxus baccata, HONG DOU
Amphoricarpos neumayeri ssp. neumayeri (aerial parts), Amphoricarpos
SHAN Taxus chinensis. Ref: 662.
neumayeri ssp. murbeckii (aerial parts). Ref: 3842.
OH O
OH
O OH
OH
5336 4,6-Di-O-acetyl hygrophorone A12
4,5-trans-4-Acetoxy-5-hydroxy-5-(1-hydroxytridecyl)-2-cyclopenten-1-one
5332 2,6-Diacetyl-3,4-diisobutyryl-1-O-octylglucopyranoside
C26H44O10 (516.63). Pharm: Antibacterial (gram-positive methicillinresistant Staphylococcus aureus ATCC33591, MIC = 128g/mL, control
C22H36O6 (396.53). Colorless oil, []D23 = +53.0 (c = 0.940, MeOH). Pharm:

Antifungal (Cladosporium cucumerinum, 20g, IZA = 23mm2, 40g, IZA =
40mm2). Source: Hygrophorus persoonii. Ref: 3800.
Gentamicin, MIC = 2g/mL). Source: AI SHENG XIONG GUO

O
Arctostaphylos pumila (stem). Ref: 5060.

O
O
OH
O
O
5337 4,5-Di-O-acetyl hygrophorone A14

4,5-trans-4-Acetoxy-5-hydroxy-5-(1-acetoxypentadecyl)-2-cyclopenten-1-one
O
O
C24H40O6 (424.58). Colorless oil. Pharm: Antifungal (Cladosporium
cucumerinum, 20g, IZA = 2mm2, 40g, IZA = 6mm2). Source: Hygrophorus

persoonii. Ref: 3800.
O
5333 2,6-Diacetyl-3,4-dimethylbutyryl-1-O-octylglucopyranoside
C28H48O10 (544.69). Pharm: Antibacterial (gram-positive
methicillin-resistant Staphylococcus aureus ATCC33591, MIC = 64g/mL;
O
OH
O
control Gentamicin, MIC = 2g/mL). Source: AI SHENG XIONG GUO

O
Arctostaphylos pumila (stem). Ref: 5060.
5338 4,6-Di-O-acetyl hygrophorone B14
4,5-cis-4-Acetoxy-5-hydroxy-5-(1-acetoxypentadecyl)-2-cyclopenten-1-one
O
O
C24H40O6 (424.58). Colorless oil. Source: Hygrophorus olivaceoalbus. Ref:
3800.
O
O
O
O
O
O
O
OH
O
5334 12,15-Diacetyl-13(21)-epoxyeurycomanone
C24H28O12 (508.48). Source: Eurycoma sp. Ref: 4556.
5339 1,4-Di-O-acetyl hygrophorone E10

1-(2,5-Diacetoxy-1-hydroxy-cyclopent-3-enyl)-undecan-1-one C20H32O6
O
HO
OH
(368.47). Colorless oil. Source: Hygrophorus latitabundus. Ref: 3800.
O
OH
O
O
O
O
OH
O
O
84
5344 1S,13-Diacetyloxy-4S-hydroxy-6R-(3-)furancarbonyloxy-9S-cinna-
1-(2,5-Diacetoxy-1-hydroxy-cyclopent-3-enyl)-tridecan-1-one C22H36O6
moyloxy--dihydroagarofuran
(396.53). Colorless oil, []D23 = +80.3 (c = 0.395, MeOH). Source:
C33H38O11 (610.66). Yellow oil, []D = +87.5 (c = 4.20, CHCl3). Pharm:
Hygrophorus latitabundus. Ref: 3800.
Cytotoxic inactive (hmn Bel7402, HL-60, A549 and mouse P388, all IC50 >
100mol/L). Source: Euonymus nanoides (seed: yield = 0.0035%dw). Ref:
1129.
O
OH

O
OH O
1-(2,5-Diacetoxy-1-hydroxy-cyclopent-3-enyl)-pentadecan-1-one C24H40O6
(424.58). Colorless oil. Source: Hygrophorus latitabundus. Ref: 3800.
O
OH
5345 4',6''-Diacetyl puerarin
C25H26O11 (502.48). Source: GE GEN Pueraria lobata [Syn. Pueraria

thunbergiana; Pueraria pseudohirsuta]. Ref: 2.
5342 Diacetyl montanin D

2
C24H30O8 (446.50). Pharm: Insect antifeedant (Spodoptera litura, 10g/cm ,

antifeedant activity = (672)%, control Azadirachtin A, 0.5g/cm2,
antifeedant activity = (792)%; Plutella xylostella, 10g/cm2, antifeedant
O
O
activity = (622)%, control Azadirachtin A, 0.5g/cm 2, antifeedant activity
OH
OH
OH
5346 3",6"-O,O-diacetylsaikosaponin b2
C46H72O15 (865.08). Source: WEN CHUAN CHAI HU Bupleurum
wenchuanense. Ref: 2247.
O
O
= (712)%). Source: RONG MAO XIANG KE KE Teucrium tomentosum
OH
H
O
OH
O
O
5343 2'',6''-O-Diacetyloninin
Yellow amorphous powder, []D25 = + 9.3 (c = 0.55, MeOH). Pharm:
DA DOU Glycine max (Soybean phytochemical concentrate: yield =

0.0039%dw). Ref: 4630.
HO
OH
OH
C22H20O9 (428.40). Pharm: Platelet aggregation inhibitor. Source: QUAN

YUAN YE HUA JIAO Zanthoxylum integrifoliolum. Ref: 2176.
O
O
OO
HO
OH
5347 3,5-Diacetyltambulin
O
O
O
O
O
OH
O O
OH
Cytotoxic (in vitro, Hs740T, ED50 = 7.61g/mL; Hs756T, ED50 =

DU145, ED50 = 4.18g/mL; LNCaP-FGC, ED50 = 22.12g/mL). Source:
OO
Formononetin-7-O-(2'',6''-O-diacetyl)glucopyranoside C26H26O11 (514.49).
8.89g/mL; Hs578T, ED50 = 5.44g/mL; Hs742T, ED50 = 25.53g/mL;
H
HO
85
5348 7,9-Diacetyltaxayuntin
5353 Diandraflavone
10-Benzoyloxy-2,4-diacetoxy-5,20-epoxy-1,7,9,13-tetrahydrox-11(
C29H34O11 (558.59). Pharm: Antioxidant (selectively inhibits superoxide anion
151)-abeo-taxene C31H40O11 (588.66). mp 242~243C; 266~268C. Source:
generation, hmn neutrophils, stimulated by fMLP/CB, IC50 = 10g/mL).
DUAN YE HONG DOU SHAN Taxus brevifolia, YUN NAN HONG DOU
Source: ER RUI HE LIAN DOU Drymaria diandra [Syn. Drymaria cordata
SHAN Taxus yunnanensis. Ref: 662.
ssp. diandra] (whole herb: yield = 0.00003%). Ref: 4758.
O
OH
OH
HO
HO
HO
HO
HO
HO
OH
O
HO
OH
O
O
5354 (3S)-3-O-(3',4'-Diangeloyl--D-glucopyranosyloxy)-6-hydroperoxy-3,7-dimethylocta-1,7-diene
C26H40O10 (512.60). Colorless oil. []D20 = 5.1 (c = 0.15, CHCl3). Source:
5349 Diallyl tetrasulfide
DONG FENG CAI Doellingeria scaber [Syn. Aster scaber] (aerial parts). Ref:
[2444-49-7] C6H10S4 (210.40). Source: DA SUAN Allium sativum. Ref: 2.
4102.
HO
S S
S S
OO
O
OH
5350 2,3-Diaminobutyric acid

C4H10N2O2 (118.14). Source: DUO HUA HUANG JING Polygonatum
cyrtonema [Syn. Polygonatum multiflorum], MO GU Agaricus campestris.
Ref: 6, 660.
OH
5355 (3S)-3-O-(3',4'-Diangeloyl--D-glucopyranosyloxy)-7-hydroperoxy-3,7-dimethylocta-1,5-diene
C26H40O10 (512.60). Colorless oil. []D20 = 13.1 (c = 0.48, CHCl3). Source:
DONG FENG CAI Doellingeria scaber [Syn. Aster scaber] (aerial parts). Ref:
4102.
O
OH
H2N
HO
NH2
OO
OH
OH
O
5351 L-,-Diaminobutyric acid
OH
2,4-Diaminobutyric acid C4H10N2O2 (118.14). mp 205C (dec). Pharm:

Causes chronic ammonia toxicosis (liver damage, tingle and tic, blocks
5356 3,6-Diangeloyloxy-10-hydroxy-8-methoxyeremophilenolide
displace of carbamoyl of ornithine). Source: DUO HUA HUANG JING
C26H36O8 (476.57). Colorless gum, []D20 = 109.8 (c = 0.56, CHCl3). Source:
Polygonatum cyrtonema [Syn. Polygonatum multiflorum], LIN SHENG
TU ER FENG XIE JIA CAO Cacalia ainsliaeflora. Ref: 5428.
SHAN LI DOU Lathyrus sylvestris, MO GU Agaricus campestris, SU GEN

OH
XIANG WAN DOU Lathyrus latifolius, Acacia sp. Ref: 6, 658, 660.
O
O
NH2
O
O
OH
H2N
5357 Diangoutengjian I
5352 ,-Diaminopropionic acid
C3H8N2O2 (104.11). mp () 193C, () 110~120C. Source: WANG GUA ZI
C22H28N2O4 (384.48). Colorless block crystals, mp 190~191C. Source: DIAN

GOU TENG Uncaria yunnanensis. Ref: 869.
Trichosanthes cucumeroides. Ref: 6.

O
H2N
OH
NH2
N
H H
O
O
N
H
H
OH
86
5358 Dianoside A
5362 Dianoside E
[91652-87-8] C42H66O15 (810.99). Pharm: Analgesic. Source: CHANG E QU MAI
[91652-23-2] C42H66O16 (826.98). Source: BIAN SE SHI ZHU Dianthus
Dianthus superbus var. longicalycinus, BIAN SE SHI ZHU Dianthus versicolor,
versicolor. Ref: 1530, 1531, 1532, 1533.
QU MAI Dianthus superbus. Ref: 658, 1530, 1531, 1532, 1533, 4450, 5501.
OH
H
H
HO
OO
OH
OH
HO
HO
H
O
HO
OH
H
OH
OH
OH
OH
OH
OO
OO
OH
OH
OO
OH
OH
OH
OH
5359 Dianoside B
C54H86O25 (1135.27). Pharm: Antihepatotoxin (aglucon is active component,
5363 Dianoside F
liver damage caused by CCl4); analgesic (mus, acetic acid-induced writhing
model, InRt = 68%). Source: BIAN SE SHI ZHU Dianthus versicolor, QU
versicolor. Ref: 1530, 1531, 1532, 1533.
MAI Dianthus superbus. Ref: 1530, 1531, 1532, 1533, 5501.

OH
H
HO
OO
OH
OH
HO
OH
OH
H
HO
OO
OH
OH
O OH
HO
OH
OH
OH
OH
OH
5364 Dianoside G
OH
OH
OO
HO
OH
[96333-09-4] C48H76O20 (973.13). Source: CHANG E QU MAI Dianthus

superbus var. longicalycinus, BIAN SE SHI ZHU Dianthus versicolor. Ref:
OH
1530, 1531, 1532, 1533, 4450.

5360 Dianoside C
versicolor. Ref: 1530, 1531, 1532, 1533.
OH
OO
HO
OH
OH
HO
H
OH
H
OH
OO
OH
OO OH
OH
OH
OH
OH
OH
HO
OH
5361 Dianoside D
versicolor. Ref: 1530, 1531, 1532, 1533.
5365 Dianoside H
versicolor. Ref: 1530, 1531, 1532, 1533.
OH
O
H
HO
H
HO
O
H
OH
O O
OH
OH
O O OH
OH
OH
OH
OH
O
H
HO
OH
OH
OH
OH
OH
HO
O O
HO
H
H
H
O
OH
HO
OO
OH
OH
OH
87
5366 Dianthalexine
[85914-62-4] C14H9NO3 (239.23). Pharm: Antifungal. Source: SHE XIANG
OH HN
SHI ZHU Dianthus caryophyllus. Ref: 658, 1521.
O
HN
O
HO
O
O
NH
N
H
NH
5370 Dianthin F
C30H37N5O5 (547.66). Pale yellow powder, []D21 = 16.0 (c = 0.03, MeOH).
5367 Dianthin C
C36H48N6O7 (676.82). Pale yellow powder, []D21 = 50 (c = 0.17, MeOH).
Pharm: Cytotoxic (in vitro, HepG2, IC50 = 17.17g/mL; Hep3B, IC50 >
Source: QU MAI Dianthus superbus (aerial parts: yield = 0.0005%dw). Ref:

4765.
20g/mL; MCF7, IC50 > 20g/mL; A549, IC50 > 20g/mL; MDA-MB-231,
H
N
IC50 > 20g/mL; control Doxorubicin, HepG2, IC50 = 0.19g/mL; Hep3B,
IC50 = 0.31g/mL; MCF7, IC50 = 1.21g/mL; A549, IC50 = 0.19g/mL;
MDA-MB-231, IC50 = 0.73g/mL). Source: QU MAI Dianthus superbus
(aerial parts: yield = 0.0033%dw). Ref: 4765.
O
HN
O
O
OH
NH
5371 Dianthoside
Maltol-3-O--D-glucopyranoside [20847-13-6] C12H16O8 (288.26). Source:

NH
NH
NH
N
H
H
N
HN
O
O
SHI ZHU Dianthus chinensis, JIN JI WEI BA CAO GEN Macrothelypteris

oligophlebia, REN SHEN Panax ginseng [Syn. Panax schinseng]. Ref: 1238,
1488, 1529.
5368 Dianthin D
C36H53N7O8 (711.87). Pale yellow powder, []D21 = 19.6 (c = 0.10, MeOH).

Pharm: Cytotoxic (in vitro, HepG2, IC50 > 20g/mL; Hep3B, IC50 > 20g/mL;
HO
OO
OH
MCF7, IC50 > 20g/mL; A549, IC50 > 20g/mL; MDA-MB-231, IC50 >
OH
20g/mL; control Doxorubicin, HepG2, IC50 = 0.19g/mL; Hep3B, IC50 =
OH
0.31g/mL; MCF7, IC50 = 1.21g/mL; A549, IC50 = 0.19g/mL;

5372 Dianthramine
[136945-65-8] C14H11NO6 (289.25). Pharm: Antifungal. Source: SHE XIANG
SHI ZHU Dianthus caryophyllus. Ref: 522, 658.
N
HN
O
O
HN
N
O
OH
OH
O
HN
O
NH
N
H
N
H
O
OH
OH
OH
5373 Diarylheptanoid CPB-51-262-1

C20H22O5 (342.40). Brown solid, []D25 = 81.13 (c = 0.03, MeOH). Pharm:
Cytotoxic inactive (MTT assay, HT29 cell line, MCF7 cell line). Source: HU
5369 Dianthin E
21
C30H44N6O7 (600.72). Pale yellow powder, []D = 30.5 (c = 0.02, MeOH).

Pharm: Cytotoxic (in vitro, HepG2, IC50 = 2.37g/mL; Hep3B, IC50 >
TAO QIU Juglans mandshurica (root). Ref: 4321.

H
20g/mL; MCF7, IC50 > 20g/mL; A549, IC50 > 20g/mL; MDA-MB-231,
IC50 > 20g/mL; control Doxorubicin, HepG2, IC50 = 0.19g/mL; Hep3B,

IC50 = 0.31g/mL; MCF7, IC50 = 1.21g/mL; A549, IC50 = 0.19g/mL;
OH
O
OH
88
5379 1,1'-Dibenzene-6',8',9'-trihydroxy-3-allyl-4-O--D-glucopyra-
C20H24O4 (328.41). Yellow oil, []D25 = 39.07 (c = 0.21, MeOH). Pharm:
noside
Cytotoxic inactive (MTT assay, HT29 cell line, MCF7 cell line). Source: HU
C24H30O9 (462.50). Colorless glue. Source: DA YE HOU PO Magnolia
TAO QIU Juglans mandshurica (root). Ref: 4321.
rostrata. Ref: 2030.
OH
OH
OH
O
O
OH

C21H26O5 (358.44). Brown oil, []D21 = 7.1 (c = 0.42, MeOH). Pharm:
OH
HO
Cytotoxic (MTT assay, HT29 cell line, IC50 = 41.3g/mL; MCF7 cell line,
IC50 = 50g/mL)[4321]. Source: HU TAO QIU Juglans mandshurica (root). Ref:
OH
OH
4321.
O
OH
5380 Dibenzofuran
C12H8O (168.20). Source: CHUAN XU DUAN Dipsacus asperoides. Ref:

OH
HO
660.
5376 ()-Diasesamin-di--lactone
C20H14O8 (382.33). Colorless needles (Me2CO), mp 188~189C, []D26 =
47.4 (c = 0.1, CHCl3). Source: PI ZHEN XING YAO HUA Wikstroemia
lanceolata (stem and root). Ref: 4947.
O
O
O
H
O
5381 6-O--L-(2''-O-,3''-O-Dibenzoyl,4''-O-cis-p-coumaroyl)rhamno-
H
O
pyranosylcatalpol
C44H46O18 (862.85). Source: FEI LV BIN SHI ZI Gmelina philippensis (aerial

parts). Ref: 3954.
5377 Diatoxanthin
C40H54O2 (566.88). Pharm: Anti-carcinogenic (inhibits 50nmol/L
12-O-tetradecanoyl phorbol 13-acetate (TPA)-stimulated 32P-incorporation

into the phospholipids of HeLa cells, 25g/mL, InRt = 48.2%)[4256]. Source:
HO
OO
ER JIAO DUO JIA ZAO Peridinium bipes. Ref: 4256.

OH
O O
OH
O
OH
OH
O
O
H
OH
OH
5382 6-O--L-(2''-O-,3''-O-Dibenzoyl,4''-O-trans-p-coumaroyl)rhamnopyranosylcatalpol
OH
5378 Diayangambin
Lirioresinol dimethyl ether [21453-68-9] C24H30O8 (446.50). Pharm:
parts). Ref: 3954.
Cytotoxic (Meth-A sarcoma cell line, ED50 > 10g/mL, LLC cell line, ED50 >
10g/mL)[3510]. Source: QING HAO Artemisia apiacea [Syn. Artemisia
O
O
carvifolia; Artemisia caruifolia] (aerial parts). Ref: 3510.

HO
O
O
O
H
H
O
O
O
OO
H
O
O O
O
O
H
OH
OH
O
OH
OH
OH
89
5383 2,7-Dibenzoyl-5,20-epoxy-1-hydroxy-4,9,10,13-tetra-
5387 5,3'-Dibenzoyloxy-3,6,7,4'-tetramethoxyflavone
acetoxytax-11-ene
C33H26O10 (582.57). mp 220~222C. Pharm: Cytotoxic (in vitro, Col2, ED50 >
C42H48O14 (776.84). Source: DUAN YE HONG DOU SHAN Taxus brevifolia.
20g/mL; hTERT-RPE1, ED50 = 4.3g/mL; HUVEC, ED50 > 20g/mL; KB,
Ref: 662.
ED50 > 20g/mL; HUVEC, ED50 > 20g/mL; Lu1, ED50 = 6.5g/mL). Source:
HUANG JING YE Vitex negundo. Ref: 4699.
O
O
O
O
O
O
HO
O
O
5388 6-O--L-(2''-O-,3''-O-Dibenzoyl)rhamnopyranosylcatalpol
5384 Dibenzoylgagaimol
[38753-71-8] C35H42O9 (606.72). mp 192~197C. Source: LUO MO
Metaplexis japonica. Ref: 6.

parts). Ref: 3954.
OH
O
O
OH
O
OH
O
O
O O
OH
O
OH
OH
O
H
OH
OH
OH
HO
OH
5385 3,7-Dibenzoyloxy-6-hydroxy-tropane
C22H23NO5 (381.43). mp 220C, []D25 = +10 (c = 0.1, EtOH). Source:
Erythroxylon alaternifolium (leaf). Ref: 3999.
C35H40O16 (716.70). Pale yellow powder. Source: FEI LV BIN SHI ZI

Gmelina philippensis (aerial parts). Ref: 3954.
O
HO
O
O
OO
OH O
H
O
O
O
H
OH
OH
O
OH
OH
OH
5386 3,29-O-Dibenzoyloxykarounidiol
C43H54O4 (634.91). Colorless needles, mp 149~152C (n-hexane), []D = +9.1
(c = 0.17, CHCl3). Source: FENG GUA Gymnopetalum integrifolium (fruit).
Ref: 4189.
C35H40O16 (716.70). Pale yellow powder. Source: FEI LV BIN SHI ZI
Gmelina philippensis (aerial parts). Ref: 3954.
O
H
O
O
OO
O
O OH
H
O
H
OH
OH
O
OH
OH
OH
90
5391 Dibenzyl disulphide
5395 Di(benzyltrithio)methane
C14H14S2 (246.40). Yellow amorphous solid. Pharm: Antifungal (plant
C15H16S6 (388.68). Orange amorphous solid. Pharm: Antifungal (plant
pathogenic fungi Cladosporium sphaerospermum, MIC = 0.1g, control
Nystatin, MIC = 1.0g; Cladosporium cladosporioides, MIC = 1.0g,
Nystatin, MIC = 1.0g; Cladosporium cladosporioides, MIC = 5.0g,
Nystatin, MIC = 1.0g); antineoplastic (mechanism-based yeast bioassay for
Nystatin, MIC = 1.0g); antineoplastic (mechanism-based yeast bioassay for
DNA-modifying agents, mutant yeast Saccharomyces cerevisiae: RS 188N
(rad+), IC12 = 332g/mL; RS 321, IC12 = 66g/mL; RS 52YK (rad 52Y), IC12
= 16g/mL, control Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL).
= 67g/mL, control Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL).
Source: SUAN CHOU MU JI CAO Petiveria alliacea (root, stem and leaf).
Source: SUAN CHOU MU JI CAO Petiveria alliacea (root, stem and leaf).
Ref: 5159.
Ref: 5159.
5392 Dibenzyl sulphide

C14H14S (214.33). Yellow oil. Pharm: Antifungal (plant pathogenic fungi
5396 Dibothrioclinin I
Cladosporium sphaerospermum, MIC = 1.0g, control Nystatin, MIC = 1.0g;
C30H28O6 (484.55). Colorless block crystals, mp > 300C, []D19 = +24 (c =
Cladosporium cladosporioides, MIC = 1.0g, Nystatin, MIC = 1.0g);
0.05, CHCl3). Source: MAO DA DING CAO Gerbera piloselloides. Ref:
antineoplastic (mechanism-based yeast bioassay for DNA-modifying agents,
2564.
mutant yeast Saccharomyces cerevisiae: RS 188N (rad+), IC12 = 402g/mL;
RS 321, IC12 = 381g/mL; RS 52YK (rad 52Y), IC12 = 412g/mL, control
Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL). Source: SUAN CHOU
MU JI CAO Petiveria alliacea (root, stem and leaf). Ref: 5159.

H
O
5397 Dibothrioclinin II
C30H28O6 (484.55). Colorless plate crystals, mp > 300C, []D19 = 0 (c =
5393 Dibenzyl tetrasulphide
0.045, CHCl3). Source: MAO DA DING CAO Gerbera piloselloides. Ref:
C14H14S4 (310.52). Orange amorphous solid. Pharm: Antifungal (plant
2564.
Nystatin, MIC = 1.0g; Cladosporium cladosporioides, MIC = 10.0g, Nystatin,
MIC = 1.0g); antineoplastic (mechanism-based yeast bioassay for

(rad+), IC12 = 328g/mL; RS 321, IC12 = 53g/mL; RS 52YK (rad 52Y), IC12 =
H
O
104g/mL, control Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL).

Source: SUAN CHOU MU JI CAO Petiveria alliacea (root, stem and leaf). Ref:
5159.
5398 Di-p-bromobenzoate of tetrahydrodeoxyoxolucidine B

C44H59Br2N3O4 (853.79). []D21.5 = 30.5 (c = 0.89, CHCl3). Source:
GUANG LIANG SHI SONG Lycopodium lucidulum. Ref: 3927.
Br
5394 Dibenzyl trisulphide

C14H14S3 (278.46). Yellow amorphous solid. Pharm: Antifungal (plant
pathogenicfungi Cladosporium sphaerospermum, MIC = 1.0g, control Nystatin,
MIC = 1.0g; Cladosporium cladosporioides, MIC = 1.0g, Nystatin, MIC =

H
1.0g); antineoplastic (mechanism-based yeast bioassay for DNA-modifying

H
H
N
H O
H
O
control Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL). Source: SUAN

CHOU MU JI CAO Petiveria alliacea (root, stem and leaf). Ref: 5159.
S
H
N
agents, mutant yeast Saccharomyces cerevisiae: RS 188N (rad+), IC12 =

73g/mL; RS 321, IC12 = 64g/mL; RS 52YK (rad 52Y), IC12 = 62g/mL,
Br
91
5399 (E)-10,15-Dibromo-9-hydroxy-chamigra-1,3(15),7(14)-triene
5405 Dibutyl uralsaponin A ester
C15H20Br2O (376.13). Source: LUE DA AO DING ZAO Laurencia majuscula.
Inflasaponin IV; Glycyrrhetic acid-3-O--D-6''-n-butyl-glucuronopyranosyl-
Ref: 5191.
(12)--D-6'-n-butyl-glucuronopyranoside C50H78O16 (935.17). Colorless

powder, mp 234~236C. Source: GAN CAO Glycyrrhiza uralensis, ZHANG
GUO GAN CAO Glycyrrhiza inflata. Ref: 301, 880.
HO
O
Br
OH
Br
5400 (Z)-10,15-Dibromo-9-hydroxychamigra-1,3(15),7(14)-triene
C15H20Br2O (376.13). Source: LUE DA AO DING ZAO Laurencia majuscula.
OO
Ref: 5191.
OH
O
HO
OH
O
O
OH
Br
Br
OH
OH
5406 1,3-Di-O-(E)-caffeoyl-4-O-galloyl--D-glucopyranose
5401 5,3'-Dibutanoyloxy-3,6,7,4'-tetramethoxyflavone
11.7g/mL; hTERT-RPE1, ED50 = 0.6g/mL; HUVEC, ED50 > 20g/mL; KB,
[4699]
ED50 = 0.5g/mL; HUVEC, ED50 = 0.8g/mL; Lu1, ED50 = 1.7g/mL)
C31H28O16 (656.56). Yellow amorphous powder, []D15 = 100.4 (c = 0.7,

MeOH). Source: GE XUN Balanophora japonica (aerial parts: yield =
0.1069%, underground part: yield = 0.0859%). Ref: 4101.
O
O
O
O
O
HO
OO
O
HO
OH
OH
OH
OH HO
HO
OH
5407 1,2-Di-O-(E)-caffeoyl--D-glucopyranose
5402 2,6-Dibutyl-p-cresol
C14H22O2 (222.33). Source: MIAN MA Dryopteris filix-mas. Ref: 1534.
MeOH). Source: GE XUN Balanophora japonica (underground part: yield =

0.0287%). Ref: 4101.
OH
OH
OH
OO
HO
OH
OH
OH
OO
O
5403 Dibutyl oxalate
OH
[2050-60-4] C10H18O4 (202.25). Source: REN SHEN Panax ginseng [Syn.

Panax schinseng]. Ref: 2.
O
O
OH
5408 1,3-Di-O-(E)-caffeoyl--D-glucopyranose
O
O
5404 Dibutyl phthalate

0.0014%). Ref: 4101.
OH
OH
[84-74-2] C16H22O4 (278.35). Source: NIU XI Achyranthes bidentata, HUA

DONG LAN CI TOU Echinops grijsii. Ref: 582, 660.
OH
OO
O
O
O
OH
OH
O
O
OH
O
OH
92
5409 3,6-Di-O-caffeoyl-(/)-glucose
5413 1,4-Di-O-caffeoylquinic acid
C24H24O12 (504.45). Source: SHEN SHENG XUAN GOU ZI Rubus sanctus.
C25H24O12 (516.46). mp 229~230C. Source: CANG ER Xanthium sibiricum
Ref: 3421.
[Syn. Xanthium strumarium]. Ref: 6.

O
HO
OH
O
O
HO
OH
HO
OH
OH
OH
OH
OH
O
HO
HO
OH
HO
5414 3,4-Di-O-caffeoylquinic acid

5410 1,3-Di-O-(E)-caffeoyl-4,6-(S)-HHDP--D-glucopyranose
Isochlorogenic acid B [14534-61-3] C25H24O12 (516.46). Pharm: Platelet
aggregation inhibitor (rat, 500g/mL, induced by ADP, InRt = 75%, induced
by collagen, InRt = 42%); promotes release of prostacyclin PGI2 (rat,
0.0092%). Ref: 4101.
10mol/L, 190.6%); increases coronary flow; Increases spread and mobility

of macrophage (mus); anti-HIV (HIV-1 integradase inhibitor, inhibits
OH
replication of HIV); anrtineoplastic (mus, melanotic carcinoma B16, inhibits
OH
HO
OO
HO
HO
inhibits lipid peroxidization). Source: CU ZHUANG KA FEI Coffea robusta,
OH
O
SAI ER WEI YA SHI CAO Achillea alexandri-regis, XIAO GUO KA FEI

O
OH
HO
formation of melanin); antioxidant (cytoblast and microsome in hepatic cells,
Coffea arabica, ZHI ZI Gardenia jasminoides [Syn. Gardenia florida],
Artemisia sp. Ref: 2, 626, 658, 1034, 1573, 1574, 1575, 1576, 2545.
OH
HO
OH
HO
OH
OH
HO
O
5411 3,4-Di-O-caffeoyl-5-O-(3-hydroxy-3-methyl) glutaroyl quinic acid

C31H32O16 (660.59). Source: ZHI ZI Gardenia jasminoides [Syn. Gardenia
florida]. Ref: 2, 626.
OH
5415 3,4-Di-O-caffeoylquinic acid methyl ester
O
HO
O
HO
C26H26O12 (530.49). Pharm: Antiallergic (hyaluronidase inhibitor (activated

OH
O
O
O
OH
OH
OH
hyaluronidase by compound 48/80, 0.2mmol/L, InRt = 31%, 76% inhibition

of control DSCG)[3924]. Source: QUAN YUAN YE TE SA JU Tessaria
integriforia (aerial parts), XIAO LONG YE KUO BAO JU Baccharis
dracunculifolia (aerial parts). Ref: 3924, 4184.

OH
OH
OH
OH
HO
OH
HO
OH
HO
5412 3,5-Di-O-caffeoyl-4-O-(3-hydroxy-3-methyl)glutaroylquinic acid

O
O
O
HO
5416 Dicapryl phthalate

O
HO
[117-84-0] C24H38O4 (390.57). Source: SAN QI Panax pseudo-ginseng var.

notoginseng [Syn. Panax notoginseng]. Ref: 2.
OH
O
O
O
HO
OH
O
OH HO
O
OH
OH
93
5417 ()-Dicentrine
5422 Dichotomine A
[517-66-8] C20H21NO4 (339.39). Pharm: Analgesic; sedative; antitrypa-
C14H12N2O3 (256.26). Yellow powder, []D27 = 9.7 (c = 0.85, MeOH).
nosomal and cytotoxic (Trypanosoma brucei brucei , IC50 = 14.6mol/L,
Pharm: -Hexosaminidase release inhibitor inactive (RBL-2H3 cells); TNF-
Suramin, IC50 = 0.06mol/L; hmn cervixcarcinoma cell HeLa, IC50 =
release inhibitor inactive (RBL-2H3 cells, antigen-IgE-mediated); IL-4 release
35mol/L)
[4969]
. Source: HE BAO DI BU RONG Stephania dicentrinifera,
WU YE TENG Cassytha filiformis, XI XIAO HE BAO MU DAN Dicentra
inhibitor inactive (RBL-2H3 cells, antigen-IgE-mediated). Source: YIN CHAI

HU Stellaria dichotoma var. lanceolata (root: yield = 0.0014%dw). Ref: 4761.
pusilla. Ref: 658, 4969.

OH
H
N
N
OH
O
O
O
5418 2,4-Dichloro-6-aminopyridine
5423 Dichotomine B
C5H4Cl2N2 (163.01). mp 271C. Source: KU SHU PI Picrasma quassioides
[Syn. Picrasma ailanthoides]. Ref: 6.
Pharm: -Hexosaminidase release inhibitor inactive (RBL-2H3 cells); TNF-

release inhibitor inactive (RBL-2H3 cells, antigen-IgE-mediated); IL-4 release
Cl

H2N
Cl
5419 2',2'-N,N-Dichloromethyltetrandrine
C40H46Cl2N2O62+ (721.73). Source: FANG JI Stephania tetrandra. Ref: 2.
OH
N
OH
HO
H
N
O
H
N
5424 Dichotomine C
Cl
Cl
Pharm: -Hexosaminidase release inhibitor (RBL-2H3 cells, IC50 =

O
62mol/L); TNF- release inhibitor (RBL-2H3 cells, antigen-IgE-mediated,
IC50 = 19mol/L); IL-4 release inhibitor (RBL-2H3 cells,
5420 Dichotomide I
antigen-IgE-mediated, IC50 = 15mol/L). Source: YIN CHAI HU Stellaria
C18H17N3O4 (339.35). Yellow powder. Pharm: -Hexosaminidase release
dichotoma var. lanceolata (root: yield = 0.0016%dw). Ref: 4761.
inhibitor inactive (RBL-2H3 cells); TNF- release inhibitor inactive

(RBL-2H3 cells, antigen-IgE-mediated); IL-4 release inhibitor inactive
(RBL-2H3 cells, antigen-IgE-mediated). Source: YIN CHAI HU Stellaria
HO
H
N
dichotoma var. lanceolata (root). Ref: 4761.
OH
N
O
O
H
N
O
N
H
N
5425 Dichotomine D
O
C18H20N2O4 (328.37). Yellow powder, []D27 = 1.8 (c = 0.75, CHCl3). Pharm:
5421 Dichotomide II
-Hexosaminidase release inhibitor inactive (RBL-2H3 cells); TNF- release
C18H15N3O4 (337.34). Yellow powder, []D19 = +7.2 (c = 0.30, CHCl3). Pharm:
inhibitor inactive (RBL-2H3 cells, antigen-IgE-mediated); IL-4 release
-Hexosaminidase release inhibitor inactive (RBL-2H3 cells); TNF- release
inhibitor inactive (RBL-2H3 cells, antigen-IgE-mediated); IL-4 release

H
N
HO
H
N
O
O
H
N
O
OH
N
O
O
94
5426 Dichotomitin
5430 Dichotomoside D
3',4'-Dimethoxy-5',5-dihydroxy-6,7-methylenedioxyisoflavone C18H14O8
C34H48O13 (664.75). White powder, []D27 = +7.4 (c = 0.30, MeOH). Pharm:
(358.31). Yellowish rhomboid crystals, mp 249~251C. Source: BAI HUA
-Hexosaminidase inhibitor (RBL-2H3 cells, IC50 = 64mol/L, control
SHE GAN Iris dichotoma, JUAN QIAO YUAN WEI Iris potaninii
Ketotifen fumarate IC50 = 216mol/L); tumor necrosis factor- inhibitor
(underground part). Ref: 69, 4235.
(TNF-) (RBL-2H3 cells, IC50 = 16mol/L); interleukin-4 inhibitor

(RBL-2H3 cells, IC50 = 34mol/L); antiallergic (effective against the
late-phase reactions in type I allergy than in the immediate phase). Source:
O
OH
YIN CHAI HU Stellaria dichotoma var. lanceolata (root: yield = 0.0002%).
Ref: 2571.
O
OH
OH
O
5427 Dichotomoside A
-Hexosaminidase inhibitor inactive (RBL-2H3 cells, 100mol/L, InRt =
OH
C26H32O13 (552.54). White powder, []D27 = 2.3 (c = 0.30, MeOH). Pharm:
OH
HO
OH
(1.00.7)%, control Ketotifen fumarate, InRt = (19.11.3)%). Source: YIN

CHAI HU Stellaria dichotoma var. lanceolata (root: yield = 0.0013%). Ref:
2571.
OH
O
O
OH
O
OH
HO
5431 Dichotomoside E
OH

2571.
HO
OH
OH
O
5428 Dichotomoside B
OH
O
HO
OH

2571.
OH
O
O
OH
O
OH
HO
5432 Dichroanal A
rel-(4aS,9R,9aS)-8-formyl-1,2,3,4,4a,9a-hexahydro-5,6,9-trihydroxy-7-isopro
OH
pyl-1,1,4a-trimethylfluorene C20H28O4 (332.44). Source: ER SE HUA SHU

WEI CAO Salvia dichroantha. Ref: 1909.
OH
HO
OH
5429 Dichotomoside C
C30H40O13 (608.65). White powder, []D27 = +5.5 (c = 0.20, MeOH). Source:
YIN CHAI HU Stellaria dichotoma var. lanceolata (root: yield = 0.0009%).
Ref: 2571.
OH
O
5433 Dichroanal B
OH
O
OH
O
OH
HO
4aS*-8-formyl-2,3,4,4a-tetrahydro-5,6-dihydroxy-7-isopropyl-1,1,4a-trimethy
l-1H-fluorene C20H26O3 (314.43). Source: ER SE HUA SHU WEI CAO
Salvia dichroantha. Ref: 1909.
OH
OH
OH
OH
95
5434 Dichroanone
5439 Dicliripariside C
4aS*-2,3,4,4a-tetrahydro-6-hydroxy-7-isopropyl-1,1,4a-trimethyl-5,8(1H)-flu
C29H34O15 (622.59). Yellowish powder, mp 238~240C, []D10 = 1.3 (c =
orene-dione C19H24O3 (300.40). Source: ER SE HUA SHU WEI CAO Salvia
0.016, MeOH:pyridine = 1:1). Source: HE AN GOU GAN CAI Dicliptera
dichroantha. Ref: 1909.
riparia. Ref: 1945.
OH
OH
O
OH
OO
OO
OH
OH
OH
OH OH
5435 -Dichroine
Isofebrifugine C16H19N3O3 (301.35). mp 129~130C. Pharm: Antimalarial;
inhibits heart (rbt, iv, in vitro); antihypertensive (anesthetic cat, iv); uterine
5440 Dicoumarin
stimulant (anesthetic dog in vivo, pregnant rbt in vitro, rat in vitro). Source:
Dicoumarol [66-76-2] C19H12O6 (336.30). mp 288~289C. Pharm:
CHANG SHAN Dichroa febrifuga, SAN XING XIU QIU Hydrangea
Antineoplastic (inhibits cellular proliferation of EAC, ID50 of synthesis of
umbellata. Ref: 4, 6, 658.
nucleic acid = 11.5g/mL); platelet aggregation inhibitor; rodenticide;

antithrombotic (intravenous thrombus, pulmonary embolism, heart infarction
H H
N
and infarction caused by atrial fibrillation); toxin (bleeding). Source: BAI

XIANG CAO MU XI Melilotus albus, HONG CHE ZHOU CAO Trifolium
N
O
HO
pratense, MU XU Medicago sativa, PI HAN CAO Melilotus suaveolens,
Anthoxanthum sp. Ref: 4, 5, 6, 658.

5436 -Dichroine
OH
Febrivugine [24159-07-7] C16H19N3O3 (301.35). mp 139~140C. Pharm:
OH
Antimalarial (amoeba); antipyretic; uterine stimulant (anesthetic dog in vivo,

pregnant rbt or rat, in vitro); emetic; LD50 (mus, orl) = 2.5~3.0mg/kg. Source:
O O
CHANG SHAN Dichroa febrifuga. Ref: 658.

5441 3,6-Di-O-p-coumaroyl--D-fructofuranosyl 6-O-acetyl--D-glucoO
OH
pyranoside
C32H36O16 (676.63). Light yellow amorphous solid, []D23 = +23.4 (c = 0.25,
N
HN
MeOH). Source: JIAO YU Canna edulis (rhizome). Ref: 3836.

OH
5437 Dicliripariside A
HO
C32H48O14 (656.73). Yellowish powder, mp 104~106, []D10 = +0.127 (c =

0.11, MeOH). Source: HE AN GOU GAN CAI Dicliptera riparia. Ref: 1945.
O
HO
HO
O
OH
OH
OH
O
O
O
O
O
O
O O O
OO
5442 2,3-Dicresol
HO
OH OH
[526-75-0] C8H10O (122.17). Source: DANG GUI Angelica sinensis. Ref: 2.
HO
OH OH
OH
5438 Dicliripariside B
C31H36O16 (664.62). Yellow powder, mp 210~212C, []D10 = 0.9 (c = 0.01,
MeOH:pyridine = 1:1). Source: HE AN GOU GAN CAI Dicliptera riparia.
5443 Dictafolin A
Ref: 1945.
C11H12O3 (192.22). Colorless oil, []D = +62.3 (c = 0.015, Me2CO), []D =

O
OH
O
+30.08 (c = 0.02, CHCl3). Source: XIA YE BAI XIAN Dictamnus

angustifolius. Ref: 1912.
O
OO
OO
OH
OH
OH
OH OH
O
O
96
5444 Dictafolin B
5448 Dictamnoside G
C8H10O4 (170.17). Yellowish oil. Source: XIA YE BAI XIAN Dictamnus
C27H46O14 (594.66). Source: BAI XIAN PI Dictamnus dasycarpus (root
angustifolius. Ref: 1912.
cortex). Ref: 3068.
OH
OH
O
O
H
OO
HO
5445 Dictamnine
C12H9NO2 (199.21). mp 132C. Pharm: Antibacterial; antifungal; contracts
O
OH
OH
OH
blood vessels (blood vessel of rbt ear, in vitro); uterine stimulant (rbt and gpg);
OH
O
OH
OH
OH
stimulates heart (frog heart in vitro, in low dose). Source: A NUO TI HUA
5449 Dictamnoside H
JIAO Zanthoxylum arnottianum, BAI XIAN PI Dictamnus dasycarpus (root
C21H36O8 (416.52). White amorphous powder, []D24 = 13.2 (c = 0.10
cortex: content = 0.12%)[5501], CHU YE HUA JIAO Zanthoxylum ailanthoides,
MeOH). Source: BAI XIAN PI Dictamnus dasycarpus (root cortex). Ref:
CHU YE HUA JIAO PI Zanthoxylum ailanthoides, DE KA RUI HUA JIAO
3068.
OH
Zanthoxylum decaryi, RI BEN BAI SONG FENG CAO Boenninghausenia

albiflora var. japonica, YAN JIAO CAO Boenninghausenia albiflora, ZHU
YE JIAO Zanthoxylum planispinum, ZHU YE JIAO GEN Zanthoxylum
planispinum. Ref: 6, 658, 5501.
HO
HO
HO
OH
O
OH
5450 Dictamnoside I
3068.
OH
5446 Dictamnoside A
C21H36O9 (432.52). Pharm: Immunoenhancer (in vitro, stimulates proliferation
of T-cells, 0.00001mol/L, P<0.001). Source: BAI XIAN PI Dictamnus
dasycarpus (root cortex). Ref: 3068.
HO
HO
HO
HO
OH
O
OH
OH
5451 Dictamnoside J
O
H
OH
HO

3068.
OH
OH
OH
OH
5447 Dictamnoside B
OH
O
HO
HO
HO
OH
C21H36O9 (432.52). Source: BAI XIAN PI Dictamnus dasycarpus (root

cortex). Ref: 3068.
OH
5452 Dictamnoside K
OH
OH

3068.
OH
OH
OH
HO
OH
OH
OH
HO
HO
HO
OH O
O
OH
OH
97
5453 Dictamnoside L
5458 Dictysine
Ref: 16.
3068.
OH
OH
OH
OH
H
HO
HO
HO
O O
5459 2,7-Dideacetyl-2,7-dibenzoyl-taxayunnanine F
OH
C40H46O13 (734.80). mp 203~205C. Source: DUAN YE HONG DOU SHAN
5454 Dictamnoside M
24
C27H48O14 (596.68). White amorphous powder, []D = 24.0 (c = 0.10
Taxus brevifolia. Ref: 662.

3068.
O
HO
OH
O
O
HO
HO
HO
HO
O
HO
OH
OH
HO
HO
O
O
OH
5455 Dictamnoside N
5460 7,13-Dideaceyl-9,10-debenzoyltaxchinin C
C29H38O10 (546.62). mp 162C, [] D = 15 (CHCl3). Source: DUAN YE
3068.

H
HO
H
HO
HO
HO
HO
OH
O O
OH OH
HO
OH
HO
O
O
5456 Dictangustine A
O
O
C12H9NO3 (215.21). Yellowish powders (Me2CO), mp > 280C. Source: XIA

YE BAI XIAN Dictamnus angustifolius. Ref: 1912.
5461 N,O-Dideacyl-N-methylpachysandrine A
O
C25H46N2O (390.66). mp 126~150C. Source: XUE SHAN LIN Pachysandra
HO
terminalis. Ref: 6.
N
5457 -Dictyopterol
C15H24O (220.36). Pharm: NO production inhibitor (mus peritoneal
macrophages, induced by LPS, 100mol/L, InRt = (51.53.5)%, control
L-NMMA, 100mol/L, InRt = (79.20.9)%, p<0.01). Source: PING E SHU
Curcuma zedoaria [Syn. Curcuma aeruginosa]. Ref: 4150.
OH
H
OH
5462 3,5-Didecanoylpyridine
C25H41NO2 (387.61). Source: YU XING CAO Houttuynia cordata. Ref: 2428.
O
H
N
98
5463 Didehydro-3'-hydroxyaglaiastatin
5468 5,6-Didehydropygmaeocin A
[259143-58-3] C31H28N2O7 (540.58). Pharm: Insecticidal (neonate larvae of
[122590-06-1] C20H20O6 (356.38). Yellow crystals (MeOH), mp 211~213C.
Spodoptera littoralis, LC50 = 5.70mg/L, EC50 = 0.31mg/L; control
Source: QIAN JIE CAO Pygmaeopremna herbacea [Syn. Premna herbacea].
Azadirachtin, LC50 = 0.9mg/L, EC50 = 0.04mg/L). Source: Aglaia duperreana.
Ref: 3119.
Ref: 2376.
O
OH N
OH
N
O
O
O
HO
O
5464 7,8-Didehydrocimigenol 3-O--D-xylopyranoside
5469 1,10-Didehydrosalviarin
C35H54O9 (618.82). Source: XING AN SHENG MA Cimicifuga dahurica
C20H20O5 (340.38). Crystals (n-hexaneCHCl 3), mp 186~188C, [] D25 =
200.2 (c = 1.0, CHCl3). Source: Salvia wagneriana (aerial parts). Ref: 4976.
O
OH
OH
OO
OH
OH
H
H
OH
5465 2,3-Didehydrocinnzeylanone
C20H28O7 (380.44). Source: YIN DU E LI Persea indica (aerial parts). Ref: 5128.
5470 Didehydrostemofoline
Asparagamine A C22H27NO5 (385.46). Pharm: Insecticidal (neonate larvae of
OH O
HO
OH
HO
Spodoptera littoralis, LC50 = 0.8mg/L, EC50 = 0.5mg/L). Source: XIAO QIU

BAI BU Stemona collinsae Ref: 3409.
O
OH
5466 7,8-Didehydro-27-deoxyactein
C37H54O10 (658.84). White crystals, mp 260~262C (CH3CN/H2O). Source:
SHENG MA Cimicifuga foetida. Ref: 2427.
O
N
O
O
5471 Didehydrotuberostemonine
C22H29NO4 (371.48). Colorless acicular crystals, mp 176~177C. Source: BAI
BU Stemona tuberosa. Ref: 673.
OO
OH
OH
OH
O
O
O
N
5467 5,6-Didehydroferruginol
C20H28O (284.45). Amorphous solid, mp 145C, []D25 = +35.3 (c = 1.0,
CHCl3). Source: CHANG GENG CU FEI Cephalotaxus harringtonia var.
5472 3,4-Didehydroxy-3'-deoxycapsanthin
drupacea. Ref: 5401.
(5'R)-3,4-Didehydro-,-caroten-6'-one C40H54O (550.88). Source: HONG
OH
HAI JIAO Capsicum annuum (fruit: yield = 0.000013%). Ref: 3007.

O
99
5473 13,15-Dideoxyaconitine
5478 7,2'-Didesacetoxy austrospicatine
[77757-14-3] C34H47NO9 (613.75). Colorless rhomboid crystals, mp
C37H51NO8 (637.82). Source: XI MA LA YA HONG DOU SHAN Taxus
167~169C, []D25 = +16.4 (c = 0.07, ethanol). Source: SONG PAN WU

O
TOU Aconitum sungpanense, ZHUA KUI GUA YE WU TOU Aconitum

[4678]
hemsleyanum var. leueanthus (root: yield = 0.0022%dw)
. Ref: 107, 4678.
O
H
O
H
O
N
H
O O
O
HO
5479 (rel)-1,2-Di-(2,4-dihydroxy-6-methoxybenzoyl)-3,4-di-(4-methoxyphenyl)-cyclobutane
C34H32O10 (600.63). Pale amorphous solid, []D23.5 = +17.2 (c = 0.29, CHCl3).
5474 3,6-Dideoxy-10-hydroxypseudoanisatin
Source: CHANG YE GE NA XIANG Goniothalamus gardneri (aerial parts).
C15H22O5 (282.34). Colorless amorphous. Source: Illicium merrillianum
Ref: 5096.
(pericarp). Ref: 5113.
O
HO
HO
OH
O
OH
OH
HO
5480 rel-(1,2)-Di-(2,6-dimethoxy-4-hydroxy)-benzoyl-rel-(3,4)-di5475 1,4-Dideoxy-1,4-imino-arabinitol
phenylcyclobutane
C5H11NO3 (133.15). Source: SANG ZHI Morus alba. Ref: 2170.
C34H32O8 (568.53). White crystalline solid, mp 213C, []D21 = +17.5 (c = 0.5,
HO
MeOH). Source: BAI DIAN FENG CHE ZI Combretum albopunctatum
HO
OH
O
O
5476 4,20-Dideoxyphorbol 12,13-bis(isobutyrate)
HO
OH
[250258-01-6] C28H40O6 (472.63). Oil, []D = +54 (c = 0.74, CHCl3). Source:
DUN YE DA JI Euphorbia obtusifolia var. obtusifolia. Ref: 2365.

O
5481 1,3-Di-O-[2',2'-di-(p-phenylene) isopropylidene] glycerol
C18H20O3 (284.36). White powder. Source: XI NANG MA WEI ZAO

O
Sargassum parvivesiculosum. Ref: 2591.
H
H
OH
O H
O
HO
5477 Diderroside
[86989-19-7] C19H28O13 (464.43). Pharm: Antitrypanosomal (trypomastigotes
5482 Didrovaltratum
of Trypanosoma cruzi, in vitro, IC50 = 84.9g/mL, control Gentian violet, IC50
Dihydrovaltrate [18296-45-2] C22H32O8 (424.50). Pharm: Sedative. Source:
= 7.5g/mL). Source: Calycophyllum spruceanum. Ref: 3439.
ZHI ZHU XIANG Valeriana jatamansii [Syn. Valeriana wallichii]. (rhizome
O O
H
HO
and root: yield = 0.000013%dw)[4672], Valeriana sp. Ref: 658, 4672.

O
O
O
O
O
HO
H
OO
OH
OH
OH
O
O
O
O
100
5483 8-Diebenzoylpaeoniflorin
5488 20S,22R,23S,24R-16,23;22,25-Diepoxy-cycloartane-3,23,24-triol
C16H24O10 (376.36). Amorphous white powder, []D = 9.6 (c = 1.0, MeOH).
3-O-(6-O-trans-isoferuloyl--D-glucopyranosyl)-(12)--D-glucopyranos
Source: CHI SHAO Paeonia lactiflora wild. Ref: 722.
yl-(12)--D-xylopyranoside
HO
O
OH
Immunosuppressant (mouse allogeneic mixed lymphocyte reaction,
suppresses the proliferation of lymphocytes, IC50 = 99.6mol/L). Source:

Cimicifuga sp. (rhizome). Ref: 4330.
O
OH
OH
OH
OH
5484 Dieckol
OH
OH
[88095-77-6] C36H22O18 (742.57). Amorphous powder, mp > 300C. Pharm:

Antifibrinolysis (2-macroglobulin, IC50 = 5.0g/mL, 2-fibrinolysin, IC50 =
0.8g/mL) [955]; antioxidant (DPPH scavenger, IC50 = 6.2mol/L, control
OO
Ascorbic acid, IC50 = 10.3mol/L)[4376]. Source: HEI KUN BU Ecklonia
OH OH
kurome, Brown alga Ecklonia stolonifera. Ref: 955, 4376.
HO
HO
OO
OH
OH
HO
HO
OH
OH
OH
HO
OH
OH
O
O
OH
OH
OH
OH
5489 20S,22R,23S,24R-16,23;22,25-Diepoxy-cycloartane-3,23,24-triol
O
OH
OO
OH
3-O--D-glucopyranosyl-(12)--D-glucopyranosyl-(12)--D-xylopyranoside
Immunosuppressant (mouse allogeneic mixed lymphocyte reaction,
5485 Diellagic acid rhamnoside (14) glucopyranoside
suppresses the proliferation of lymphocytes, IC50 = 55.6mol/L). Source:
C40H30O24 (894.67). Yellowish amorphous powder. Source: SHI LIU XIN
Cimicifuga sp. (rhizome). Ref: 4330.
CAI Punica granatum. Ref: 1942.
O
OH
OH
OH
OH
O
HO
O O
OO
OH
OH
OH
OO
OH
OH
HO
OH
OH
HO
O
O
OH OH
OH
OH
5486 Z-4,9-Diene-2,3,7-trithiadeca-7-oxide
OH
C7H12OS3 (208.37). Colorless oil liquid. Source: DA SUAN Allium sativum.
OH
Ref: 2118.
OO
HO
OH
5490 16,22R;21,23S-Diepoxy-21S,24-dihydroxy-5-stigmasta-8,14diene-3,28-dione
C29H40O6 (484.64). Colorless oil, []D = +26.6 (c = 0.3, CH2Cl2). Source: JI
NEI YA BAN JIU JU Vernonia guineensis. Ref: 3412.
5487 ()-3,4-Di-epi-3,7-trifara-9,14-diene
HO
C15H24 (204.36). Source: YE TAI Trocholejeunea sandvicensis. Ref: 735.
OH
H
H
H
O
101
5491 (13R,14S)-ent-8,13;14,15-Diepoxy-13-epi-labdan-3-one
5497 2,19;15,16-Diepoxy-neo-clerodan-3,13(16),14-trien-18-oic acid
C20H32O3 (320.48). Colorless needles (MeOH), mp 145~146C, [] D25 = 26.0 (c
C20H26O4 (330.43). Colorless oil, []D20 = +6.1 (c = 0.26, CHCl3) Source:
= 0.5, CHCl3). Source: HAI QI Excoecaria agallocha (root). Ref: 5114.
SHAN XING KUO BAO JU Baccharis flabellata. Ref: 1921.
O
O
5492 1,10,4,5-Diepoxyglechoman-8,12-olide
OH
C15H20O4 (264.32). Pharm: Cytotoxic (in vitro, P388, IC50 = 94g/mL)[5162].

Source: XIAO MEI WEI QIN Smyrnium olusatrum (fruit). Ref: 5162.
O
5498 1,4,4,5-Diepoxy-10,11H-xantha-12,8-olide
CHANG YE TIAN MING JING Carpesium longifolium (aerial parts: yield =
0.0003%dw). Ref: 4736.
5493 16,22R;21,23S-Diepoxy-3-O--D-glucopyranosyloxy-21S,24-di-
hydroxy-5-stigmasta-8,14-dien-28-one
C35H52O11 (648.80). Yellowish powder (acetone), mp 187~188C, []D = 80 (c =
0.7, MeOH). Source: JI NEI YA BAN JIU JU Vernonia guineensis. Ref: 3412.
HO
O
O
OH
H
H
5499 1,1-Diethoxy-n-nonane
C13H28O2 (216.37). Source: CU LIU GUO Hippophae rhamnoides. Ref: 2.
HO
OO
OH
OH
OH
5494 5H-1,10:3,4-Diepoxyguaia-11(13)-en-6,12-olide
C15H18O4 (262.31). Pharm: Cytotoxic (KB ATCC CCL17, IC50 = 4.3g/mL).
5500 1,1-Diethoxy-n-tetradecane
Source: Warionia saharae. Ref: 5399.
O
O
O
O
5495 1,10,4,5-Diepoxy-6-hydroxyglechoman-8,12-olide
C15H20O5 (280.32). White needle crystals (MeOH), mp 165~168C. Source:
XIAO MEI WEI QIN Smyrnium olusatrum (fruit). Ref: 5162.
5501 Diethylene glycol monobenzoate

C11H14O4 (210.23). Colorless oil. Source: TAN XIANG Santalum album
(heartwood). Ref: 4468.
O
O
O
O
O
OH
OH
5496 1,10,4,5-Diepoxy-8-hydroxyglechoman-8,12-olide
C15H20O5 (280.32). Pharm: Cytotoxic (in vitro, P388, IC50 = 88g/mL). Source:
XIAO MEI WEI QIN Smyrnium olusatrum (fruit). Ref: 5162.
O
OH
5502 Diethylphthalate
[84-66-2] C12H14O4 (222.24). bp 295C. Pharm: Anthelmintic; detumescent;
LD50 (rbt, orl) = 1.0g/kg. Source: SHUI QIN Oenanthe javanica. Ref: 6, 658.
O
O
O
O
O
O
102
5503 Diethyl sulfide
5508 2,9-Di-(-furancarbonyloxy)-4,6,15-trihydroxy-1-(2)-methyl-
3-Thiapentane; Ethyl sulfide [352-93-2] C4H10S (90.19). Source: SHENG
butanoyloxy-dihydro--agarofuran
JIANG Zingiber officinale. Ref: 2.
C30H38O12 (590.63). Colorless oil, []D25 = +30.0 (c = 0.13, CHCl3) Source:

OU ZHOU WEI MAO Euonymus europaeus (seed). Ref: 4162.
S
O
HO
5504 Difengpin
4-Allyl-2,6-dimethoxyphenyol cinnamate C20H20O4 (324.38). Colorless

granular crystals, mp 153~155C (petroleum spiritacetic acid). Source: DI
FENG PI Illicium difengpi. Ref: 354.

H
HO
OH
O
H
5509 ,-Digalactosyl-'-linolenic-glyceride
C33H56O14 (676.81). Red oil liquid. Source: SU MI Setaria italica. Ref: 2112.
5505 (1E,22Z)-1,22-Diferuloyloxydocosane
C42H62O8 (694.96). Inseparable mixture with (1E,24Z)-1,24-Diferuloyloxy-
HO
HO
OO
OH
tetracosane, yellow oil. Source: SHAN ZHU ZI Garcinia multiflora (stem).

HO
HO
Ref: 4708.
OH
OH
OO
OH
O
O
O
OH
5510 m-Digallic acid
[536-08-3] C14H10O9 (322.23). mp 268~270C (dec). Source: A LA BO JIAO

JIN HE HUAN Acacia nilotica, MANG GUO Mangifera indica. Ref: 6, 5375.
HO
O
OH
HO
O
5506 (1E,24Z)-1,-24-Diferuloyloxytetracosane
C44H66O8 (723.01). Inseparable mixture with (1E,22Z)-1,22-
HO
OH
HO
Diferuloyloxydocosane, yellow oil. Source: SHAN ZHU ZI Garcinia

multiflora (stem). Ref: 4708.
OH
5511 m-Digalloyl acid
OH
C14H10O9 (322.23). Colorless colloid. Source: LUAN SHU Koelreuteria
paniculata. Ref: 677.

O
OH
OH
OH
O
HO
O
OH
O
OH
HO
5507 Diffractaic acid

[436-32-8] C20H22O7 (374.39). mp 189~190C. Pharm: Antineoplastic
5512 p-Digalloyl acid
(inhibits a tumor which induces Epstein-Barr virus activation). Source:
C14H10O9 (322.23). Source: LUAN SHU Koelreuteria paniculata. Ref: 677.
SONG LUO Usnea longissima, HUAN JIE SONG LUO Usnea diffracta.
OH
Ref: 6, 658, 660.
O
O
OH
OH
OH
OH
HO
O
OH
O
OH
103
5513 ()-2,3-Digalloyl-4-(E)-caffeoyl-L-threonic acid
5517 1,4-Di-O-galloylglucose
C27H22O16 (602.47). Dark brown amorphous powder, mp 215~217C, []D20 =
C20H20O14 (484.37). Source: AN MO LE Phyllanthus emblica (branch and
38 (c = 0.05, MeOH). Source: DENG TAI SHU Cornus controversa [Syn.
leaf). Ref: 3094.
Bothrocaryum controversum] (leaf). Ref: 3918.

OH
OH
OH
OH
HO
OH
OH
OH
OH
O
HO
OO
OH
OH
HO
HO
HO
OH
OH
5518 1,6-Di-O-galloyl--glucose
OH
5514 1,6-Digalloyl-2-cinnamoyl-glucose
C20H20O14 (484.37). []D25 = 22 (c = 0.1, MeOH). Pharm: Antifungal
C29H26O15 (614.52). Source: DA HUANG Rheum officinale, TANG GU TE
(Candida albicans ATCC2091, MIC > 200g/mL, control Amphotericin B,
DA HUANG Rheum tanguticum, ZHANG YE DA HUANG Rheum palmatum.
MIC = 1g/mL; Candida albicans 32, MIC = 25g/mL, Amphotericin B,
Ref: 2, 660.
MIC = 4g/mL; Candida albicans 19, MIC = 12.5g/mL, Amphotericin B,

MIC = 2g/mL)[5021]; cytotoxic inactive (MIC > 200g/mL)[5021]. Source: AN
OH
MO LE Phyllanthus emblica (fruit juice)[3094], DA HUANG Rheum officinale,
OH
HO
OH
OO
HO
OH
ZHANG YE DA HUANG Rheum palmatum, TANG GU TE DA HUANG

Rheum tanguticum, Baseonema acuminatum (leaf). Ref: 2, 660, 3094, 5021.
OH
O
OH
OH
OH
HO
O
O
OH
O
HO
O
5515 3,5-Di-O-galloyl-4-O-digalloylquinic acid
OO
OH
OH
C35H28O22 (800.60). Pharm: Anti-AIDS; reverse transcriptase inhibitor (hmn
OH
O
OH
immunodeficiency virus). Source: YAN FU ZI Rhus chinensis [Syn. Rhus

semialata]. Ref: 658.
5519 3,6-Di-O-galloylglucose
OH
C20H20O14 (484.37). mp 185C (dec). Source: AN MO LE Phyllanthus
HO
HO
O
HO
emblica (leaf, branch)[3094], CAO YUAN LAO GUAN CAO Geranium

O
O
O
O
HO
O
HO
OH
HO
emblica, YOU GAN MU PI Phyllanthus emblica. Ref: 6, 3094.
OH
OH
HO
OH
pratense, QUAN SHEN Polygonum bistorta, YOU GAN YE Phyllanthus
HO
O
HO OH
HO
O OH
O
OH
OH
HO
5516 1,3-Di-O-galloyl--D-glucopyranose
OH
OH
C20H20O14 (484.37). Yellow amorphous powder, []D15 = +17.3 (c = 0.7,

0.0353%). Ref: 4101.
Nicocitin C20H20O14 (484.37). Source: SHAN ZHU YU Cornus officinalis

[Syn. Macrocarpium officinale]. Ref: 2.
O
HO
OH
OO
OH
OH
OH
HO
O
OH
OH
HO
HO
OH
OH
OH
5520 2,3-Di-O-galloyl-D-glucose
OH
OH
OH
OH
OH
104
5521 1,2-Di-O-galloyl-4,6-O-(S)-hexahydroxydiphenoyl--D-glucopyra-
5524 Digitonin
nose
[11024-24-1] C56H92O29 (1229.34). Pharm: Antibacterial; antifungal. Source:
C34H26O22 (786.57). Pharm: Antioxidant (SOD-like activity, EC50 =
MAO DI HUANG Digitalis purpurea. Ref: 658.
76.3mol/L, control Gallic acid, EC50 = 31.7mol/L, L-Ascorbic acid, EC50 =

34.6mol/L); antioxidant (DPPH free radical scavenger, EC50 = 1.27mol/L,
control Gallic acid, EC50 = 5.88mol/L, L-Ascorbic acid, EC50 = 6.25mol/L).

Source: HU TAO REN Juglans regia. Ref: 3408.
HO
HO
OH
OO
HO
HO
HO
OH
O
O
O
OH
HO
OH
OH
OH
HO
HO
OO
O
OH
OH
OH
OH
OO
O
H
H OH
OH
OH
HO
OH
OH
HO
HO
O
OH
OH
OH
OH
5522 Digiferrugineol
1-Hydroxy-2-hydroxymethyl anthraquinone C15H10O4 (254.24). Pharm:
Cytotoxic (KB, ED50 > 25g/mL, control Doxorubicin, ED50 = 0.12g/mL;
5525 Digitoxigenin
Hep3B, ED50 = 3.85g/mL, Doxorubicin, ED50 = 0.14g/mL; Colon205,
(17)-Card-20(22)-enolide [143-62-4] C23H34O4 (374.53). Mp 253C. Source:
ED50 > 25g/mL, Doxorubicin, ED50 = 0.10g/mL; HeLa, ED50 =
FU SHOU CAO Adonis amurensis. Ref: 6.
24.5g/mL, Doxorubicin, ED50 = 0.11g/mL)[4369]; cytotoxic (hmn

nasopharyngeal epidermoid carcinoma cells, in vitro); antibacterial
O
O
(Bacillus subtilis, Escherichia coli). Source: BAI YAN TENG Morinda

parvifolia, GUANG JING QIAN CAO Rubia wallichiana (stem), HU CI
Damnacanthus indicus, JIN JI LE Cinchona ledgeriana, QIAN CAO GEN
H
Rubia cordifolia, XIU MAO DI HUANG Digitalis ferruginea, Cinchona sp.

Ref: 658, 660, 4369.
H
HO
OH
OH
5526 Digitoxin
HO
[71-63-6] C41H64O13 (764.96). Long and thin rectangular lamellar crystals
(ethanol), containing 0.5 or 1 H2O. pure crystals, mp 256~257C, []D20 =
+48 (c = 1.2, dioxane). Pharm: Cardiotonic; LD50 (gpg, orl) = 600mg/kg, (cat,
orl) = 0.18mg/kg, (cat, iv) = 0.4mg/kg. Source: MAO DI HUANG Digitalis
purpurea (dried leaf: content = 0.0226%[5508]), MAO HUA MAO DI HUANG
Digitalis lanata. Ref: 658, 5508.
5523 Diginatin
O
[52589-12-5] C29H44O9 (536.67). Pharm: Cardiotonic; toxin (vertebrate).
Source: MAO HUA MAO DI HUANG Digitalis lanata. Ref: 1521.

O
OH
H
H
OO
H
OO
OH
OO
OH
OH
OO
OH
HO
OH
HO
OH
OH
105
5527 Digitoxose
5531 6,8-Di-C--glucosylchrysin
C6H12O4 (148.16). mp 110~112C. Source: LUO MO ZI Metaplexis japonica.
6,8-Di--glucopyranosyl-5,7-dihydroxy-2-phenyl-4H-1-benzopyran-4-one
Ref: 6.
C27H30O14 (578.53). Amorphous powder. Pharm: Anti-inflammatory inactive

(in vivo, carrageenan-induced rat paw edema). Source: Lychnophora ericoides
(fresh leaf ). Ref: 5040.
O
OH
HO
HO
O
OH
OH
OH
HO OH
5528 5,6-O--D-Diglucopyranosylangelicin
pyridine). Pharm: Antiproliferation inactive (hmn mononuclear cells involving
HO
O
OH
OH
OH
OH
T lymphocytes, B lymphocytes, and macrophages isolated from peripheral

blood, 100mol/L; control Cyclosporine, IC50 = 12nmol/L). Source: LAN YU
5532 Digoniodiol
LUO YE RONG Ficus ruficaulis var. antaoensis (leaf: yield = 0.00023%fw).
C26H26O7 (450.49). Colorless prisms, mp 166~168C, []D23 = 35.5 (c =
Ref: 4794.
0.11, MeOH). Pharm: Cytotoxic (HepG2, IC50 = 6.83g/mL, control

Doxorubicin, IC50 = 0.38g/mL; Hep3B, IC50 = 20.15g/mL, Doxorubicin,
IC50 = 0.36g/mL; MDA-MB-231, IC50 = 6.80g/mL, Doxorubicin, IC50 =
O
O
HO
HO
HO
1.20g/mL; NCF-7, inactive). Source: TAI WAN GE NA XIANG

Goniothalamus amuyon (stem and leaf). Ref: 5056.
OH
HO
HO
HO
HO H
OH
H
O
O
H
5529 3,5-Di-O-(-glucopyranosyl)cyanidin 6''-O-4,6'''-O-1-cyclic malate

C31H33O19+ (709.60). Source: SHE XIANG SHI ZHU Dianthus caryophyllus
H OH
(petal). Ref: 5118.

5533 Digoxin
OH
OH
O
HO
[20830-75-5] C41H64O14 (780.96). Scattering tetrahedral or pentahedral

trioblique lamellar crystals (diluting ethanol or diluting pyridine), mp
260~265C (some dec). Pharm: Cardiotonic. Source: MAO HUA MAO DI
HUANG Digitalis lanata. Ref: 658.
O
HO
OO
OH OH
OH
OH
OH
OH
OH
OH
OH
O OH
H
OO
5530 3,5-Di-O-(-glucopyranosyl)pelargonidin 6''-O-4,6'''-O-1-cyclic
malate
C31H33O18 + (693.60). Source: SHE XIANG SHI ZHU Dianthus caryophyllus

(petal). Ref: 5118.
OH
OH
5534 Digupigan A
4-Hydroxy-3-methoxyphenyl--D-xylopyranosyl(16)--D-glucopyranoside
OH
O
HO
OO
O
OH
HO
OH

Source: GOU QI GEN PI Lycium chinense, GUAN CANG ZHU Atractylodes
japonica (fresh rhizome). Ref: 2451, 4310.
OH
OH
OH
OH
O
OO
OO
OH
OH
OH
OH
OH
OH
OH
106
5535 (12R,12''R)-Diheraclenol
5540 3,14-Dihydroangustine
C32H30O11 (590.59). Pale-yellow amorphous solid, [] D19.1 = +28.31 (c = 0.36,
CHCl3). Pharm: Platelet aggregation inhibitor inactive (rbt platelets, 4.5nmol/L
PAF-induced, 350mol/L AA-induced, 5mol/L ADP-induced, 240mol/L).
Source: BAI YUN HUA Heracleum rapula (fresh root). Ref: 4997.

O
O
O
O
O
OH
HO
O
N
H
N
O
5536 5,3'-Dihexanoyloxy-3,6,7,4'-tetramethoxyflavone
5541 18,19-Dihydroangustine
20g/mL; hTERT-RPE1, ED50 = 0.4g/mL; HUVEC, ED50 = 11.1g/mL; KB,
O
O
O
O
O
O
5537 Dihydroacanthospermal A
C23H32O8 (436.51). Amorphous gum. Pharm: Antineoplastic (mus, P388, in
5542 3,14-Dihydroangustoline
vivo); cytotoxic (KB in vitro, ED50 = 2.6g/mL). Source: GUANG CI BAO
C20H19N3O2 (333.39). Pharm: Antibacterial (in vitro: Staphylococcus aureus,
JU Acanthospermum glabratum. Ref: 661.

HO
O

O
HO
N
H
O
O
5538 9(H)-9-Dihydro-19-acetoxy-10-deacetylbaccatin III

C31H40O12 (604.66). Source: JIANG GUO ZI SHAN Taxus baccata. Ref: 662.
O
HO
O
O
O
O
HO
HO
OH
Dehydroxypodorhizol; ()-Yatein C22H24O7 (400.43). []D20 = 26.8 (c = 1,

CHCl3). Pharm: Antineoplastic; cytotoxic (inhibition of TPA-induced ornithine
O
H
OH
5543 Dihydroanhydropodorhizol
decarboxylase activity with cultured mouse epidermal 308 cells)[5038]; CYP3A4

inhibitor and CYP2D6 inhibitor (in vitro, CYP3A4, IC50 = 1mol/L; CYP2D6, IC50
= 95.7mol/L; control Ketoconazole, CYP3A4, IC50 = 0.72mol/L; control
Quinidine, CYP2D6, IC50 = 0.082mol/L)[4797]. Source: BEI MEI YA BAI Thuja
OH
occidentalis, BI CHENG QIE Piper cubeba (fruit: yield = 0.00017%dw), E SHEN
5539 Dihydroagarofuran
Anthriscus sylvestris, HONG CHAI HU Bupleurum scorzonerifolium (root), LIAN
[5956-09-2] C15H26O (222.37). Bp 135C/8mmHg. Source: CHEN XIANG
YE TONG Hernandia Sonora [Syn. Hernandia ovigera] (seed), Juniperus sp. Ref:
Aquilaria agallocha. Ref: 6, 13.
658, 3498, 4797, 5030, 5038, 5499.

O
O
O
H
O
O
107
5544 2,3-Dihydroauriculatin
5550 3-Dihydrocadambine
C25H26O6 (422.48). Source: SAI NEI JIA ER CI TONG Erythrina
3-19-(S)-Dihydrocadambine [54483-84-0] C27H34N2O10 (546.58). White
senegalensis, Erythrina vogelii. Ref: 1521, 4421.
amorphous powder, mp 144~145C (dec), []D = 91 (c = 0.097, methanol).

Pharm: Antihypertensive (strong and enduring, rat, iv 0.1mg/kg, arterial blood
OH
OH
HO
O
pressure is lowered by 20mmHg); antihypertensive (anesthetized and

conscious spontaneously hypertensive rats)[5341]; antibacterial (in vitro:
Staphylococcus aureus, Bacillus subtilis, Bacillus coli, Bacillus diphtheriae,
Streptococcus sp., Salmonella sp., Bacillus proteus, Aspergillus niger, Bacillus

lactis, Klebsiella pneumoniae); antileishmanial. Source: GOU TENG Uncaria
rhynchophylla [Syn. Nauclea rhynchophylla], HUA GOU TENG Uncaria
sinensis. Ref: 2, 902, 961, 2178, 5341.
5545 Dihydroazorellolide
C20H32O2 (304.48). Colorless needles, mp 121~122C, []D
19.8
= +27.84 (c =
0.58, CHCl3). Source: YIN HUA YAO XIAO YING QIN Azorella cryptantha
HO
N
H
N
H
OH
O H
O
HO
O
OH
OH
5546 Dihydrobaicalin
C21H20O11 (448.39). Source: HUANG QIN Scutellaria baicalensis. Ref: 2.
O
HO
5551 Dihydrocalodenin B
C30H22 O9 (526.50). Pharm: Antibacterial (MDR Staphylococcus aureus:
RN4220 strain, MIC = 8g/mL = 15mol/L, control Erythromycin, MIC
O O
= 128g/mL; XU212 strain, MIC = 8g/mL = 15mol/L, control
OH
OH
OH
Tetracycline, MIC = 128g/mL; SA-1199-B strain, MIC = 8g/mL =
HO
OH
OH
15mol/L, control Norfloxacin, MIC = 32g/mL); cytotoxic (MCF7
5547 2,3-Dihydrobenzofuran-2-(4'-hydroxy-3'-methoxyphenyl)-3--Lrhamnopyranosyloxymethyl-7-methoxy-5-propanol
C26H34O10 (506.55). Brownish amorphous powder, [] D25 = 10 (c = 0.1,
MeOH). Pharm: Antifungal inactive (Candida albicans, MIC > 200g/mL;
breast cancer cells, MTT method, IC50 = (357)mol/L, control

Doxorubicin, IC50 = (0.10.001)mol/L). Source: CHANG E JIN LIAN
MU PI Ochna macrocalyx, SANG DAO BU SHI MU Brackenridgea
zanguebarica. Ref: 5372.
OH
control Amphotericin B, MIC = 1~4g/mL); antibacterial inactive. Source:

Baseonema acuminatum (leaf). Ref: 5021.
HO
O
OH
O
HO
O
OH
OO
OH
OH
OH
HO
OH OH
5548 1,2-Dihydrobis(de-O-methyl)-curcumin
5552 3'',4''-Dihydrocapnolactone
C19H18O4 (310.35). Pharm: Cytotoxic (Colon26-L5, ED50 = 62.6mol/L;
C19H20O5 (328.37). White needles, mp59~62C. Source: JI XIAO XIAO YUN
HT1080, ED50 > 100mol/L). Source: YUN NAN CAO KOU Alpinia
XIANG MU Micromelum minutum (leaf). Ref: 3467.
blepharocalyx (seed: yield = 0.00070%). Ref: 3042.

O
OH
O
OH
HO
5553 Dihydrocapsaicin
5549 Dihydrobungeanool
C18H29NO3 (307.44). Source: LA JIAO Capsicum frutescens (fruit: mean
C18H31NO2 (293.45). Pharm: Anti-PAF. Source: Zanthoxylum sp. Ref: 2176.
content of 3 batch samples = 29.9%[5508]) Ref: 6, 15, 1521, 5508.

O
O
N
H
OH
O
HO
N
H
108
5554 Dihydrocarpalasionin
5560 11,12-Dihydrochiloscyphone
C22H30O8 (422.48). mp 258~265C. Source: ZHOU YE XIANG CHA CAI
(+)-(1S,7S,7aS)-2,3,5,6,7,7a-Hexahydro-7,7a-dimethyl-1-(2-methylpropanony
Isodon rugosus [Syn. Rabdosia rugosa]. Ref: 4067.
l)-1H-indene C15H24O (220.36). Colorless oil. Source: DONG YA ZHI YE
TAI Lepidozia fauriana (essential oil). Ref: 5209.
H
O
OH
5561 ()-Dihydroclusin
OH
C22H26O7 (402.45). Pharm: CYP3A4 inhibitor and CYP2D6 inhibitor (in vitro,
CYP3A4, IC50 = 0.8mol/L; CYP2D6, IC50 > 100mol/L; control
5555 Dihydrocarveol
Ketoconazole, CYP3A4, IC50 = 0.72mol/L; control Quinidine, CYP2D6,
C10H18O (154.25). Source: GAN DI HUANG Rehmannia glutinosa [Syn.
IC50 = 0.082mol/L). Source: BI CHENG QIE Piper cubeba (fruit: yield =
Rehmannia glutinosa f. huechingensis]. Ref: 2.
0.00017%dw). Ref: 4797.

O
HO
OH
OH
O
O
5556 Dihydrocarveol acetate

O
C12H20O2 (196.29). Source: JIU LI XIANG Murraya paniculata [Syn.
Chalcas paniculata]. Ref: 11.
5562 Dihydroconcuressine
C24H42N2 (358.62). mp 93~94C. Source: ZHI XIE MU PI Holarrhena
antidysenterica. Ref: 6.
5557 Dihydrocatalpol
C15H24O10 (364.35). Source: GAN DI HUANG Rehmannia glutinosa [Syn.
OH
H
HO
5563 Dihydroconessine
C24H42N2 (358.62). mp 190~191C. Source: ZHI XIE MU PI Holarrhena
H
HO
OO
OH
OH
antidysenterica. Ref: 6.
N
OH
5558 Dihydrochelerythrine
[6880-91-7] C21H19NO4 (349.39). mp 160~165C. Source: FEI LONG
ZHANG XUE Toddalia asiatica [Syn. Toddalia aculeata; Paullinia asiatica].
H
H
Ref: 6.
O
5564 Dihydroconiferyl alcohol
4-Hydroxy-3-methoxyphenylpropanol [2305-13-7] C10H14O3 (182.22). Pharm:
Lettuce cotyledon factor. Source: WO JU Lactuca sativa, YI ZHU QIAN MA

Urtica dioica. Ref: 658, 660.
5559 11,12-Dihydrochiloscypholone
(+)-(1S,3aR,7S,7aS)-2,3,3a,4,5,6,7,7a-Octahydro-3a-hydroxyl-7,7a-dimethyl1-(2-methylpropanonyl)-1H-indene C15H26O2 (238.37). Colorless oil. Source:
DONG YA ZHI YE TAI Lepidozia fauriana (essential oil). Ref: 5209.
OH
HO
5565 Dihydroconiferyl ferulate

C20H22O6 (358.39). Pale yellow semi-solid. Source: LUO TUO HAO
OH
Peganum nigellastrum (aerial parts). Ref: 3945.

O
O
O
HO
O
OH
109
5566 4'-Dihydroconsabatine
5570 11,13-Dihydrocostunolide
C20H31NO4 (349.47). Oil. Source: Convolvulus sabatius ssp. sabatius (ground
C15H22O2 (234.34). Pharm: Cytotoxic (in vitro, HepG2, CD50 = 75g/mL;
root and rhizome). Ref: 5292.
HeLa, CD50 = 85g/mL; OVCAR-3, CD50 = 75g/mL; control Cisplatin,

HepG2, CD50 = 2.8g/mL; HeLa, CD50 = 5.2g/mL; OVCAR-3, CD50 =
3g/mL). Source: MU XIANG Saussurea lappa [Syn. Aucklandia lappa]
(root: yield = 0.024%dw). Ref: 4720.

O
HO
H
O
OH
5567 6-Dihydrocornic acid

MeOH). Source: JI SU ZI Cornus capitata [Syn. Dendrobenthamia capitata]
(root). Ref: 5177.
HO
HO
5571 3-O-Dihydrocoumaroyl--amyrin
C39H58O3 (574.90). Oil, []D25.9 = +49.5 (c = 0.65, CHCl3). Source: MU MA
HUANG Casuarina equisetifolia. Ref: 2300.
H
H
O
O
H
HO
O
O
H
O
OH
HO
OH
OH
5568 6-Dihydrocornic acid

MeOH). Source: JI SU ZI Cornus capitata [Syn. Dendrobenthamia capitata]
(root). Ref: 5177.
HO
HO
5572 Dihydrocubebin
()-Dihydrocubebin [24563-03-9] C20H22O6 (358.39). Pharm: CYP3A4
inhibitor and CYP2D6 inhibitor (in vitro, CYP3A4, IC50 = 9.5mol/L;
CYP2D6, IC50 = 17.5mol/L; control Ketoconazole, CYP3A4, IC50 =
0.72mol/L; control Quinidine, CYP2D6, IC50 = 0.082mol/L)[4797];
antibacterial (Mycobacterium smegmatis). Source: BI CHENG QIE Piper
cubeba (fruit: yield = 0.001%dw)[4797], JI NEI YA HU JIAO Piper guineense.

O
Ref: 658, 4797.
O
O
HO
OH
OH
OH
OH
OH
5569 Dihydrocorynantheine
C22H28N2O3 (368.48). Pharm: CVS activity (tested in both conscious and
anaesthetized normotensive rats, arterial pressure in both types of rats fell
substantially, while heart rate of only anaesthetized rats also decreased).
Source: CHANG HUA GOU TENG Uncaria longiflora, DUO MAI GOU
TENG Uncaria nervosa, FEI ZHOU GOU TENG Uncaria africana, GOU
TENG Uncaria rhynchophylla [Syn. Nauclea rhynchophylla], GUI YA NA
GOU TENG Uncaria guianensis, HOU YE GOU TENG Uncaria callophylla,
TUO YUAN GOU TENG Uncaria elliptica, XIA GOU TENG Uncaria
5573 Dihydrocucurbitacin B
23,24-Dihydrocucurbitacin B C32H48O8 (560.73). Pharm: Cytotoxic (hmn
cancer lines NUGC-3, IC50 = 3.26g/mL, hmn cancer lines HONE-1, IC50 =
1.55g/mL)[4267]; anti-inflammatory (carrageenan-induced mouse paw edema,
4mg/kg, InRt = 46% at 3h and InRt = 36% at 5h)[4970]. Source: TA YOU XIE
GUA Cayaponia tayuya (root), NAN TOU QIU HAI TANG Begonia
nantoensis (rhizome). Ref: 4267, 4970.
attenuata, XIN XING GOU TENG Uncaria cordata. Ref: 2, 5341.
O
O
HO
N
H H
O
H
H
HO
O
O
OH
110
5574 Dihydrocucurbitacin E
5579 Dihydrocyperaquinone
C32H46O8 (558.72). Pharm: Cytotoxic (hmn cancer lines NUGC-3, IC50 =
[41555-17-3] C14H12O4 (244.25). mp 113~114C. Source: PIAO FU CAO
8.60g/mL, hmn cancer lines HONE-1, IC50 = 2.68g/mL). Source: NAN
Fimbristylis dichotoma. Ref: 6.
TOU QIU HAI TANG Begonia nantoensis (rhizome). Ref: 4267.

O
HO
H
O
HO
OH
O
O
5580 Dihydrodaidzin
()-Dihydrodaidzin; 7-O--D-Glucopyranosyl-4'-hydroxyisoflavanone

MeOH). Pharm: Cytotoxic (in vitro, Hs740T, ED50 = 17.37g/mL; Hs756T,
5575 Dihydrocucurbitacin F
C30H48O7 (520.71). mp 155~157C. Source: DA ZI XUE DAN Hemsleya
macrosperma, LUO GUO DI Hemsleya amabilis, PENG XIAN XUE DAN
Hemsleya pengxianensis. Ref: 6, 554, 660, 1521.
OH
ED50 = 14.92g/mL; Hs578T, ED50 = 28.23g/mL; Hs742T, ED50 =

33.57g/mL; DU145, ED50 = 9.16g/mL; LNCaP-FGC, ED50 = 32.45g/mL).
Source: DA DOU Glycine max (Soybean phytochemical concentrate: yield =
0.0080%dw). Ref: 4630.
O
H
O
HO
OH
HO
HO
HO
OH
OH
OH
5581 2,3-Dihydrodauriporphine
HO
C20H19NO5 (353.38). mp 141.0~142.0C. Source: BIAN FU GE GEN

5576 Dihydrocucurbitacin F-25-acetate
C32H50O8 (562.75). mp 266~268C. Source: CHANG GUO XUE DAN
Hemsleya dolichocarpa (tuberoid: mean content collected in Aug. to Nov. =

3.46%[5508]), DA ZI XUE DAN Hemsleya macrosperma, LUO GUO DI
Hemsleya amabilis, PENG XIAN XUE DAN Hemsleya pengxianensis. Ref: 6,
554, 660, 5508.

O
OH
H
O
HO
O
OH
5582 Dihydrodehydrodiconiferyl alcohol

O
2,3-7-O-Methylcedrusin C20H24O6 (360.41). []D20 = +0.0 (c = 0.10,

MeOH). Source: HUANG JING ZHONG ZI Vitex negundo (seed: yield =
0.0012%), YUE NAN LIE LAN Bursera tonkinensis (root). Ref: 4791, 5336.
HO
C15H24O2 (236.36). Pharm: NO production inhibitor inactive (mus peritoneal
HO
5577 4S-Dihydrocurcumenone
OH
HO
O

5583 Dihydrodehydrodiconiferyl alcohol 4'-O--D-glucoside

(2R,3S)-2,3-Dihydro-2-(4'-hydroxy-3'-methoxyphenyl)-3-hydroxymethyl-7-m
OH
ethoxy-5-benzofuranpropanol 4'-O--D-glucopyranoside C26H34O11 (522.55).
Amorphous powder, []D26 = 15.0 (c = 0.20, MeOH); []D25 = 20.7 (c =

0.10, MeOH). Source: LAN SHAI PIAO Sambucus sieboldiana (leaf), SHAN
FAN GEN Symplocos caudata. Ref: 2535, 4192.
5578 Dihydrocuspidiol
Antifungal (TLC-based assay, Cladosporium cucumerinum, MIQ = 0.01g;

control Miconazole, MIQ = 1g). Source: Fagara xanthoxyloides. Ref: 5385.
HO
OH
O
OH
OO
OH
HO
OH
HO
C14H22O3 (238.33). Colorless oil, []D23 = 11 (c = 0.1, CHCl3). Pharm:
O
OH
111
5584 Dihydrodehydrodiconiferyl alcohol 9'-O-glucoside
5589 (Z)-4,5-Dihydro-6,7-trans-dihydroxy-3-butylidene phthalide
C27H36O10 (520.58). Colorless crystals, []D25 = 15.5 (c = 2.0, MeOH).
C12H16O4 (224.26). Source: CHUAN XIONG Ligusticum chuanxiong [Syn.
Source: RI BEN AN XI XIANG JING PI Styrax japonica. Ref: 2546.
Ligusticum wallichii]. Ref: 2.
HO
O
OH
OH
OH
HO
O
OH
OH
O
HO
5590 (Z)-4,5-Dihydro-6,7-cis-dihydroxy-3-butylidene phthalide

O
Senkyunolide I [94596-28-8] C12H16O4 (224.26). Source: CHUAN XIONG
5585 3,4-Dihydro-15-dehydrolactucopicrin
Ligusticum chuanxiong [Syn. Ligusticum wallichii], GAO BEN Ligusticum
C23H22O7 (410.43). Source: JU QU Cichorium intybus. Ref: 736.
sinense. Ref: 2, 660.
OH
HO
OH
O
O
5591 5,6-Dihydro-1,7-dihydroxy-3,4-dimethoxy-2-methyldibenz[b,f]
oxepin
C17H18O5 (302.33). Colorless crystalline solid (CHCl 3), mp 215~217C
5586 (R)-2,3-Dihydro-7-demethylrobustigenin
(R)-5,7-Dihydroxy-2',4',5'-trimethoxyisoflavanone C18H18O7 (346.34).
Source: CAI BAN YANG TI JIA Bauhinia variegata (root cortex). Ref: 3468.
OH
Amorphous powder, []D = 28 (c = 0.1, MeOH). Source: Erythrina sacleuxii
(stem cortex). Ref: 5097.

HO
O
HO
O
O
5592 2,3-Dihydro-5,7-dihydroxy-2,6-dimethyl-8-(3-methyl-2-butenyl)OH
4H-1-benzopyran-4-one
C16H20O4 (276.34). Pale-yellow acicular crystals, mp 122~124C, [] D25 =
92.8 (c = 0.13, CHCl3). Source: BAI BEI YE Mallotus apelta. Ref: 755.
5587 Dihydro-deoxyarteannuin B
C15H22O2 (234.34). Oil. Source: HUANG HUA HAO Artemisia annua (aerial
OH
parts). Ref: 5224.
HO
5593 2,3-Dihydro-5,7-dihydroxy-2,8-dimethyl-6-(3-methyl-2-butenyl)4H-1-benzopyran-4-one
5588 6'',7''-Dihydro-5',5'''-dicapsaicin
C36H54N2O6 (610.84). Light yellow oil. Pharm: Antioxidant
OH
(ADP/Fe2+-induced liposomal lipid peroxidation, IC50 = 10mol/L; control

Capsaicin, IC50 = 10mol/L; Vitamin E, IC50 = 250mol/L)
[4710]
. Source:
HONG HAI JIAO Capsicum annuum (fruit: yield = 0.00024%). Ref: 4710.
O
O
N
H
HO
5594 (3S,5S,6R,3'R,6'R)-5,6-Dihydro-5,6-dihydroxylutein
C40H58O4 (602.91). Source: DA HUA JU Dendranthema grandiflorum (petal).
Ref: 3865.
HO
OH
HO
O
H
N
OH
HO
OH
112
5595 4',5'-Dihydro-11,5'-dihydroxy-4'-methoxytephrosin
5600 2,3-Dihydro-7,7''-dimethoxyamentoflavone
C24H26O10 (474.47). Colorless solid, []D20 = +1.7 (c = 0.1, acetone). Pharm:
C32H24O10 (568.54). Yellow powder, mp > 290C, []D 24.5 = +5.10 (c = 0.29,
Antineoplastic (Inhibition of DMBA-induced preneoplastic lesions in vitro,
C5H5N). Source: YUN NAN SUI HUA SHAN Amentotaxus yunnanensis (leaf
MMOC assay, IC50 = 9.1mol/L; control Sulforaphane, IC50 = 11mol/L).
and twig: yield = 0.00178%dw). Ref: 4707.
Source: DU HUI MAO DOU Tephrosia toxicaria (stem: yield =

0.00016%dw). Ref: 4718.
OH
OH
O
O
OH
OH
O
H
O
OH
OH
OH
5601 (2R,3S)-Dihydro-2-(3',5'-dimethoxy-4'-hydroxyphenyl)-7-meth5596 (2S,3S,1'S,2'R)-and(2S,3S,1'R,2'R)-2,3-Dihydro-5-(1',2'-di-
oxy-5-acetyl-benzofuran
hydroxypropyl)-2-(3,4-dimethoxyphenyl)-7-methoxy-3-methylbenzofuran
C20H22O7 (374.39). Yellowish resin, []D25 = 9.6 (c = 1.80, MeOH). Source:
C21H26O6 (374.44). Yellow oil, []D25 = +3.5 (c = 1.036, CHCl3). Source:
JUAN BAI Selaginella tamariscina (whole herb). Ref: 4828.
DUAN ROU MAO MA DOU LING Aristolochia pubescens. Ref: 2359.

O
OH
HO
O
5597 (2S,3S,1'S,2'R)-and(2S,3S,1'R,2'R)-2,3-Dihydro-5-(1',2'-dihydroxypropyl)-2-(4-hydroxy-3-methoxyphenyl)-7-methoxy-3-methylbenzofuran
25
C20H24O6 (360.41). Yellow oil, []D = +3.6 (c = 1.024, CHCl3). Source:

DUAN ROU MAO MA DOU LING Aristolochia pubescens. Ref: 2359.
OH
O
OH
O
O
HO
HO
OH
5602 3,4-Dihydro-6,7-dimethoxy-2-methyl-isoquinoline
C12H16NO2+ (206.27). Colorless crystalline, mp 184.5~187.5C. Source:
XIAO HUA MU BAN SHU Xylopia parviflora (bark and root). Ref: 3794.
O
N
5603 9,10-Dihydro-7,8-dimethyl-2-(1-methylethyl)phenanthren-3-ol
C19H22O (266.39). Yellowish gum. Source: XIU QIU SHU WEI CAO Salvia
5598 2,3-Dihydro-5,7-dihydroxy-2,6,8-trimethyl-4H-1-benzopyran-
hydrangea (root). Ref: 5447.
4-one
OH
OH
HO
5599 (Z')-3,8-Dihydro-6,6';7,3'-diligustilide
[106533-38-4] C24H30O4 (382.50). Source: CHUAN XIONG Ligusticum
chuanxiong [Syn. Ligusticum wallichii]. Ref: 2.
5604 Dihydroechioidinin
C16H14O5 (286.29). Colorless needles (CHCl3), mp 200~201C, []D28 =
19.7 (c = 0.13, MeOH). Source: LAN JI CHUAN XIN LIAN Andrographis
echioides. Ref: 2379.
H
H
OH
O
OH
113
5605 Dihydroenmein
5610 5,6-Dihydroeurycomalactone
C20H28O6 (364.44). mp 282 (dec), 240~242C, []D = 114 (C5H5N). Source:
MAO GUO XIANG CHA CAI Isodon trichocarpa. Ref: 4067.
O
H
O
HO
HO
OH
5611 13,18-Dihydroeurycomanol
OH
5606 Dihydro-epi-deoxyarteannuin B
OH
H
C15H22O2 (234.34). Source: HUANG HUA HAO Artemisia annua (aerial

HO
OH
parts). Ref: 5224.
OH
OH
HO
5612 3,4-Dihydro-excelsin
O
C26H40O8 (480.60). Source: GAO CHU Ailanthus excelsa. Ref: 2051.

OH
HO
OH
5607 11,13-Dihydro-3-epizaluzanin C
O
H
O
H

(root: yield = 0.00034%dw). Ref: 4720.
5613 (+)Dihydrofisetin
(+)-Fustin [20725-03-5] C15H12O6 (288.26). White needles (MeOH), mp
228~229C, []D25 = +28.3 (c = 0.9, 50% acetoce). Pharm: Antibacterial
(Pseudomonas maltophilia, Enterobacter cloacae); antiviral (HSV-1); NADH
HO
oxidase inhibitor; succinic oxidase inhibitor; anti-rheumatoid arthritis (oral

H
administration 30mg/kg, significantly decreased rheumatoid arthritis (RA)
and C-reactive protein (CRP) factors in Freund's complete adjuvant)[5460].

O
Source: JI CAI Capsella bursa-pastoris, HUANG LIAN YA Pistacia
5608 5,6-Dihydroergosterol
chinensis, LIN BEI ZI Toxicodendron succedaneum [Syn. Rhus succedanea],
Ergosta-7,22-dien-3-ol C28H46O (398.68). mp 176~177C. Source: CHA YE
QI ZI Rhus verniciflua [Syn. Toxicadendron verniciflum], YE QI SHU YE
Camellia sinensis [Syn. Thea sinensis], LING ZHI Ganoderma lucidum (dried
Rhus sylvestris, Rhus sp., Schinopsis sp., Platanus sp., Tilia sp. Ref: 6, 658,
sporocarp: yield = 0.00075%). Ref: 6, 4603.
5460
OH
HO
OH
OH
O
H
HO
5614 ()Dihydrofisetin
()-Fustin C15H12O6 (288.26). mp 228C. Source: HUANG LIAN YA
5609 3,4-Dihydroeurycomalactone
HO
OH
Pistacia chinensis, LIN BEI ZI Toxicodendron succedaneum [Syn. Rhus

succedanea], JI CAI Capsella bursa-pastoris, YE QI SHU YE Rhus sylvestris.
Ref: 6.
OH
O
O
HO
OH
OH
114
5615 Dihydrofoliamenthin
5620 8,9-Dihydroganoderic acid J methyl ester
[22314-48-3] C26H38O12 (542.59). Source: SHUI CAI Menyanthes trifoliata,
C31H46O7 (530.71). Colorless prisms (MeOHH 2O), mp 202~205C, [] D25 =
SHUI CAI GEN Menyanthes trifoliata. Ref: 6.
+52 (c = 0.22, MeOH). Source: LING ZHI Ganoderma lucidum (dried

HO
O
H
HO
H
O
OH
O
O
OH
OH
O
H
5621 Dihydrogenistin
OH
5616 -Dihydrofucosterol
C29H50O (414.72). Source: ZE QI Euphorbia helioscopia. Ref: 6.
()-Dihydrogenistin; 7-O--D-Glucopyranosyl-5,7,4'-trihydroxyisoflavanone
C21H22O10 (434.4). Yellow amorphous powder, []D25 = 23.7 (c = 0.50, MeOH).
Pharm: Cytotoxic (in vitro, Hs740T, ED50 = 15.12g/mL; Hs756T, ED50 =
12.24g/mL; Hs578T, ED50 = 15.36g/mL; Hs742T, ED50 = 30.8g/mL; DU145,
ED50 = 10.25g/mL; LNCaP-FGC, ED50 = 41.58g/mL). Source: DA DOU
Glycine max (Soybean phytochemical concentrate: yield = 0.013%dw). Ref: 4630.
HO
HO
H
H
OO
HO
OH
OH
HO
OH
5617 Dihydrofukinolide
5622 Dihydrogrindelaldehyde
[41059-95-4] C22H32O6 (392.50). Source: FENG DOU CAI Petasites
C20H34O2 (306.49). Colorless gum. Pharm: Cytotoxic (MCF7, ED 50 =
japonicus. Ref: 6.
3.5g/mL). Source: Colophospermum mopane (bark and seed). Ref: 5147.
O
O
5623 Dihydrogrindelic acid
C20H34O3 (322.49). Colorless gum. Source: Colophospermum mopane (bark

and seed). Ref: 5147.
5618 Dihydrogadesine
C23H37NO6 (423.55). White amorphous powder. Source: QIN LING CUI
OH
QUE HUA Delphinium giraldii. Ref: 2506.

H
OH
O
OH
5624 ()-Dihydroguaiaretic acid
H
N
H
C20H26O4 (330.43). Source: MEI ZHOU SAN BAI CAO Saururus cernuus. Ref: 3959.
OH
OH
HO
5619 8,9-Dihydroganoderic acid J
C30H44O7 (516.68). Colorless prisms (MeOHH 2O), mp 205~208C, [] D25 =

O
+24 (c = 0.04, MeOH). Source: LING ZHI Ganoderma lucidum (dried

OH
5625 Dihydroharman
O
O
H
H
[525-41-7] C12H12N2 (184.24). Source: SHA ZAO SHU PI Elaeagnus

O
OH
angustifolia. Ref: 6.
OH
O
N
H
115
5626 2,3-Dihydro-7-hydroxy-2S*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7-
5631 2,3-Dihydro-7-hydroxy-2S*,3R*-dimethyl-2-[4-methyl-5-(4-
nonadien-6-onyl]-furo[3,2-c]coumarin
methyl-2-furyl)-3(E),7-pentenyl]-furo[2,3-b]chromone
C24H28O5 (396.49). Oil, []D21 = 0 (c = 0.7, CHCl3). Source: DUO SAN A
C24H26O5 (394.47). Colorless oil, []D22 = 0 (c = 0.7, CHCl3). Source: DUO
WEI Ferula ferulaeoides (root). Ref: 4117.
SAN A WEI Ferula ferulaeoides (root: yield = 0.06%). Ref: 4193.

O
HO
HO
O
O
5632 2,3-Dihydro-7-hydroxy-2R*,3R*-dimethyl-2-[4-methyl-5-(4methyl-2-furyl)-3(E)-pentenyl]-furo[3,2-c]coumarin
5627 2,3-Dihydro-7-hydroxy-2S*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7-
nonadienyl]-furo[2,3-b]chromone
C24H30O4 (382.50). Colorless oil, []D22 = 0 (c = 0.2, CHCl3). Source:

O
DUO SAN A WEI Ferula ferulaeoides (root: yield = 0.05%). Ref: 4193.
O
HO
O
HO
5633 2,3-Dihydro-7-hydroxy-2S*,3R*-dimethyl-2-[4-methyl-5-(4methyl-2-furyl)-3(E)-pentenyl]-furo[3,2-c]coumarin
5628 2,3-Dihydro-7-hydroxy-2R*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7-
C24H26O5 (394.47). Oil, []D23 = 0 (c = 0.6, CHCl3). Pharm: NO production
nonadienyl]-furo[3,2-c]coumarin
inhibitor (macrophage-like cell line RAW264.7 activated by LPS/IFN-, IC50
= (87.511.7)mol/L)[2574]; cytotoxic inactive (MTT assay, 3~100mol/L, did
not demonstrate any significant cytotoxicity upon LPS/IFN- treatment for

24h.)[2574]. Source: DUO SAN A WEI Ferula ferulaeoides (root), FU KANG
A WEI GEN Ferula fukanensis. Ref: 2574, 4117.
O
O
O
HO
O
HO
5629 2,3-Dihydro-7-hydroxy-2S*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7
5634 (2R,3S)-2,3-Dihydro-7-hydroxy-2-(4'-hydroxy-3'-methoxyphenyl)-
3-hydroxymethyl-5-benzofuranpropanol 4'-O--D-glucopyranoside

Source: LAN SHAI PIAO Sambucus sieboldiana (leaf). Ref: 4192.
OH
HO
OH
OH
OO
HO
OH
O
O
OH
OH
5630 2,3-Dihydro-7-hydroxy-2R*,3R*-dimethyl-2-[4-methyl-5-(4-
5635 (2S,3R)-2,3-Dihydro-7-hydroxy-2-(4'-hydroxy-3'-methoxyphenyl)-
methyl-2-furyl)-3(E),7-pentenyl]-furo[2,3-b]chromone
3-hydroxymethyl-5-benzofuranpropanol 4'-O--D-glucopyranoside
C24H26O5 (394.47). Colorless oil, []D22 = 0 (c = 0.7, CHCl3). Source: DUO

SAN A WEI Ferula ferulaeoides (root: yield = 0.02%). Ref: 4193.

Source: LAN SHAI PIAO Sambucus sieboldiana (leaf). Ref: 4192.
OH
HO
OH
OO
HO
OH
OH
O
O
OH
OH
116
5636 (7S,8R)-Dihydro-3'-hydroxy-8-hydroxy-methyl-7-(4-hydroxy-3-
1mmol/L, StRt = (31~60)%; Allium cepa, 1mol/L, StRt = (31~60)%, 10mol/L,
methoxyphenyl)-1'-benzofuranpropanol
StRt = (10~30)%, 100mol/L, StRt = (10~30)%, 1mmol/L, InRt = (31~60)%).
C19H22O6 (346.38). Yellowish oil, []D20 = 5.3 (c = 1.0, MeOH). Source:
Source: XI YANG JIE GU MU Sambucus nigra. Ref: 5217.

OH
TAN XIANG Santalum album (heartwood). Ref: 4468.

O
OH
OH
OH
HO
O
HO
5641 (2R-trans) 2,3-Dihydro-2-(4-hydroxy-3-methoxyphenyl)-3-(hydroxymethyl)-7-methoxy-5-benzofuranpropanol acetate
OH
5637 2,3-Dihydro-4-hydroxy-2-indole-3-acetonitrile
C22H26O7 (402.45). Pharm: Plant growth stimulatory or inhibitory activity
C10H8N2O2 (188.19). Orange yellow crystals, mp 150~152C. Source: BAN
(radicle length: Lactuca sativa, 1mol/L, StRt = (10~30)%, 10mol/L, StRt =
LAN GEN Isatis indigotica. Ref: 855.
(31~60)%, 100mol/L, StRt = (31~60)%, 1mmol/L, StRt > 61%; Raphanus

sativus, 1mol/L, StRt = (31~60)%, 10mol/L, StRt > 61%, 100mol/L, StRt
= (10~30)%, 1mmol/L, InRt = (10~30)%; Allium cepa, 1mol/L, StRt =
OH
(10~30)%, 10mol/L, StRt = (31~60)%, 100mol/L, StRt = (10~30)%,

O
1mmol/L, StRt = (10~30)%). Source: XI YANG JIE GU MU Sambucus nigra.
N
H
Ref: 5217.
5638 4,5-Dihydro-5'-hydroxy-4'-methoxy-6,12-dehydro--toxicarol
C24H24O9 (456.45). Yellow needles, mp 215~218C, []D20 = +0.1 (c = 0.1,
O
O
CHCl3:MeOH = 1:1). Source: SAN LIE XUE TONG Macaranga triloba
OH
(leaf). Ref: 3756.
OH
5642 8,9-Dihydro-5-hydroxy-6-(2-methylbutanoyl)-4-phenyl-8-(prop-1-
OH
O
O
en-2-yl)furo[2,3-h]chromen-2-one
O
OH
C25H24O5 (404.47). Source: TIE LI MU Mesua ferrea (blossom). Ref: 3870.
5639 (2R-trans)-2,3-Dihydro-2-(4-hydroxy-3-methoxyphenyl)-3-(hy-
OH
droxymethyl)-7-hydroxy-5-benzofuran-propanol
C19H22O6 (346.38). Pharm: Plant growth stimulatory or inhibitory activity
(radicle length: Lactuca sativa, 1mol/L, StRt = (31~60)%, 10mol/L, StRt =
5643 8,9-Dihydro-5-hydroxy-6-(3-methylbutanoyl)-4-phenyl-8-(prop-1-
(10~30)%, 100mol/L, StRt = (31~60)%, 1mmol/L, StRt = (10~30)%;
en-2-yl)furo[2,3-h]chromen-2-one
Raphanus sativus, 1mol/L, StRt = (31~60)%, 10mol/L, StRt = (31~60)%,
100mol/L, StRt = (10~30)%, 1mmol/L, InRt = (10~30)%; Allium cepa,

1mol/L, StRt = (31~60)%, 10mol/L, StRt or InRt < 10%, 100mol/L, StRt
= (10~30)%, 1mmol/L, InRt > 61%). Source: XI YANG JIE GU MU
Sambucus nigra. Ref: 5217.

OH
OH
O
OH
HO
5644 (2R,3R)-2,3-Dihydro-2-(4-hydroxyphenyl)-5-methoxy-3-methyl-7HO
propenylbenzofuran
C19H20O3 (296.37). Colorless oil, []D25 = +358 (c = 1.91, MeOH). Source:
5640 (2R-trans)-2,3-Dihydro-2-(4-hydroxy-3-methoxyphenyl)-3-(hy-
TE LI NI DA HU JIAO Piper aequale. Ref: 1910.
droxymethyl)-7-methoxy-5-benzofuran-propanol
C20H24O6 (360.41). Pharm: Plant growth stimulatory or inhibitory activity (radicle
length: Lactuca sativa, 1mol/L, StRt = (31~60)%, 10mol/L, StRt = (31~60)%,
100mol/L, StRt or InRt < 10%, 1mmol/L, InRt > 61%; Raphanus sativus,
1mol/L, StRt > 61%, 10mol/L, StRt = (31~60)%, 100mol/L, StRt = (31~60)%,
O
HO
O
117
5645 Dihydroimpranine
5650 Dihydroisodocarpin
(17R,20S,22R)-5-Impra-15,16-ene-3,6-diol C28H47NO2 (429.69).
C20H28O5 (348.44). mp 220~226C. Source: ZHOU YE XIANG CHA CAI
Amorphous powder, []D25 = 32 (c = 0.08, MeOH). Source: XI BEI MU
Isodon rugosus [Syn. Rabdosia rugosa]. Ref: 4067.
Fritillaria imperialis. Ref: 3372.

H
H
H
HO
H
H
OH
OH
5651 Dihydroisomorellin
5646 Dihydro--ionone
[1064-70-6] C33H38O7 (546.67). mp 167C. Source: TENG HUANG Garcinia
C13H22O (194.32). bp 126~129C/12mmHg. Source: GUI HUA Osmanthus
morella. Ref: 6.
fragrans. Ref: 6.
O
OH
5647 2,3-Dihydroirigenin
C18H18O8 (362.34). Pale yellow amorphous powder, []D = 0 (c = 0.5, MeOH).
Source: SHE GAN Belamcanda chinensis (rhizome). Ref: 4128.
5652 (+)-Dihydroisorhamnetin
C16H14O7 (318.29). Pharm: Antioxidant inactive (Takamatsu DCFH method,
Vitamin C, IC50 = (1.90.7)g/mL, Trolox, IC50 = (1.40.5)g/mL)[3850];
cytotoxic (XTT assay, HL-60 cells, IC50 > 50.0g/mL; control NDGA, IC50 =
OH
O
OH
myelomonocytic HL-60 cells, control NDGA, IC50 = (0.70.3)g/mL,
HO
(2.60.2)g/mL, Vitamin C, IC50 > 10.0g/mL, Trolox, IC50 >

10.0g/mL)[3850]. Source: SAN CHI LA RUI A Larrea tridentata (leaf), WU
YA GUO Dillenia indica. Ref: 1521, 3850.
O
OH
5648 Dihydroisoalantolactone
11,13-Dihydroisoalantolactone C15H22O2 (234.34). mp 171~172C. Pharm:
HO
Anthelmintic (effect and toxicity similar to santonin); cytotoxic inactive

OH
(SMMC-7721 IC50 = (174.520.2)g/mL, Vincristine IC 50 =
OH
(30.352.23)g/mL; HO-8910 IC50 = (169.216.3)g/mL, Vincristine IC 50 =
(20.741.91)g/mL; LO2 hmn hepatocytes cell IC50 = (713.323.1)g/mL,
5653 Dihydroisotanshinone I
Vincristine IC50 = (17.250.91)g/mL)[5422]. Source: CHANG YE TIAN
C18H14O3 (278.31). Source: DAN SHEN Salvia miltiorrhiza. Ref: 2.
MING JING Carpesium longifolium (aerial parts: yield = 0.001%dw)
[4736]
JIN FEI CAO Inula japonica, TU MU XIANG Inula helenium. Ref: 6, 658,
O
O
1521, 4736, 5422.

O
O
O
5654 Dihydroisotanshinone II
11,16-Oxy-18,20-dinor-1,3,5(10),6,8,11-abietahexaene-13,14-dione C18H14O3
5649 Dihydroisocucurbitacin B
C32H48O8 (560.73). Colorless acicular crystals, mp 235~237C. Source: XIN
YE CHI BO Thladiantha cordifolia. Ref: 425.
O
HO
CAO Salvia glutinosa (root). Ref: 2384.
O
OH
O
(278.31). Red crystals (MeOH), mp 247~249C. Source: JIAO ZHI SHU WEI
OH
O
O
O
118
5655 7,8-Dihydroisoxuxuarine F
5658 2',3'-Dihydro-jatamansin
Cangorosin B C58H76O8 (901.25). Yellow amorphous solid. Source: QIU SHI
C19H22O5 (330.38). Amorphous powder, []D25 = +53.6 (c = 0.8, MeOH).
MEI DENG MU Maytenus chuchuhuasca(bark). Ref: 4295.
Source: Niphogeton ternata. Ref: 4156.
HO
O
5659 Dihydrokaempferol-3-O--L-rhamnopyranoside
O
Engeletin; Engelitin [572-31-6] C21H22O10 (434.40). Colorless massive
crystals, mp 169~171C. Pharm: Antimalarial (Plasmodium falciparum PoW,

IC50 > 50g/mL, control Chloroquine diphosphate, IC50 = (0.0060.002)g/mL;
Dd2, IC50 < 50g/mL, Chloroquine diphosphate, IC50 = (0.0630.01)g/mL)[5208].
Source: BA QIA Smilax china [Syn. Smilax japonica], TU FU LING Smilax
glabra, WU CI KE YA SHU Andira inermis (leaf). Ref: 714, 2192, 5208.

O
OH
O
HO
5656 7,8-Dihydroisoxuxuarine G
C58H76O8 (901.25). Yellow amorphous solid. Source: QIU SHI MEI DENG
OH
MU Maytenus chuchuhuasca(bark). Ref: 4295.
OH
OH OH
O
O
5660 Dihydrokaranone
C15H22O (218.34). Source: BAI MU XIANG Aquilaria sinensis, CHEN
XIANG Aquilaria agallocha. Ref: 13.
HO
O
O
O
5661 Dihydrokoumine
C20H24N2O (308.43). Source: GOU WEN Gelsemium elegans. Ref: 14.
5657 2,3-Dihydroixocarpalactone B
N
H
C28H40O8 (504.63). White amorphous powder, mp 178~180C, []D20 = 93
(c = 0.089, CH3CN). Pharm: Quinone reductase inducer (mus Hepa 1c1c7

cells, CD = (3.811.47)mol/L, IC50 = (96.92.4)mol/L, CI = 20, positive
control Sulforaphane, CD = (0.360.17)mol/L, IC50 = (9.92.1)mol/L, CI =
28). Source: FEI CHENG SUAN JIANG Physalis philadelphica (stem and
leaf). Ref: 4337.
5662 Dihydrolophirone C
C30H24O8 (512.52). Yellow crystals, mp 187~188C (Me2CO), []D25 = 18 (c
= 0.6, Me2CO). Source: Ochna afzelii (stem cortex). Ref: 5153.
OH
OH
OH
O
HO
OO
H
H
H
H
OH
OH
O
OH
OH
119
5663 Dihydrolucidine A
5668 2,3-Dihydro-7-methoxy-2S*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7-
C30H51N3O (469.76). Source: GUANG LIANG SHI SONG Lycopodium
lucidulum. Ref: 3927.

H
N
H H H
H
H
5669 2,3-Dihydro-7-methoxy-2S*,3R*-dimethyl-2-[4-methyl-5-(4-meth-
yl-2-furyl)-3(E)-pentenyl]-furo[3,2-c]coumarin
C25H28O5 (408.50). Oil, []D23 = 0 (c = 0.6, CHCl3). Pharm: NO production
5664 Dihydrolucidine B
C30H51N3O (469.76). Source: GUANG LIANG SHI SONG Lycopodium
H
H
H
= (27.84.6)mol/L)[2574]; inhibits the inducible nitric oxide synthase (iNOS)

gene expression (LPS/IFN- treatment increased the level of iNOS mRNA
expression, and the compound inhibits this increase, dose-dependent
manner)[2574]; cytotoxic inactive (MTT assay, 3~100mol/L, did not
H
N
H H H
inhibitor (macrophage-like cell line RAW264.7 activated by LPS/IFN-, IC50
demonstrate any significant cytotoxicity upon LPS/IFN- treatment for

24h.)[2574]. Source: DUO SAN A WEI Ferula ferulaeoides (root), FU KANG
A WEI GEN Ferula fukanensis. Ref: 2574, 4117.

H
5665 Dihydromelilotoside
3-(2-O--D-Glucosylphenyl)propanoic acid [24696-05-7] C15H20O8 (328.32).
Colorless thin lamellar (ethyl acetate), mp 144~145C. Pharm: Antiulcerative
(rat, ip, 8g/kg, inhibits 5-HT induced ulcer, InRt = 40%). Source: GUI ZHI
5670 14,15-Dihydro-15-methoxy-3-epicaryoptin
Cinnamomum cassia [Syn. Cinnamomum aromaticum], PI HAN CAO
C27H40O10 (524.61). Viscous mass, []D = 57.4 (CHCl3). Source: KU LANG
Melilotus suaveolens. Ref: 6, 1155.
SHU Clerodendrum inerme (leaf). Ref: 5261.

O
OH
HO
OO
OH
OH
OH
5666 2,3-Dihydro-7-methoxy-2S*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7-
O
O
nonadien-6-onyl]-furo[3,2-c]coumarin
23
C25H30O5 (410.51). Oil, []D = 0 (c = 0.7, CHCl3). Source: DUO SAN A
5671 2,3-Dihydro-3-methoxyixocarpalactone A
O
O
(c = 0.088, CH3CN), artifact generated during the extraction and isolation

procedure. Pharm: Quinone reductase inducer (mus Hepa 1c1c7 cells, CD =
5667 2,3-Dihydro-7-methoxy-2R*,3R*-dimethyl-2-[4,8-dimethyl-3(E),7nonadienyl]-furo[3,2-c]coumarin
(18.634.29)mol/L, IC50 > 20mol/L, positive control Sulforaphane, CD =

(0.360.17)mol/L, IC50 = (9.92.1)mol/L, CI = 28). Source: FEI CHENG
SUAN JIANG Physalis philadelphica (stem and leaf). Ref: 4337.
OH
OH

O
H
O
O
O
OH
OH O
O
H
120
5672 2,3-Dihydro-3-methoxyixocarpalactone B
5676 ()-2,3-Dihydro-2-(1-methylethenyl)-5-benzofurancarboxylic acid
C29H42O9 (534.65). White amorphous powder, mp 190~192C, []D20 = 117 (c =
methyl ester
0.076, CH3CN), artifact generated during the extraction and isolation procedure.
[69703-22-6] C13H14O3 (218.25). Source: BAI HUA LONG DAN Gentiana
Pharm: Quinone reductase inducer (mus Hepa 1c1c7 cells, CD =
algida. Ref: 704.
(10.154.18)mol/L, IC50 = (106.60.2)mol/L, CI = 10, positive control

Sulforaphane, CD = (0.360.17)mol/L, IC50 = (9.92.1)mol/L, CI = 28). Source:
FEI CHENG SUAN JIANG Physalis philadelphica (stem and leaf). Ref: 4337.
OH
OH
OO
5677 Dihydromethysticin
[19902-91-1] C15H16O5 (276.29). Pharm: Antispasmodic. Source: KA WA HU
H
H
JIAO Piper methysticum. Ref: 658.
O
OH
5673 2,3-Dihydro-4'''-O-methyl amentoflavone
H O
C31H22O10 (554.51). Yellow crystals, mp 231~232C (dec), []D25 = 0.53 (c

= 1.33, MeOH). Source: NAN YIN DU SU TIE SHU GUO Cycas beddomei.
Ref: 2540.
5678 Dihydromikanolide
[23758-04-5] C15H16O6 (292.29). Pharm: Antifungal (Candida albicans).
OH
Source: WEI GAN JU Mikania scandens. Ref: 658.

O
HO
O
OH
HO
5679 Dihydromorin
OH
[18422-83-8] C15H12O7 (304.26). mp 226~228C. Pharm: Cytotoxic
5674 1,5-Dihydro-1-methyl-2-amino-imidazol-4-one
(cyclooxygenase-1 inhibitor, IC50 = 20.4g/mL); cytotoxic (mouse
C4H7N3O (113.12). Yellowish crystalline powder, mp > 300C (H2O). Source:
mammary organ culture assay, 82% at 10g/mL). Source: DA DA HE MIAN
CU WEN HAI LONG Trachyrhamphus serratus. Ref: 4583.
BAO GUO Artocarpus dadah, SANG ZHI Morus alba. Ref: 6, 5038.
HO
O
HO
OH
N
NH2
OH
OH
5675 3,4-Dihydro-methylcatalpol
5680 Dihydronepetalactone
Pharm: Antitrypanosomal (Trypanosoma brucei rhodesiense, IC50 =
[17672-81-0] C10H16O2 (168.24). Source: JIA JING JIE Nepeta cataria, MU
73.0g/mL, control Melarsoprol, IC50 = 0.0033g/mL; Trypanosoma cruzi,
TIAN LIAO Actinidia polygama. Ref: 6.
IC50 > 90g/mL, control Benznidazole, IC50 = 0.70g/mL); antileishmanial
(Leishmania donovani, IC50 = 12.7g/mL, control Miltefosine, IC50 =

0.32g/mL); antimalarial (Plasmodium falciparum, IC50 > 50g/mL, control
Artemisinin, IC50 = 0.002g/mL); cytotoxic (L6 cells, IC50 > 90g/mL,
control Podophyllotoxin, IC50 = 0.0075g/mL). Source: LIN PIAN XUAN

SHEN Scrophularia lepidota (root). Ref: 5251.
O
5681 Dihydroniloticin
HO
HO
OH
OH
HO
OH
OH
121
5682 Dihydronortoxiferine I
5686 Dihydroosthenon
C38H40N4 (552.77). Free alkali: amorphous powder, bitter acid
C14H14O4 (246.27). Pharm: Antineoplastic (Raji cells, antitumor promotor, in
salt (acetonewater): mp 300C (dec). Pharm: Antibacterial (Bacillus coli,
vivo, inhibits TPA-induced EBV-EA activation, compound concentration =
Bacillus pyocyaneus, and Staphylococcus aureus, 0.8~3.0mg/mL); antifungal
500mol ratio/32 pmol TPA: EBV-EA-positive cells = (14.71.2)%
(Candida albicans, 0.8~3.0mg/mL). Source: A FU ZE ER MA QIAN ZI
(viability > 80%), -Carotene, EBV-EA-positive cells = (34.31.1)%
Strychnos afzelii, CHANG HUA XU MA QIAN ZI Strychnos dolichothyrsa,
(viability >80), Curcumin, EBV-EA-positive cells = (22.81.8)% (viability
YA MA XUN MA QIAN ZI Strychnos amazonica. Ref: 661.
> 80%), compound IC50 = 176mol ratio/32 pmol TPA, -Carotene, IC50 =
400mol ratio/32 pmol TPA, Curcumin, IC50 = 341mol ratio/32 pmol TPA).
N
H
N
H
H
Source: Citrus hassaku. Ref: 5048.
H
H
H
H
5687 Dihydrooxolucidine A
C30H51N3O2 (485.76). []D21.5 = +3.9 (c = 0.79, CHCl3). Source: GUANG

LIANG SHI SONG Lycopodium lucidulum. Ref: 3927.
5683 2'',3''-Dihydroochnaflavone
H
OH
C30H20O10 (540.48). mp > 300C, []D20 = +6.8 (c = 0.2, MeOH). Source: JIN
H
LIAN MU Ochna integerrima (leaf). Ref: 5133.
N
H H H
OH
O
HO
H
N
OH
O
OH
H
H
5688 Dihydrooxolucidine B
C30H51N3O2 (485.76). Source: GUANG LIANG SHI SONG Lycopodium
OH
H
OH
H
5684 2'',3''-Dihydroochnflavone 7''-O-methyl ether

C31H22O10 (554.51). mp 180~182C, []D20 = +7.7 (c = 0.2, MeOH). Source:
N
H H H
JIN LIAN MU Ochna integerrima (leaf). Ref: 5133.

H
OH
O
HO
5689 11,13-Dihydroparthenolide
C15H22O3 (250.34). Pharm: Cytotoxic (in vitro, SMMC-7721, IC50 >

O
O
OH
200g/mL; HO-8910, IC50 = 158g/mL; control Vincristine, SMMC-7721,

IC50 = 30.35g/mL; HO-8910, IC50 = 20.74g/mL)[4736]. Source: CHANG YE
OH
TIAN MING JING Carpesium longifolium (aerial parts: yield = 0.0007%dw).

Ref: 4736.
5685 Dihydrooroxylin A
Dihydrooroxylin [18956-18-8] C16H14O5 (286.29). Source: HUANG QIN
Scutellaria baicalensis. Ref: 2.
O
O
5690 Dihydroperilla alcohol

HO
C10H18O (154.25). Source: ZI SU YE Perilla frutescens var. arguta. Ref: 2.

OH
O
OH
122
5691 Dihydrophaseic acid 4'-O--D-glucopyranoside
5696 Dihydropseurata F
(1'R,3'R,5'R,8'S)-Epi-dihydrophaseic acid -D-glucoside C21H32O10 (444.48).
C22H32O7 (408.50). mp 268~273C. Source: CHUAN ZANG XIANG CHA
Brown transparent gum, []D = 5.0 (c = 0.16, MeOH). Source: E LI Persea
CAI Isodon pharicus. Ref: 4067.
americana [Syn. Persea gratissima] (seed), HUA NAN WU ZHU YU Evodia
austrosinensis. Ref: 3796, 5052.
OH
O
HO
OO
OH
OH
5697 4,5-Dihydropyrocurzerenone
OH
OH
OH
O
OH
[59462-26-9] C15H18O (214.31). Crystals (pet. ether), mp 65~66C, []D17 =

OH
28 (c = 0.84, CHCl3). Source: JI JI Chloranthus serratus. Ref: 3122.
5692 2,3-Dihydrophilonotisflavone
[124615-13-0] C30H20O12 (572.49). Source: ZE XIAN Philonotis fontana. Ref:
3120.
O
OH
HO
HO
OH
C10H13NO2 (179.22). Yellowish needles. Source: GUANG JIN QIAN CAO

OH
5698 (3,4,5)-4,5-Dihydro-3-(1-pyrryl)-4,5-dimethyl-2(3H)-furanone
Desmodium styracifolium (stem and leaf). Ref: 4907.
OH
OH
OH
5693 2,4-Dihydrophthalic anhydride
C8H6O3 (150.14). Source: DANG GUI Angelica sinensis. Ref: 2.

5699 Dihydroquercetin
Distylin; Taxifolin [480-18-2] C15H12O7 (304.26). Yellow powder, mp
240~242C, mp 221~222C, []D = +44.1 (c = 1.0, Me2CO). Pharm:

Anti-inflammatory (modulator of cytokine network: reduces IFN--induced
ICAM-1 protein, as well as mRNA expression in hmn keratinocytes)[4416].

5694 Dihydropinosylvin
Source: BA DAN XING REN Prunus amygdalus, BAI HUA YING SHAN
[14531-52-3] C14H14O2 (214.27). Pharm: Antifungal (Pyricularia grisea, EC50
HONG Rhododendron mucronatum, MAN SHAN HONG Rhododendron
= 44g/mL, EC90 = 55g/mL; Cladosporium herbarum, EC50 = 32g/mL,
dauricum, YING SHAN HONG Rhododendron mucronulatum, XIAN HE
EC90 = 209g/mL; Fusarium avenaceum, EC50 = 56g/mL, EC90 = 131g/mL;
CAO GEN Agrimonia pilosa var. japonica, HUANG LIAN YA Pistacia
Alternaria citri, EC50 = 89g/mL, EC90 > 200g/mL; Botrytis cinerea, EC50 =
chinensis, TU FU LING Smilax glabra, XIAO YE HONG GUANG SHU
69g/mL, EC90 = 77g/mL)[3751]; antibacterial. Source: SHAN YAO
Knema globularia, Pinus maritime (bark). Ref: 4, 6, 336, 411, 416, 2209,
Dioscorea batatas [Syn. Dioscorea opposita], Stemona cf. pierrei
4416.
(underground parts), Pinus sp. Ref: 658, 3751.

OH
O
OH
OH
HO
OH
OH
OH
5700 Dihydroresveratrol
5695 5,6-Dihydropiperlonguminine
C14H14O3 (230.47). Pharm: Antibacterial (Escherichia coli and
C16H21NO3 (275.35). Pharm: Antifungal (Cladosporium sphaerospermum,
Staphylococcus aureus); antifungal (Cladosporium cladosporioides and
MIA = 5.0g, control Nystatin, MIA = 0.5g). Source: LIU TU HU JIAO
Trichophyton mentagrophytes). Source: Morus sp. Ref: 658.
Piper tuberculatum (seed). Ref: 5102.

OH
O
O
O
OH
HO
123
5701 11,13-Dihydroreynosin
5706 3,4-Dihydrosamaderine C
C15H22O3 (250.34). Pharm: Cytotoxic (in vitro, HepG2, CD50 > 100g/mL;
C19H26O7 (366.41). Pale yellow amorphous solid, []D = 18 (c = 0.022,
HeLa, CD50 > 100g/mL; OVCAR-3, CD50 = 95g/mL; control Cisplatin,
CHCl3). Pharm: Cytotoxic (non-small cell lung cancer NCI-H266, LC50 =
20.9g/mL; colon cancer HCC-2998, LC50 = 26.1g/mL, HCT116, LC50 =
35.9g/mL; HCT15, LC50 = 8.55g/mL; CNS cancer SF539, LC50 =
(root: yield = 0.0015%dw). Ref: 4720.
21.8g/mL, U251, LC50 = 9.42g/mL; melanoma LOX IMVI, LC50 =

7.09g/mL, MI4, LC50 = 11.0g/mL, SK-MEL-5, LC50 = 8.42g/mL; renal
OH
cancer A498, LC50 = 18.1g/mL, ACHN, LC50 = 10.9g/mL; prostate cancer

DU-145, LC50 = 50.8g/mL). Source: MA DAO HUANG LIAN SHU
H
H
Samadera madagascariensis (leaf). Ref: 5334.
HO
OH
5702 Dihydrorobinetin
O
O
HO
[70460-55-8] C15H12O7 (304.26). mp 246C; 225~226C. Source: CI HUAI
HUA Robinia pseudoacacia. Ref: 6.
5707 Dihydrosamidin
OH
HO
Dimidin [10182-81-7] C21H24O7 (388.42). mp 117~119C (methanol), []D =
OH
+19 (c = 1.0); []D = +63 (c = 1.0, dioxane). Pharm: Anti-adrenaline;

antihypercholesterolemic (rbt, inhibits rise of cholesterol and lecithin);
OH
OH
vasodilator. Source: CHI A MI Ammi visnaga, ZHANG GUO QIN

Phlojodicarpus sibiricus. Ref: 658, 661.
5703 16,17-Dihydrorostronol F
C20H32O4 (336.48). Pharm: Cytotoxic inactive (hmn leukemia cell HL-60,
10mol/L). Source: JIE XING YE TAI Jungermannia truncata. Ref: 4201.
O
O
HO
OH
O
OH
5708 Dihydrosanguinarine
[3606-45-9] C20H15NO4 (333.35). mp 191C. Pharm: Antibacterial
(antiphlogosis, using source plant XIAO HUA ZI JING, Fumaria parviflora);
5704 Dihydrorugosanin
20
C22H30O7 (406.48). mp 234~239C, []D = 197.6 (c = 0.21, C5H5N).

Source: ZHOU YE XIANG CHA CAI Isodon rugosus [Syn. Rabdosia
rugosa]. Ref: 4067.
O
(whole herb: mean content of 5 origins = 0.049%)[5508], DUI YE YUAN HU

Corydalis ledebouriana, HUA LING CAO Eschscholzia californica, JU HUA
HUANG LIAN Corydalis pallida, JU ZI JIN Corydalis gigantea, WEI LAN
QIU GUO ZI JIN Fumaria vaillantii, XIAO HUA QIU GUO ZI JIN Fumaria
O
H
parviflora, YING SU KE Papaver somniferum. Ref: 6, 658, 5508.
H
O
similar action with sanguinarin. Source: BAI QU CAI Chelidonium majus
OH
O
O
5705 5,6-Dihydrosamaderine A
C18H20O6 (332.36). White amorphous solid, []D = +75 (c = 0.032, CHCl3).
5709 3,4-Dihydro-1,2-secomicrominutinin
Source: MA DAO HUANG LIAN SHU Samadera madagascariensis (leaf).
C14H14O5 (262.26). Amorphous, []D26 = +6.0 (c = 1.0, MeOH). Source:
Ref: 5334.
XIAO GAN Micromelum falcatum. Ref: 2421.

O
HO
O
OH
H
H
OH
H
O
124
5710 3,4-Dihydro-1,2-secomicrominutinin-9-O-glucoside
5715 Dihydro--sitosteryl ferulate
C20H24O10 (424.41). Amorphous, []D26 = +11.5 (c = 1.0, MeOH). Source:
C39H60 O4 (592.91). mp 155~156C. Source: MI PI KANG Oryza sativa.
Ref: 6.
O
OH
H
H
O H
O
O
HO
OH
OH
O
OH
H
O
HO
5716 Dihydrositsirikine
5711 3,4-Dihydro-1,2-secomicrominutinin methyl ester
C15H16O5 (276.29). Amorphous, []D26 = 3.6 (c = 0.5, CHCl3). Source:
[6519-26-2] C21H28N2O3 (356.47). Source: CHANG CHUN HUA

Catharanthus roseus [Syn. Vinca rosea; Lochera rosea]. Ref: 2.
OH
N
H H
H
H
O
OH
H
5717 Dihydroskullcapflavone I
5712 Dihydrosecurinine
[1878-04-2] C13H17NO2 (219.29). mp 58~60C. Source: YI YE QIU
21.7 (c = 0.15, MeOH). Source: TIAO WEN CHUAN XIN LIAN
Securinega suffruticosa. Ref: 6.
Andrographis lineata. Ref: 3390.
O
H
O
OH
OH
5713 Dihydrosinapyl ferulate
5718 Dihydrosolidagenone
C21H24O7 (388.42). Pale yellow semi-solid. Source: LUO TUO HAO
C20H30O3 (318.46). Source: MAN JING ZI Vitex trifolia. Ref: 746.
Peganum nigellastrum (aerial parts). Ref: 3945.

O
O
O
OH
OH
HO
O
H
5714 Dihydro--sitosteryl ferulate
[83-45-4] C39H60O4 (592.91). mp 156~157C. Source: MI PI KANG Oryza

5719 (+)-8,9-Dihydrostepharine
sativa. Ref: 6.
C18H21NO3 (299.37). Colorless needles (MeOH), []D = +141.4 (c = 0.0055,

MeOH). Source: HOU KE GUI Cryptocarya chinensis (wood). Ref: 3092.
H
H
O
O
HO
H
O
H
O
NH
H
125
5720 22-Dihydrostigmast-4-en-3,6-dione
5723 1,2-Dihydrotanshiquinone
C29H46O2 (426.69). mp 170~171C. Source: LING Trapa bispinosa. Ref: 6.
1,2-Dihydrotanshinone C18H14O3 (278.31). Red acicular crystals (benzene),

mp 169C. Source: DAN SHEN Salvia miltiorrhiza, GAN XI SHU WEI CAO
Salvia przewalskii. Ref: 721, 4538.
O
O
H
H
O
O
5721 15,17-Dihydrotanshinone I
C18H14 O3 (278.31). Pharm: immunosuppressant (lymphocyte
5724 11,13-Dihydro-taraxinic acid-1'-O--D-glucopyranoside
transformation assay control group concanavalin A, 5g/mL, InRt =
C21H30O9 (426.47). Colorless needle crystals (EtOHEt 2O), mp 175~177C,
28%; 20g/mL, InRt = 28%; 80g/mL, InRt = 49%, control
[]D21 = 52.0 (CH3OH, c = 0.450). Source: DAO LUAN YE PU GONG
Dexamethasone, 50g/mL, InRt = 63%). Source: ZHAN LONG JIAN
YING GEN Taraxacum obovatum, YUAN JING HUAN YANG SHEN Crepis
Veronicastrum sibiricum (aerial parts). Ref: 4260.
napifera. Ref: 2216, 5357.
HO
O O
O
OH
O
OH
OH
5725 ,'-Dihydro-3,5,3',4'-tetrahydroxy-4,5'-diisopentenylstilbene
5722 Dihydrotanshinone I
C24H30O4 (382.5). Amorphous solid. Pharm: Antioxidant (linoleic acid
15,16-Dihydrotanshinone I C18H14O3 (278.31). Pharm: Antibacterial
solution, inhibition rate constant K inh = 110000L/(mols)). Source: GUANG
(Staphylococcus aureus, hmn Mycobacterium tuberculosis H37Rv, MIC =
GUO GAN CAO Glycyrrhiza glabra (leaf: yield = 0.06%fw). Ref: 4685.
1.5g/mL); antiallergic (inhibits degranulation of mast cell RBL-2H3,

dose-dependent, IC50 = (14.32.1)mol/L)[4939], MAO A inhibitor (hmn
OH
recombinant MAO A, IC50 = 23mol/L); iNOS inhibitor (RAW267.4 cells,

LPS-induced, IC50 = 2.4mol/L)[5032]; acetylcholinesterase(AChE) inhibitor
HO
(IC50 = 1.0mol/L, Argentatin A, IC50 = 42.8mol/L)[4944]. Source: DAN
OH
SHEN Salvia miltiorrhiza (dried root: mean content = 0.079%[5508]), GAN XI

[5508]
SHU WEI CAO Salvia przewalskii (dried root: content = 0.067%)
OH
HONG GEN CAO Salvia prionitis (dried root: content = 0.067%)[5508],
5726 ,'-Dihydro-3,5,3',4'-tetrahydroxy-5'-isopentenyl stilbene
HUANG HUA SHU WEI CAO Salvia flava (dried root: content =
C19H22O4 (314.38). Yellow oil. Pharm: Antioxidant (linoleic acid solution,
0.001%)[5508], JI YE SHU WEI CAO Salvia bulleyana (dried root: content =
inhibition rate constant K inh = 90000L/(mols)). Source: GUANG GUO GAN
0.002%)[5508], LI SE SHU WEI CAO Salvia castanea (dried root: content =
CAO Glycyrrhiza glabra (leaf: yield = 0.25%fw). Ref: 4685.
0.031%)[5508], MAO DI HUANG SHU WEI CAO Salvia digitaloides (dried

root: content = 0.001%)[5508], NAN DAN SHEN Salvia bowleyana (dried root:
OH
content = 0.004%)[5508], NI DAN SHEN Salvia sinica (dried root: content =

0.006%)[5508], SAN YE SHU WEI CAO Salvia trijuga (dried root: content =
0.031%)[5508], YUN NAN SHU WEI CAO Salvia yunnanensis (dried root:
HO
content = 0.019%)[5508], ZI DAN SHEN Salvia przewalskii var. mandarinorum
OH
(dried root: content = 0.120%) [5508]. Ref: 2, 658, 4939, 4944, 5032, 5508.
OH
5727 3'',4''-DihydrothonningineC
O
C24H24O8 (440.45). Colorless oil. Source: Millettia thonningii. Ref: 2326.
O
O
O
O
OH
126
5728 2,3-Dihydro-3,6,7-trihydroxy-1-H-benzo[b]pyran-4-one
5733 12-Dihydrousararotenoid A
C9H8O5 (196.16). Yellow powder, []D23 = 8.0 (c = 0.50, MeOH). Source:
C18H14O8 (358.31). Pharm: Antimalarial inactive (antiplasmodial,
HUA TAO SHU Trewin nudiflora (seed crust). Ref: 4894.
chloroquine-resistant W2 strain of Plasmodium falciparum, IC50 > 100mol/L,

control Chloroquine, IC50 = 0.094mol/L, control Quinine, IC50 =
0.209mol/L; chloroquine-sensitive D6 strain of Plasmodium falciparum, IC50
HO
OH
HO
> 100mol/L, control Chloroquine, IC50 = 0.009mol/L, control Quinine, IC50

= 0.044mol/L). Source: Millettia usaramensis ssp. usaramensis. Ref: 3454.
O
O
H
O
5729 ,'-Dihydro-3,5,4'-trihydroxy-4,5'-diisopentenylstilbene
C24H30O3 (366.5). Orange-yellow oil. Pharm: Antioxidant (linoleic acid
OH
OH
5734 Dihydrovalepotriate
OH
C22H32O8 (424.50). mp 62~63C. Source: ZHI ZHU XIANG Valeriana

jatamansii [Syn. Valeriana wallichii]. Ref: 6.
HO
O
OH
O
O
5730 ,'-Dihydro-3,5,4'-trihydroxy-5'-isopentenylstilbene
C19H22O3 (298.39). Amorphous solid. Pharm: Antioxidant (linoleic acid
H
O
O
5735 3,4-Dihydroverbenalin
C17H26O10 (390.39). Amorphous powder (CH3OH), mp 209~211C. Source:
OH
MA BIAN CAO Verbena officinalis. Ref: 787.

O
O
HO
OH
O
H
5731 ,'-Dihydro-3,5,3'-trihydroxy-4'-methoxy-5'-isopentenylstilbene
C20H24O4 (328.41). Colorless oil. Pharm: Antioxidant (linoleic acid solution,
inhibition rate constant K inh = 80000L/(mols)). Source: GUANG GUO GAN
CAO Glycyrrhiza glabra (leaf: yield = 0.35%fw). Ref: 4685.
HO
O
OH
OH
OH
5736 Dihydroverticillatine
OH
O
H
HO
N
O
H
O
OH
OH
OH
5732 Dihydrotutin
C15H20O6 (296.32). Source: RI BEN MA SANG Coriaria japonica (seed). Ref:
5737 Dihydrovindolinine
4497.

O
HO
O
O
O
OH
N
H
127
5738 14,15-Dihydrovirosecurinine
5743 1'',2''-Dihydroxanthohumol C
C13H17NO2 (219.29). Yellow oil, []D20 = +280 (c = 0.1, EtOH). Source: YI
(2E)-1-(3,4-Dihydro-5-hydroxy-7-methoxy-2,2-dimethyl-2H-1-benzopyran-6-
YE QIU Securinega suffruticosa (branch leaf). Ref: 4818.
yl)-3-(4-hydroxyphenyl)-2-propen-1-one C21H22O5 (354.41). Orange solid.

Source: PI JIU HUA Humulus lupulus (strobile). Ref: 4789.
O
H
OH
OH
5739 2,3-Dihydrowithaferin A
C28H40O6 (472.63). Pharm: Acetylcholinesterase (AChE) inhibitor (IC50 =
5744 7',8'-Dihydroxuxuarine A
(5003)mol/L, control Galanthamine IC 50 = (8.20.0)mol/L, Eserine
IC50 = (0.850.00)mol/L); BChE inhibitor inactive. Source: CUI MIAN
SHUI QIE Withania somnifera. Ref: 2563.

O
OH
H
O
O
H
H
HO
O
O
OH
5740 24,25-Dihydrowithanolide A
C28H40O6 (472.63). Source: CUI MIAN SHUI QIE Withania somnifera (leaf).
5745 7',8'-Dihydroxuxuarine D
Ref: 5329.
H
OH
O
O
H
H
OH
HO
O
5741 11,13-Dihydroxanthalongin
C15H22O3 (250.34). Source: JIN FEI CAO Inula japonica. Ref: 5422.
H
O
H
O
O
OH
O
5746 (2S)-2',4'-Dihydroxy-2''-(1-hydroxy-1-methylethyl)dihydrofuro
[2,3-h]-flavanone
C20H20O6 (356.38). Yellow powder. Pharm: Cytotoxic (aromatase inhibitor, a
5742 Dihydroxanthohumol
,-Dihydroxanthohumol C21H24O5 (356.42). Pharm: Anti-inflammatory (NO
production inhibitor, in vitro, macrophage RAW264.7 cells, induced by
LPS/IFN-, IC50 = 23mol/L, without showing cytotoxicity at concentrations
lower than 10mol/L, cell viability > 95%)[4795]. Source: PI JIU HUA
Humulus lupulus (strobile). Ref: 4789, 4795.
promising lead as potential cancer chemopreventive agents)[5038]; aromatase

inhibitor (in vitro, IC50 = 0.1mol/L; control Aminoglutethimide, IC50 =
6.4mol/L)[3090]. Source: GOU SHU Broussonetia papyrifera. Ref: 3090, 5038.
HO
OH
HO
OH
O
OH
OH
128
5747 6,12-Dihydroxy-5,8,11,13-abietetraen-7-one
5751 8,10-Dihydroxy-9-acetoxythymol 3-O-tiglate
6,12-Dihydroxyabieta-5,8,11,13-tetraen-7-one [140923-35-9] C20H26O3
C17H22O6 (322.36). []D21 = 1.6 (c = 1.5, CHCl3). Source: PEI LAN
(314.43). []D25 = 9.0 (c = 1.0, CHCl3). Pharm: Antibacterial
Eupatorium fortunei (aerial parts). Ref: 3077.
(Staphylococcus aureus, MIC = 7.8g/mL (MCC > 250g/mL), control

Tetracycline, MIC = 1.56g/mL; Bacillus subtilis, MIC > 250g/mL,
Tetracycline, MIC = 1.56g/mL; Enterococcus faecalis, MIC = 7.8g/mL
(MCC > 250g/mL), Tetracycline, MIC = 1.56g/mL; Listeria

monocytogenes, MIC = 7.8g/mL (MCC >250g/mL), Tetracycline, MIC <
HO
O
OH
0.39g/mL; Salmonella enteriditis, MIC > 250g/mL, Tetracycline, MIC =

1.56g/mL; Escherichia coli, MIC > 250g/mL, Tetracycline, MIC =
1.56g/mL; Shigella sonnei, MIC > 250g/mL, Tetracycline, MIC =
6.25g/mL)[5401]; antifungal (Candida albicans, MIC > 250g/mL,
Miconazole, MIC = 8g/mL; Candida krusei, MIC > 250g/mL,
Miconazole, MIC = 2g/mL)[5401]. Source: CHANG GENG CU FEI
Cephalotaxus harringtonia var. drupacea, DU SONG SHI Juniperus rigida.
5752 16,24-Dihydroxy-12-acetoxy-25,26,27-trinor-16,24-cycloartan-23-one 3-O--L-arabinopyranoside

C34H52O10 (620.79). White powder (MeOH), mp 257~259C, []D = 102.1
(c = 0.18, MeOH). Source: XING AN SHENG MA Cimicifuga dahurica
Ref: 6, 5401.
OH
OH
OH
OH
OO
OH
OH
OH
5748 Dihydroxyacetone
[96-26-4] C3H6O3 (90.08). Source: CU vinegar. Ref: 6.
OH
HO
5753 3',19-Dihydroxyaglaine C
C36H42N2O10 (662.74). []D20 = 103.4 (c = 0.43, CHCl3). Source: MI ZI
LAN Aglaia odorata. Ref: 2289.
5749 2',4'-Dihydroxyacetophenone
OH
H N
[89-84-9] C8H8O3 (152.15). Source: DANG GUI Angelica sinensis. Ref: 2.
HO
OH
N
H
OH
H O
HO
OH
5750 3',4'-Dihydroxyacetophenone
[1197-09-7] C8H8O3 (152.14). White tiny cluster acicular crystals, mp
5754 3,4-Dihydroxyallylbenzene 4-O-[-L-rhamnopyranosyl-(16)]-
119~121C. Pharm: Platelet aggregation inhibitor (induced by ADP,
-D-glucopyranoside
0.5mg/mL); CVS activity (anesthetic dog iv, 40mg/kg, increases coronary
C21H30O11 (458.47). White amorphous powder. Source: JIAN YE LONG XUE
flow, reduces consumption of oxygen in myocardium, increases cerebral
SHU Dracaena cochinchinensis. Ref: 832.
blood flow, lowers blood pressure, and slows heart rate); inhibits vasomotion
(induced by KCl, 1.0mg/kg); anti-inflammatory inactive (no significant
OH
OO
inducers; no significant inhibitory effects on TNF- formation from
O
OH
inhibitory effects on mast cells and neutrophils stimulated with various

OH OH
OH
O
OH
OH
RAW264.7 stimulated with LPS and N9 microglial cells stimulated with

LPS/INF-)[3054]. Source: BAI WEI Cynanchum atratum (root)[3054], JU HUA
Chrysanthemum morifolium [Syn. Dendranthema morifolium], TU MAO
DONG QING Ilex pubescens var. glaber. Ref: 661, 3054.
5755 3,7-Dihydroxy amorph-4-ene 3-acetate

C17H28O3 (280.41). Colorless oil, []D = 9.4 (c = 0.1, CHCl3). Source:
HUANG HUA HAO Artemisia annua (seed). Ref: 3435.
OH
OH
O
O
OH
129
5756 4,10-Dihydroxyaromadendrane
5761 6,4'-Dihydroxy aurone 4-O-rutinoside
C15H26O2 (238.37). Source: JU DA MI ZI LAN Aglaia grandis (leaf). Ref:
C27H30O14 (578.53). mp 228C. Source: SI ZI TAN Pterocarpus santalinus
3947.
(wood). Ref: 3889.

OH
HO
OH
HO
OO
HO
OH OH
OO
HO
O
OH
OH
5757 2,13-Dihydroxyaromadendr-1(10)-en-9-one
25
C15H22O3 (250.34). Needles (acetone), mp 145~146C, []D = 128 (c = 0.6,
5762 2,6-Dihydroxybenzoic acid
CHCl3). Pharm: Insecticidal (adult Cylas formicarius elegantulus,
C7H6O4 (154.12). Source: HU ZHANG Polygonum cuspidatum. Ref: 4186.
0.04mg/insect, 24h mortality = 10%, 48h mortality = 20%, 72h mortality =

70%)[5140]. Source: Curvularia lunata. Ref: 5140.
O
HO
OH
OH
OH
O
H
H

Protocatechuic acid [99-50-3] C7H6O4 (154.12). mp 199~200C, 195~196C.
HO
Pharm: DPPH scavenger (SC50 = 11mol/L)[4247]; antioxidant (in vitro, DPPH

5758 13,14-Dihydroxyaromadendr-1(10)-en-9-one
C15H22O3 (250.34). Oil, []D = 160 (c = 1.0, CHCl3). Pharm: Insecticidal
(adult Cylas formicarius elegantulus, 0.04mg/insect, 24h mortality = 10%,
48h mortality = 40%, 72h mortality = 80%)[5140]. Source: Curvularia lunata.
Ref: 5140.
scavenger, 0.1mg/mL, ScRt = 86.5%)[3015]; antioxidant (superoxide anion

radical scavenger, superoxide dismutase method, IC50 for Formazan formation
activity = 7.2mol/L)[4247]; prostaglandin synthetase activator; antiasthmatic
(gpg, asthma induced by histamine); antibacterial (Staphylococcus albus,
Staphylococcus aureus, Diplococcus pneumoniae, -Streptococcus, Bacillus
coli, Bacillus pyocyaneus, Bacillus proteus and Hemophilus influezae);
antifungal (ash fungi); antihepatotoxin; anti-inflammatory; anti-venom;
OH
antitussive (dispels phlegm, mus, orl, 4.86mg); reduces consumption of

oxygen in myocardium; LD50 (mus, ip) = 896.4mg/kg. Source: AI NA
XIANG Blumea balsamifera (leaf and twig: mean content = 0.0077%)[5508],
H
OH
BAI YE TENG Cryptolepis sinensis, BAN XIA Pinellia ternata, CHUAN

XIONG Ligusticum chuanxiong [Syn. Ligusticum wallichii], DAN SHEN
Salvia miltiorrhiza (dried root: content = 0.047%[5508]), DIAN NAN HONG
5759 ent-16,17-Dihydroxyatisan-3-one
HOU KE Calophyllum polyanthum (seed: yield = 0.0056%dw)[4767], GAN XI
C20H32O3 (320.48). Colorless needles. Source: DA GUO DA JI Euphorbia
SHU WEI CAO Salvia przewalskii (dried root: content = 0.340%[5508]), GE
wallichii (root). Ref: 4585.
YE MI HOU TAO Actinidia rubricaulis var. coriacea (ripe fruit: content =

0.34%)[5508], GUI ZHI Cinnamomum cassia [Syn. Cinnamomum aromaticum]
OH
OH
0.0069%[5508]), HONG GEN CAO Salvia prionitis (dried root: content =

0.038%[5508]), HONG PI YUN SHAN Picea koraiensis, HU HUANG LIAN
H
O
(twig: content scope of 41 origins = 0.0015%~0.0164%, mean content =
Picrorhiza kurrooa, HU ZHANG Polygonum cuspidatum, HUA NAN MI
HOU TAO Actinidia glaucophylla (ripe fruit: content = 0.40%)[5508], HUANG

HUA SHU WEI CAO Salvia flava (dried root: content = 0.464%[5508]), JI YE
5760 ent-3,(13S)-Dihydroxyatis-16-en-14-one
SHU WEI CAO Salvia bulleyana (dried root: content = 0.296%[5508]), JIN
C20H30O3 (318.46). White powder. Source: DA GUO DA JI Euphorbia
HUA MI HOU TAO Actinidia chrysantha (ripe fruit: content = 0.17%)[5508],
wallichii (root). Ref: 4585.
JIN MAO GOU Cibotium barometz [Syn. Polypodium barometz] (rhizome:

mean content of 4 origins = 0.0284%)[5508], JING LI MI HOU TAO Actinidia
callosa var. henryi (ripe fruit: content = 0.32%)[5508], JU AN Eucalyptus
HO
O
H
HO
grandis, KUO YE MI HOU TAO Actinidia latifolia (ripe fruit: content =

0.18%)[5508], LAN YU BAI JI Bletilla formosana (whole herb), LI SE SHU
WEI CAO Salvia castanea (dried root: content = 0.336%)[5508], LI ZHI CAO
Salvia plebeia, LU SHAN SHI WEI Pyrrosia sheareri, LU XIAN CAO
130
Pyrola calliantha [Syn. Pyrola rotundifolia ssp. chinensis], MANG QI GU
5767 1,6-Di-O-p-hydroxybenzoyl--D-glucopyranoside
Dicranopteris pedata [Syn. Polypodium pedatum; Dicranopteris dichotoma],
C20H20O10 (420.38). Source: ZI YE Catalpa ovata (fallen leaf). Ref: 4290.
MAO DI HUANG SHU WEI CAO Salvia digitaloides (dried root: content =
OO
content = 0.14%)[5508], MEI WEI MI HOU TAO Actinidia deliciosa (ripe fruit:
content = 0.16%)[5508], MI HOU LI Actinidia arguta (ripe fruit: content =
OH
0.140%)[5508], MAO HUA MI HOU TAO Actinidia eriantha (ripe fruit:
OH
HO
OH
0.26%)[5508], MI HOU TAO Actinidia chinensis (ripe fruit: content =

0.11%)
[5508]
, MU TIAN LIAO Actinidia polygama (ripe fruit: content =
O
OH
5768 2-O-(3,4-Dihydroxybenzoyl)-2,4,6-trihydroxyphenylacetic acid
0.31%)[5508], MU ZEI MA HUANG Ephedra equisetina, NAN DAN SHEN
C15H12O8 (320.26). Solid. Source: LI CHUN HUA Papaver commutatum [Syn.
Salvia bowleyana (dried root: content = 0.217%)[5508], NAN FANG OU SHI
Papaver rhoeas] (petal). Ref: 4965.
NAN Erica australis, NI DAN SHEN Salvia sinica (dried root: content =
OH
0.088%)[5508], PU HUANG Typha angustata, QUAN CHI QIANG WEI Rosa
canina, SAN YE SHU WEI CAO Salvia trijuga (dried root: content =
[5508]
0.147%
), SANG HUANG Phellinus igniarius (sporocarp: yield =
0.0008%dw)[4747], SI JI QING Ilex chinensis [Syn. Ilex purpurea], XIAN REN
OH
HO
ZHANG Opuntia dillenii (fresh stem: yield = 0.00041%), XIU MAO JI

SHENG Taxillus levinei, XUAN FU HUA Inula britannica, YUN NAN SHU
WEI CAO Salvia yunnanensis (dried root: content = 0.059%)[5508], ZANG
HONG HUA Crocus sativus (petal: yield = 0.00016%), ZI HUA JING TIAN
Hylotelephium mingjinianum, ZONG LV PI Trachycarpus fortunei (petiole
and fibre of sheath, roasted petiole: mean content of 5 origins = 0.033%)[5508],
occurs in many plants (various higher plants: e.g. Fagopyrum spp. and Alnus
spp. etc). Ref: 2, 4, 6, 308, 527, 559, 658, 660, 1521, 3015, 4247, 4500, 4747,
4767, 5501, 5508.
OH
OH
5769 3,4-Dihydroxybenzyl alcohol-4-glucoside

C13H18O8 (302.28). Source: YE LI ZHI YE Pyrus calleryana. Ref: 6.
HO
OO
OH
OH
HO
OH
OH
5770 3,6-Di(4-hydroxy) benzyl-2,5-dioxopiperazine

C18H18N2O4 (326.36). Source: DONG CHONG XIA CAO Cordyceps sinensis
HO
OH
H
N
HO
HO
N
H

[99-10-5] C7H6O4 (154.12). Light-yellow crystals, mp 232~233C, mp 176~178C.
Source: SHAN ZHU YU Cornus officinalis [Syn. Macrocarpium officinale] (fruit:
yield = 0.0028%dw)[9], ZE QI Euphorbia helioscopia. Ref: 6, 9.
O
OH
5771 1,3-Di(4-hydroxybenzyl)-4-methoxy-9,10-dihydrophenanthrene2,7-diol
C29H26O5 (454.53). Source: LAN YU BAI JI Bletilla formosana (whole herb).
Ref: 4500.
OH
OH
HO
OH
HO
OH
5765 2,4-Dihydroxy-1,4-benzoxazin-3-one
OH
C8H7NO4 (181.15). Source: LAO SHU LE Acanthus ilicifolius. Ref: 2080.

5772 2'-(o,m-Dihydroxybenzyl) sweroside
OH
[201598-65-4] C23H26O12 (494.46). Yellow amorphous powder, mp
OH
101~103C, []D20 = 86 (c = 6.349, MeOH). Source: BAI HUA LONG

DAN Gentiana algida. Ref: 704.
5766 2,4-Dihydroxy-1,4-benzoxazin-3-one-2-O--D-glucopyranoside
C14H17NO9 (343.29). Source: LAO SHU LE Acanthus ilicifolius. Ref: 2080.
OH
N
OO
HO
OH
O
HO
OH
OH
OH
OH
O
O
OH
OH
131
5773 2,6-Dihydroxybetulinic acid
5777 (3S,5R,6S,7R)-5,6-Dihydroxy-1,7-bis(4-hydroxyphenyl)-de-O-
C30H48O5 (488.71). Colorless amorphous solid, mp 223~225C (MeOH).
methylcentrolobine
Source: Leandra chaetodon (whole herb). Ref: 5411.
C19H22O5 (330.38). Yellow amorphous solid. Pharm: Cytotoxic (mixture with

(3S,5S,6R,7R)-5,6-Dihydroxy-1,7-bis(4-hydroxyphenyl)-de-O-methylcentrolo
bine: Colon26-L5, ED50 = 49.4mol/L, control 5-FU, ED50 = 0.53mol/L;
HT1080, ED50 = 83.7mol/L, 5-FU, ED50 = 8.0mol/L). Source: YUN NAN
O
HO
CAO KOU Alpinia blepharocalyx (seed). Ref: 3048.
OH
OH
HO
HO
OH
O
OH
5774 (3R,5R)-3,5-Dihydroxy-1,7-bis-(3,4-dihydroxyphenyl)heptane
OH
C19H24O6 (348.4). Viscous syrup, []D23 = +4.0 (c = 0.10, MeOH). Pharm:

Cytotoxic (in vitro, HL-60, IC50 = 1.8g/mL; HSC-2, IC50 = 54g/mL; HGF,
IC50 > 250g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2, IC50 =
24g/mL; HGF, IC50 > 200g/mL). Source: JIAN GEN SHU Tacca chantrieri
[Syn. Tacca minor; Tacca esquirolii] (rhizome: yield = 0.02%dw). Ref: 4609.
OH
5778 (3S,5S,6R,7R)-5,6-Dihydroxy-1,7-bis(4-hydroxyphenyl)-de-Omethylcentrolobine
C19H22O5 (330.38). Yellow amorphous solid. Pharm: Cytotoxic (mixture with
(3S,5R,6S,7R)-5,6-Dihydroxy-1,7-bis(4-hydroxyphenyl)-de-O-methylcentrolo
bine: Colon26-L5, ED50 = 49.4mol/L, control 5-FU, ED50 = 0.53mol/L;
OH
HO
OH
HO
OH
HT1080, ED50 = 83.7mol/L, 5-FU, ED50 = 8.0mol/L). Source: YUN NAN

CAO KOU Alpinia blepharocalyx (seed). Ref: 3048.
OH
HO
O
5775 (3R,5R)-3,5-Dihydroxy-1,7-bis(3,4-dihydroxyphenyl)heptane
3-O--D-glucopyranoside
OH
C25H34O11 (510.54). Amorphous solid, []D23 = 8.0 (c = 0.10, MeOH).
OH
Pharm: Cytotoxic (in vitro, HL-60, IC50 = 3g/mL; HSC-2, IC50 = 92g/mL;
HGF, IC50 = 189g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2,
IC50 = 24g/mL; HGF, IC50 > 200g/mL). Source: JIAN GEN SHU Tacca
5779 (3S,5S,6S,7R)-5,6-Dihydroxy-1,7-bis(4-hydroxyphenyl)-4-de-O-
chantrieri [Syn. Tacca minor; Tacca esquirolii] (rhizome: yield = 0.0022%dw).
methylcentrolobine
Ref: 4609.
C19H22O5 (330.38). Yellow amorphous solid, []D25 = +28.5 (c = 0.040,

MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 44.2mol/L, control 5-FU,
HO
HO
HO
HO
ED50 = 0.53mol/L; HT1080, ED50 > 100mol/L, 5-FU, ED50 = 8.0mol/L).

O
Source: YUN NAN CAO KOU Alpinia blepharocalyx (seed: yield =
OH
OH
HO
OH
0.00025%dw). Ref: 3048.
OH
HO
OH
O
5776 (3R,5R)-3,5-Dihydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)
OH
heptane 3-O--D-glucopyranoside
OH
23
C27H38O11 (538.6). Amorphous solid, []D = 18.0 (c = 0.10, MeOH).

Pharm: Cytotoxic (in vitro, HL-60, IC50 > 10g/mL; HSC-2, IC50 = 198g/mL;
HGF, IC50 > 250g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2,
5780 (3S,5S)-3,5-Dihydroxy-1,7-bis(4-hydroxyphenyl)heptane
chantrieri [Syn. Tacca minor; Tacca esquirolii] (rhizome: yield =
HT1080, ED50 = 94.4mol/L). Source: YUN NAN CAO KOU Alpinia
0.00072%dw). Ref: 4609.
HO
HO
O
HO
HO
OH
O
OH
OH
OH
O
OH
HO
OH
132
5781 (3R,5R)-3,5-Dihydroxy-1,7-bis(4-hydroxyphenyl)heptane 3-O--D-
5786 2,4'-Dihydroxy-5-carboxy-dibenyl ether
glucopyranoside
C13H10O5 (246.22). Source: MAO GUO QI Acer nikoense (stem cortex). Ref:
C25H34O9 (478.54). Amorphous solid, []D23 = 8.0 (c = 0.10, MeOH). Pharm:
4304.
Cytotoxic (in vitro, HL-60, IC50 > 10g/mL; HSC-2, IC50 = 157g/mL; HGF,
OH
IC50 = 213g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2, IC50 =
[Syn. Tacca minor; Tacca esquirolii] (rhizome: yield = 0.0026%dw). Ref:
OH
4609.
O
HO
HO
HO
OH
5787 3,15-Dihydroxy cedrane
OH
OH

OH
HO
OH
OH
5782 4,7-Dihydroxy-3-butylphthalide
C12H14O4 (222.24). White plate crystals, mp 211C. Source: CHUAN XIONG
Ligusticum chuanxiong [Syn. Ligusticum wallichii]. Ref: 2156.
H
OH
5788 4,4-Dihydroxychalcone
C15H12O3 (240.26). Pharm: Cytotoxic inactive (Colon26-L5, HT1080,
100mol/L)[3042]. Source: YUN NAN CAO KOU Alpinia blepharocalyx (seed:
OH
yield = 0.00013%). Ref: 3042.
5783 (3S),4-Dihydroxybutyric acid

OH
C4H8O4 (120.11). Colorless oil, []D25 = 12.3 (c = 0.02, H2O). Pharm:

Tyrosinase inhibitor inactive (in vitro). Source: ZANG HONG HUA Crocus
HO
sativus (petal: yield = 0.0023%). Ref: 3015.

O
5789 5,7-Dihydroxychromone
OH
[31721-94-5] C9H6O4 (178.15). Pharm: Antibacterial (gram-positive bacteria);
HO
OH
Anti-HIV (inhibits HIV replication, H9 Lymphocytic Cells, IC50
5784 (4R)-3,14-Dihydroxycadin-10(15)-ene
(concentration that inhibits uninfected H9 cell growth by 50%) > 25g/mL,
C15H26O2 (238.37). Gum. Pharm: Insecticidal (adult Cylas formicarius
EC50 = 18.65g/mL, TI = 1.34, control AZT IC50 = 500g/mL, EC50 =
elegantulus, 0.27mg/insect, 24h, mortality = 85%, 48h mortality = 100%,
0.0007g/mL, TI = 710000)[4267]. Source: SANG YE Morus alba, SHUI FEI
control Farnesyl methyl ether, 0.27mg/insect, 24h, mortality = 85%, 48h
JI Silybum marianum, LUO HUA SHENG Arachis hypogaea, NAN TOU
mortality = 100%). Source: BAI JIANG JUN Beauveria bassiana. Ref: 3949.
QIU HAI TANG Begonia nantoensis (rhizome). Ref: 658, 4267.

OH
HO
HO
OH
5790 12,21-Dihydroxycimigenol 3-O--L-arabinopyranoside
5785 1,3-Dihydroxy-2-carbomethoxy-9,10-anthraquinone 3-O--prime-
C35H56O11 (652.83). Amorphous solid, []D27 = +10.0 (c = 0.10, MeOH).
veroside
Pharm: Cytotoxic (HSC-2 cells, IC50 = 222mol/L, control Etoposide, IC50 =
C27H28O15 (592.52). Yellow powder, []D = 184.9 (c = 0.08, MeOH).
24mol/L; HGF cells, IC50 = 265mol/L)[4158]. Source: ZONG ZHUANG
Source: MA LAI BAN DAO RAN MU SHU Saprosma scortechinii (stem and
SHENG MA Cimicifuga racemosa (rhizome). Ref: 4158.
24
OH
leaf). Ref: 4219.

O
OH
OH
H
O
OH
OO
OO
O
OH
OH
OH
OH
OH
OH
OH O O
OH
OH
H
OH
133
5791 3-(3'',4''-Dihydroxy-trans-cinnamoyloxy)-D-friedo-olean-14-en-
5795 1,6-Dihydroxycostic acid ethyl ester
28-oic acid
C39H54O6 (618.86). Amorphous solid, mp 196~198C, []D27 = 22 (c = 0.04,
MeOH). Pharm: Antioxidant (in vitro: DPPH free radical scavenger, IC50 =
(291)mol/L, control BHA, IC 50 = (442)mol/L; superoxide scavenger,
IC50 = (3061)mol/L, control PG IC 50 = (1062)mol/L; PEP inhibitor,
(root: yield = 0.0015%dw). Ref: 4720.
IC50 = (0.2500.021)mol/L, control Bacitracin, IC 50 = (129.33.3)mol/L).

Source: GANG MAO CHENG LIU Tamarix hispida (aerial parts). Ref: 4923.
OH
O
H
H
HO
H
O
HO
O
OH
O
OH
5796 5,7-Dihydroxycoumarin
C9H6O4 (178.15). Pharm: EBV-EA inhibitor (TPA-induced, IC50 = 477 Mol
ratio/32 pmol TPA, control -Carotene, IC50 = 400 Mol ratio/32 pmol TPA).
Source: YUAN DONG JIU LI XIANG Murraya siamensis (leaf). Ref: 5255.
OH
5792 (ent-2,7,13E) 2,7-Dihydroxy-3,13-clerodadien-15-oic acid

C20H32O4 (336.48). Source: GAO YI ZHI HUANG HUA Solidago altissima.
Ref: 1521.
HO
5797 7,8-Dihydroxycoumarin-7-O--D-glucuronide
C15H14O10 (354.27). Brown solid, []D20 = 75.11 (c = 1.35, MeOH). Source:
HO
OH
O
OH
BIAN TAI Bazzania trilobata. Ref: 3860.

OH
OH
OO
OH
5793 ()-12,16-Dihydroxy-cis-cleroda-3,13-dien-15-oic acid-15,16-olide
OH
C20H28O5 (348.44). Source: GE LUN BI YA BA DOU Croton schiedeanus
OH

5798 (8S)-8,9-Dihydroxycuminyl -D-glucopyranoside
O
O
Source: ZI RAN QIN Cuminum cyminum (fruit). Ref: 4243.

OH
HO
OO
OH
OH
OH
OH
HO
OH
5794 1-6-Dihydroxycostic acid

C15H22O4 (266.34). Colorless gum, []D20 = +12.0 (c = 0.1, MeOH). Pharm:
5799 3,23(R or S)-dihydroxycycloart-24-en-26-oic acid
Cytotoxic inactive (KB ATCC CCL17, 20g/mL). Source: Warionia saharae.
C30H48O4 (472.71). Shining crystals (CHCl3MeOH), mp 279~281 [] D30 =
Ref: 5399.
+49 (c = 0.52, CHCl3). Source: MANG GUO Mangifera indica. Ref: 1868.
O
OH
H
H
H
OH
O
OH
HO
OH
OH
134
5800 2-(1,4-Dihydroxycyclohexanyl)-acetic acid
5806 8,12-Dihydroxydielmentha-5,9-diene-7,11-dione
C8H14O4 (174.20). Colorless snow-like crystals (MeOHH 2 O), mp 163~165C.
C20H28O4 (332.44). Source: TAI WAN CUI BAI Calocedrus macrolepis var.
Source: MA YE QIAN LI GUANG Senecio cannabifolius. Ref: 4809.
formosana (leaf). Ref: 4298.

O
OH
HO
OH
O
OH
HO
5801 3(),8()-Dihydroxydec-9-en-4,6-yne-1-O--D-glucopyranoside
25
C16H22O8 (342.35). Pale yellow oil, []D = 45.3 (c = 0.75, CH3OH). Pharm:
12-Lipoxygenase inhibitor (10g/mL, InRt = 8.11%; 30g/mL, InRt =
25.81%; control Baicalein, 10g/mL, InRt = 56.23%). Source: DAN ZI HAO
Artemisia monosperma. Ref: 5249.
HO
5807 3,4-Dihydroxydihydroagarofuran
C15H26O3 (254.37). mp 176C. Source: CHEN XIANG Aquilaria agallocha.
Ref: 6, 13.
OH
HO
OH
H
OH
OH
OH
5808 (4S,8S)-8,9-Dihydroxy-8,9-dihydrocarvone 9-O--D-glucopyranoH
side
OH
5802 erythro-Dihydroxydehydrodiconiferyl alcohol
Source: SHI LUO ZI Anethum graveolens (fruit). Ref: 4177.

O
OH
HO
OH
O
O
OH
H H
O
OH
OH
OH
OH OH
OH
5809 (4S,8R)-8,9-Dihydroxy-8,9-dihydrocarvone
5803 threo-Dihydroxydehydrodiconiferyl alcohol
Source: GE LU ZI Carum carvi (fruit). Ref: 4153.
H
HO
OH
OH
H
OH
OH
OH
HO
5804 (5S,6S)-5,6-Dihydroxy-4''-de-O-methylcentrolobine
C19H22O5 (330.38). Source: YUN NAN CAO KOU Alpinia blepharocalyx
(seed: yield = 0.00025%[3035]; yield = 0.00118%[3042]). Ref: 3035, 3042.
HO
5810 (4S,8S)-8,9-Dihydroxy-8,9-dihydrocarvone
C10H16O3 (184.24). Amorphous powder, []D25 = 7 (c = 0.2, MeOH). Source:
GE LU ZI Carum carvi (fruit), SHI LUO ZI Anethum graveolens (fruit). Ref:
4153, 4177.
OH
HO
OH
O
HO
OH
5805 1,6-Dihydroxy-3-deoxyminwanensin
C15H24O6 (300.35). Source: Illicium merrillianum (pericarp). Ref: 4257.
O
5811 (3S,6R)-6,7-Dihydroxy-6,7-dihydrolinalool
C10H20O3 (188.27). Amorphous powder, []D21 = +22 (c = 0.1, CHCl3), []D21
= +24 (c = 0.2, MeOH). Source: HU SUI ZI Coriandrum sativum. Ref: 4302.
HO
OH
OH
OH
OH
HO
OH
135
5812 (3S,6S)-6,7-Dihydroxy-6,7-dihydrolinalool
5817 (3R,5R)-3,5-Dihydroxy-1-(3,4-dihydroxyphenyl)-7-(4-hydroxy-
C10H20O3 (188.27). Amorphous powder, []D21 = 29 (c = 0.3, CHCl3), []D21
phenyl)heptane 5-O--D-glucopyranoside
= 15 (c = 0.3, MeOH). Source: HU SUI ZI Coriandrum sativum. Ref: 4302.

Pharm: Cytotoxic (in vitro, HL-60, IC50 = 5.5g/mL; HSC-2, IC50 =
155g/mL; HGF, IC50 > 250g/mL; control Etoposide: HL-60, IC50 =
OH
HO
0.2g/mL; HSC-2, IC50 = 24g/mL; HGF, IC50 > 200g/mL). Source: JIAN
GEN SHU Tacca chantrieri [Syn. Tacca minor; Tacca esquirolii] (rhizome:
OH
yield = 0.00027%dw). Ref: 4609.
5813 (3S,6R)-6,7-Dihydroxy-6,7-dihydrolinalool-3-O--D-glucopyrano-
HO
side
HO
C16H30O8 (350.41). Amorphous powder, []D21 = +6 (c = 0.1, MeOH). Source:

HU SUI ZI Coriandrum sativum. Ref: 4302.
HO
OH
HO OH
HO
OH
HO
OH
HO
O
HO
5818 1,6-Dihydroxy-2,4-dimethoxyanthraquinone V
OH
C16H12O6 (300.27). Yellow acicular crystals, mp 205~207C. Source: BA JI

TIAN Morinda officinalis. Ref: 228, 8.
OH
5814 (3S,6S)-6,7-Dihydroxy-6,7-dihydrolinalool-3-O--D-glucopyrano-
OH
side

Source: HU SUI ZI Coriandrum sativum. Ref: 4302.
HO
O
HO
OH
OH
HO
5819 6,3'-Dihydroxy-2,4-dimethoxybenzophenone
C15H14O5 (274.28). Source: SHAN ZHU ZI Garcinia multiflora (stem: yield =
OH
0.0022%dw). Ref: 4708.

OH
5815 3,5-Dihydroxy-1-(3,4-dihydroxyphenyl)-7-(4-hydroxyphenyl)heptane
OH
HO
C19H24O5 (332.4). Viscous syrup, []D23 = +1.7 (c = 0.12, MeOH). Pharm:
Cytotoxic (in vitro, HL-60, IC50 = 2.1g/mL; HSC-2, IC50 = 54g/mL; HGF,
IC50 = 162g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2, IC50 =

5820 2',3'-Dihydroxy-4',6'-dimethoxychalcone
[Syn. Tacca minor; Tacca esquirolii] (rhizome: yield = 0.0052%dw). Ref:
C17H16O5 (300.31). Red crystals, mp 124~126C. Source: TIAN ZI YU PAN
4609.
Uvaria dulcis (leaf). Ref: 3928.

OH
OH
HO
OH
OH
O
OH
HO
5816 (3R,5R)-3,5-Dihydroxy-1-(3,4-dihydroxyphenyl)-7-(4-hydroxy-
phenyl)heptane 3-O--D-glucopyranoside
25

5821 2',4'-Dihydroxy-4,6'-dimethoxychalcone
158g/mL; HGF, IC50 = 220g/mL; control Etoposide: HL-60, IC50 =
C17H18O5 (302.33). Colorless needles (MeOH), mp 171C, mp 175~176C).
Ref: 5096.
yield = 0.0014%dw). Ref: 4609.

HO
HO
HO
HO
HO
O
O
OH
OH
HO
OH
OH
136
5822 -2'-Dihydroxy-4,4'-dimethoxydihydrochalcone
5827 1,3-Dihydroxy-6,7-dimethoxy-2,8-diprenylxanthone
C17H18O5 (302.33). Colorless needles (C6H6-EtOAc), mp 94C, []D25 =
C25H28O6 (424.50). Yellow powder, mp 91~92C. Pharm: Cytotoxic (hmn
76.84 (c = 0.001015, MeOH). Source: MENG MAI ROU DOU KOU
small cell lung cancer NCI-H187 cell line, IC50 = (3.691.27)g/mL,
Myristica malabarica (heartwod). Ref: 3906.
control Ellipticine, IC50 = (0.350.15)g/mL). Source: QIAO MU

ZHUANG HUANG NIU MU Cratoxylum arborescens (stem cortex). Ref:
5061.
OH
OH
OH
5823 2',3'-Dihydroxy-4',6'-dimethoxydihydrochalcone
C17H18O5 (302.33). Light yellow crystals, mp 141~142C. Source: TIAN ZI
OH
YU PAN Uvaria dulcis (leaf). Ref: 3928.

5828 (2S)-5,2'-Dihydroxy-7,5'-dimethoxyflavanone
OH
C17H16O6 (316.31). Pharm: AChE inhibitor (in vitro, IC50 = (28.05.0)mol/L,

OH
control Galanthamine, IC50 = (32.22.5)mol/L)[4333]; BChE inhibitor (in vitro,

IC50 = (7.95.0)mol/L, control Galanthamine, IC50 = (163.05.0)mol/L).
Source: CU YING MAO DIAN ZI CAO Onosma hispida (whole herb). Ref:
4333.
5824 2',4'-Dihydroxy-4,6'-dimethoxydihydrochalcone
C17H16O5 (300.31). Yellow plates (MeOH), mp 161~163C, mp 158~159C.
Ref: 5096.
HO
O
OH
5829 5,3'-Dihydroxy-7,4'-dimethoxyflavone
HO
[32174-62-2] C17H14O6 (314.30). Source: CHI YANG Alnus japonica. Ref:

OH
1521.
5825 (2R,3S)-(+)-3',5-Dihydroxy-4',7-dimethoxydihydroflavonol
OH
C17H16O7 (332.31). Colorless powder from MeOH, mp 183.5~184.0C, []D24

= 156 (c = 0.2, MeOH). Source: HOU PI SHU Lannea grandis [Syn. Lannea
OH
coromandelica]. Ref: 739.
O
O
OH
5830 5,8-Dihydroxy-6,7-dimethoxyflavone
OH
OH
OH
5826 (2R,3R)-4',7-Dihydroxy-2',5-dimethoxydihydroflavonol
Cytotoxic (Bel7402, ED50 > 10g/mL, control Camptothecin, ED50 =
OH
0.06g/mL; BGC823, ED50 > 10g/mL, Camptothecin, ED50 = 0.09g/mL;

HCT8, ED50 > 10g/mL, Camptothecin, ED50 = 0.14g/mL; A549, ED50 >
5831 5,7-Dihydroxy-8,2'-dimethoxyflavone-7-O--D-glucopyranoside
10g/mL, Camptothecin, ED50 = 0.09g/mL; MCF7, ED50 > 10g/mL,
C23H24O11 (476.44). Yellow needles (MeOH), mp 248~249C (dec), []D25 =
Camptothecin, ED50 = 0.01g/mL). Source: GOU JI Cudrania
252.5 (c = 0.075, MeOH). Source: KE AI HUANG QIN Scutellaria
cochinchinensis (root). Ref: 5338.
amabilis (root: yield = 0.0027%dw). Ref: 2072.
OH
OO
HO
O
OH
O
HO
OH
OH
OH
OH
137
5832 4',7-Dihydroxy-2',5-dimethoxyflavonol
5837 1,7-Dihydroxy-3,9-dimethoxy pterocarpene
C17H14O7 (330.30). Yellow powder. Pharm: Cytotoxic (Bel7402, ED50 >
C17H14O6 (314.30). Colorless acicular crystals, mp 210~214C. Source:
10g/mL, control Camptothecin, ED50 = 0.06g/mL; BGC823, ED50 >
HONG HUA YAN HUANG QI Hedysarum multijugum. Ref: 2224.
10g/mL, Camptothecin, ED50 = 0.09g/mL; HCT8, ED50 > 10g/mL,

Camptothecin, ED50 = 0.14g/mL; A549, ED50 > 10g/mL, Camptothecin,
ED50 = 0.09g/mL; MCF7, ED50 > 10g/mL, Camptothecin, ED50 =
OH
0.01g/mL). Source: GOU JI Cudrania cochinchinensis (root). Ref: 5338.

OH
OH
HO
O
OH
O
5838 5,7-Dihydroxy-3',4'-dimethoxyspiro{2H-1-benzopyran-7'-bicyclo
5833 7,4'-Dihydroxy-2',5'-dimethoxyisoflav-3-ene
[4.2.0]octa[1,3,5]-trien}-4-one
C17H16O5 (300.31). Amorphous powder. Pharm: Antimalarial (antiplasmodial
C18H16O6 (328.32). Yellow gum, []D25 = +56.0 (c = 0.035, MeOH). Source:
in vitro, Plasmodium falciparum, W2 strain, IC50 = (27.71.8)mol/L,
HE CAO YE JIA BEI FANG FENG Ledebouria graminifolia (tuber). Ref:
control Quinine, IC50 = (0.210.01)mol/L; D6 strain, IC50 =
3368.
(18.21.1)mol/L, Quinine, IC50 = (0.0420.002)mol/L). Source: A BI XI

NI YA CI TONG Erythrina abyssinica (root cortex). Ref: 5420.
HO
O
O
HO
O
OH
OH
O
5839 3',4-Dihydroxy-3,5'-dimethoxystilbene
C16H16O4 (272.30). Brown oil. Source: Scilla nervosa (bulb). Ref: 2381.
5834 2',7-Dihydroxy-4',5'-dimethoxyisoflavone
C17H14O6 (314.30). Yellow crystals from methanol, mp 238~240C. Pharm:
Hepatoprotective (mus primary cultured hepatocytes, antihepatotoxin induced
O
HO
by D-galactosamine (GalN), 100mol/L, InRt = (25.91.6)%, weak, control

Silybin, 100mol/L, InRt = (77.05.5)%)[4095]. Source: GUANG BU DING
OH
GONG TENG Erycibe expansa, JIANG ZHEN XIANG Dalbergia odorifera.

Ref: 716, 4095.
HO
O
O
O
HO
5835 3',7-Dihydroxy-4',6-dimethoxyisoflavone
5840 1,3-Dihydroxy-4,5-dimethoxyxanthone
[22804-53-1] C15H12O6 (288.26). mp 274~275C. Source: ZHANG YA CAI
Swertia pseudochinensis. Ref: 6.
C17H14O6 (314.30). Source: XIANG DOU Dipteryx odorata (callus and root),
OH
Glycyrrhiza sp. Ref: 2431, 4475.
HO
HO
OH
O
O
O
O
5836 1,3-Dihydroxy-5,6-dimethoxy-2-methyl-9,10-anthraquinone
C17H14O6 (314.30). Yellow powder (acetone), mp >228C. Source: NAN
C15H12O6 (288.26). Pharm: Cytotoxic (P388 ED50 = 4.74g/mL, control
SHAN HUA Prismatomeris tetrandra (root). Ref: 4521.
Mithramycin ED50 = 0.06g/mL, HT29 ED50 = 7.28g/mL, Mithramycin

ED50 = 0.08g/mL). Source: TAI WAN LV DAO TENG HUANG Garcinia
OH
linii. Ref: 4094.

O
OH
OH
O
O
HO
O
138
5847 1,3-Dihydroxy-4,5-dimethoxyxanthone-1-O--D-glucopyranoside
C15H12O6 (288.26). Source: YUAN ZHI Polygala tenuifolia. Ref: 2.
C21H22O11 (450.40). mp 269~274C (dec). Source: ZHANG YA CAI Swertia

pseudochinensis. Ref: 6.
OH
O
O
HO
OH
HO
OH
OH
OH

linii. Ref: 4094.
5848 1,3-Dihydroxy-4,5-dimethoxyxanthone-3-O--D-glucopyranoside
C21H22O11 (450.40). mp 264~266C. Source: ZHANG YA CAI Swertia
OH
pseudochinensis. Ref: 6.
O
O
HO
OH
O
OO
HO
C15H12O6 (288.26). Pharm: Antifungal (Aspergillus fumigatus CBS113.26,
O
O
OH
OH
OH
MIC80 = 16g/mL, control Amphotericin B, MIC80 = 8g/mL; Aspergillus

flavus IHEM37.19, MIC80 = 8g/mL, Amphotericin B, MIC80 = 8g/mL;
Aspergillus niger IHEM2951, MIC80 = 31g/mL, Amphotericin B, MIC80 =
5849 5,4'-Dihydroxy-8-(3,3-dimethylallyl)-2''-hydroxymethyl-2''-meth-
16g/mL; Aspergillus terreus 5029.2000, MIC80 = 62g/mL; Amphotericin B,
ylpyrano[5,6:6,7]isoflavone
MIC80 = 16g/mL; Candida albicans ATCC663.90, MIC80 = 62g/mL;
C25H24O6 (420.47). Yellow amorphous powder, mp 205~207C, []D20 = 7.8
Amphotericin B, MIC80 = 1g/mL). Source: SU GE LAN HU TONG
(c = 0.1, MeOH). Source: CI TONG Erythrina variegata [Syn. Erythrina
Calophyllum caledonicum (stem cortex). Ref: 4995.
indica] (stem cortex: yield = 0.000024%fw). Ref: 2269.
OH
O
O
OH
HO
OH
OH
C15H12O6 (288.26). Source: CHAN YI TENG Securidaca inappendiculata

(stem). Ref: 5238.
O
5850 5,4'-Dihydroxy-8-(3,3-dimethylallyl)-2''-methoxyisopropylfurano
OH
[4,5:6,7]isoflavone
HO
C26H26O6 (434.49). Yellow amorphous powder, mp 101~102C. Source: CI

O
O
O
TONG Erythrina variegata [Syn. Erythrina indica] (stem cortex: yield =

0.000012%fw). Ref: 2269.
C15H12O6 (288.26). Yellow powder, mp 251~252C (dec). Source: HUANG
HAI TANG Hypericum ascyron. Ref: 2398.
O
OH
O
HO
O
O
OH
OH
139
5851 3,9-Dihydroxy-4-(3,3-dimethylallyl)[6aR,11aR]-pterocarpane
5856 5,7-Dihydroxy-6,8-dimethyl-3-(4'-hydroxy-3'-methoxybenzyl)
C20H20O4 (324.38). Yellow gum, []D25 = 41 (c = 0.3, MeOH). Pharm:
chroman-4-one
Cytotoxic (KB, IC50 = (60.88.0)mol/L, control Helenalin, IC50 =
C19H20O6 (344.37). Source: MAI DONG Ophiopogon japonicus. Ref: 2044.
(0.640.08)mol/L, Melphalan, IC50 = (6.00.5)mol/L; Mono-Mac-6,

IC50 > 75mol/L, Helenalin, IC50 = (3.10.3)mol/L; Jurkat-T, IC 50 =
(61.17.7)mol/L, Helenalin, IC50 = (1.140.08)mol/L, Melphalan, IC50 =
HO
OH
(9.10.8)mol/L). Source: Bituminaria morisiana (leaf). Ref: 5077.

O
OH
5857 4',6'-Dihydroxy-3',5'-dimethyl-2'-methoxychalcone
HO
C18H18O4 (298.34). Source: YANG PU TAO YE Syzygium samarangense. Ref:

H
4100.
OH
5852 1-[2',4'-Dihydroxy-3',5'-di-(3''-methylbut-2''-enyl)-6'-methoxy]-
HO
phenylethanone
C19H26O4 (318.42). Source: SHA TANG MU Acronychia pedunculata. Ref:
2373.
OH
5858 7-(5',6'-Dihydroxy-3',7'-dimethylocta-2',7'-dienyloxy)-coumarin
C19H22O5 (330.38). Pharm: Antibacterial; smooth muscle relaxant;
OH
anticoagulant; photosensitive agent; ichthyotoxin; toxin. Source: Zanthoxylum

sp. Ref: 2176.
OH
OH
O
5853 6,7-Dihydroxy-1,1-dimethyl-N-ethyl-1,2,3,4-tetrahydroisoquinoline

25
C13H19NO2 (221.30). Amorphous brownish solid, 184 dec (MeOH), []D =
OH
+13 (c = 0.70, MeOH). Source: GONG XING MA DOU LING Aristolochia

arcuata. Ref: 2037.
5859 1,4-Dihydroxy-2-(3',7'-dimethyl-1'-oxo-2'-E,6'-octadienyl)benzene
C16H20O3 (260.34). White amorphous powder. Pharm: Antifungal (TLC
bioautographic assay, Cladosporium cladosporioides, MA = 1.0g, control
HO
Miconazole, MA = 1.0g; Cladosporium sphaerospermum, MA = 1.0g,
HO
Miconazole, MA = 1.0g). Source: CU YE MAI HU JIAO Piper

crassinervium. Ref: 3440.
5854 6,7-Dihydroxy-1,1-dimethyl-N-(6'-fructopyranosyl)-1,2,3,4-tetrahydroisoquinoline
C17H25NO7 (355.39). Amorphous brownish solid, 105 dec (MeOH), []D25 =
OH
44 (c = 0.26, MeOH). Source: GONG XING MA DOU LING Aristolochia

arcuata. Ref: 2037.
O
HO
OH
OH
HO
OH
5860 1,4-Dihydroxy-2-(3',7'-dimethyl-1'-oxo-2'-Z,6'-octadienyl)benzene
OH
OH

5855 6,7-Dihydroxy-1,1-dimethyl-N-(2'-glyceryl)-1,2,3,4-tetrahydroiso-
quinoline
C14H21NO4 (267.33). Amorphous brownish solid, 174 dec. (MeOH), []D25 =

arcuata. Ref: 2037.
OH
HO
HO
OH
OH
OH
140
5861 2,7-Dihydroxy-1,6-dimethylpyrene
5866 4,4'-Dihydroxydiphenyl methane
C18H16O2 (264.33). Source: JIAN DENG XIN CAO Juncus acutus. Ref: 1965.
[620-92-8] C13H12O2 (200.24). Source: TIAN MA Gastrodia elata. Ref: 2.

OH
OH
HO
HO
5867 3,7-Dihydroxy-2,5-diundecylnaphthoquinone
C32H50O4 (498.75). Yellow powder, mp 75~77C. Pharm: Cytotoxic inactive
5862 6,7-Dihydroxy-1,1-dimethyl-1,2,3,4-tetrahydroisoquinoline
C11H15NO2 (193.25). Amorphous brownish solid, 250 dec (MeOH), []D =
(in vitro, HL-60, IC50 > 100g/mL; Bel7402, IC50 > 100g/mL; HeLa, IC50 >
+13 (c = 0.61, Me2CO). Source: GONG XING MA DOU LING Aristolochia
100g/mL; U937, IC50 > 100g/mL; control Colchicine, HL-60, IC50 =
arcuata. Ref: 2037.
1.6g/mL; Bel7402, IC50 = 0.4g/mL; HeLa, IC50 = 0.1g/mL; U937, IC50 =
25
0.1g/mL). Source: LA ZHU GUO Aegiceras corniculatum (stem and twig:
HO
yield = 0.000025%). Ref: 4746.

NH
HO
O
HO
5863 1,3-Dihydroxy-6,7-dimethylxanthone-1-O--D-glucoside
C21H22O9 (418.40). Yellowish massive crystals, mp 262~265C. Source: HE
OH
SHOU WU Polygonum multiflorum. Ref: 292.

HO
5868 1,2-Dihydroxy-8(9)-ene-p-menthane
C10H18O2 (170.25). Yellowish oil. Source: JING JIE Schizonepeta tenuifolia
OO
HO
[Syn. Nepeta tenuifolia]. Ref: 2158.
OH
OH
OH
OH
OH
5864 (E)-4,4'-Dihydroxy-7,7'-dioxolign-8(8')-ene
C18H16O4 (296.33). Off-white powder. Pharm: Antioxidant inactive
(Takamatsu DCFH method, myelomonocytic HL-60 cells, control NDGA,
5869 (13S)-9,18-Dihydroxy-9-epi-10-epi-ryanodine
IC50 = (0.70.3)g/mL, Vitamin C, IC50 = (1.90.7)g/mL, Trolox, IC50 =
C25H35NO11 (525.56). Crystals (CHCl3:Me2CO = 3:1), mp 190C, []D = +10
(1.40.5)g/mL); cytotoxic (XTT assay, HL-60 cells, IC50 > 50.0g/mL;
(c = 0.35). Pharm: Cardiac contraction inhibitor (guinea-pig papillary muscle,
control NDGA, IC50 = (2.60.2)g/mL, Vitamin C, IC50 > 10.0g/mL, Trolox,
causes a prolongation of the latency time and decrease of contraction force,
IC50 > 10.0g/mL). Source: SAN CHI LA RUI A Larrea tridentata (leaf). Ref:
EC50 = 390nmol/L). Source: QU CHONG CAO Spigelia anthelmia (aerial
3850.
parts). Ref: 5139.

O
OH
HO
HO
OH
HO
HO
OH OH
5865 (Z)-4,4'-Dihydroxy-7,7'-dioxolign-8(8')-ene
C18H16O4 (296.33). Pharm: Antioxidant inactive (Takamatsu DCFH method,
myelomonocytic HL-60 cells, control NDGA, IC50 = (0.70.3)g/mL,
OH
N
H
OH
O
Vitamin C, IC50 = (1.90.7)g/mL, Trolox, IC50 = (1.40.5)g/mL); cytotoxic
5870 9,20-Dihydroxy-9-epi-10-epi-ryanodine
(XTT assay, HL-60 cells, IC50 > 50.0g/mL; control NDGA, IC50 =
C25H35NO11 (525.56). Crystals (CHCl3:MeOH = 3:1), mp 178C, []D = +4 (c
(2.60.2)g/mL, Vitamin C, IC50 > 10.0g/mL, Trolox, IC50 > 10.0g/mL).
= 0.1). Source: QU CHONG CAO Spigelia anthelmia (aerial parts). Ref:
Source: SAN CHI LA RUI A Larrea tridentata (leaf). Ref: 3850.
5139.
OH
OH
O
HO
N
H
O
O
OH
OH
HO OH OH
OH
OH
141
5871 4,8-Dihydroxyepipinoresinol
5876 10,19-Dihydroxy-15,16-epoxy-8(17),13(16),14-nor-ent-labdatriene
C20H22O8 (390.39). Amorphous powder, mp 128~130C, []D27 = +36.8 (c =
C19H28O3 (304.43). Colorless oil, [] D25 = 4.1 (c = 0.21, CHCl3). Pharm:
0.29, MeOH). Source: YUN NAN TIE SHAN Tsuga dumosa (heartwood).
Phytotoxin (Raphidocelis subcapitata, IC50 = 2.84mol/L). Source: FU YE
Ref: 4568.
YAN ZI CAI Potamogeton natans. Ref: 5184.

O
OH
OH
HO
H
HO
H
OH
5877 3,4-Dihydroxy-15,16-epoxy-12-oxo-cleroda-13(16),14-dien
C20H30O4 (334.46). Source: Croton hovarum. Ref: 4552.
HO
5872 6,18-Dihydroxy-7,8-epoxy-9-epi-ent-pimara-15-ene
C20H32O3 (320.48). Source: TENG CANG CHI MEI Gibberella fujikuroi. Ref:
3916.
HO
HO
H
HO
5878 3,4-Dihydroxy-15,16-epoxy-12-oxo-cleroda-13(16),14-dien-9-oal
OH
5873 9,18-Dihydroxy-7,8-epoxy-9-epi-ent-pimara-15-ene
C20H32O3 (320.48). Source: TENG CANG CHI MEI Gibberella fujikuroi. Ref:
3916.
O
H
HO
OH
HO
5879 5,17-Dihydroxy-6,7-epoxy-1-oxo-3-O-sulfate-witha-24HO
enolide
C28H40O10S (568.69). mp 158C, []D30 = +59.40 (c = 0.25, MeOH). Source:
5874 3,4-Dihydroxy-3',6'-epoxy-1',2',5',6'7',8'-hexahydro-6'-methyl-16'-
CUI MIAN SHUI QIE Withania somnifera (leaf). Ref: 5329.
nor-,-carotene-1',8'-dione
C40H56O5 (616.89). Reddish solid. Source: MU LI (Oyster) Crassostrea gigas.
Ref: 4515.
O
OH
O
O
O
HO
O
HO
OH
OH
5880 (20S,22R)-5,27-Dihydroxy-6,7-epoxy-1-oxowitha-2,24-dieno5875 19,20-Dihydroxy-15,16-epoxy-8(17),13(16),14-ent-labdatriene
lide
C20H30O3 (318.46). Colorless oil, [] D = 20.4 (c = 0.38, CHCl3). Pharm:
C28H38O6 (470.61). Source: CUI MIAN SHUI QIE Withania somnifera (root).
Phytotoxin (Raphidocelis subcapitata, IC50 = 18.45mol/L). Source: FU YE
Ref: 4198.
25
YAN ZI CAI Potamogeton natans. Ref: 5184.

OH
HO
O
H
HO
OH
H
O
142
5881 1,7-Dihydroxy-4,20-epoxy-2,5,9,10,13-pentaacetoxytax-
5886 1,8-Dihydroxyeudesman-3,7(11)-dien-8,12-olide
11-ene
C15H20O4 (264.32). White needle crystals (MeOH), mp 193~195C. Pharm:
Cytotoxic (in vitro, P388, IC50 = 60g/mL). Source: XIAO MEI WEI QIN
Ref: 662.
Smyrnium olusatrum (fruit). Ref: 5162.

O O
OH
O O
O
O
O
O
O
OH
OH
OH O
5887 1,8-Dihydroxyeudesman-4(15),7(11)-dien-8,12-olide
C15H20O4 (264.32). White prism crystals (MeOH), mp 178~180C. Pharm:
5882 1,9-Dihydroxy-4,20-epoxy-2,5,7,10,13-penta-acetoxytax11-ene
Cytotoxic (in vitro, P388, IC50 = 65g/mL). Source: XIAO MEI WEI QIN
Smyrnium olusatrum (fruit). Ref: 5162.
OH
OH
O
Ref: 662.
O
O
O
O OH
O
O
O
O
OH O
5888 1,4-Dihydroxyeudesman-11-ene
C15H26O2 (238.37). []D17 = 25 (c = 0.13, CHCl3). Pharm: Cytotoxic
(inhibits growth of Bel7402 cell, 0.0001mol/L, InRt = 34.4%, control
Etoposide, InRt = 96.0%). Source: YI NIAN PENG Erigeron annuus (aerial
parts). Ref: 5073.
5883 6,10-Dihydroxyeremophila-7(11),8(9)-dien-12,8-olide
OH
C15H20O4 (264.32). Source: Ligularia virgaurea ssp. oligocephala (whole

herb). Ref: 4981.
HO
OH
5889 1,4-Dihydroxyeudesman-11-ene
C15H26O2 (238.37). Colorless oil, []D17 = 29 (c = 0.13, CHCl3). Source: YI

OH
NIAN PENG Erigeron annuus (aerial parts). Ref: 5073.

OH
5884 3,5-Dihydroxy-(22E)-ergosta-7,22-dien-6-one
C28H44O3 (428.66). Source: Pleurotus eryngii. Ref: 4183.
H
OH
H
5890 3,4-Dihydroxy-5H,11H-eudesman-6,12-olide
C15H24O4 (268.36). Source: Ferula sinaica (leaf). Ref: 5145.
H
HO
OH
O
HO
HO
O
O
5885 3,5-Dihydroxyergost-7-en-6-one
C28H46O3 (430.68). Colorless amorphous solid, []D30 = +28.6 (c = 0.04,
MeOH). Source: Pleurotus eryngii. Ref: 4183.
5891 1,4-Dihydroxyeudesman-5,6,7,11H-12,6-olide
C15H24O4 (268.36). Colorless oil, []D25 = +31 (c = 0.5, CHCl3). Source: JIA
NA LI HAO Artemisia canariensis. Ref: 2332.
H
OH
H
HO
OH
O
H
H
OH
O
O
143
5892 (1R,5S,6S,7S,10R)-1,6-Dihydroxyeudesman-4-one
5897 (3S,6R)-6,7-Dihydroxy-6,7-dihydrolinalool-3-O--D-(3-O-
C14H24O3 (240.35). Colorless oil, []D17 = +25 (c = 0.13, CHCl3). Source: YI
Potassium sulfo)-glucopyranoside
NIAN PENG Erigeron annuus (aerial parts). Ref: 5073.
C16H29O11S (429.47). Amorphous powder, []D21 = 14 (c = 0.3, MeOH).

Source: HU SUI ZI Coriandrum sativum. Ref: 4302.
OH
HO
H
O
O
S
OH
HO
5893 13,21-Dihydroxyeurycomanol
OH
OH
OH
5898 (2E,6E,10E,14Z)-17,20-Dihydroxygeranylnerol
C20H34O3 (322.49). Source: ZHONG BIN JU Tithonia diversifolia (aerial
OH
OH
HO
OH
parts). Ref: 4622.
OH
OH
OH
HO
O
HO
H
O
OH
HO
5894 7,4'-Dihydroxyflavan
(2S)-7,4'-Dihydroxyflavan [82925-54-0] C15H14O3 (242.28). Pharm:
5899 3,17-Dihydroxy-16-[(O--D-glucopyranosyl-(14)-O-(2-O-3,4-
Antibacterial (phytopathogenic bacteria, Corynebacterium betae and
dimethoxybenzoyl--D-xylopyranosyl)-(13)-2-O-acetyl--L-arabinopyr
Corynebacterium fascians); antifungal (Botrytis cinerea, ED50 = 65g/mL);
anosyl)oxy]cholest-5-en-22-one
aromatase inhibitor inactive (in vitro, IC50 > 40mol/L; control
C54H80O21 (1065.23). Pharm: Cytotoxic (HL-60 cells, IC50 = 0.016mol/L).
[3090]
Aminoglutethimide, IC50 = 6.4mol/L)
. Source: GOU SHU Broussonetia
Source: Ornithogalum saundersiae (bulb: yield = 0.00007%). Ref: 3030.
papyrifera[3090]. Ref: 658, 3090.

O
OH
HO
O
H
H
HO
HO
H O HO
5895 4',7-Dihydroxyflavone
[2196-14-7] C15H10O4 (254.24). Source: BAI CI HUA ZI Sophora viciifolia,
OH
H
O
OH
HO
OH
ZHANG GUO GAN CAO Glycyrrhiza inflata, YUN NAN GAN CAO
Glycyrrhiza yunnanensis. Ref: 2, 561, 660.
5900 3,-17-Dihydroxy-16-[(O--D-glucopyranosyl-(14)-O-(2-OOH
HO
3,4,5-trimethoxybenzoyl--D-xylopyranosyl)-(13)-2-O-acetyl--L-arabi
nopyranosyl)oxy]cholest-5-en-22-one
C55H82O22 (1095.25). Pharm: Cytotoxic (HL-60 cells, IC50 = 0.014mol/L).

Source: Ornithogalum saundersiae (bulb: yield = 0.00011%). Ref: 3030.
O
5896 5,4'-Dihydroxyflavone-6-C--D-glycosylrhamnoside-7-O-glycoside
C33H40O19 (740.68). mp 194~196C. Source: HUANG JING Polygonatum
sibiricum. Ref: 6.
HO
OH
OO
OH
OH
OH
O
OO
HO
OH
OH
H
HO
HO
HO HO
O
OH
OH
OH
OH OHOH
OH
HO
O
O
O
O
144
5901 1,3-Dihydroxy-5-O--D-glucopyranosylxanthone-4-sulfonate
5906 (3R,5S)-3,5-Dihydroxy-1-(4-hydroxy-3,5-dimethoxyphenyl)-
C19H17O13S (485.40). Yellow powder, mp > 360C, []D31.2 = +38.10 (c =
7-(4-hydroxy-3-methoxyphenyl)heptane
0.033, MeOH). Pharm: Cytotoxic (P388 cell line, ED50 = 15.69mol/L; control
C22H30O7 (406.48). Colorless oil, []D24 = 0 (c = 0.55, CHCl3). Source:
VP-16, ED50 = 0.064mol/L). Source: YUAN BAO CAO Hypericum
sampsonii (whole herb). Ref: 3861.

O
OH
OH
OH
O
OO
HO
OH
OH
OH
HO
OH
O S O
O
5907 2,3-Dihydroxy-1-(4-hydroxy-3,5-dimethoxyphenyl)-1-propanone
OH
5902 (1S,4S,5R,7R,10R)-11,14-Dihydroxyguai-3-one 11-O--D-glucopyranoside

C21H36O8 (416.52). Colorless needles (MeOH), mp 98~100C, []D22 = +34 (c
C11H14O6 (242.23). Amorphous white powder, []D25 = 0 (c = 0.5, CHCl3).

Source: TIAN XIAN GUO Ficus beecheyana [Syn. Ficus erecta var.
beecheyana] (root: yield = 0.012%dw). Ref: 4657.
= 0.5, MeOH). Source: CANG ZHU Atractylodes lancea, GUAN CANG

ZHU Atractylodes japonica (fresh rhizome). Ref: 4310, 4348.
HO
O
O
OH
OH
HO
O
O
H
HO
OO
OH
5908 2,6-Dihydroxy-4-[(E)-5-hydroxy-3,7-dimethylocta-2,7-dienyloxy]
benzophenone
OH
OH
C23H26O5 (382.46). Yellow amorphous powder, []D25 = 20 (c = 0.2, MeOH).
5903 (3S*,4S*,5R*)-(E)-3,4-Dihydroxy-2-(hexa-2,4-diynyliden)-1,6-di-
Source: YUAN BAO CAO Hypericum sampsonii (whole herb). Ref: 4055.
oxaspiro-(4,5)decane
C14H16O4 (248.28). []D24 = 19.8 (c = 0.22, EtOH). Source: JIN SE MU JU
HO
Matricaria aurea. Ref: 2301.

HO
OH
OH
OH
O
O
5909 2,6-Dihydroxy-4-[(E)-7-hydroxy-3,7-dimethylocta-2-enyloxy]5904 1,3-Dihydroxy-2-hexanoylamino-(4E)-heptadecene
benzophenone
C23H46NO3 (383.62). Colorless gummy solid, []D25 = 19.1 (c = 0.021,
C23H28O5 (384.48). Yellow amorphous powder, []D25 = +30 (c = 0.3, MeOH).
pyridine). Source: QI ZHOU YI ZHI HAO Conyza canadensis [Syn. Erigeron
Source: YUAN BAO CAO Hypericum sampsonii (whole herb). Ref: 4055.
canadensis]. Ref: 4249.

HO
O
N
O
OH
OH
OH
OH
5905 3,3'-Dihydroxy-2-(4-hydroxybenzyl)-5-methoxybibenzyl
C22H22O4 (350.42). Colorless needles. Pharm: Antiallergic -Hexosaminidase
inhibitor (rat basophilic RBL-2H3 cells, inhibits release of -hexosaminidase,
100mol/L, InRt = (98.41.6)mol/L, p<0.01; 300mol/L control Ketotifen
fumarate, InRt = (72.50.9)mol/L, p<0.01). Source: SHOU ZHANG SHEN
5910 5,7-Dihydroxy-3-(3-hydroxy-4-methoxy-benzyl)-6-methoxychroman-4-one
C18H18O7 (346.34). []D20 = 16.0 (c = 0.20, MeOH). Pharm: Angiogenesis
inhibitor (IC50 = 0.5g/mL, control Retinoic acid, IC50 = 0.3g/mL). Source:
DU JUAN LAN Cremastra appendiculata (bulb). Ref: 4937.
Gymnadenia conopsea (tuber). Ref: 5022.

O
HO
OH
O
OH
HO
OH
OH
O
145
5911 1-[2,4-Dihydroxy-3-(3-hydroxy-2-methoxy-3-methylbutyl)-6-meth-
5916 3,7-Dihydroxy-3'-(2-hydroxy-3-methyl-3-butenyl)-5,6,4'-trimeth-
oxyphenyl]-3-(4-hydroxyphenyl)propenone
oxyflavone
C22H26O7 (402.45). Yellow powder. Pharm: Anti-inflammatory (NO
C23H24O8 (428.44). Yellow gummy solid, []D25 = +33.3 (c = 0.03, MeOH).
production inhibitor, in vitro, macrophage RAW264.7 cells, induced by
Pharm: Prolyl endopeptidase inhibitor (flavobacterium origin, IC50 =
LPS/IFN-, IC50 = 6.5mol/L, without showing cytotoxicity at concentrations
(2330.003)mol/L, control Z-pro-prolinal, IC50 = (0.8840.025)mol/L)[4179];
lower than 10mol/L, cell viability > 95%). Source: PI JIU HUA Humulus
thrombin inhibitor inactive (bovine source, control Leupeptin, IC50 =
lupulus (strobile). Ref: 4795.
(45.40.03)mol/L). Source: JIA LIAN QIAO Duranta repens (whole herb).

Ref: 4179.
OH
HO
O
HO
OH
OH
O
O
OH
O
5912 (3R,5R)-3,5-Dihydroxy-1-(4-hydroxy-3-methoxyphenyl)-7-(3,4dihydroxyphenyl)heptane 3-O--D-glucopyranoside

25
OH
5917 5,7-Dihydroxy-3'-(2-hydroxy-3-methyl-3-butenyl)-3,6,4'-trimeth-
oxyflavone
C23H24O8 (428.44). Yellow gummy solid, []D25 = +18.5 (c = 0.05, MeOH).
209g/mL; HGF, IC50 > 250g/mL; control Etoposide: HL-60, IC50 =
Pharm: Prolyl endopeptidase inhibitor (flavobacterium origin, IC50 =
(4500.02)mol/L, control Z-pro-prolinal, IC50 = (0.8840.025)mol/L) ;
yield = 0.0013%dw). Ref: 4609.
HO
HO
Ref: 4179.
HO
OH
OH
HO
OH
HO
OH
O
O
OH
5913 (3R,5R)-3,5-Dihydroxy-1-(4-hydroxy-3-methoxyphenyl)-7-(4-
OH
hydroxyphenyl)heptane 3-O--D-glucopyranoside
5918 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
C19H12O7 (352.30). Light pink granular crystals, mp > 300C. Source: DA
Pharm: Cytotoxic (in vitro, HL-60, IC50 > 10g/mL; HSC-2, IC50 = 160g/mL;
DING CAO Gerbera anandria [Syn. Leibnitzia anandria]. Ref: 141.
HGF, IC50 > 250g/mL; control Etoposide: HL-60, IC50 = 0.2g/mL; HSC-2,
chantrieri [Syn. Tacca minor; Tacca esquirolii] (rhizome: yield = 0.0020%dw).
Ref: 4609.
OH
HO
HO
OH
O
HO
OH
OH
OH
5919 5,4'-Dihydroxy-[2''-(1-hydroxy-1-methylethyl)dihydrofurano](7,8:5'',4'')flavanone
OH
HO
5914 1,8-Dihydroxy-4-hydroxymethyl anthraquinone
C20H20O6 (356.38). Pale yellow solid, []D20 = 99 (c = 0.1, MeOH). Source:

ZHEN YE XUE TONG Macaranga conifera. Ref: 1929.
C15H10O5 (270.24). Source: LEI GONG TENG Tripterygium wilfordii. Ref: 2.

OH
OH
HO
OH
O
OH
5915 3,6-Dihydroxy-2-hydroxymethyl-9,10-anthraquinone
OH
C15H10O5 (270.24). Yellow powder. Source: MA LAI BAN DAO RAN MU
5920 2,3-Dihydroxy-2-(1-hydroxytridecyl)-4-methoxycyclopentanone
SHU Saprosma scortechinii (stem and leaf). Ref: 4219.
C19H36O5 (344.50). Source: Hygrophorus persoonii. Ref: 3800.
OH
OH
HO
O
OH
OH
O
OH
146
5921 7,8-Dihydroxy-isobutyryl-thymol
5926 1,7-Dihydroxy-2-isoprenyl-3-methoxyxanthone
C14H20O5 (268.31). Straw yellow oil. Source: XIAN MAI XUAN FU HUA
1,7-Dihydroxy-3-methoxy-2-(3-methylbut-2-enyl)xanthone C19H18O5 (326.35).
Inula nervosa. Ref: 795.
Pharm: Antioxidant (DPPH scavenger, 10mol/L, ScRt = 15%, control BHT,

10mol/L, ScRt = 43%)[5319]; antibacterial inactive (MRSA)[4735]; cytotoxic (in
vitro, HL-60, IC50 = 23.6mol/L)[4715]; antitubercular (Mycobacterium
OH
OH
tuberculosis,MIC > 200g/mL, inactive)[4358]. Source: DAO NIAN ZI Garcinia
mangostana (fruit), DAO NIAN ZI Garcinia mangostana (fruit hull), HEI
XIAN TIAO TENG HUANG Garcinia nigrolineata (leaf: yield = 0.0001%dw),
OH
TIAN SHAN ZHU ZI Garcinia dulcis (fruit), TIAN SHAN ZHU ZI Garcinia
5922 (1R,2R)-ent-1,2-Dihydroxyisopimara-8(14),15-diene
dulcis (flower). Ref: 3066, 4422, 4358, 4715, 4735, 5319.
C20H32O2 (304.48). Crystals, mp 132~133C, []D20 = 16.5 (c = 2.51). Source:
OH
O
OH
JI RUAN RONG TAI Trichocolea mollissima. Ref: 3489.

O
OH
5927 2,5-Dihydroxy-3-isoprenyl-6-(3-methylbut-3-en-1-ynyl)benza-
HO
ldehyde
H
C17H18O3 (270.33). Source: MAO REN GE JUN Stereum hirsutum. Ref: 3930.
OH
H
O
5923 1,14-Dihydroxyisopimara-7,15-diene
C20H32O2 (304.48). Amorphous powder, []D = 16.0 (c = 0.6, CHCl3).
OH
Pharm: Antifungal (TLC bioautographic assay, plant pathogenic fungus

Cladosporium cucumerinum, MA= 25-50g, yeast Candida albicans, MA=
25-50g). Source: PU FU QIANG DAO YAO Hypoestes serpens. Ref: 3438.
5928 16,17-Dihydroxy-ent-kauran-19-al
C20H32O3 (320.48). Pharm: Antioxidant (inhibits superoxide anion generation,
fMLP/CB, IC50 = (2.771.71)g/mL, control DPI, IC 50 = (0.130.06)g/mL,
p<0.001)[4950]; platelet aggregation selected inhibitor (washed rabbit platelets,
200mol/L: 100mol/L AA induced, InRt = 9.6%; 10g/mL collagen induced,
OH
InRt = 17.6%; 1ng/mL PAF induced, InRt = 5.5%; 0.05U/mL thrombin
OH
induced, InRt = 0.0%)[4654]. Source: FAN LI ZHI Annona squamosa (stem:

yield = 0.0010%fw). Ref: 4950, 4654.
OH
OH
5924 3,19-Dihydroxy-8(9),15-isopimaradien-7-one
25
C20H30O3 (318.46). Colorless oil, []D = +52 (c = 0.06, CHCl3). Source: CE
BAI ZHI JIE Thuja orientalis [Syn. Platycladus orientalis; Biota orientalis]
(branch). Ref: 3022.
H
O
5929 16,17-Dihydroxy-ent-kauran-19-al
C20H32O3 (320.48). Pharm: Platelet aggregation inhibitor inactive (washed
rabbit platelets, 200mol/L: 100mol/L AA induced, InRt = 0.5%; 10g/mL
collagen induced, InRt = 4.9%; 1ng/mL PAF induced, InRt = 10.3%;
HO
0.05U/mL thrombin induced, InRt = 3.2%)[4654]; antioxidant (inhibits
superoxide anion generation, fMLP/CB, IC50 = (6.493.31)g/mL, control DPI,
HO
IC50 = (0.130.06)g/mL, p<0.001) [4950]; antiproliferative and cytotoxic (in vitro,
5925 1,5-Dihydroxy-2-isoprenyl-3-methoxyxanthone
L-929, GI50 = 50g/mL; K562, GI50 = 50g/mL; HeLa, CC50 = 50g/mL;
1,5-Dihydroxy-3-methoxy-2-(3-methylbut-2-enyl)-xanthone C19H18O5
control Paclitaxel, L-929, GI50 = 0.1g/mL; K562, GI50 = 0.01g/mL; HeLa,
(326.35). Pharm: Antibacterial inactive (MRSA). Source: DAO NIAN ZI
CC50 = 0.01g/mL)[4770]. Source: FAN LI ZHI Annona squamosa (stem: yield
Garcinia mangostana (fruit hull), HEI XIAN TIAO TENG HUANG Garcinia
= 0.0012%fw), MU LAN
nigrolineata (leaf: yield = 0.0008%dw). Ref: 3066, 4735.
Ref: 4654, 4770, 4950.
(3)
OH
OH
O
H
O
OH
OH
Bruguiera gymnorrhiza (stem: yield = 0.00011%).
147
5930 ()-16,17-Dihydroxy-16-kauran-19-oic acid
5934 ent-11,15-Dihydroxy-16-kaurene
Diterpenoid SP II C20H32O4 (336.48). mp 260~262C. Pharm:
C20H32O2 (304.48). Pharm: Cytotoxic inactive (hmn leukemia cell HL-60,
Antihypertensive (rat, orl, 50mg/(kgd)); anti-inflammatory (caused by
10mol/L). Source: JIE XING YE TAI Jungermannia truncata. Ref: 4201.
formalin, 300mg/kg orl, regression of edema 38%, caused by protein,

300mg/kg orl, regression of edema 53%); antioxidant (inhibits superoxide
HO
anion generation, fMLP/CB, IC50 = (3.070.33)g/mL, p<0.001, control DPI,

IC50 = (0.130.06)g/mL, p<0.001)[4950]; platelet aggregation inhibitor
OH
inactive (washed rabbit platelets, 200mol/L: 100mol/L AA induced, InRt =
7.2%; 10g/mL collagen induced, InRt = 2.3%; 1ng/mL PAF induced, InRt =
8.9%; 0.05U/mL thrombin induced, InRt = 0.4%)[4654]. Source: JIAO XI
XIAN Siegesbeckia gummifer, TU DANG GUI Aralia cordata, XIAN GENG
XI XIAN Siegesbeckia orientalis var. pubescens [Syn. Siegesbeckia
C20H32O2 (304.48). Amorphous, []D22 = 48.5 (c = 2.89). Source: JIE XING

[4654]
pubescens], FAN LI ZHI Annona squamosa (stem: yield = 0.00047%fw)
YE TAI Jungermannia truncata. Ref: 4201.
Ref: 2, 6, 658, 660, 661, 4654, 4950.

OH
OH
OH
OH
H
O
OH
5931 16,17-Dihydroxy-ent-kauran-19-oic acid

C20H32O4 (336.48). Pharm: Cytotoxic inactive (Lu1, Col2, KB, LNCaP,
hTERT-RPE1, HUVEC; control Taxol, ED50 = 0.002g/mL, 0.003g/mL,
0.0005g/mL, 0.001g/mL, 0.004g/mL, 0.008g/mL, respectively). Source:
CHCl3). Pharm: Cytotoxic (BST test, weak active). Source: DONG JIN BA
Parinari sprucei (leaf). Ref: 4991.
DOU Croton tonkinensis (leaf). Ref: 4444.
OH
OH
H
HO
H
HO
OH
5932 16,17-Dihydroxy-ent-kauran-19-oic acid

C20H32O4 (336.48). Pharm: Antioxidant (inhibits superoxide anion generation,
5937 16,17-Dihydroxy-ent-9(11)-kauren-19-oic acid
fMLP/CB, IC50 = (0.790.14)g/mL, p<0.001, control DPI, IC 50 =
C20H30O4 (334.46). Source: MU LAN
[4950]
(0.130.06)g/mL, p<0.001)
platelet aggregation inhibitor inactive
(3)
Bruguiera gymnorrhiza (stem: yield
= 0.00075%) Ref: 4770.
(washed rabbit platelets, 200mol/L: 100mol/L AA induced, InRt = 14.9%;

10g/mL collagen induced, InRt = 8.6%; 1ng/mL PAF induced, InRt = 14.4%;
OH
OH
0.05U/mL thrombin induced, InRt = 6.8%)[4654]. Source: FAN LI ZHI Annona

squamosa (stem: yield = 0.0013%fw). Ref: 4950, 4654.
HO
O
OH
OH
H
5938 7,12-Dihydroxykaurenolide
C20H28O4 (332.44). Pharm: Plant growth regulator. Source: XI HU LU
OH
Cucurbita pepo. Ref: 658.
5933 16,17-Dihydroxy-ent-9(11)-kauren-19-al
C20H30O3 (318.46). White amorphous solid, []D20 = +4.8 (c = 0.3, CHCl3).
Source: MU LAN
(3)
OH
Bruguiera gymnorrhiza (stem: yield = 0.00028%) Ref:
4770.
H
OH
OH
H
O
H
O
OH
O
148
5939 7,14-Dihydroxykaur-16-en-15-one
5943 ent-8,9-Dihydroxylabda-13(16),14-dien-1-one
C20H32O3 (320.48). Colorless oil, [] D20 = +13.6 (c = 0.21, CHCl3). Source:
(c = 0.3, CHCl3). Pharm: Anti-inflammatory (inhibits LPS-induced NF-B
JIE MAO TAI Blepharostoma trichophyllum. Ref: 3843.
activation in murine macrophage RAW264.7 cells, IC50 = 0.11mol/L; control

Parthenolide, IC50 = 2.34mol/L); NO production inhibitor (IC50 =
0.26mol/L; control Parthenolide, IC50 = 2.01mol/L). Source: DONG JIN
BA DOU Croton tonkinensis (leaf: yield = 0.00054%dw). Ref: 4724.
O
OH
OH
OH
O
OH
5940 ent-7,18-Dihydroxykaur-16-en-3-one
5944 12,17-Dihydroxylabda-13(E)-ene
C20H30O3 (318.46). Syrup, []D = 45.8 (c = 0.5, CHCl3). Source: MU ER
C20H36O2 (308.51). mp 161~163C, []D20 = 15.42 (c = 1.18, CHCl3).
DU MA CAO Sideritis moorei (aerial parts). Ref: 5295.
Pharm: Cytotoxic inactive (in vitro, BT474, CHAGO, HepG2, Kato3,

SW620: > 10g/mL). Source: GUANG YE BA DOU Croton oblongifolius
[Syn. Croton laevigatus]. Ref: 5363.
O
HO
OH
OH
5941 14,15-Dihydroxyklaineanone
OH
C20H28O8 (396.44). Pharm: Cytotoxic (KB cells, IC50 = 0.38g/mL, P388 cells,
IC50 = 0.29g/mL)[4556]; plant growth inhibitor (Cucumber seedling, root
growth, IC50 = (2.50.5)mol/L, shoot growth, IC50 = (22.70.5)mol/L; Rice
seedling, root growth, IC50 > 200mol/L, shoot growth, IC50 >
200mol/L)[5215]. Source: CHANG YE KUAN MU Eurycoma longifolia (leaf),
Eurycoma sp. Ref: 4556, 5215.
5945 2,3-Dihydroxy-labda-8(17),12(E),14-triene
C20H32O2 (304.48). White solid, mp 69~70C, []D20 = 6.96 (c = 1.0, CHCl3).
Pharm: Cytotoxic (Kato3, IC50 = 2.2g/mL, control Doxorubicin
hydrochloride, IC50 = 1.7g/mL; SW620, IC50 = 2.7g/mL, Doxorubicin
OH
HO
OH
hydrochloride, IC50 = 1.1g/mL; BT474, IC50 = 4.6g/mL, Doxorubicin

OH
OH
O
H
hydrochloride, IC50 = 0.08g/mL; HepG2, IC50 = 3.7g/mL, Doxorubicin

hydrochloride, IC50 = 0.9g/mL; CHAGO, IC50 = 3.3g/mL, Doxorubicin
hydrochloride, IC50 = 2.3g/mL). Source: GUANG YE BA DOU Croton
oblongifolius [Syn. Croton laevigatus] (stem cortex). Ref: 5121.
5942 12,17-Dihydroxylabda-7,13(E)-diene
C20H34O2 (306.49). mp 109~111C, []D20 = 7.55 (c = 1.06, CHCl3). Pharm:
HO
Cytotoxic (in vitro, BT474, IC50 = 2.5g/mL, control Doxorubicin

hydrochloride, IC 50 = 0.08g/mL; CHAGO, IC50 = 6.1g/mL, Doxorubicin
HO
hydrochloride, IC 50 = 2.3g/mL; HepG2, IC50 = 5.3g/mL, Doxorubicin

hydrochloride, IC 50 = 0.9g/mL; Kato3, IC50 = 0.6g/mL, Doxorubicin
hydrochloride, IC 50 = 1.7g/mL; SW620, IC50 = 6.1g/mL, Doxorubicin
hydrochloride, IC 50 = 1.1g/mL). Source: GUANG YE BA DOU Croton
oblongifolius [Syn. Croton laevigatus]. Ref: 5363.
5946 26,27-Dihydroxy-lanosta-7,9(11),24-trien-3,16-dione
C31H46O4 (482.71). mp 136~139C. Source: LING ZHI Ganoderma lucidum.
Ref: 2235.
H
OH
OH
OH
O
OH
149
5947 3,9-Dihydroxylanost-24-en-26-ol
5952 3,23-Dihydroxy-lup-20(29)-ene-28-O--L-rhamnopyranosyl-
C30H50O3 (458.73). White amorphous powder, []D27 = +5.0 (c = 0.003,
(14)--D-glucopyranosyl-(16)--D-glucopyranoside
CHCl3). Source: MEI LI TENG HUANG Garcinia speciosa (bark). Ref:
C47H78O17 (915.14). Source: BAI TOU WENG Pulsatilla chinensis. Ref: 2.
3762.
O
H
H
OH
HO
OO
HO
HO
OH
H
OH
OH
OO
5948 (7,8-cis-8,8'-trans)-2',4'-Dihydroxyl-3,5-dimethoxyl-lariciresinol
C20H24O6 (360.41). Light-brown powder, mp 220~223C (dec). Source: FEI
O
OH
OH
OH
OH
OH OH
SHU Torreya grandis (aril). Ref: 4836.
5953 2,3-Dihydroxylup-20(29)-en-28-oic acid
OH
C30H48O4 (472.71). Source: SAN YE MU TONG Akebia trifoliata (stem). Ref:

O
4545.
HO
OH
O
5949 5,4'-Dihydroxyl-6,7-dimethoxyl-8-C-[-D-xylocopyranosyl-(12)]-
HO
-D-glucopyranosyl flavone
OH
H
25
C28H32O15 (608.56). Yellow amorphous powder, mp 173~175C, []D =
HO
44.9 (c = 0.60, MeOH). Source: SHI DAN CAO Corallodiscus flabellatus

[Syn. Didissandra flabellat] (whole herb). Ref: 4830.
O
5954 12,19-Dihydroxymanoyl oxide

8,13-Epoxy-14-labdene C20H34O3 (322.49). Amorphous, []D26 = +13.1 (c =
OH
0.21, CHCl3). Source: TAI WAN SHAN MU Cunninghamia konishii (wood).
Ref: 4176.
O
HO
HO
OH
O
OH
OH
OO
OH
HO
OH
OH
5955 5,9-Dihydroxymatrine
5950 1,8-Dihydroxy-3-(3'-hydroxy-butoxy) xanthone
[72362-00-6] C15H24N2O3 (280.37). Source: XI XIAN Siegesbeckia orientalis.
C17H16O6 (316.31). Yellow columnar crystals (CHCl3MeOH), mp 269~270C.
Ref: 2.
Source: CHUAN DONG ZHANG YA CAI Swertia davidii. Ref: 2480.

OH
OH
OH
O
N
HO
5951 3,23-Dihydroxy-lup-20(29)-ene-28-O--D-glucopyranosyl-(16)C41H68O13 (768.99). Source: BAI TOU WENG Pulsatilla chinensis. Ref: 2.
H
N
-D-glucopyranoside
H
OH
5956 (3R,6R,7E,9R)-3,9-Dihydroxy-4,7-megastigmadiene
C13H22O2 (210.32). Colorless oil, [] D25 = +25.9 (c = 0.53, CH2Cl2). Pharm:
Phytotoxin (inhibits germination and growth of Lactuca sativa)[3776]. Source:
PA KE YE XIANG SHU Cestrum parqui (leaf). Ref: 3776.

H
H
HO
H
OH
HO
OO
OH
OH
HO H
O
OH
OH
OH
OH
HO
150
5957 (3S,7E,9R)-3,9-Dihydroxy-5,7-megastigmadiene
5963 3,5-Dihydroxy-4-methoxybenzoic acid
C13H22O2 (210.32). Colorless oil, [] D25 = 97.9 (c = 0.48, CH2Cl2). Pharm:
C8H8O5 (184.15). Source: DIAN NAN HONG HOU KE Calophyllum
Phytotoxin (inhibits germination and growth of Lactuca sativa). Source: PA
polyanthum (seed: yield = 0.0022%dw). Ref: 4767.

O
KE YE XIANG SHU Cestrum parqui (leaf). Ref: 3776.
OH
HO
HO H
O
HO
OH
5964 3,4-Dihydroxy-5-methoxybenzoic acid methyl ester-4-sulfate
5958 (2R,6R,9R)-2,9-Dihydroxy-4-megastigmen-3-one
C13H22O3 (226.32). Colorless oil, [] D25 = +102.7 (c = 0.56, CH2Cl2). Pharm:
C9H9O8S (277.23). Amorphous powder. Source: HU ZHANG Polygonum

cuspidatum. Ref: 4186.

OH
HO
HO
O
O
O
S
5959 (3R,4R,6S)-3,6-Dihydroxy-1-menthene
C10H18O2 (170.25). Colorless needles, mp 166~168C (CH3OH). Pharm:
5965 2,6-Dihydroxy-4-methoxybenzophenone
Antibacterial (Staphylococcus aureus, antibacterial circle < 12mm; Bacillus
Cotoin C14H12O4 (244.25). Source: DUO ZHI ZHI TENG HUANG Garcinia
subtilis, antibacterial circle = 13~16mm; Escherichia coli, antibacterial
virgata (stem cortex). Ref: 3874.
circle > 17mm). Source: JIAN YE TOU WU GEN Ligularia sagitta. Ref:
OH
5382.
OH
HO
HO
5966 rel-1-(4,6-Dihydroxy-2-methoxy)-benzoyl-rel-2-(2,6-dimethoxy4-hydroxy)-benzoyl-rel-(3,4)-diphenylcyclobutane
5960 2,4'-Dihydroxy-3'-methoxyacetophenone
C33H30O8 (554.60). Yellowish amorphous solid, mp 210C, []D21 = +19.3 (c
= 0.1, MeOH). Source: BAI DIAN FENG CHE ZI Combretum albopunctatum
OH

O
O
O
O
HO
OH
OH
O
OH
5961 1,6-Dihydroxy-2-methoxyanthraquinone
C15H10O5 (270.24). Orange-red needles, mp 178~180C. Source: BA JI TIAN
Morinda officinalis. Ref: 8.
O
OH
5967 3-(,4-Dihydroxy-3-methoxybenzyl)-4-(hydroxy-3-methoxybenzyl)
tetrahydrofuran
C20H24O6 (360.41). Yellow colloid. Source: YUN NAN HAN XIAO Michelia
HO
O
5962 3,9-Dihydroxy-4-methoxy-benzo[4,5]furo[3,2-c]chromen-6-one
HO
OH
C16H10O6 (298.25). Brown amorphous solid. Source: SHUI LIU DOU

Pongamia pinnata (fruit). Ref: 3767.
5968 2',6'-Dihydroxy-4'-methoxychalcone
O
HO
OH
C16H14O4 (270.29). mp 161~162C. Source: ZHEN CAI Litsea pungens. Ref: 6.

OH
O
OH
OH
151
5969 2',6'-Dihydroxy-4'-methoxydihydrochalcone
5974 1,5-Dihydroxy-3-methoxy-6',6'-dimethyl-2H-pyrano(2',3':6,7)-4-
C16H16O4 (272.30). Pharm: Germination inhibitor (spores of Pityrogramma
(3-methylbut-2-enyl)xanthone
calomelanos, 50mol/L). Source: DIAO ZHANG GEN PI Lindera umbellata
C24H24O6 (408.46). Yellow needles, mp 217~218C. Source: YUN NAN
[Syn. Lindera erythrocarpa], LIU HUANG TIE XIAN JUE Adiantum
SHAN ZHU ZI Garcinia cowa (stem: yield = 0.0008%dw). Ref: 916.
sulphureum, Notholaena sp. Ref: 658.

O
O
OH
OH
O
OH
OH
5970 4,7-Dihydroxy-2-methoxy-9,10-dihydro-phenanthrene
5975 2,7-Dihydroxy-8-methoxy-3,6-diundecyldibenzofuran-1,4-dione
(stem). Ref: 5171.
C35H52O6 (568.8). Dark red solid (CHCl3), mp 65~66C. Pharm: Cytotoxic

inactive (in vitro, HL-60, IC50 > 100g/mL; Bel7402, IC50 > 100g/mL; HeLa,
OH
IC50 > 100g/mL; U937, IC50 > 100g/mL; control Colchicine, HL-60, IC50 =
OH
5971 5,4'-Dihydroxy-2'-methoxy-8-(3,3-dimethylallyl)-2'',2''-dimethylpyrano[5,6:6,7]isoflavanone

yield = 0.00005%). Ref: 4746.
O
20
C26H28O6 (436.51). Yellow oil, []D = 7.6 (c = 0.1, MeOH). Source: CI
OH
TONG Erythrina variegata [Syn. Erythrina indica] (stem cortex: yield =

0.00001%fw). Ref: 2269.
HO
O
O
5976 2,8-Dihydroxy-7-methoxy-3,9-diundecyldibenzofuran-1,4-dione
C35H52O6 (568.8). Dark red solid (CHCl3), mp 88~89C. Pharm: Cytotoxic
inactive (in vitro, HL-60, IC50 > 100g/mL; Bel7402, IC50 > 100g/mL; HeLa,
OH
IC50 > 100g/mL; U937, IC50 > 100g/mL; control Colchicine, HL-60, IC50 =
O
OH

5972 5,2'-Dihydroxy-3-methoxy-6,7-(2'',2''-dimethylchromene)-8-
yield = 0.000058%). Ref: 4746.
(3''',3'''-dimethylallyl)-flavanone
Jayacanol 3-methyl ether C26H28O6 (436.51). Pale yellow crystals (methanol),
mp 128.8~129.2C, []D20 = 12.69 (c = 0.670 , CH2Cl2). Source:
HO
OH
Lonchocarpus atropurpureus. Ref: 2423.

O
O
O
HO
5977 8,10-Dihydroxy-6-methoxyeremophil-7(11)-en-12,8-olide
C16H24O5 (296.37). Colorless plates, mp 181~182C (Me2CO). Source: JIAN

YE TOU WU GEN Ligularia sagitta. Ref: 5382.
O
OH
OH
5973 4',5''-Dihydroxy-6''-methoxy-4'',4''-dimethyl-4'',5''-dihydro-
OH
O
6''H-pyrano[2'',3'':7,8]-isoflavone
C21H20O6 (368.39). White amorphous powder, mp 226~228C, []D25 = 12 (c =

O
0.05, MeOH). Pharm: Cytotoxic (KB, IC50 > 75mol/L, control Helenalin, IC50 =
(0.640.08)mol/L, Melphalan, IC50 = (6.00.5)mol/L; Mono-Mac-6, IC 50 >
75mol/L, Helenalin, IC50 = (3.10.3)mol/L; Jurkat-T, IC50 > 75mol/L,
5978 (2S),3',4'-Dihydroxy-7-methoxy flavan
Helenalin, IC50 = (1.140.08)mol/L, Melphalan, IC50 = (9.10.8)mol/L).
C16H16O4 (272.30). Amorphous powder. Source: LIN JING ZHONG ZI WEN
Source: Bituminaria morisiana (leaf). Ref: 5077.
SHU LAN Crinum bulbispermum (bulb). Ref: 3997.

OH
OH
HO
O
OH
O
O
O
152
5979 (2S)-4',7-Dihydroxy-3'-methoxyflavan
5983 4,5-Dihydroxy-7-methoxyflavonol 3-O--D-xylopyranosyl-(12)-
C16H16O4 (272.30). Source: LONG XUE SHU Dracaena draco (stem cortex).
O-[-L-rhamnopyranosyl-(16)]--D-glucopyranoside
Ref: 4696.
C33H40O19 (740.68). Pale-yellow amorphous powder, []D24 = 47.6 (c = 0.21,

CHCl3MeOH, 1:1). Pharm: Cytotoxic inactive (HSC-2, HGF). Source: YE
XIANG SHU Cestrum nocturnum (leaf: yield = 0.0044%fw). Ref: 3023.
HO
OH
OH
5980 (2S)-7,2'-Dihydroxy-5-methoxyflavanone 7-O--D-glucuronopyranoside
OH
C22H22O11 (462.41). Colorless needles (MeOH), mp 190~191C (dec), []D25
HO
= 116.8 (c = 0.052, MeOH). Source: KE AI HUANG QIN Scutellaria
HO
amabilis (root: yield = 0.0052%dw). Ref: 2072.
O O
HO
HO
HO
OO
HO HO
OH
HO
OH
5984 7,6'-Dihydroxy-3'-methoxyisoflavone
C16H12O5 (284.27). Yellowish crystals (Me2CO), mp 250~252C. Source: TU
OO
OH
OH
FU LING Smilax glabra. Ref: 416.

OH
HO
5981 5,4'-Dihydroxy-7-methoxyflavone-3-O-[-L-rhamnopyranosyl
(13)-O--L-rhamnopyranosyl(16)-O--D-glucopyranoside]
O
HO
C34H42O19 (754.70). Yellow powder, mp 210~212C, []D20 = 41.99 (c = 0.5,

MeOH). Pharm: Inhibitory activity against NFAT transcription (IC50 >
100mol/L, control Cyclosporin A, IC50 = (0.290.01)mol/L). Source:
5985 4,7-Dihydroxy-5-methoxyl-6-methyl-8-formyl-flavan
HUA CHA BIAO Ribes fasciculatum var. chinense. Ref: 2536.
C18H18O5 (314.34). Yellowish rhomboid crystals, mp 137~139C. Source: JIA

YING ZHAO Desmos cochinchinensis [Syn. Desmos chinensis]. Ref: 121.
OH
O
HO
OH O
OH
OO
OH
OH
O OH
OH
OH
5986 5,7-Dihydroxy-6-methoxy-3-(4-methoxybenzyl)chroman-4-one
OH
C18H18O6 (330.34). Yellow vitreous solid, []D = 100 (c = 0.025 , MeOH).

Source: Scilla dracomontana. Ref: 2327.
OH OH
HO
5982 4,5-Dihydroxy-7-methoxyflavonol 3-O-[6-O-(E)-3,5-dimethoxy-4hydroxycinnamoyl--D-glucopyranosyl]-(12)-O-[-L-rhamnopyranos-
O
OH
yl-(16)]--D-glucopyranoside
C45H52O24 (976.9). Pale-yellow amorphous powder, []D24 = 29.2 (c = 0.26,
CHCl3-MeOH, 1:1). Pharm: Cytotoxic inactive (HSC-2, HGF). Source: YE
XIANG SHU Cestrum nocturnum (leaf: yield = 0.0062%fw). Ref: 3023.
C18H14O8 (358.31). Pharm: NO production inhibitor (LPS-induced,

concentration-dependent manner, IC50 = 61.6mol/L or 40.4mol/L); PGE2
production inhibitor (LPS-induced, concentration-dependent manner, IC50 =
OH
32.8mol/L or 30.3mol/L). Source: XIAO YE JU HAO Tanacetum
5987 5,3'-Dihydroxy-4'-methoxy-7-methoxycarbonylflavonol
microphyllum (aerial parts). Ref: 4918.

OH
OH
O
HO
HO
HO
O O
HO
O
HO
HO
HO
O
O
O
O
HO
OH
OH
OH
153
5988 2,4-Dihydroxy-6-methoxy-3-methylacetophenone
5994 3,8-Dihydroxy-4-methoxy-2-oxo-2H-1-benzopyran-5-carboxylic
C10H12O4 (196.20). Light brown acicular crystals, mp 190C Source: YUE
acid
XIAN DA JI Euphorbia ebracteolata. Ref: 678.
C11H8O7 (252.18). Yellowish acicular crystals, mp 277~279C. Source: DA

DING CAO Gerbera anandria [Syn. Leibnitzia anandria]. Ref: 141.
OH
OH
OH
OH
O
5989 2,4-Dihydroxy-6-methoxy-3-methylacetophenone-4-O--D-glu-
HO
copyranoside
5995 6,7-Dihydroxy-3-methoxy-8-[2-oxo-2H-1-benzopyran-7-(O--
C16H22O9 (358.35). Hoar acicular crystals, mp 198C. Source: YUE XIAN DA
D-glucopyranosyl)-8-yl]-2H-1-benzopyran-2-one
JI Euphorbia ebracteolata. Ref: 678.
Gulsamanin C25H22O13 (530.45). mp 192~193C. Source: YOU RUI XIANG

Daphne oleoides. Ref: 2278.
HO
OH
HO
HO
HO
OO
OH
OH
OH
OO
OH
OH
OH
5990 1,3-Dihydroxy-2-methoxymethylanthraquinone
5996 5,8-Dihydroxy-2-[2-(4'-methoxyphenyl) ethyl]chromone
C16H12O6 (300.27). Source: GUANG JING QIAN CAO Rubia wallichiana
C18H16O5 (312.33). Colorless acicular crystals, mp 172~180C. Source: BAI
(stem). Ref: 4369.
MU XIANG Aquilaria sinensis. Ref: 13.
OH
OH
OH
O
OH
O
OH
5991 7,3'-Dihydroxy-4'-methoxy-8-methylflavan
5997 2-(3',5'-Dihydroxy-4'-methoxyphenyl)-3-methoxy-5-hydroxy
[87733-81-1] C17H18O4 (286.33). Pharm: Larvacide (larva of Eurema hecabe
benzofuran
mandarina, antifeedant). Source: LONG XUE SHU Dracaena draco (stem
C16H14O6 (302.29). Colorless acicular, mp 219~221C. Source: XIAO YE
cortex)
[4696]
, SHI SUAN Lycoris radiata [Syn. Amaryllis radiata]. Ref: 658,
MAI MA TENG Gnetum parvifolium [Syn. Gnetum indicum]. Ref: 193.

O
HO
4696.
O
OH
HO
OH
O
OH
5998 14,18-Dihydroxy-13-methoxy-8,11,13-podocarpatriene
5992 1,6-Dihydroxy-3-methoxy-8-methylxanthone
C18H26O3 (290.41). Yellow amorphous solid, []D18 = +5.3 (c = 0.42, CHCl3).
C15H12O5 (272.26). Yellow powder, mp 210~212C (dec). Source: HE CAO
Source: TAI WAN SHAN Taiwania cryptomerioides (bark). Ref: 4182.

O
YE JIA BEI FANG FENG Ledebouria graminifolia (tuber). Ref: 3368.

O
OH
OH
H
HO
HO
5999 1,14-Dihydroxy-13-methoxy-8,11,13-podocarpatriene-2,7-dione
5993 1,8-Dihydroxy-5-methoxy-3-methylxanthone
C18H22O5 (318.37). Yellow amorphous solid, []D24 = 35.0 (c = 0.17,
C15H12O5 (272.26). Yellow needles (CHCl3), mp.214~215C. Source: RI BEN
CHCl3). Source: TAI WAN SHAN Taiwania cryptomerioides (bark). Ref:
XIAO HE YI Pyrenula japonica, Ref: 2362.
4182.
OH
OH
OH
O
OH
O
O
154
6000 3,14-Dihydroxy-13-methoxy-8,11,13-podocarpatrien-7-one
6004 2',7-Dihydroxy-4'-methoxy-8-prenylflavan 2',7-di-O--D-gluco-
C18H24O4 (304.39). Yellow amorphous solid, []D24 = 9.4 (c = 0.35, CHCl3).
pyranoside
C33H44O14 (664.71). Amorphous powder, []D = 91.1 (c = 0.25, MeOH).

Pharm: Antioxidant (hmn LDL, inhibits CuSO4-induced oxidation of hmn
LDL, 10.0nmol/mL, relative lag time = 0.850.07, positive control Quercetin,
0.5nmol/mL, assigned relative lag time = 1.0)[3507]; DPPH scavenger (IC50 =
505nmol/mL, positive control Quercetin, IC50 = 3.7nmol/mL)[3507]. Source:

OH
HO
SANG YE Morus alba (leaf: yield = 0.0013%), SANG BAI PI Morus alba.
Ref: 3507, 2513.
O O
HO
OH
6001 (2S)-2',4'-Dihydroxy-7-methoxy-8-prenylflavan
C21H24O4 (340.42). Pharm: Aromatase inhibitor inactive (in vitro, IC50 >
40mol/L; control Aminoglutethimide, IC50 = 6.4mol/L). Source: GOU SHU
OO
HO
OH
O OH
OH
OH
Broussonetia papyrifera. Ref: 3090.
OH
6005 (4S)-4,8-Dihydroxy-5-methoxy--tetralone
C11H12O4 (208.22). Source: DONG BEI HU TAO Juglans mandshurica var.
OH
O
sieboldiana (fruit). Ref: 4492.
O
OH
OH
H
OH
6002 2',4'-Dihydroxy-7-methoxy-8-prenylflavan
C21H24O4 (340.42). Amorphous powder, []D = 1.6 (c = 1.0, MeOH). Pharm:
Antioxidant (hmn LDL, inhibits CuSO4-induced oxidation of hmn LDL,
0.5nmol/mL, relative lag time = 0.810.10, positive control Quercetin,
[3507]
0.5nmol/mL, assigned relative lag time = 1.0)
; DPPH scavenger (IC50 =
603nmol/mL, positive control Quercetin, IC50 = 3.7nmol/mL)
[3507]
. Source:
6006 (4R)-5,8-Dihydroxy-4-methoxy--tetralone
C11H12O4 (208.22). Amorphous powder, []D = 0 (CHCl3). Source: DONG
BEI HU TAO Juglans mandshurica var. sieboldiana (fruit). Ref: 4492.
SANG BAI PI Morus alba, SANG YE Morus alba (leaf: yield = 0.0003%).
Ref: 2513, 3507.
HO
O
OH
OH
OH
6007 (4S)-5,8-Dihydroxy-4-methoxy--tetralone
C11H12O4 (208.22). Amorphous powder, []D = 0 (CHCl3). Source: DONG
BEI HU TAO Juglans mandshurica var. sieboldiana (fruit). Ref: 4492.
6003 2',7-Dihydroxy-4'-methoxy-8-prenylflavan
C21H24O4 (340.42). Amorphous powder, []D = 5.5 (c = 1.0, MeOH). Pharm:
OH
OH
Antioxidant (hmn LDL, inhibits CuSO4-induced oxidation of hmn LDL,

0.5nmol/mL, relative lag time = 1.700.25, positive control Quercetin,
0.5nmol/mL, assigned relative lag time = 1.0)[3507]; DPPH scavenger (IC50 =
137nmol/mL, positive control Quercetin, IC50 = 3.7nmol/mL)[3507]. Source:
SANG YE Morus alba (leaf: yield = 0.0018%), SANG BAI PI Morus alba.
Ref: 2513, 3507.
HO
6008 2,3-Dihydroxy-4-methoxy-6,6,9-trimethyl-6H-dibenzo[b,d]pyran
C17H17O4 (286.33). Oil. Pharm: Anti-HIV-1 (binds to chemokine receptor
CCR5, IC50 = 33mol/L). Source: Wigandia urens (stem). Ref: 3474.
OH
HO
OH
O
155
6009 1,3-Dihydroxy-2-methoxy xanthone
6015 1,4-Dihydroxy-2-methylanthraquinone
C14H10O5 (258.23). Colorless acicular crystals (chloroformmethanol), mp
[2589-39-1] C15H10O4 (254.24). Pharm: Anthelmintic (termites). Source: YOU
162~164C, mp 174~176C, mp 176~178C. Source: HUANG HUA YUAN
MU Tectona grandis. Ref: 658.
ZHI Polygala arillata, JIA HUANG HUA YUAN ZHI Polygala fallax [Syn.
OH
OH
Polygala aureocauda] (root and stem: yield = 0.00043%)[4683]. Ref: 382,

4683.
O
OH
O
OH
[21891-63-4] C15H14O4 (254.24). Orange red crystals. Source: CANG BAI
6010 1,6-Dihydroxy-7-methoxyxanthone
CHENG GOU FENG Diploclisia glaucescens, SI SHI MAO DI HUANG
Digitalis schischkinii, DONG FANG YANG DI HUANG Digitalis orientalis,
GAN XI SHU WEI CAO Salvia przewalskii, YI DA LI JUE MING ZI Cassia
italika. Ref: 2100, 2102, 2104, 2105, 2270.
linii. Ref: 4094.

O
OH
OH
O
O
HO
6011 1,7-Dihydroxy-3-methoxy xanthone

Gentisin [437-50-3] C14H10O5 (258.23). mp 266~267C. Pharm: Mutagen
(Salmonella typhimurium). Source: BA XI HU TONG Calophyllum
brasiliense, HUANG LONG DAN Gentiana lutea, TIE LI MU Mesua ferrea,
YUAN ZHI Polygala tenuifolia, ZHANG YA CAI Swertia pseudochinensis,
ZHEN YE TENG HUANG Garcinia eugenifolia. Ref: 2, 6, 658.
O
OH
C15H10O4 (254.24). Pharm: Cytotoxic (KB, ED50 > 25g/mL, control
Doxorubicin, ED50 = 0.12g/mL; Hep3B, ED50 > 25g/mL, Doxorubicin,
ED50 = 0.14g/mL; Colon205, ED50 > 25g/mL, Doxorubicin, ED50 =
0.10g/mL; HeLa, ED50 > 25g/mL, Doxorubicin, ED50 = 0.11g/mL).
Source: GUANG JING QIAN CAO Rubia wallichiana (stem). Ref: 4369.
OH
HO
OH
6018 5,7-Dihydroxy-6-(2-methylbutanoyl)-8-[(E)-3,7-dimethylocta-2,6-
(stem). Ref: 5238.

O
OH
dienyl]-4-phenyl-2H-chromen-2-one
OH
C30H34O5 (474.60). Yellow crystals, mp 89~90C. Pharm: Antibacterial
HO
(Enterococcus faecalis 18292, MIC = 8g/mL; Enterococcus faecalis 19250, MIC

= 8g/mL); antibacterial (Staphylococcus aureus 18268, MIC = 32g/mL;
O
O
Staphylococcus aureus 17380, MIC = 8g/mL; Staphylococcus aureus 17592, MIC
= 64g/mL; Staphylococcus aureus 18110, MIC = 64g/mL; Staphylococcus
aureus 17547, MIC = 32g/mL; Staphylococcus aureus 17728, MIC = 16g/mL;
(stem). Ref: 5238.
Staphylococcus aureus 3012, MIC = 16g/mL; Staphylococcus aureus 414, MIC =
16g/mL; Staphylococcus epidermidis 3112, MIC = 4g/mL; Staphylococcus
O
OH
HO
epidermidis 2515, MIC = 8g/mL; Staphylococcus saprophyticus 3010, MIC =

32g/mL; Staphylococcus simulans 214, MIC = 4g/mL); antimalarial
(Plasmodium falciparum D10 (CQ-S), IC50 = (2.750.45)g/mL, control
6014 1,3-Dihydroxy-5-methoxyxanthone-4-sulfonate
Chloroquine, IC50 = (0.0110.004)g/mL; W2 (CQ-R), IC50 = (1.170.61)g/mL,
C14H9O8S (337.29). Yellow needles, mp > 360C. Pharm: Cytotoxic (P388 cell
control Chloroquine, IC50 = (0.2290.090)g/mL). Source: TIE LI MU Mesua
line, ED50 = 3.46mol/L; control VP-16, ED50 = 0.064mol/L). Source:
ferrea (blossom). Ref: 3870.
YUAN BAO CAO Hypericum sampsonii (whole herb). Ref: 3861.

O
OH
OH
O
O
HO
OH
O S O
O
O
O
156
6019 5,7-Dihydroxy-6-(3-methylbutanoyl)-8-[(E)-3,7-dimethylocta-2,6-
6022 1-[2',4'-Dihydroxy-3'-(3''-methylbut-2''-enyl)-5'-(1'''-ethoxy-3'''-
methylbutyl)-6'-methoxy]phenylethanone
C21H32O5 (364.49). Source: SHA TANG MU Acronychia pedunculata. Ref: 2373.

O
O
HO
OH
O
OH
OH
6023 4,6-Dihydroxy-3-[3'-methyl-2'-butenyl]-5-[4''-hydroxy-3''-methyl6020 5,7-Dihydroxy-8-(2-methylbutanoyl)-6-[(E)-3,7-dimethylocta-2,6-
2''-butenyl]-cinnamic acid
C19H24O5 (332.40). Colorless oil. Source: DAN ZI HAO Artemisia
C30H34O5 (474.60). Colorless crystals, mp 90~92C. Pharm: Antibacterial
monosperma. Ref: 5249.
(Enterococcus faecalis 18292, MIC = 8g/mL; Enterococcus faecalis

19250, MIC = 8g/mL); antibacterial (Staphylococcus aureus 18268, MIC =
4g/mL; Staphylococcus aureus 17380, MIC = 64g/mL; Staphylococcus

aureus 17592, MIC = 2g/mL; Staphylococcus aureus 18110, MIC =
4g/mL; Staphylococcus aureus 17547, MIC = 2g/mL; Staphylococcus
OH
HO
OH
aureus 17728, MIC = 2g/mL; Staphylococcus aureus 3012, MIC = 2g/mL;

OH
Staphylococcus aureus 414, MIC = 16g/mL; Staphylococcus epidermidis

3112, MIC = 2g/mL; Staphylococcus epidermidis 2515, MIC = 2g/mL;
Staphylococcus saprophyticus 3010, MIC > 128g/mL; Staphylococcus
simulans 214, MIC = 2g/mL); antimalarial (Plasmodium falciparum D10
(CQ-S), IC 50 = (11.215.40)g/mL, control Chloroquine, IC50 =
(0.0110.004)g/mL; W2 (CQ-R), IC 50 = (8.382.52)g/mL, control
Chloroquine, IC 50 = (0.2290.090)g/mL). Source: TIE LI MU Mesua
ferrea (blossom). Ref: 3870.
6024 (E)-1-[2,4-Dihydroxy-3-(3-methyl-2-butenyl)phenyl]-3-(2,2-dimethyl-8-hydroxy-2H-benzopyran-6-yl)-2-propen-1-one
6'',6''-Dimethylpyrano(2'',3'':4,5)-3'-,-dimethylallyl-2',3,4'-trihydroxychalcon
e [151135-83-0] C25H26O5 (406.48). Yellow acicular crystals (chloroform or
hexane), mp 153~156C. Pharm: Antileishmanial (Leishmania sp., 20g/mL,
InRt = 32%). Source: GUANG GUO GAN CAO Glycyrrhiza glabra,
ZHANG GUO GAN CAO Glycyrrhiza inflata, GAN CAO Glycyrrhiza
uralensis. Ref: 1002, 1154.
O
HO
OH
O
HO
OH
OH
6021 5,7-Dihydroxy-8-(3-methylbutanoyl)-6-[(E)-3,7-dimethylocta-2,6dienyl]-4-phenyl-2H-chromen-2-one
6025 (E)-1-[2,4-Dihydroxy-3-(3-methyl-2-butenyl)phenyl]-3-(4-hydroxy-3-[3-methyl-2-butenyl)phenyl]-2-propen-1-one
3,3'-Di-(,-dimethylallyl)-2',4,4'-trihydroxychalcone [151135-82-9] C25H28O4
(392.50). Yellow acicular crystals (methanolwater), mp 134~137C. Pharm:
Antileishmanial (Leishmania sp., 20g/mL, InRt = 90%). Source: GUANG
HO
GUO GAN CAO Glycyrrhiza glabra, ZHANG GUO GAN CAO Glycyrrhiza
inflata, GAN CAO Glycyrrhiza uralensis. Ref: 1002, 1154.
OH
OH
HO
OH
157
6026 6-(2',3'-Dihydroxy-3'-methylbutyl)-7-acetoxy-2H-1-benzopyran-2- one
6031 1,7-Dihydroxy-2,3-methylenedioxyxanthone
C16H18O6 (306.32). White clustered crystals (MeOH), mp 171~172C. Source: CI
C14H8O6 (272.22). Colorless acicular crystals (chloroformmethanol), mp
YI YE HUA JIAO Zanthoxylum dimorphophyllum var. spinifolum. Ref: 2121.
224~226C, mp 245~247C, mp 243~245C. Pharm: Aldose reductase

inhibitor (eye lens). Source: HUANG HUA YUAN ZHI Polygala arillata, JIA
O
O
HUANG HUA YUAN ZHI Polygala fallax [Syn. Polygala aureocauda] (root
OH
and stem: yield = 0.00135%)[4683]. Ref: 345, 658, 4683.
OH
6027 2,3-Dihydroxy-2-methyl-butyolactone
O
HO
OH
O
C5H8O4 (132.12). White granular crystals (acetone). Pharm: Cytotoxic
(stronger). Source: DA YE BAI TOU WENG Anaphalis margaritacea,
GUAN GUANG MU Tsoongiodendron odorum. Ref: 2177, 3853.

6032 7,4'-Dihydroxy-8-methylflavan
HO
C16H16O3 (256.30). Pharm: Antibacterial (phytopathogenic bacteria,

Corynebacterium betae and Corynebacterium fascians); antifungal (Botrytis
HO
cinerea, ED50 = 32g/mL). Source: LONG XUE SHU Dracaena draco. Ref:
658.
OH
6028 2,5-Dihydroxymethyl-3,4-dihydroxypyrrolidine
C6H13NO4 (163.17). Pharm: Glucosidase I and -, -glucosidase inhibitor
HO
(insect); insect antifeedant (armyworms). Source: MAO YU TENG Derris

elliptica. Ref: 658.
HO
HO
OH
6033 6,7-Dihydroxy-1-methyl-N-(6'-fructopyranosyl)-1,2,3,4-tetrahyOH
N
H
droisoquinoline
C16H23NO7 (341.36). Amorphous brownish solid, 105 dec (MeOH), []D25 =
6029 2,3-Dihydroxymethyl-4-(3',4'-dimethoxyphenyl)--butyrolactone
arcuata. Ref: 2037.
C14H18O6 (282.30). Colorless needles. Source: LIAN QIAO Forsythia

O
HO
suspensa. Ref: 2520.

HO
OH
HO
OH
OH
OH
OH
O
O
6034 4,7-Dihydroxy-10-methyl-3,4,7,8,9,10-hexahydro-oxecin-2-one
C10H16O4 (200.24). Colorless crystals (MeOHCHCl 3), mp 203~204C, [] D29

6030 8-(3,4-Dihydroxy-2-methylene-butanoyloxy)-dehydro-melitensin
= 55 (c = 0.036, MeOH). Pharm: Antimalarial inactive (Plasmodium
C20H26O7 (378.43). Pharm: Antifungal (Aspergillus niger, MIC = 0.25g/mL,
falciparum K1, 20g/mL; control Dihydroartemisinin, IC50 = 1.2ng/mL).
control Miconazole, MIC = 1.5g/mL; Aspergillus ochraceus, MIC =
Source: YONG CHONG CAO Cordyceps militaris. Ref: 4784.
0.125g/mL, Miconazole, MIC = 1.5g/mL; Aspergillus versicolor, MIC =
0.125g/mL, Miconazole, MIC = 2g/mL; Aspergillus flavus, MIC = 1g/mL,
Miconazole, MIC = 0.5g/mL; Penicillium ochrochloron, MIC = 0.25g/mL,
OH
Miconazole, MIC = 2g/mL; Penicillium funiculosum, MIC = 0.5g/mL,

Miconazole, MIC = 2g/mL; Trichoderma viride, MIC = 0.25g/mL,
OH
Miconazole, MIC = 2g/mL; Cladosporium cladosporioides, MIC =
6035 (1R,4R,4aS,7aS)-4,7-Dihydroxymethyl-1-hydroxyl-1,4,4a,7a-tetra-
0.5g/mL, Miconazole, MIC = 0.03g/mL; Alternaria alternata, MIC =
hydrocyclopenta-6-ene[e]pyran-3-one
0.25g/mL, Miconazole, MIC = 0.5g/mL). Source: Centaurea thessala ssp.
C10H14O5 (214.22). Colorless gum, []D25 = +32.0 (c = 0.30, CHCl3). Source:
drakiensis (aerial parts), Centaurea attica ssp. attica (aerial parts). Ref: 5115.
GUANG YAO DA HUANG HUA Cymbaria mongolica. Ref: 2001.
OH
OH
H
O
OH
O
H
H
HO
HO
O
O
OH
158
6036 2,5-Dihydroxy-6-methyl-7-methoxyflavanone
6041 1,4-Dihydroxy-2-(7'-methyl-3'-methylene-1'-oxo-4',7'-peroxide-
[186906-54-7] C17H16O5 (300.31). Source: YUAN ZHI YE AO ZHOU CHA
octyl)benzene
Leptospermum polygalifolium ssp. Polygalifolium (foliage). Ref: 3485.

OH

OH
OH
6037 2,5-Dihydroxy-8-methyl-7-methoxyflavanone
[186906-53-6] C17H16O5 (300.31). Source: YUAN ZHI YE AO ZHOU CHA
OH
Leptospermum polygalifolium ssp. Polygalifolium (foliage). Ref: 3485.
6042 10,13-Dihydroxy-9-methyl-15-oxo-20-nor-kauran-19-oic acid

-lactone
O
OH
C20H28O4 (332.44). Pale-yellow crystals, mp 85~88C, [] D25 = 68.0 (c =

0.1, MeOH). Pharm: Cytotoxic (Lu1, Col2, KB, LNCaP, hTERT-RPE1, ED50
= 10-20g/mL, HUVEC, ED50 > 20g/mL; control Taxol, ED50 = 0.002g/mL,
OH
0.003g/mL, 0.0005g/mL, 0.001g/mL, 0.004g/mL, 0.008g/mL,

respectively). Source: Parinari sprucei (leaf). Ref: 4991.
6038 (1R,4R,4aS,7aS)-4,7-Dihydroxymethyl-1-methoxyl-1,4,4a,7a-tetraOH
O
OH
H
HO
O
H
6043 3,12-Dihydroxy-13-methyl-8,10,13-podocarpanetriene
O
H
C18H26O2 (274.41). Semi solid, []D25 = 12.6 (c = 0.5, MeOH). Source: MA
FENG SHU Jatropha curcas (aerial parts). Ref: 4287.
6039 (1R,4S,4aS,7aS)-4,7-Dihydroxymethyl-1-methoxyl-1,4,4a,7a-tetra-
OH
HO
HO
H
6044 3,12-Dihydroxy-13-methyl-6,8,11,13-podocarpatetraen
O
H
HO
C18H24O2 (272.39). Yellow oil, []D20 = +86.7 (c = 0.91, acetone). Pharm:
Cytotoxic (in vitro, pulmonary adenocarcinoma A549 cells, IC50 =

31.8mol/L; hepatocarcinoma Bel 7402 cells, IC50 = 22.9mol/L; gastric
6040 7-(2',6'-Dihydroxy-7'-methyl-3'-methyleneocta-7'-en-1-oxy)-8-
carcinoma BGC823 cells, IC50 = 21.1mol/L; colorectal adenocarcinoma
methoxycoumarin
HCT8 cells, IC50 = 21.8mol/L; ovarian cancer A2780 cells, IC50 =
23.7mol/L). Source: YI YE QIU Securinega suffruticosa (callus). Ref: 4544.

sp. Ref: 2176.
OH
O
OH
OH
O
O
HO
159
6045 3,12-Dihydroxy-13-methyl-5,8,11,13-podocarpatetraen-7-one
6050 2,3-Dihydroxy-30-noroleana-12,20(29)-dien-28-oic acid
C18H22O3 (286.37). Pale yellow oil, []D20 = 56.6 (c = 0.09, acetone). Pharm:
Cytotoxic (in vitro, pulmonary adenocarcinoma A549 cells, IC50 =
Source: SAN YE MU TONG Akebia trifoliata (stem). Ref: 4545.
31.6mol/L; hepatocarcinoma Bel 7402 cells, IC50 = 26.5mol/L; gastric

carcinoma BGC823 cells, IC50 = 20.0mol/L; colorectal adenocarcinoma
HCT8 cells, IC50 = 22.0mol/L; ovarian cancer A2780 cells, IC50 =
21.8mol/L). Source: YI YE QIU Securinega suffruticosa (callus). Ref: 4544.
HO
OH
OH
HO
6051 2,3-Dihydroxy-30-noroleana-12,20(29)-dien-28-oic acid

HO

6046 2,7-Dihydroxy-1-methyl-5-vinylphenanthrene
OH
HO
OH
H
HO
HO
6052 2,3-Dihydroxynortropane
6047 9,12-Dihydroxy-15-nonadecenoic acid
C7H13NO2 (143.19). Colorless powder, []D = 33.9 (c = 0.32, H2O). Pharm:
-Glucosidase inhibitor inactive (control 1-Deoxynojirimucin, IC50 =

0.98mmol/L, Fagoming, IC50 = 15mmol/L). Source: SANG SHI Morus alba.
OH
OH
O
OH
Ref: 4161.
HN
H
OH
6048 2,5-Dihydroxy-3-(nonadec-14-enyl)-benzoquinone
OH
C25H40O4 (404.60). Yellow brown crystals (MeOH), mp 138~139C, []D25 =

40 (c = 1.0, CH2C12). Source: PI ZHEN DU JING SHAN Maesa lanceolata
(fruit). Ref: 3464.
6053 2,3-Dihydroxynortropane
-Glucosidase inhibitor inactive (control 1-Deoxynojirimucin, IC50 =
0.98mmol/L, Fagoming, IC50 = 15mmol/L). Source: SANG SHI Morus alba.
Ref: 4161.
O
HN
OH
HO
OH
OH
6049 3,15-Dihydroxy-18-norabieta-3,8,11,13-tetraene
C19H26O3 (302.42). White-brown powder, []D24 = +23.5 (c = 2.9, MeOH).
Pharm: Cytotoxic (KB, IC50 > 66mol/L, control Podophyllotoxin, IC50 =
6054 3,6-exo-Dihydroxynortropane
0.014mol/L); antibacterial (Bacillus cereus, MIC = 423.84mol/L; control
Chloramphenicol, MIC = 6.19mol/L). Source: GAO MEI YING BAN
-Glucosidase inhibitor (IC50 = 33mmol/L, control 1-Deoxynojirimucin, IC50
Crossopetalum gaumeri (root). Ref: 3969.
= 0.98mmol/L, Fagoming, IC50 = 15mmol/L). Source: SANG SHI Morus alba.
OH
Ref: 4161.
HN
OH
HO
OH
H
160
6055 2,3-Dihydroxy-28-norurs-12,17,19(20),21-tetraen-23-oic cid
6060 3,22-Dihydroxyolean-12-en-29-oic acid
C29H40O4 (452.64). White amorphous powder, []D28.6 = +19.8 (c = 0.21,
C30H48O4 (472.71). Pharm: DPPH scavenger inactive (for 40mol/L DPPH
MeOH). Pharm: Cytotoxic (SGC cell, EC50 = 10.2mol/L). Source: DI YU
radical, SC50 > 40mol/L). Source: SUO LA MU Salacia prinoides [Syn.
Sanguisorba officinalis. Ref: 5304.
Salacia chinensis] (stem). Ref: 4378.

O
OH
OH
H
HO
HO
HO
O
OH
6061 3,15-Dihydroxy-olean-12-en-16-one
6056 3,7-Dihydroxy-5-octanolide
Eriocarpin A; 3,15-Dihydroxy-olean-12(13)-en-16-one C30H48O3 (456.72).
C8H14O4 (174.20). White powder, mp 93.5~94.0C, []D26 = 24.4 (c = 0.086,
Colorless acicular crystals (MeOH), mp 195~197C, [ ] D20 = +0 (c =
EtOH). Source: YE YA CHUN Euscaphis japonica. Ref: 2204.
0.011, MeOH). Source: MAO GUO YU TENG Derris eriocarpa, YUN NAN
GE TENG Pueraria peduncularis. Ref: 665, 2262.
OH
OH
O
6057 3,11-Dihydroxy-olean-12-ene
C30H50O2 (442.73). White crystals (acetone), easily soluble in CHCl3 and
MeOH, mp 192~196C. Source: SI CHUAN QING FENG TENG Sabia
schumanniana (aerial parts). Ref: 4883.
H
HO
OH
6062 3,16-Dihydroxy-olean-12-en-15-one
C30H48O3 (456.72). Colorless acicular crystals mp 218~220C. Source: YUN
NAN GE TENG Pueraria peduncularis. Ref: 853.
HO
H
H
H
HO
OH
HO

C30H48O4 (472.71). Source: SAN YE MU TONG Akebia trifoliata (stem). Ref: 4545.
6063 6,10-Dihydroxy-1-oxoeremophila-7(11),8(9)-dien-12,8-olide
C15H18O5 (278.31). Source: Ligularia virgaurea ssp. oligocephala (whole
herb). Ref: 4981.
O
HO
OH
H
HO
OH
OH
6064 4,10-Dihydroxy-3-oxo-8-isobutyryloxyguaia-11(13)-en-12,6-olide
C19H26O7 (366.41). Pharm: Cytotoxic (antiproliferative, Col2 cells, IC50 =
()-Maslinic acid; Crategolic acid [4373-41-5] C30H48O4 (472.71). mp ()
18.9g/mL); cytotoxic (cellular differentiation inducer, hmn promyelocytic leukemia
263~265C. Source: DA ZAO Ziziphus jujuba, HUO XIANG Agastache
HL-60 cells, 4g/mL, activity denotes percentage of cells differentiated = 32.4%);
rugosus, SAN YE MU TONG Akebia trifoliata (stem), YANG MEI SHU PI
cytotoxic (MMOC model, inhibits DMBA-induced preneoplastic lesion formation,
Myrica rubra (bark: yield = 0.00083%). Ref: 2, 660, 1247, 4163, 4545.
10g/mL, rel-InRt = 48.7%, control DMBA, rel-InRt =100%). Source: ZHONG

BIN JU Tithonia diversifolia (aerial parts: yield = 0.0063%dw). Ref: 4622.
OH
HO
H
HO
HO
OH
H
O
O
161
6065 16,17-Dihydroxy-3-oxo-19-nor-ent-kaur-4-ene
6070 2,19-Dihydroxy-3-oxo-12-ursen-28-oic acid
C19H28O3 (304.43). Pharm: Antibacterial (Staphylococcus aureus, MIC <
C30H46O6 (502.70). Pharm: Immunosuppressant (hmn mononuclear cells
1.5mg/mL; Bacillus cereus and Pseudomonas aeruginosa, MIC =
antiproliferation, involving T lymphocytes, B lymphocytes, and macrophages
2.0~3.0mg/mL; Escherichia coli, inactive). Source: Antennaria geyeri (aerial
isolated from peripheral blood, IC50 = 40.0mol/L; control Cyclosporine A, IC50 =
parts). Ref: 3853.
0.012mol/L). Source: TAI WAN PI PA Eriobotrya deflexa (leaf). Ref: 3064.

OH
OH
HO
OH
6066 16,17-Dihydroxy-15-oxo-ent-kaur-19-oic acid
OH
HO
C20H30O5 (350.46). Brownish solid, mp 137~142C, []D25 = +5.0 (c = 0.1,
6071 3,19-Dihydroxy-6-oxo-urs-12-en-23-ol-28-oic acid
MeOH). Pharm: Cytotoxic inactive (Lu1, Col2, KB, LNCaP, hTERT-RPE1,
C30H46O6 (502.70). Source: BI LU GOU TENG Uncaria tomentosa. Ref: 5341.
HUVEC; control Taxol, ED50 = 0.002g/mL, 0.003g/mL, 0.0005g/mL,

0.001g/mL, 0.004g/mL, 0.008g/mL, respectively). Source: Parinari
HO
sprucei (leaf). Ref: 4991.

H
H
HO
OH
OH
H
HO
HO
OH
6067 16,17-Dihydroxy-15-oxo-ent-kaur-19-oic acid methyl ester
6072 5,7-Dihydroxy-2',3',4',5',6'-pentamethoxyflavone
C21H32O5 (364.49). White solid, mp 187~193C (dec), []D25 = +27.0 (c = 0.1,
C20H20O9 (404.38). Pharm: Anti-HIV-1 inactive. Source: TAI GUO ZHI ZI
MeOH). Pharm: Cytotoxic inactive (Lu1, Col2, KB, LNCaP, hTERT-RPE1,
Gardenia thailandica (leaf and twig). Ref: 4963.
HUVEC; control Taxol, ED50 = 0.002g/mL, 0.003g/mL, 0.0005g/mL,
0.001g/mL, 0.004g/mL, 0.008g/mL, respectively). Source: Parinari

sprucei (leaf). Ref: 4991.
H
O
O
HO
OH
OH
O
O
OH
6073 3,4-Dihydroxyphenethoxy-O--L-rhamnopyranosyl-(13)--D-(2-
H
O
O-acetyl-4-O-caffeoyl)-galactopyranoside
6068 2,3-Dihydroxy-19-oxo-18,19-seco-urs-11,13(18)-dien-28-oic acid
C31H38O16 (666.64). White amorphous powder, []D28 = 43.34 (c = 0.47, MeOH).
C30H46O5 (486.70). White amorphous powder. Source: FEI LONG ZHANG
Source: LAI JIANG TENG Brandisia hancei (whole herb). Ref: 4569.
XUE Toddalia asiatica [Syn. Toddalia aculeata; Paullinia asiatica] (stem).

Ref: 4561.
OH
HO
O
HO
O
HO
O
OH
O
HO
OO
O
O
OH
O O
OH
HO
OH OH
6074 3,5-Dihydroxyphenethyl alcohol 3-O--glucopyranoside

6069 3,19-Dihydroxy-6-oxo-urs-12-en-23-al-28-oic acid
C30H44O6 (500.68). Source: BI LU GOU TENG Uncaria tomentosa. Ref: 5341.
Pharm: Antioxidant (DPPH scavenger, DPPH radical 15mol/L: 10mol/L,

ScRt = 41.4%; control BHA, 10mol/L, ScRt = 23.0%; Vitamin E, 10mol/L,
HO
ScRt = 41.1%). Source: JIA HUI SE JIU LI XIANG PO PO NA Veronica

H
H
HO
H
H
O
OH
thymoides ssp. pseudocinerea. Ref: 3846.

HO
OO
OH
OH
OH
OH
OH
162
6075 (E)-4-(3,4-Dihydroxyphenyl)but-3-en-2-one
6079 3,4-Dihydroxyphenylethanol-8-O-[4-O-trans-caffeoyl--D-apio-
C10H10O3 (178.19). Pharm: Cytotoxic (in vitro, A549, IC50 > 0.28mol/L;
furanosyl(13)]--D-glucopyranosyl-(16)]--D-glucopyranoside
BGC823, IC50 = 0.243mol/L; MCF7, IC50 = 0.141mol/L; Bel7402, IC50 =
C34H44O20 (772.72). Yellow-white amorphous powder, has accessibility,
0.153mol/L; Ketr3, IC50 = 0.245mol/L; HCT8, IC50 = 0.227mol/L; control
easily soluble in water and methanol, []D25 = 65.6 (c = 0.09, MeOH).
Topotican, A549, IC50 = 0.0032mol/L; BGC823, IC50 = 0.0043mol/L;
Source: SHI DAN CAO Corallodiscus flabellatus [Syn. Didissandra
MCF7, IC50 = 0.0018mol/L; Bel7402, IC50 = 0.0012mol/L; Ketr3, IC50 =
flabellat]. Ref: 2460.
0.0049mol/L; HCT8, IC50 = 0.0015mol/L). Source: SANG HUANG

Phellinus igniarius (sporocarp: yield = 0.0062%dw). Ref: 4747.
OO
HO
OH
O
HO
OH OH
HO
OH
OO
OH
HO
O OH
OH OH
OH
OH
O
6076 3,4-Dihydroxyphenylethanol-8-O-[-D-apiofuranosyl(12)]--D-
6080 3,4-Dihydroxyphenylethanol-8-O-[(5-O-vanilloyl)--D-apiofura-
glucopyranoside
nosyl(12)]--D-glucopyranoside
C27H34O15 (598.56). White amorphous powder, has accessibility, easily
easily soluble in water and methanol, []D = 59.3 (c = 0.14, MeOH).
soluble in water and methanol, []D25 = 54.8 (c = 0.42, MeOH). Source: SHI
DAN CAO Corallodiscus flabellatus [Syn. Didissandra flabellat]. Ref: 2463.
25

HO
HO
HO
OH
OO
OH
OH
O
O
HO
OH
OO
OH
OH
OH
O
O
OH
OH OH
OH OH
6081 3,4-Dihydroxyphenylethyl alcohol glucoside

6077 3,4-Dihydroxyphenylethanol-8-O-[-D-apiofuranosyl(13)]--D-
2-(3,4-Dihydroxy-phenyl)-ethyl-O--D-glucopyranoside C14H20O8 (316.31).
glucopyranoside
Pharm: Antioxidant (DPPH scavenger, DPPH radical 15mol/L: 10mol/L,
ScRt = 41.4%; control BHA, 10mol/L, ScRt = 23.0%; Vitamin E, 10mol/L,
easily soluble in water and methanol, []D = 61.6 (c = 0.16, MeOH).
ScRt = 41.1%)[3846]; antioxidant (hydroxyl radical scavenger, IC50 =
55.9mol/L, control Ascorbic acid, IC50 = 51.8mol/L, superoxide anion
radical scavenger, IC50 = 86.5mol/L, Ascorbic acid, IC50 = 86.2mol/L)[4289].
25
Source: HUANG LIAN Coptis chinensis, JIA HUI SE JIU LI XIANG PO PO

NA Veronica thymoides ssp. pseudocinerea, XI ZANG HU HUANG LIAN
HO
OH
Picrorhiza scrophulariiflora (root)[4289]. Ref: 2, 3846, 4289.
HO
OO
OH
OH
OH OH
OH
OO
HO
OH
OH
6078 3,4-Dihydroxyphenylethanol-8-O-[-D-apiofuranosyl(13)--D-
OH
OH
OH
glucopyranosyl(16)]--D-glucopyranoside
easily soluble in water and methanol, []D25 = 70.5 (c = 0.12, MeOH).
6082 5,8-Dihydroxy-2-(2-phenylethyl)chromone
C17H14O4 (282.30). Colorless lump crystals, mp 159~160C. Source: BAI MU
HO
OO
OH
OH
HO
O OH
OH OH
OO
OH
OH
O
O
OH
OH
OH
OH
163
6083 6,8-Dihydroxy-2-(2-phenylethyl)chromone
6089 7'-(3',4'-Dihydroxyphenyl)-N-[(4-methoxyphenyl)ethyl]propenamide
C17H14O4 (282.30). Colorless needles, mp 218~220C (MeOH). Source:
C18H19NO4 (313.36). Colorless solid. Pharm: -Glucosidase inhibitor (type VI,
CHEN XIANG Aquilaria agallocha. Ref: 4173.
IC50 = 103.58mol/L, control 1-Deoxynojirimycin, IC50 = 300mol/L);

thrombin inhibitor inactive; -glucuronidase inhibitor inactive. Source: YUN
O
OH
NAN TU SI ZI Cuscuta reflexa. Ref: 4155.

O
HO
OH
6084 6,7-Dihydroxy-2-(2-phenylethyl)-5,6,7,8-tetrahydrochromone
C17H18O 4 (286.33). Brown amorphous solid,
[]D25 =
15.1 (c = 1.0, MeOH).
Source: BAI MU XIANG Aquilaria sinensis (withered wood). Ref: 4339.
N
H
HO
6090 1,3-Di-p-hydroxyphenyl-4-penten-1-one
C17H16O3 (268.32). Pharm: Cytotoxic (in vitro, HOG.R5, CC50 = 20.6g/mL
(76.8mol/L), control Ellipticine, HOG.R5, IC50 = 0.02g/mL (0.08mol/L));
cytotoxic inactive (KB, Col2, LNCaP, Lu1, HUVEC, IC50 > 20g/mL);
OH
anti-HIV (IC50 = 20g/mL (74.6mol/L)). Source: TIAN MEN DONG

O
OH
Asparagus cochinchinensis [Syn. Asparagus lucidus] (dried root: yield =

0.00005%dw). Ref: 3009.
O
6085 1'-O--D-(3,4-Dihydroxyphenyl)-ethyl-6'-O-vanilloyl-glucopyranoside
C22H26O11 (466.45). White amorphous powder, having hygroscopicity, mp
145~147C, []D25 = 42.1 (c = 0.41, MeOH). Source: SHI DAN CAO
Corallodiscus flabellatus [Syn. Didissandra flabellat] (whole herb). Ref: 4849.
O
O
OO
OH
OH
HO
OH
OH
OH
HO
6091 3-(3,4-Dihydroxyphenyl)propanoic acid

C9H10O4 (182.18). Pharm: Tyrosine kinase inhibitor (IC50 = 418mol/L,
interleukin-2 inducible T-cell kinase). Source: MO LEI NAN YANG SHEN
Polyscias murrayi. Ref: 5252.
OH
6086 2-(2,4-Dihydroxyphenyl)-6-hydroxybenzofuran
C14H10O4 (242.23). Pharm: Antioxidant (rat brain homogenate lipid
peroxidation test, IC50 = 0.2mol/L, control EGCg, IC50 = 0.07mol/L).
Source: TONG XING LIE PIAN HU ZHI ZI Lespedeza homoloba. Ref: 2356.
HO
OH
HO
OH
6092 3-(3,4-Dihydroxyphenyl)-1-propanol
OH
C9H12O3 (168.19). Source: TAI WAN CUI BAI Calocedrus macrolepis var.
formosana (leaf). Ref: 4297.

OH
HO
OH
OH
6087 1-(3',5'-Dihydroxyphenyl)-2-(4''-hydroxyphenyl)-ethane-1,2-diol
Source: HU ZHANG Polygonum cuspidatum. Ref: 4186.
OH
OH
6093 3,4-Dihydroxyphenylpropanol -D-glucopyranoside

OO
HO
OH
OH
HO
OH
OH
HO
OH
OH
6088 1-(2,4-Dihydroxyphenyl)-3-(4-hydroxyphenyl)propane
C15H16O3 (244.29). Brown powder, mp 92~93C. Pharm: Aromatase inhibitor
inactive (in vitro, IC50 > 40mol/L; control Aminoglutethimide, IC50 =
6.4mol/L). Source: GOU SHU Broussonetia papyrifera. Ref: 3090.
HO
OH
6094 3-(3,4-Dihydroxyphenyl)-2-propen-1-ethanoate
C11H14O4 (210.23). Pharm: -Glucosidase inhibitor inactive (type VI, control
1-Deoxynojirimycin, IC50 = 0.3mmol/L); thrombin inhibitor inactive;
-glucuronidase inhibitor inactive[4155]. Source: YUN NAN TU SI ZI Cuscuta
reflexa. Ref: 4155.
OH
O
HO
OH
164
6095 3-(3,4-Dihydroxyphenyl)-2-propenoic acid (Z,E)-2-(3,4-dihydroxy-
6100 17,20R-Dihydroxypregnan-3,16-dione
phenyl) ethenyl ester
C21H32O4 (348.49). Colorless acicular crystals (Me2CO), []D26 = 106.3 (c =
[55486-06-1] C17H14O6 (314.29). Yellow acicular crystals (methanolwater),
0.31, CHCl3). Source: YA LUO CHUN Cipadessa baccifera. Ref: 745.
mp 183~185C (dec). Pharm: Xanthinoxidase inhibitor (in vitro, IC50 =

0.021g/mL). Source: JIAN ZI SU Perilla frutescens var. acuta [Syn. Perilla
HO
frutescens var. purpurascens]. Ref: 1006.
OH
O
OH
H
O
OH
HO
OH
6101 15,20-Dihydroxy-4-pregnen-3-one
C21H32O3 (332.49). Source: HONG HUA Carthamus tinctorius. Ref: 2.
6096 3-(3,4-Dihydroxyphenyl)-2-propenoic acid (Z,E)-2-(3,5-dihydroxy-
HO
phenyl) ethenyl ester

[130233-90-8] C17H14O6 (314.29). Yellow thinly crystals (methanolwater),
mp 188~190C. Pharm: Xanthinoxidase inhibitor (in vitro, IC50 =

0.124g/mL). Source: JIAN ZI SU Perilla frutescens var. acuta [Syn. Perilla
H
H
OH
frutescens var. purpurascens]. Ref: 1006.

6102 (2S)-7,4'-Dihydroxy-3'-prenylflavan
OH
HO
C20H22O3 (310.4). Brown powder, mp 116~117C. Pharm: Aromatase inhibitor

inactive (in vitro, IC50 > 40mol/L; control Aminoglutethimide, IC50 =
OH
6.4mol/L). Source: GOU SHU Broussonetia papyrifera. Ref: 3090.
O
OH
OH
6097 Dihydroxypicrotoxinin
C15H18O8 (326.31). Colorless needles, mp 260~262C, []D17 = 65 (c = 1.34,
HO
EtOH) Source: Anamirta cocculus. Ref: 1876.

O
6103 1-(2,4-Dihydroxy-3-prenylphenyl)-3-(4-hydroxyphenyl)-propane
Anticancer Benzenoid PMV70P691-003 C20H24O3 (312.41). Brown powder,
O
O
H
H
mp 115~116C. Pharm: Aromatase inhibitor inactive (in vitro, IC50 >
OH
H
40mol/L; control Aminoglutethimide, IC50 = 6.4mol/L)[3090]; cytotoxic
OH
(antioxidant assay)[5038]. Source: GOU SHU Broussonetia papyrifera. Ref:
OH
3090, 5038.
6098 ent-16,18-Dihydroxy-8(14)-pimaren-15-one
C20H32O3 (320.48). Viscous oil, []D26 = 9.1 (c = 0.55, MeOH). Source: HAI
NAN JIAN MU Dysoxylum hainanense. Ref: 750.
OH
HO
OH
OH
H
6104 2',3'-Dihydroxy-1'-propoxypseudolarate B
OH
6099 1,13-Dihydroxy-8,11,13-podocarpatriene
23
C17H24O2 (260.38). Yellow amorphous solid, []D = 3.1 (c = 0.55, CHCl3).
Me2CO). Source: TU JING PI Pseudolarix amabilis [Syn. Larix amabilis;

Pseudolarix kaempferi] (root cortex: yield = 0.000047%dw). Ref: 4637.

O
OH
OH
O
O
O H
O
OH
O
O
OH
165
6105 3,9-Dihydroxypterocarp-6a-ene
6109 5,11-Dihydroxy-ros-15-ene
C15H10O4 (254.24). Pharm: Antioxidant (rat brain homogenate lipid
C20H34O2 (306.49). []D20 = +68 (c = 0.23, CHCl3). Source: Gackstroemia
peroxidation test, IC50 = 0.2mol/L, control EGCg, IC50 = 0.07mol/L);
decipiens. Ref: 3907.
Antiallergic (50mg/kg, InRt = 49.6%, control EGCg, InRt = 12.8%). Source:
HO
TONG XING LIE PIAN HU ZHI ZI Lespedeza homoloba. Ref: 2356.
HO
H
OH
6110 5,12-Dihydroxy-ros-15-ene
OH
6106 20,23-Dihydroxy-3-[(O--L-rhamnopyranosyl-(12)--L-arabi-

OH
nopyranosyl)oxy]lupan-28-oic acid 28-O--L-rhamnopyranosyl-(14)O--D-glucopyranosyl-(16)--D-glucopyranosyl ester
Source: BAI TOU WENG Pulsatilla chinensis. Ref: 3086.

OH
HO
6111 3,4-Dihydroxyrottlerin
H
[24650-82-6] C31H30O9 (546.58). mp 200C. Source: LV SONG QIU MAO

Mallotus philippinensis. Ref: 6.
H
H
OH
OO
HO
HO
HO
OH
O O HO
HO
OH
H
O
HO
OH
O
O
O
OH
OH HO
HO
OH OH
OH OH
OH
OH
OH
6107 (22S)-3,22-Dihydroxy-1-[(-L-rhamnopyranosyl)oxy]cholest5,24-dien-16-yl -D-glucopyranoside

Cytotoxic (HL-60 cells, IC50 > 10mol/L, control Etoposide, IC50 = 0.025mol/L).
Source: XIA FENG XIN ZI Galtonia candicans (bulb). Ref: 4116.
OH
6112 1,2-Dihydroxyrutaecarpine
C18H13N3O3 (319.32). Yellow amorphous solid. Source: Bouchardatia
neurococca. Ref: 3445.
OH
OH
O O
N
H
H
OH OH
O
H
HO
HO
HO
O
OH
OH
OH
6113 12,25-Dihydroxy-16-scalaren-24,25-olide
OH
C25H38O4 (402.58). Source: Cacospongia scalaris. Ref: 1521.
6108 5,4'-Dihydroxy-3--L-rhamnosyl-(1''3')--D-xylopyranosyloxy-
HO
OH
bibenzyl
O
O
C25H32O11 (508.53). Amorphous yellowish color, >179C(glass transition),
20
[]D = 39 (c = 0.235, MeOH). Pharm: Antioxidant (DPPH scavenger, IC50

= (8.930.94)g/mL; control Ascorbic acid, IC50 = (2.490.32)g/mL; Caffeic
acid, IC50 = (1.780.03)g/mL; Chlorogenic acid, IC50 = (1.280.38)g/mL).
Source: SUAN YE PO LUO MEN SHEN Tragopogon porrifolius (subaerial
parts). Ref: 5307.
6114 1,6-Dihydroxy-4H-1,10-secoeudesma-5(10),11(13)-dien-12,8- olide

C15H22O4 (266.34). Pharm: Cytotoxic (SMMC-7721 IC50 =
OH
(52.221.25)g/mL, Vincristine IC50 = (30.352.23)g/mL; HO-8910 IC50 =

(21.322.64)g/mL, Vincristine IC50 = (20.741.91)g/mL)[5422]. Source: JIN
OH
FEI CAO Inula japonica. Ref: 5422.
OO
OO
OH
HO
OH
OH
OH OH
OH
166
6115 (1R)-1,11--Dihydroxy-3,4-seco-lupa-4(23), 20(29)-diene-3,28-dioic
6119 3,21-Dihydroxyserrat-14-en-24-ol
acid 3,11-lactone 28-O--L-rhamnopyranosyl-(14)--D-glucopyranosyl
C30H50O3 (458.73). Source: QIAN CENG TA Huperzia serrata [Syn.
Lycopodium serratum] (whole herb: yield = 0.0001%dw). Ref: 4729.
C48H74O19 (955.11). White needles, mp 232~234C []D14 = +11.7 (c = 0.5,

MeOH). Source: CI WU JIA Acanthopanax senticosus [Syn. Eleutherococcus
OH
H
senticosus]. Ref: 469.
O
OH
HO
OH
O
HO
OH
OH
OH
OO
OO
OO
OH
OH
OH
OH
H
OH OH
6116 3,21-Dihydroxyserrat-14-ene-24,29-diol
HO
OH
OH
H
OH

OH
H
HO
OH
OH
6117 3,21-Dihydroxyserrat-14-en-24-oic acid
HO
C30H48O4 (472.71). White powder (CHCl3CH 3OH), mp 304~306C, []D20 =

0.6 (c = 0.78, C5D5N). Source: QIAN CENG TA Huperzia serrata [Syn.
6122 3,21-Dihydroxyserrat-14-en-16-one
16-Oxo-21-episerratenediol C30H48O3 (456.72). Source: QIAN CENG TA

Huperzia serrata [Syn. Lycopodium serratum] (whole herb: yield =
OH
H
0.000084%dw), SHEN JIN CAO Lycopodium japonicum [Syn. Lycopodium

clavatum]. Ref: 1410, 2811, 4729.
OH
H
HO
O
OH
O
HO
6123 7,22S-Dihydroxysitosterol
C29H53O3 (446.72). White powder, mp 183~185C Source: MA BIAN CAO
Verbena officinalis. Ref: 2173.
OH
OH
H
H
H
H
HO
OH
HO
H
OH
167
6124 1,2-Dihydroxyspirosta-5,25(27)-dien-3-yl O--D-rhamno-
6127 (25R)-1,2-Dihydroxyspirost-5-en-3-yl O--L-rhamnopy-
pyranosyl-(12)--L-galactopyranoside
ranosyl-(12)--D-galactopyranoside
Source: Cestrum sendtenerianum (leaf). Ref: 5105.
HO
H
HO
HO
OH
OH
HO
HO
HO
OO
OO
OH
OH
OH
OH
OO
OO
OH OH
OH OH
6125 1,2-Dihydroxyspirosta-5,25(27)-dien-3-yl O--L-rhamnopyra-
6128 (25R)-2,17-Dihydroxyspirost-5-en-3-yl O--D-glucopyranos-
nosyl-(12)-O-[-D-glucopyranosyl-(14)]--D-galactopyranoside
yl-(13)-O--D-glucopyranosyl-(12)-O-[-D-xylopyranosyl-(13)]-O-
-D- glucopyranosyl-(14)--D-galactopyranoside
Pharm: Cytotoxic (HL-60, IC50 = 7.7g/mL, control Etoposide, IC50 =
C56H90O29 (1227.32). Amorphous powder, []D24 = 57 (c = 0.2,
0.75g/mL). Source: Cestrum sendtenerianum (leaf). Ref: 5105.
CHCl3-MeOH, 1:1). Pharm: Cytotoxic (HSC-2 cells, LD50 = 5.5g/mL; HGF,

LD50 = 34g/mL)[3023]; cytotoxic (in vitro, HSC-2, LD50 = 4.4g/mL; control
HO
OH
OO
nocturnum (leaf: yield = 0.0077%fw). Ref: 3023, 4667.
OH
HO
Doxorubicin, LD50 = 2.5g/mL)[4667]. Source: YE XIANG SHU Cestrum
OO
OH
OH
OH
OH
HO
HO
HO
OO
O HO
O
HO
HO OH HO
OO
HO
HO
OH
OH OH
6126 (25R)-1,2-Dihydroxy-5-spirostan-3-yl O--L-rhamnopyranosyl-(12)--D-galactopyranoside

25

OH
O O
O O HO
HO
OH
OO
OH
H
OH
OH
6129 (25R)-2,15-Dihydroxyspirost-5-en-3-yl O--D-glucopyranosyl(13)-O--D-glucopyranosyl-(12)-O-[-D-xylopyranosyl-(13)]-O--D

-glucopyranosyl-(14)--D-galactopyranoside
C56H90O29 (1227.32). Amorphous powder, []D24 = 60 (c = 0.13,
CHCl3:MeOH, 1:1). Pharm: Cytotoxic (HSC-2 cells, LD50 = 4.4g/mL; HGF,
LD50 = 22g/mL). Source: YE XIANG SHU Cestrum nocturnum (leaf: yield

= 0.0071%fw). Ref: 3023.
OH
HO
H
HO
HO
OO
OH
OH
OO
H
O
O HO
HO
HO
HO
OH OH
HO
OH HO
O
HO
OH
O
HO
OH
O O
OO
O
OH
HO
OH
OO
HO
OH
H
H
OH
168
6130 (25R)-2,17-Dihydroxyspirost-5-en-3-yl O--D-glucopyranosyl-
6134 2,13(S)-Dihydroxystemodane
(12)-O-[-D-xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--D-
C20H34O2 (306.49). Needles, mp 157~159C, []D27 = +11.9 (c = 0.78,
galactopyranoside
MeOH). Source: DAO GEN MEI Rhizopus oryzae. Ref: 3781.
C50H80O24 (1065.18). Amorphous powder, []D24 = 70.8 (c = 0.13,

OH
CHCl3:MeOH, 1:1). Pharm: Cytotoxic (HSC-2 cells, LD50 = 13g/mL; HGF,

LD50 = 58g/mL). Source: YE XIANG SHU Cestrum nocturnum (leaf: yield
= 0.0070%fw). Ref: 3023.
HO
H
H
O
O
HO
HO
HO
OH
O O
O HO
O
HO
OHHO
HO
OO
H
H
OH
OO
OH
H
6135 6,13(S)-Dihydroxystemodan-2-one
C20H32O3 (320.48). Needles, mp 191~193C, []D27 = +55.6 (c = 4.5, CHCl3).
Source: DAO GEN MEI Rhizopus oryzae. Ref: 3781.
OH
HO
OH
OH
H
H
6131 1,2-Dihydroxy-5-spirost-25(27)-en-3-yl O--L-rhamnopyranosyl-(12)--D-galactopyranoside

OH
6136 7,17-Dihydroxystemod-12-en-2-one
C20H30O3 (318.46). Needles, mp 220~225C, []D27 = 10.9 (c = 2.8, Me2CO).
OH
HO
H
HO
HO
OO
OH
OH
6137 3,5-Dihydroxy-stilbene-3-O-neohesperidoside
OH
OH
C26H32O11 (520.54). White powder, mp 184~186C, []D20 = 100 (c = 0.045,

MeOH). Source: QIAN LIE LIN MAO JUE Dryopteris sublaeta. Ref: 4879.
OO
OH
OH OH
OO
HO
6132 9,10-Dihydroxystearic acid
OH
C18H36O4 (316.49). Source: BI MA ZI Ricinus communis. Ref: 658.

HO
OH
OH
OH
OO
O
OH OH
OH
6138 2,23-Dihydroxy-3-sulfoxyolean-12-en-28-oic acid

O--D-glucopyranosyl-(16)--D-glucopyranosyl ester sodium salt
6133 2,13(R)-Dihydroxystemodane
C20H34O2 (306.49). Plates, mp 235~237C, []D = +16.5 (c = 0.38, MeOH).
C42H67NaO18S (915.05). Amorphous solid, []D27 = +14.0 (c = 0.10, MeOH).
27
HO
H
H
OH
Na HO
O
O
H
OH
OO
OO
HO
OH
OH
OH
OH
OH
OH
169
6139 2,23-Dihydroxy-3-sulfoxyolean-12-en-28-oic acid O--L-rham-
6144 N-(1',4'-Dihydroxy-1',2',3',4'-tetrahydronaphthyl)-propyl-N-di-
nopyranosyl-(14)-O--D-glucopyranosyl-(16)--D-glucopyranosyl
phenylmethyl-N-3,3-dimethylbutylamine
ester sodium salt
C32H41NO2 (471.69). Colorless filamentary needles mp 148.5C. Source: YI
C48H77NaO22S (1061.19). Amorphous solid, []D27 = 8.0 (c = 0.10, MeOH).
BEI MU Fritillaria pallidiflora. Ref: 2116.
Na HO
H
OH
OO
HO
OO
OH
OH
OH
OH
OH
OH
OH
HO
6145 (4R)-4,8-Dihydroxy--tetralone
C10H10O3 (178.19). Source: DONG BEI HU TAO Juglans mandshurica var.
sieboldiana (fruit). Ref: 4492.
OH OH
6140 2,5-Dihydroxy-7,9,10,13-tetraacetoxy-4(20),11-taxadiene
OH
C28H40O10 (536.63). Source: AO DA LI YA HONG DOU SHAN Austrotaxus
spicata, SU MEN DA LA HONG DOU SHAN Taxus sumatrana (twig and

leaf)[4800]. Ref: 662, 4800.
O O
H
OH
O O
6146 3,5-Dihydroxy-6,7,3',4'-tetramethoxyflavone
O
O
OH
H
H OH
Quercetagetin-6,7,3',4'-tetramethyl ether C19H18O8 (374.35). Source: HUANG

HUA HAO Artemisia annua. Ref: 2, 660.
6141 (1S,4S,8S)-8,9-Dihydroxytetrahydrocarvone

OH
OH
OH
OH
6147 5,3'-Dihydroxy-3,7,4',5'-tetramethoxyflavone
C19H18O8 (374.35). Amorphous. Source: NIAN MAO LIAO Polygonum
6142 (1S,4S,8S)-8,9-Dihydroxytetrahydrocarvone 9-O--D-gluco-
viscosum (whole herbs). Ref: 3955.
pyranoside
OH

O
O
OH
HO
OH
H
OH
OH
6148 5,3'-Dihydroxy-6,7,4',5'-tetramethoxyflavone
OH
6143 10,14-Dihydroxy-10(14),11(13)-tetrahydro-8,9-didehydro-3-
C19H18O8 (374.35). Pharm: Antioxidant (ferric thiocyanate method,
deoxyzaluzanin C 10-O--D-glucopyranoside
0.5mmol/L, peroxidation value = 11.4%, control BHA, 0.5mmol/L,
C21H30O9 (426.47). Solid, []D
25.8
= 41.8 (c = 0.63, MeOH). Source: KAN
CHA JIA MAO LIAN CAI Picris kamtschatica. Ref: 1932.

HO
OH
peroxidation value = 4.5%, control Vitamin E, 0.5mmol/L, peroxidation value

= 14.7%). Source: TIAN SHE CAO Lippia dulcis (aerial parts). Ref: 4508.
O
O O
H
OH
O
O
OH
OH
OH
OH
170
6149 5,7-Dihydroxy-2',3',4',5'-tetramethoxy-flavone
6154 3,22S-Dihydroxy-tirucalla-7,24-dien-23-one
C19H18O8 (374.35). Pharm: Anti-HIV-1 inactive. Source: TAI GUO ZHI ZI
C30H48O3 (456.72). White powder, mp 80~82C, []D26 = +33.3 (c = 0.45,
Gardenia thailandica (leaf and twig). Ref: 4963.
CH3OH). Source: HAI NAN JIAN MU Dysoxylum hainanense (bark). Ref:

3987.
OH
O
O
HO
OH
O
HO
6150 5,7-Dihydroxy-6,8,2',3'-tetramethoxyflavone
6155 23,26-Dihydroxy-tirucalla-7,24-dien-3-one
72.5 (c = 0.29, CH3OH). Source: HAI NAN JIAN MU Dysoxylum
hainanense (bark). Ref: 3987.
O
HO
O
O
OH
6151 3,4-Dihydroxy-6,7,3',4'-tetramethoxyflavonol
OH
OH
C19H20O7 (360.37). Source: HUANG HUA HAO Artemisia annua. Ref: 2, 660.
6156 3,19-Dihydroxy trachylobane
O
O
C20H32O2 (304.48). mp 149~150C, []D18 = 35 (c = 4, CHCl3:MeOH = 1:1).
Source: CHANG SUI BA DOU Croton macrostachys. Ref: 3983, 4552.
OH
OH
6152 (24Z)-3,27-Dihydroxy-7,24-tirucalladien-21-al
HO
C30H48O3 (456.72). Source: KU SHU PI Picrasma quassioides [Syn.
OH
Picrasma ailanthoides]. Ref: 12.
6157 217-Dihydroxy-9,10,13-triacetoxy-5-(3'-N,N-dimethylamino3'-phenyl)-propionyloxytaxa-4(20),11-diene
O
OH
C37H51NO10 (669.82). Amorphous powder, []D22 = +39 (c = 0.1, CHCl3).

Source: JIA NA DA HONG DOU SHAN Taxus canadensis (needle leaf). Ref:
3886.
H
HO
HO
6158 3',6-Dihydroxy-2,4,4'-trimethoxybenzophenone
C16H16O6 (304.30). Pale yellow solid, mp 161~162C. Source: DAO NIAN ZI
Garcinia mangostana (heartwood). Ref: 5311.
O
HO
HO
H
H OH
hainanense (bark). Ref: 3987.
31.0 (c = 0.45, CHCl3). Source: HAI NAN JIAN MU Dysoxylum
OH
O O
6153 3,25-Dihydroxy-tirucalla-7,23-diene
HO
171
6159 (2S)-5,2'-Dihydroxy-7,4',5'-trimethoxyflavanone
6163 2,6-Dihydroxy-1,5,7-trimethoxyphenanthrene
C18H18O7 (346.34). Crystalline solid, mp 192~193 C, []D25 = 8.5 (c = 0.11,
MeOH). Pharm: AChE inhibitor (in vitro, IC50 = (11.60.6)mol/L, control
(stem). Ref: 5171.
Galanthamine, IC50 = (32.22.5)mol/L); BChE inhibitor (in vitro, IC50 =

(15.72.0)mol/L, control Galanthamine, IC50 = (163.05.0)mol/L). Source:
CU YING MAO DIAN ZI CAO Onosma hispida (whole herb). Ref: 4333.
HO
OH
OH
HO
6164 1,3-Dihydroxy-2,4,7-trimethoxyxanthone
C16H14O7 (318.29). Yellow solid. Pharm: Cytotoxic (in vitro antiproliferative
activity, LoVo, IC50 = (34.62.3)mol/L, control Doxorubicin, IC 50 =
6160 5,3'-Dihydroxy-6,7,4'-trimethoxyflavanone
(0.040.005)mol/L; LoVo/Doxo, IC50 = (39.51.8)mol/L, Doxorubicin,
C18H18O7 (346.34). Pharm: Cytotoxic (in vitro, PC12, GI50 = 2.27g/mL,
IC50 = (10.20.1)mol/L). Source: PU TONG YUAN ZHI Polygala vulgaris.
control Cisplatin, GI50 = 0.111g/mL; HCT116, GI50 = 2.87g/mL, control
Ref: 4246.
Cisplatin, GI50 = 0.794g/mL). Source: DAN YE MAN JING ZI Vitex
rotundifolia [Syn. Vitex trifollia var. simplicifolia] (seed: yield = 0.0017%dw).
Ref: 4623.
O
O
OH
OH
O
OH
3,8-Dihydroxy-2,4,6-trimethoxyxanthone C16H14O7 (318.29). Pharm:

OH
Cytotoxic (P388 ED50 = 5.11g/mL, control Mithramycin ED50 = 0.06g/mL,
6161 5,2'-Dihydroxy-6,7,8-trimethoxyflavone
HT29 ED50 = 6.25g/mL, Mithramycin ED50 = 0.08g/mL)[4094]. Source:
SHAN ZHU ZI Garcinia multiflora (stem: yield = 0.000021%dw), TAI WAN
O
O
LV DAO TENG HUANG Garcinia linii, YUAN ZHI Polygala tenuifolia. Ref:
HO
2, 4094, 4708.
O
OH
OH
6162 5,6-Dihydroxy-7,3',4'-trimethoxyflavone
[25782-23-4] C18H16O7 (344.32). Pale yellow powder, mp 244~247C.
HO
Pharm: PFTase inhibitor (100g/mL,InRt = 62%, IC50 = 25g/mL)
[5378]
cytotoxic (inhibits growth of hmn cancer cells: SW620, GI50 = (9.51.0)mol/L,

control Adriamycin, GI50 = 0.34mol/L; A549, GI50 = (19.32.0)mol/L,
Adriamycin, GI50 = 0.21mol/L; PC3, GI50 = (13.41.0)mol/L, Adriamycin,
C16H14O7 (318.29). Yellow needles (EtOH), mp 165~169C Source: CHUAN
GI50 = 0.39mol/L; LOX-IMVI, GI50 = (4.90.5)mol/L, Adriamycin, GI 50 =
DONG ZHANG YA CAI Swertia davidii. Ref: 2237.
0.12mol/L; HCT15, GI50 = (8.80.6)mol/L, Adriamycin, GI50 =

0.84mol/L)[5378]; cytotoxic inactive (hmn breast cancer cell lines:
MDA-MB-231, MCF7, T47D, 20g/mL)[5378]; angiogenesis inhibitor inactive
OH
OH
(chicken embryo chorioallantoic membrane (CAM) assay, 10g)[5378];
antineoplastic (nude mouse, hmn tumor xenograft model, SW620 hmn colon
O
O
cancer cell, 0.5% tween 80, ip 60mg/(kgd), for 22 days, reduces tumor
volume 44.6% at final day and no loss of body weight; good candidate as
antitumor agents)[5378]. Source: AI YE Artemisia argyi, Thymus piperella,
6167 5,7-Dihydroxy-2,6,8-trimethylchromone
Thymbra spp. Ref: 1521, 5378.
8-Methyleugenitol C12H12O4 (220.23). Source: CUI YUN CAO Selaginella

uncinata (whole herb). Ref: 4398.
O
O
O
HO
HO
OH
OH
172
6168 7,23-Dihydroxy-3,11,15-trioxolanosta-8,20E(22)-dien-26-oic acid
6172 2,3-Dihydroxyurs-12,20(30)-dien-28-oic acid 3-O-{O--L-arabi-
nopyranosyl-(12)-O-[-D-xylopyranosyl-(13)]-D-glucopyranoside}
MeOH). Source: SHU SHE Ganoderma applanatum (sporocarp: yield =
C46H72O17 (897.08). []D25 = +28 (c = 1, MeOH). Source: CI HUA LIAN ZI
0.00057%). Ref: 4756.
CAO Alternanthera repens. Ref: 2336.

O
HO
OH
O
HO
OO
O
OH
OH
OH
OO
O
OH
HO
OH
O
OH
O
OH
OH
6169 3,19-Dihydroxyursan-28-oic acid
OH
C30H50O4 (474.73). Source: WU SE MEI Lantana camara. Ref: 744.
6173 2,3-Dihydroxyurs-12,20(30)-dien-28-oic acid 3-O-{O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(12)-O-[-D-xylopyranosyl(13)]-D-glucopyranoside}
OH
C52H82O22 (1059.22). []D25 = +19.0 (c = 1, MeOH). Source: CI HUA LIAN
OH
H
HO
ZI CAO Alternanthera repens. Ref: 2336.
HO
OH
6170 2,3-Dihydroxyurs-12,19-dien-23,28-oic acid
HO
OH
chroosepalus. Ref: 866.
OO
OO
C30H44O6 (500.68). White powder, mp 320C. Source: MAO E MEI Rubus

OH
OH
OH
H
HO
OH
6174 2,3-Dihydroxyurs-12,20(30)-dien-28-oic acid 3-O-{O--D-quino-
HO
OO
OH
OH
OH OO
OH
OH
HO
HO
vopyranosyl-(12)-O--L-arabinopyranosyl-(12)-O-[-D-xylopyranos-
yl-(13)]-D-glucopyranoside}
6171 2,3-Dihydroxyurs-12,20(30)-dien-28-oic acid 3-O-{[O--D-xylo-
pyranosyl-(13)]-D-glucopyranoside}
H
HO
H
HO
H
HO
H
HO
OO
OH
OH
OH
OH
OO
OH
OH
OH
OO
OO
OH
OH
OH
O
O
OH
OH
OO
OH
OH
OH
O
OH
173
6179 4,8-Dihydroxy-6-vanilloyloxydauc-9-ene
6175 3,19-Dihydroxyurs-12-en-24,28-dioic acid

Ilexgenin A [108524-94-3] C30H46O6 (502.70). Powder, mp > 300C,
[]D20
+30.8 (c =0.97, pyridine). Source: MAO DONG QING Ilex pubescens. Ref: 1521.
C23H32O6 (404.51). Source: YI LANG A WEI Ferula kuhistanica (root).

Ref: 3977.
HO
OH
O
OH
OH
HO
O
O
HO
HO
6176
H
O
3,19-Dihydroxyurs-12-en-28-oic acid 28--D-glucopyranosyl
6180 4,8-Dihydroxy-6-vanilloyloxydauc-9-ene
ester
C23H32O6 (404.51). Source: YI LANG A WEI Ferula kuhistanica (stem).
C36H58O9 (634.86). Pharm: Cytotoxic (HSC-2, IC50 = 50g/mL; HGF, IC50 >
Ref: 3977.
200g/mL). Source: DI YU Sanguisorba officinalis. Ref: 5160.

HO
OH
O
H
H
HO
O
O
HO
OH
OH
HO
O
O
OH
OH
6177 19,24-Dihydroxyurs-12-en-3-one-28-oic acid
6181 1,5-Dihydroxyxanthone
C30H46O5 (486.70). Colorless prisms, mp 189.5~191.0C, []D17.6 = 27.4 (c =
1.55, acetone). Source: DU JUAN HUA YE Rhododendron simsii. Ref: 749.

ED50 = 0.08g/mL)[4094]; antifungal (Aspergillus fumigatus CBS113.26, MIC80
= 16g/mL, control Amphotericin B, MIC80 = 8g/mL; Aspergillus flavus
HO
Aspergillus niger IHEM2951, MIC80 = 31g/mL, Amphotericin B, MIC80 =
H
O
IHEM37.19, MIC80 = 16g/mL, Amphotericin B, MIC80 = 8g/mL;
OH
16g/mL; Aspergillus terreus 5029.2000, MIC80 = 62g/mL; Amphotericin B,

MIC80 = 16g/mL; Candida albicans ATCC663.90, MIC80 = 62g/mL;
Amphotericin B, MIC80 = 1g/mL)[4995]. Source: FEI ZHOU HUANG GUO
OH
6178 2,19-Dihydroxyursolic acid

Tormentic acid [13850-16-3] C30H48O5 (488.71). Yellowish crystalline
powder, mp 265~269C; 273C; 288~289C, []D15 = 17.3 (c = 0.2,
pyridine); colorless crystals powder, mp 260~262C (methanolwater), 273C,
[]D = 20 (pyridine). Pharm: Antibacterial (Streptococcus var.);
[900]
hypoglycemic (rat, orl, 10mg/kg)
MU Mammea Africana, HAI TANG GUO Calophyllum inophyllum (root

cortex and nut), MEI ZHOU MAN MI PING GUO Mammea americana, SU
GE LAN HU TONG Calophyllum caledonicum (stem cortex), TAI WAN LV
DAO TENG HUANG Garcinia linii, TIE LI MU Mesua ferrea., Mesua
thwaitesii, Calophyllum spp., Garcinia spp. Ref: 1521, 3866, 4094, 4995.
. Source: BAN BIAN SU Elsholtzia

O
ciliata, CU YE XUAN GOU ZI Rubus alceaefolius, PI PA YE Eriobotrya
OH
japonica, QIANG WEI GEN Rosa multiflora, SHAN DI XIANG CHA CAI
Isodon oresbia, SHUI YANG MEI Geum japonicum, TUN XING GUO
Pygeum topengii, WU LING ZHI Trogopterus xanthipes; Pteromys volans,
O
OH
XIN ZANG JIA ZI CAO Arnebia euchroma, ZE LAN Lycopus lucidus. Ref: 6,
447, 592, 595, 606, 637, 900.
(stem). Ref: 5238.
HO
H
HO
OH
HO
HO
OH
174
6189 Diisocapryl phthalate
Euxanthone [529-61-3] C13H8O4 (238.21). Pharm: Cytotoxic (P388 ED50 =
[27554-26-3] C24H38O4 (390.57). Source: SAN QI Panax pseudo-ginseng var.
1.21g/mL, control Mithramycin ED50 = 0.06g/mL, HT29 ED50 = 3.94g/mL,
Mithramycin ED50 = 0.08g/mL)[4094]; cytotoxic inactive (hmn small cell lung
[5061]
cancer NCI-H187 cell line, control Ellipticine, IC50 = (0.350.15)g/mL)
anti-inflammatory. Source: CHAN YI TENG Securidaca inappendiculata (stem),
DA HUA GE NA XIANG Goniothalamus griffithii, MEI ZHOU MAN MI
PING GUO Mammea Americana, QIAO MU ZHUANG HUANG NIU MU

Cratoxylum arborescens (stem cortex), TAI WAN LV DAO TENG HUANG
6190 4,4'-Diketo-3-hydroxy--carotene
Garcinia linii. Ref: 658, 4094, 5061, 5238, 5453.
C40H52O3 (580.86). Source: JIN YU Carassius auratus. Ref: 6.
OH
O
HO
O
HO
C19H18O10 (406.35). Yellow amorphous powder, mp 265~266C. Source: DI ER

CAO Hypericum japonicum, HENG LI DI ER CAO Hypericum henryi. Ref: 775.
O
OH
6184 1,5-Dihydroxyxanthone-6-O--D-glucoside
6191 Diketouncaric acid

C30H42O7 (514.67). Source: CHANG HUA GOU TENG Uncaria longiflora,
TUO YUAN GOU TENG Uncaria elliptica, Uncaria thwaitesii. Ref: 5341.
HO
OO
HO
OH
OH
HO
OH
OH
OH
6185 Dihydroyashabushiketol
1,7-Diphenyl-5-hydroxy-3-heptanone C19H22O2 (282.39). Yellow oil, []D20 =
3 (c = 0.7, MeOH). Pharm: 5-Reductase inhibitor (rat prostate
5-Reductase, IC50 = (23070)mol/L, control Curcumin, IC50 > 1000mol/L,
Finasteride, IC50 = 0.01mol/L). Source: GAO LIANG JIANG Alpinia
officinarum. Ref: 5345.
O
O
6192 (Z,Z')-Diligustilide
OH
6186 3,3'-Diiodothyronine
O
C15H13I2NO4 (525.08). Source: NIU YE Bos taurus domesticus; Bubalus
bubalis. Ref: 6.
6193 Dillapiol
O
I
I
HO
Dillapiole [484-31-1] C12H14O4 (222.24). Oil, mp 29.5C, bp 285C, bp

OH
NH2
[66-02-4] C9H9I2NO3 (432.99). mp (+) 202C (dec), () 213C (dec), ()

202C (dec). Source: NIU YE Bos taurus domesticus; Bubalus bubalis. Ref: 6.
O
hexobarbital, ED50 = 1.57mg/kg). Source: DA YE XIANG RU Mosla

dianthera, GOU ZHUANG HU JIAO Piper aduncum, HUI XIANG GEN
Foeniculum vulgare, JIAN ZI SU Perilla frutescens var. acuta [Syn. Perilla
frutescens var. purpurascens], SHI LUO ZI Anethum graveolens, SU GE
OH
NH2
HO
mutation (100mol/L, Ames InRt = 43.4%); molluscacide (10mg/L); synergist

of pyrethrin; sedative; hypnotic (prolongs sleeping time induced by
6187 Diiodotyrosine
162C/11mmHg, bp 100C/0.8mmHg. Pharm: Antihepatotoxin; inhibits
LAN DANG GUI Ligusticum scoticum, TAI WAN JI NING Orthodon

formosanus, XIN HE LAN HU JIAO Piper nove-hollandae, YA DAN ZI
Brucea javanica [Syn. Brucea sumatrana; Rhus javanica], Erigeron sp. Ref: 6,
658, 900.
6188 1,5-Di-isobutyl-3,3-dimethyl[3,1,0]cyclohexadione
C16H26O2 (250.38). Source: DANG SHEN Codonopsis pilosula. Ref: 2.
O
O
O
O
175
6194 Dimelic acid
6198 7,12-Dimethoxy-8,11,13-abietatrien-11-ol
Heptanedioic acid [111-16-0] C7H12O4 (160.17). Prisms (H2O), mp
C22H34O3 (346.51). Source: DU SONG SHI Juniperus rigida. Ref: 6.
104~105C, bp 212C/10mmHg, pKa1 = 4.46, pKa2 = 5.58 (25C). Source: BI
MA ZI Ricinus communis, Anthyllis sericea. Ref: 658, 1521.

O
HO
HO
OH
6195 Dimeric 4,2',4'-trihydroxydihydrochalcone

rel-(1,2)-Di-(2,4-dihydroxybenzoyl)-rel-(3,4)-di-(4-hydroxyphenyl)-cycl
6199 7,7''-Dimethoxyamentoflavone
obutane C30H24O8 (512.52). Yellow oil. Source: FEI ZHOU BAI ZI LIAN
C32H22O10 (566.53). Source: YUN NAN SUI HUA SHAN Amentotaxus
Agapanthus africanus (root). Ref: 5279.
yunnanensis (leaf and twig: yield = 0.020%dw). Ref: 4707.

OH
HO
OH
OH
O
O
HO
OH
O
OH
OH
OH
OH
6200 2,6-Dimethoxy benzoic acid
6196 Dimer iridoid glucoside 10
C9H10O4 (182.18). Pharm: Antioxidant (hydroxyl radical scavenger, IC50 =
C37H48O23S2 (924.91). Yellow powder, []D20 = 5.7 (c = 1.00, MeOH).
1.51mol/L, control EGCG, IC50 = 0.43mol/L, superoxide anion radical
Source: JI SHI TENG Paederia scandens. Ref: 1963.
scavenger, IC50 = 3.21mol/L, control EGCG, IC50 = 0.53mol/L). Source:

XIAN MAO Curculigo orchioides (rhizome). Ref: 4499.
O
HO
O
O
S
O
O
HO
6201 3,4-Dimethoxybenzoic acid
OH
O
S
OH
Veratric acid C9H10O4 (182.18). Pharm: NO production inhibitor inactive

OH
(LPS-activated macrophage-like J774.1 cells, IC50 = 129g/mL, control

L-NMMA, IC50 = 27.4g/mL) [4473]. Source: CHANG BAN JIN LIAN HUA
Trollius macropetalus, CHOU LENG SHAN Abies nephrolepis, HE SE
OH
OH
H
O
OH H
OH
ZHONG HUA SHU Tabebuia avellanedae (inner bark), HONG CHE ZHOU
OH
CAO Trifolium pratense, JIN LIAN HUA Trollius chinensis [Syn. Trollius
6197 Dimer iridoid glucoside 12
asiaticus var. chinensis], SANG HUANG Phellinus igniarius, TAI WAN GE
C36H44O22S2 (892.87). Yellow powder, []D20 = 108.9 (c = 0.54, MeOH).
NA XIANG Goniothalamus amuyon (fresh leaf: yield = 0.00012%fw)[4686].
Source: JI SHI TENG Paederia scandens. Ref: 1963.
Ref: 660, 4473, 4686.
O
O
H
HO
OH
6202 3,5-Dimethoxybenzoic acid

C9H10O4 (182.18). Source: DIAN NAN HONG HOU KE Calophyllum
polyanthum (seed: yield = 0.0017%dw). Ref: 4767.
OH
O
OH
O
S
O
O
OH
O
OH
O
HO
OH
OH
O
O
OH
176
6203 6,7-Dimethoxy-2H-1-benzopyran-2-one
6206 -D-[5-O-(3,4-Dimethoxybenzoyl)]-apiofuranosyl-(16)--D-
[120-08-1] C11H12O4 (208.22). Pharm: -Glucosidase inhibitor (type VI, IC50
glucopyranosyl
= 0.44mmol/L, control 1-Deoxynojirimycin, IC50 = 0.3mmol/L); thrombin
inhibitor inactive; -glucuronidase inhibitor inactive[4155]. Source: YUN NAN
Source: BAN ZHEN ZHONG HUA SHU Tabebuia impetiginosa (bark). Ref:
TU SI ZI Cuscuta reflexa. Ref: 4155.
3817.
OH
O
O
6204 2,6-Dimethoxybenzoquinone
OH
OH OH
2,6-Dimethoxy-p-benzoquinone [530-55-2] C8H8O4 (168.15). Yellow needles,
OO
OH
OH
mp 260C, easy to sublimation when heated. Pharm: Cytotoxic (P388 in vitro);

Cytotoxic (K562 cells, IC50 = 25.50g/mL)[4600]; cytotoxic (P388, ED50 =
6207 2''-O-(3''',4'''-Dimethoxybenzoyl)orientin
0.12g/mL, control Mithramycin, ED50 = 0.08g/mL; HT29, ED50 =
C30H28O14 (612.55). Yellow powder, mp 202~204C, []D20 = 72.2 (c =
3.97g/mL, Mithramycin, ED50 = 0.07g/mL; A549, ED50 = 10.57g/mL,
0.054, CH3OH). Source: DUAN BAN JIN LIAN HUA Trollius ledebourii
[4947]
Mithramycin, ED50 = 0.06g/mL)
; platelet aggregation inhibitor (washed
(flower: yield = 0.00033%dw). Ref: 4743.

O
rabbit platelets, 50g/mL, 100mol/L AA-induced, AggRt = 100%, control

O
50mol/L Aspirin, AggRt = 100%; 10g/mL collagen-induced, AggRt = 100%,

100mol/L Aspirin, AggRt = 4.9%; 0.1U/mL thrombin-induced, AggRt =
100%, 100mol/L Aspirin, AggRt = 1.7%; 2ng/mL PAF-induced, AggRt =
HO
100%, 100mol/L Aspirin, AggRt = 2.1%)[5427]. Source: CHUN FU SHOU
OH OH
O
O
OH
OH
OH
CAO Adonis vernalis, CUI TU LUO FU MU Rauvolfia vomitoria, CHU BAI

PI Ailanthus altissima, CI WU JIA Acanthopanax senticosus [Syn.
Eleutherococcus senticosus], JIAN YE CEN Fraxinus szaboana [Syn.
Fraxinus chinensis var. acuminata], MI MAI E ZHANG CHAI Schefflera
venulosa (stem cortex), XIAO MAI Triticum aestivum [Syn. Triticum vulgare],
PI ZHEN XING YAO HUA Wikstroemia lanceolata (stem and root), SAN QI
CAO Gynura segetum [Syn. Gynura japonica] (rhizome). Ref: 2, 6, 658, 660,
OH
6208 2''-O-(3''',4'''-Dimethoxybenzoyl)vitexin
C30H28O13 (596.55). Pale yellow powder, mp 277~279C, []D20 = 182.7 (c
= 0.064, CH3OH). Source: DUAN BAN JIN LIAN HUA Trollius ledebourii
(flower: yield = 0.00073%dw). Ref: 4743.
O
4600, 4947, 5427.
O
OH OH
O
O
O
O
HO
OH
OH
OH
6209 2,4-Dimethoxybenzyldehyde
6205 6-O-(3,4-Dimethoxybenzoyl)-ajugol
C24H32O12 (512.52). Pharm: NO production inhibitor (LPS-activated
[613-45-6] C9H10O3 (166.18). mp 71C, bp 165C/10mmHg. Source: XIANG

GEN QIN Osmorhiza aristata var. laxa. Ref: 6.
macrophage-like J774.1 cells, IC50 = 15.1g/mL, control L-NMMA, IC50 =

27.4g/mL)[4473]. Source: HE SE ZHONG HUA SHU Tabebuia avellanedae
(inner bark). Ref: 4473.
O
O
O
O
O
6210 3-(3,4-Dimethoxybenzyl)-5,7-dihydroxychroman-4-one
O
O
HO
C18H18O6 (330.34). White powder, mp 183~185C, []D25 = 74.7 (c = 0.39,

MeOH). Source: Scilla nervosa (bulb). Ref: 2381.
OO
HO
HO
OH
OH
O
OH
OH
177
6211 [(2S,3R,4R)-4-(3,4-Dimethoxybenzyl)-2-(3,4-dimethoxyphenyl)-
6215 9,10-Dimethoxycanthin-6-one
tetrahydrofuran-3-yl]-methyl (2Z)-2-methylbut-2-en-oate
C16H12N2O3 (280.29). Source: CHANG YE KUAN MU Eurycoma longifolia
C27H34O7 (470.57). Pharm: Anti-Inflammatory (anti-oedema, control oedema
(root: yield = 0.000019%dw), Eurycoma harmandiana (root). Ref: 4728,
= (7.80.3)mg, 100g/cm2, oedema = (4.00.6)mg, p<0.05, reduction = 49%,
5137.
[4985]
Indomethacin oedema = (3.40.3)mg, p<0.05, reduction = 56%)
leukotriene biosynthesis Inhibitor (in vitro, IC50 = 10.7mol/L, p<0.05, control

Zileuton, IC50 = 10.4mol/L, p<0.05)
[5037]
. Source: GAO SHAN HUO RONG
CAO Leontopodium alpinum (root). Ref: 4985, 5037.
O
O
N
O
6216 3',5'-Dimethoxy-cinnamic acid pyrrolidine

O
C15H19NO3 (261.32). Pharm: Platelet aggregation inhibitor (rbt platelets
induced by thrombin, 100g/mL, add thrombin 0.1u/mL, AggRt =

(92.60.4)%, control AggRt = (92.60.4)%; add AA, 100mol/L, 100g/mL,
AggRt = (85.20.9)%, control AggRt = (87.80.3)%, Aspirin 50g/mL,

O
O
AggRt = (11.710.1)%; add collagen 10g/mL, 100g/mL, AggRt =

(86.91.2)%, control AggRt = (89.30.5)%, Aspirin 100g/mL, AggRt =
(81.30.5)%; add PAF 2ng/mL, 100g/mL, AggRt = (91.50.3)%, control

AggRt = (93.00.6)%). Source: TAI WAN HU JIAO Piper taiwanense (stem).
6212 [(2S,3R,4R)-4-(3,4-Dimethoxybenzyl)-2-(3,4,5-trimethoxyphen-
Ref: 4938.
yl)-tetrahydrofuran-3-yl]-methyl (2Z)-2-methylbut-2-en-oate
C28H36O8 (500.59). Colorless gum, []D20 = +20.86, (c = 0.302, MeOH).

Source: GAO SHAN HUO RONG CAO Leontopodium alpinum (root). Ref:
5037.
O
O
6217 2,6-Dimethoxy-4,4-dihydroxychalcone
O

HT1080, ED50 = 50.5mol/L)[3042]. Source: YUN NAN CAO KOU Alpinia
blepharocalyx (seed: yield = 0.00018%~0.0129%). Ref: 3042, 3048.

O
O
OH
O
HO
O
O
6213 3',5'-Dimethoxy-biphenyl-4-ol
C14H14O3 (230.27). White powder. Pharm: Cytotoxic (in vitro
6218 3,8-Dimethoxy-5,7-dihydroxy-3',4'-methylenedioxyflavone
antiproliferative activity, LoVo, IC50 > 40mol/L, control Doxorubicin, IC50
C18H14O8 (358.31). Yellow crystals. Source: RU NI WENG DAO MI ZHU
= (0.040.005)mol/L). Source: PU TONG YUAN ZHI Polygala vulgaris.
YU Melicope coodeana. Ref: 1975.
Ref: 4246.
O
O
O
HO
O
O
OH
6219 2,3-Dimethoxy-9,10-dihydroxy-N-methyl-tetrahydroprotoberbe-
HO
rine quaternary salt

6214 5,9-Dimethoxycanthin-6-one
C16H12N2O3 (280.29). Source: Eurycoma sp. Ref: 4556.
Haitinosporine C20H24NO4+ (342.42). White crystals, mp 242~245C. Source:

HAI NAN QING NIU DAN Tinospora hainanensis. Ref: 408.
O
+
OH
O
O
OH
178
6220 2,2'-Dimethoxy-3,3'-dihydroxy-5,5'-oxygen-6,6'-biphenylformic
6225 2',5'-Dimethoxyflavone
anhydride
C17H14O4 (282.30). Light yellow solid (CHCl3). Source: HUANG HUA JIU
C16H10O8 (330.25). White powder, mp 296.5~298.0C. Source: DA JI(3)
LUN CAO Primula veris [Syn. Primula officinalis] (leaf). Ref: 5275.
Euphorbia pekinensis. Ref: 360.

O
O
HO
OH
6226 3',4'-Dimethoxyflavone
6221 (1aS*,1bS*,7aS*,8aS*)-4,5-Dimethoxy-1a,7a-dimethyl-1,1a,1b,2,
C17H14O4 (282.30). White crystalline solid (CHCl3). Source: HUANG HUA
7,7a,8,8a-octahydrocyclopropa[3,4]cyclopenta[1,2-b]naphthalene-3,6-
JIU LUN CAO Primula veris [Syn. Primula officinalis] (leaf). Ref: 5275.
dione
O
C18H22O4 (302.37). Yellowish oil. Pharm: Cytotoxic (B-16 IC50 = 1.30g/mL,
control Doxorubicin IC50 = 0.03g/mL; MCF7 IC50 = 5.04g/mL,

O
Doxorubicin IC50 = 0.20g/mL; HCT8 IC50 = 2.49g/mL, Doxorubicin IC50 =

0.04g/mL; HL-60 IC50 = 1.56g/mL, Doxorubicin IC50 = 0.02g/mL; CEM
IC50 = 1.24g/mL, Doxorubicin IC50 = 0.02g/mL). Source: QIU ZHUANG
PO BU MU Cordia globosa (root). Ref: 5043.
O
6227 6,14-Dimethoxyforesticine
C26H43NO6 (465.64). White powder, []D18 = +27.2 (c = 0.31, EtOH). Source:
BAI HOU WU TOU Aconitum leucostomum. Ref: 483.
H
O
6222 3,5-Dimethoxy-2'',2''-dimethylpyrano-(5'',6'':8,7)-flavone
C22H20O5 (364.40). Viscous yellowish oil. Source: Lonchocarpus latifolius
O
H
(root). Ref: 5108.
OH
H
O
6228 (2S)-5,7-Dimethoxy-8-formylflavanone
O
O
Anticancer Flavonoid PMV70P691-016 C18H16O5 (312.33). Yellow oil, []D
= 28.0 (c = 0.10, MeOH). Pharm: Cytotoxic (in vitro, Hepa 1c1c7 mouse
hepatoma cells, IC50 > 10g/mL, CD = 2.6g/mL, CI > 3.9; control
6223 2,7-Dimethoxy-1,6-dimethyl-5-vinylphenanthrene
Sulforaphane, IC50 = 2.1g/mL, CD = 0.087g/mL, CI = 24.1)[4721]; cytotoxic
(quinone reductase induction assay in cultured Hepa1c1c7 mouse hepatoma
cells)[5038]. Source: SHUI LIU DOU Pongamia pinnata (stem cortex: yield =
0.0001%)[4721]. Ref: 4721, 5038.
O
O
6224 2,3-Dimethoxyellagic acid

3,4-Di-O-methylellagic acid C16H10O8 (330.25). mp > 300C. Source: BA
WANG BIAN Euphorbia royleana, WU JIU MU GEN PI Sapium sebiferum.
Ref: 6.
6229 (2,3-trans-3,4-trans)-3,4-Dimethoxy-(2'',3'':7,8)-furanoflavan
C19H18O4 (310.35). Needles, []D20 = +21 (c = 0.4, CH2Cl2). Source:
Lonchocarpus latifolius (root). Ref: 5108.
O
O
O
OH
OH
O
O
O
O
179
6230 (+)-5,5'-Dimethoxy-9-O--D-glucopyranosyl lariciresinol
6235 (E)-3-(3',5'-Dimethoxy-4'-hydroxybenzylidene)-2-indolinone
C28H38O13 (582.61). Pharm: Anti-HSV-1 inactive (EC50 > 172mol/L). Source:
C17H15NO4 (297.31). Yellow column crystals mp 204~206C. Source: BAN
MA LAN GEN Baphicacanthus cusia [Syn. Strobilanthes cusia]. Ref: 2577.
LAN GEN Isatis indigotica. Ref: 2119.

O
O
O
HO
HO
O
O
HO
O
OH
OH
6236 5,6-Dimethoxy-7-hydroxycoumarin
C11H10O5 (222.20). Source: HUANG HUA HAO Artemisia annua. Ref: 2.
OH
OH
6231 (+)-5,5'-Dimethoxy-9-O--D-glucopyranosyl secoisolariciresinol
HO
C28H40O13 (584.62). Source: MA LAN GEN Baphicacanthus cusia [Syn.
6237 4,4-Dimethoxy-3'-hydroxy-7,9':7',9-diepoxylignan-3-O--D-gluco-
Strobilanthes cusia]. Ref: 2577.
pyranoside
C26H32O11 (520.54). White amorphous powder, []D21 = 54.69. Source: DA
YE XIAN MAO Curculigo capitulata [Syn. Leucojum capitulata]. Ref: 2493.
OH
HO
O
HO
O
O
OH
OO
HO
OH
OH
OH
OH
OH
OH
OH
H
6238 6,8-Dimethoxy-10-hydroxyeremophil-7(11)-en-12,8-olide
6232 6,6'-Dimethoxygossypol
C17H26O5 (310.39). Colorless plates, mp 164~166C (Me2CO), [] D20 =
C32H34O8 (546.62). mp 181~184C. Source: MIAN HUA GEN Gossypium
+166.7 (c = 0.27, Me2CO). Pharm: Antibacterial (Staphylococcus aureus,
herbaceum. Ref: 6.
antibacterial circle = 13~16mm; Bacillus subtilis, antibacterial circle =

13~16mm; Escherichia coli, antibacterial circle < 12mm). Source: JIAN YE
H
OH
OH
TOU WU GEN Ligularia sagitta. Ref: 5382.
HO
OH
OH
O
O
6233 1,5-Dimethoxy-3-hydroxybenzoic acid
6239 2,6-Dimethoxy-4-(2-hydroxyethyl)phenol 1-O--D-glucopyra-
C9H10O5 (198.18). Source: MAO GUO QI Acer nikoense (stem cortex). Ref: 4304.
noside
MeOH). Source: AN MO LE Phyllanthus emblica (root). Ref: 3065.
OH
HO
HO
OH
OH
6234 5,7-Dimethoxy-3-(4-hydroxybenzyl)chroman-4-one
C18H18O5 (314.34). Acetyl-: vitreous off-white solid. Source: Scilla nervosa.
Ref: 2328.
6240 7,4'-Dimethoxy-3'-hydroxyflavone
C17H14O5 (298.30). Yellow amorphous powder, mp 128~130C (MeOH);
colorless needles (MeOH), mp 190~192C. Source: WU CI ZHU YING HUA
Calliandra inermis, XIANG HE HUAN Albizzia odoratissima (root cortex).
HO
O
HO
C16H24O9 (360.36). Off-white amorphous powder, []D20 = +19.3 (c = 0.7,
OH
Ref: 2588, 4229.

O
O
O
O
OH
180
6241 6,4'-dimethoxy-5-hydroxyflavone 7-glucoside
6246 (2S)-5,7-Dimethoxy-8-(2S-hydroxy-3-methyl-3-butenyl)-flavanone
C23H24O11 (476.44). Yellow amorphous powder. Source: AI JI ZHONG ZHI
Anticancer Flavonoid PMV70P691-017 C22H24O5 (368.43). Yellow oil, []D
YUAN WEI Iris carthaliniae. Ref: 1880.
= 22.0 (c = 0.1, MeOH). Pharm: Cytotoxic (in vitro, Hepa 1c1c7 mouse
hepatoma cells, IC50 = 19.3g/mL, CD = 4.4g/mL, CI = 4.4; control
O
HO
OO
cells)[5038]. Source: SHUI LIU DOU Pongamia pinnata (stem cortex: yield =
OH
0.00036%). Ref: 4721, 5038.
OH
Sulforaphane, IC50 = 2.1g/mL, CD = 0.087g/mL, CI = 24.1)[4721]; cytotoxic
OH
OH
6242 2,5-Dimethoxy-4-hydroxy-[2'',3'':7,8]-furanoflavan
C19H18O5 (326.35). Colorless crystals, mp 135~136, []D28 = +42.1 (c = 0.3,
HO
O
MeOH). Source: HONG E JI XUE TENG Millettia erythrocalyx. Ref: 1937.

O
6247 (2S)-5,7-Dimethoxy-8-(2S-hydroxy-3-methyl-3-butenyl)-3',4'O
methylenedioxyflavanone
C23H24O7 (412.44). Yellow oil, []D = 36.0 (c = 0.1, MeOH). Source: SHUI
OH
LIU DOU Pongamia pinnata (stem cortex: yield = 0.00018%). Ref: 4721.
6243 7,4'-Dimethoxy-5-hydroxyisoflavone
C17H14O5 (298.30). Pale yellow crystals (CHCl3: petrol = 1:2, v/v), mp
145~146C. Source: MENG MAI ROU DOU KOU Myristica malabarica
HO
O
6248 4',5-Dimethoxy-3-hydroxy-6,7-methylenedioxyisoflavone
OH
C18H14O7 (342.31). Source: JUAN QIAO YUAN WEI Iris potaninii

6244 2,4'-Dimethoxy-3'-(2-hydroxy-3-methyl-3-butenyl)acetophenone
C15H20O4 (264.32). Yellow oil, []D25 = 25.0 (c = 0.04, MeOH). Pharm:
Prolyl endopeptidase inhibitor (flavobacterium origin, IC50 =
OH
(8450.005)mol/L, control Z-pro-prolinal, IC50 = (0.8840.025)mol/L);

Ref: 4179.
6249 4,8-Dimethoxy-7-hydroxy-2-oxo-2H-1-benzopyran-5,6-dicarboxylic acid

C13H10O9 (310.22). Source: XIAO DI YU Sanguisorba minor. Ref: 3385.
O
O
HO
O
H
OH
HO
O
HO
6245 (2S)-5,7-Dimethoxy-8-(2R-hydroxy-3-methyl-3-butenyl)-flavanone
C22H24O5 (368.43). Yellow oil, []D = 33.0 (c = 0.1, MeOH). Source: SHUI
LIU DOU Pongamia pinnata (stem cortex: yield = 0.00062%). Ref: 4721.
6250 2,6-Dimethoxy-4-hydroxyphenol-1-O--D-glucopyranoside
C14H20O9 (332.31). White powder. Source: XIAO YE SHI NAN Photinia
parvifolia (stem). Ref: 4553.
OH
O
HO
O
OO
HO
OH
OH
O
OH
181
6251 3,5-Dimethoxy-4-hydroxyphenol 1-O--D-(6'-O-galloyl)glucopyra-
6256 5,7-Dimethoxy-3-(4-methoxybenzyl)chroman-4-one
noside
3-(4-Methoxybenzyl)-5,7-dimethoxychroman-4-one C19H20O5 (328.37).
C21H24O13 (484.42). Source: YANG MEI SHU PI Myrica rubra (bark: yield =
Colorless gum, []D25 = 70.6 (c = 0.38, MeOH); mp 115~117C, []D = 50
0.012%). Ref: 4163.
(c = 0.3 l, MeOH). Source: Scilla nervosa (bulb). Ref: 2328, 2381.

O
OH
O
HO
O
OO
OH
HO
OH
OH
OH
6257 4,8-Dimethoxy-1-(2-methoxyethyl)--carboline
6252 eythro-2,2'-Dimethoxy-4-(3-hydroxy-1-propenyl)-4'-(1,2,3-trihydroxypropyl) diphenyl ether
C16H18N2O3 (286.33). Source: KU SHU PI Picrasma quassioides [Syn.


O
OH
OH
HO
O
OH
6253 threo-2,2'-Dimethoxy-4-(3-hydroxy-1-propenyl)-4'-(1,2,3-trihydroxypropyl) diphenyl ether

O
6258 6,7-Dimethoxy-2-[2-(4'-methoxyphenyl)ethyl]chromone
C20H20O5 (340.38). Colorless acicular crystals, mp 88~90C. Source: BAI MU
OH
OH
HO
O
N
H
OH
O
O
6254 7,4'-Dimethoxyisoflavone
Dimethoxydaidzein [1157-39-7] C17H14O4 (282.30). Acicular crystals
6259 10,11-Dimethoxy-1-methyldeacetylpicraline-3',4',5'-trimethoxy-
(ethanol), mp 154~156C. Pharm: Cytotoxic (Raji cells); cAMP
benzoate
phosphodiesterase inhibitor (rat heart, IC50 = 2.3mol/L). Source: CI GUO
GAN CAO Glycyrrhiza pallidiflora. Ref: 900.
O
O
O
O
O
O
O
6255 5,6-Dimethoxy-2-isopropenylbenzofuran
C13H14O3 (218.25). Source: ZHAI TOU TUO WU Ligularia stenocephala
(root). Ref: 4536.
6260 6,7-Dimethoxy-N-methyl-3,4-dioxo-1(2H)-isoquinolinone
C12H11NO5 (249.23). Yellow powder, mp 185~189C. Source: BIAN FU GE
GEN Menispermum dauricum. Ref: 3792.
O
O
O
O
N
O
O
182
6261 7,9-Dimethoxy-2,3-methylendioxybenzophenanthridine
6265 5,6-Dimethoxy-8-(3'-methyl-2'-oxobutyl) coumarin
C20H15 NO4 (333.35). Pharm: Platelet aggregation inhibitor; DNA
C16H18O5 (290.32). Source: JIU LI XIANG Murraya paniculata [Syn.
isomerase inhibitor; antibacterial; cytotoxic. Source: Zanthoxylum sp. Ref:
Chalcas paniculata]. Ref: 11.
2176.
O
O
O
O
6262 3,4-Dimethoxy-3',4'-methylenedioxy-7,9'-epoxylignan-9-ol
C22H26O5 (370.45). Pharm: Antineoplastic; cathartic; sthenic; pesticide;
ichthyotoxin; muscle relaxant. Source: Zanthoxylum sp. Ref: 2176.
6266 5,7-Dimethoxy-8-(3'-methyl-2'-oxobutyl)coumarin
C16H18O5 (290.32). Pharm: Platelet aggregation inhibitor (washed rabbit
platelets, induced by thrombin, AA, collagen and PAF, 100g/mL: thrombin
= 0.1U/mL, AggRt = (77.71.1)%, control, AggRt = (80.01.1)%; AA
=100mol/L, AggRt = (00)%, p<0.001, control, AggRt = (77.01.5)%;
collagen = 10g/mL, AggRt = (00)%, p<0.001, control, AggRt =
HO
O
O
(78.31.3)%; PAF = 1ng/mL, AggRt = (60.77.8)%, p<0.01, control, AggRt

= (82.51.5)%)[5417]. Source: JIU LI XIANG Murraya paniculata [Syn.
Chalcas paniculata], QI GUO JIU LI XIANG Murraya omphalocarpa (leaf).
Ref: 11, 5417.

6263 (2S)-5,7-Dimethoxy-3',4'-methylenedioxyflavanone
C18H16O6 (328.32). Colorless needles (CHCl3 ), mp 192~194C, []D25 =
18.5 (c = 0.1, MeOH). Pharm: Antibacterial (gram-positive bacteria:
O
O
Staphylococcus aureus, 30g/mL DIZ = 7mm, Bacillus subtilis, 30g/mL

DIZ = 7mm, Bacillus sphaericus, 30g/mL DIZ = 6mm, control
Penicillin G, 30g/mL DIZ = 12, 15, 14mm, respectively; gram-negative

bacteria: Pseudomonas aeruginosa, 30g/mL DIZ = 7mm, Klebsiella
6267 2,8-Dimethoxy-6-methyl-9-oxo-9H-xanthene-1-carboxylic acid
aerogenes, 30g/mL DIZ = 7mm, Chromobacterium violaceum, 30g/mL
methyl ester
DIZ = 8mm, control Penicillin G, 30g/mL DIZ = 24, 23, 24mm,
C18H16O6 (328.32). Stable yellow needles (CHCl3), mp 219~221C. Pharm:
respectively)
[3407]
; antifungal (Aspergillus niger, 100g/mL DIZ = 8mm,
Candida albicans, 100g/mL DIZ = 7mm, Rhizopus oryzae, 150g/mL
Cytotoxic inactive (brine shrimp Artemia salina lethality assay, 20g/mL or

200g/mL). Source: Xylaria sp. Ref: 3845.
inactive, control Clotrimazole, 100g/mL DIZ = 22, 25, 24mm,
respectively)[3407] . Source: CAI BAN YANG TI JIA Bauhinia variegata
(root cortex), JI MEI YUN SHI Caesalpinia pulcherrima. Ref: 3407,

3468.
O
O
6268 5,6-Dimethoxy-N-methylphthalimide
C11H11NO4 (221.21). Source: BIAN FU GE GEN Menispermum dauricum, SHUI
LIAN YE TONG Hernandia nymphaeifolia (trunk bark). Ref: 1521, 3792.

O
O
O
6264 7,8-Dimethoxy-3',4'-methylenedioxyflavone
C18H14O6 (326.31). Yellow amorphous powder, mp 252~254C (MeOH).
Source: XIANG HE HUAN Albizzia odoratissima (root cortex). Ref: 4229.

6269 2,5-Dimethoxy-6-methyl-3-tridecyl-1,4-benzoquinone
O
O
O
C22H36O4 (364.53). Pale yellow solid, mp 54~55C. Source: PI ZHEN DU

JING SHAN Maesa lanceolata. Ref: 1860.
O
O
O
O
183
6270 10,11-Dimethoxynareline
6275 2-[4,5-Dimethoxy-5-(3-phenyl-trans-allyl)cyclohexa-3,6-dien-2-on-
C22H24N2O6 (412.45). Light yellowish oil, []D = 56 (c = 1.57, CHCl3).
1-ylmethyl]-5-hydroxy-6-methoxy-3-phenylbenzofuran
Source: DA YE TANG JIAO SHU Alstonia macrophylla (leaf: yield =
C33H30O6 (522.6). Yellow amorphous solid, mp 78~83C, []D25 = +23.6 (c =
0.0112%). Ref: 3020.
0.44, CHCl3). Pharm: Testosterone 5-reductase inhibitor (25g/mL, InRt =

0.6%, 50g/mL, InRt = 3.8%, 100g/mL, InRt = 17%; control Glycyrrhetinic
acid, 25g/mL, InRt = 31.7%, 50g/mL, InRt = 64.7%, 100g/mL, InRt =

87.1%). Source: JIAO ZHI HUANG TAN Dalbergia cochinchinensis (stem:
yield = 0.0017%dw). Ref: 4716.
H
HO O
OH
6271 (2S)-4',4'-Dimethoxy-ongokein
(2S)-5-Hydroxy-2-(1'-hydroxy-4',4'-dimethoxycyclohexyl)-7-methoxychroma
n-4-one C18H24O7 (352.39). White amorphous powder, mp 52~55C, []D =
O
O
+51 (c = 0.36). Source: EN GE MU Ongokea gore (stem cortex and root).

Ref: 5308.
O
O
O
OH
6276 2-[4,5-Dimethoxy-2-(3-phenyl-trans-allyloxy)benzyl]-5-hydroxy-6-
6272 2,3-Dimethoxy-6-(3-oxo-butyl)-7,9,10,11,11a,12-hexahydrobenzo[f]
methoxy-3-phenylbenzofuran
pyrrolo[1,2-b]isoquinoline
C33H30O6 (522.6). Amorphous solid, mp 63~68C. Pharm: Testosterone
C22H27NO3 (353.47). Colorless needles, mp 164~166C, []D25 = 71.0 (c =
5-reductase inhibitor (25g/mL, InRt = 11.5%, 50g/mL, InRt = 15.9%,
0.0011, CHCl3). Pharm: Antiviral (tobacco mosaic virus (TMV), 500g/mL,
100g/mL, InRt = 18.1%; control Glycyrrhetinic acid, 25g/mL, InRt =
InRt = 15%). Source: NIU XIN PIAO ZI Cynanchum komarovii (aerial parts).
31.7%, 50g/mL, InRt = 64.7%, 100g/mL, InRt = 87.1%). Source: JIAO
Ref: 5241.
ZHI HUANG TAN Dalbergia cochinchinensis (stem: yield = 0.0012%dw).

Ref: 4716.
O
O
OH
O
O
6273 3,4-Dimethoxyphenol -D-apiofuranosyl(16)--D-glucopyranoside
25
C19H28O12 (448.43). White powder, []D = 58.9 (c = 0.68, MeOH). Source:
SHAN FAN GEN Symplocos caudata. Ref: 2535.

O
6277 4-(3,4-Dimethoxyphenyl)-but-1,3-diene
HO
OO
C12H14O2 (190.24). Pharm: Cytotoxic (A549, IC50 > 50mol/L, control
OH
Ellipticine, IC50 = 0.8mol/L; Col2, IC50 > 50mol/L, Ellipticine, IC50 =
OH
OH
OH OH
1.6mol/L; SNU638, IC50 = 44.7mol/L, Ellipticine, IC50 = 1.6mol/L;
6274 2,4-Dimethoxyphenol 1-O--D-[5-O-(3,4-dimethoxybenzoyl)]apiofuranosyl-(16)--D-glucopyranoside

BAN ZHEN ZHONG HUA SHU Tabebuia impetiginosa (bark). Ref: 3817.
O
O
O
O
OO
O
OH
OH OH
OH
OH
HT1080, IC50 = 7,9mol/L, Ellipticine, IC50 = 1.2mol/L)[4081]; COX-2

inhibitor (RAW264.7 cells, LPS-induced PGE2 production, IC50 =
20.68mol/L, control Celecoxib, IC50 = 0.52nmol/L)[4532]. Source: YE JIANG
Zingiber cassumunar (rhizome). Ref: 4081, 4532.
O
O
184
6278 (E)-4-(3,4-Dimethoxyphenyl)but-3-en-1-O--D-glucopyranoside
6282 ()-trans-3-(3,4-Dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl]
C18H26O8 (370.40). Pale yellow gum, []D25 = 21.4 (c = 0.23, MeOH).
cyclohex-1-ene
Pharm: COX-2 inhibitor inactive (RAW264.7 cells, LPS-induced PGE2
C24H28O4 (380.49). Pharm: Cytotoxic (A549, IC50 = 12.6mol/L, control
production, IC50 > 50mol/L, control Celecoxib, IC50 = 0.52nmol/L). Source:
Ellipticine, IC50 = 0.8mol/L; Col2, IC50 = 15.5mol/L, Ellipticine, IC50 =
YE JIANG Zingiber cassumunar (rhizome). Ref: 4532.
1.6mol/L; SNU638, IC50 = 8.7mol/L, Ellipticine, IC50 = 1.6mol/L;

HT1080, IC50 = 16.1mol/L, Ellipticine, IC50 = 1.2mol/L)[4081]; COX-2
inhibitor (RAW264.7 cells, LPS-induced PGE2 production, IC50 = 2.71mol/L,
control Celecoxib, IC50 = 0.52nmol/L)[4532]. Source: YE JIANG Zingiber
O
HO
cassumunar (rhizome). Ref: 4081, 4532.
O
OH
OH
OH
6279 (E)-4-(3,4-Dimethoxyphenyl)-but-3-en-1-ol
C12H16 O3 (208.26). Pharm: COX-2 inhibitor inactive (RAW264.7 cells,
LPS-induced PGE2 production, IC50 > 50mol/L, control Celecoxib, IC50

= 0.52nmol/L). Source: YE JIANG Zingiber cassumunar (rhizome). Ref:
6283 6,7-Dimethoxy-2-(2-phenylethyl) chromone
4532.
C19H18O4 (310.35). Colorless acicular crystals, mp 118~120C. Source: BAI

MU XIANG Aquilaria sinensis. Ref: 13, 660.
OH
O
O
6280 (E)-4-(3,4-Dimethoxyphenyl)-but-3-en-1-ol acetate
C14H18 O4 (250.30). Pharm: COX-2 inhibitor inactive (RAW264.7 cells,

LPS-induced PGE2 production, IC50 > 50mol/L, control Celecoxib, IC50
= 0.52nmol/L). Source: YE JIANG Zingiber cassumunar (rhizome). Ref:
6284 3,4,l-O-3,4-Dimethoxy-phenylethyl-6-O-cinnamoyl--D-gluco-
4532.
pyranose
C27H34O11 (534.57). Pharm: Cytotoxic (EAC, T/C = 240%; P388, ED50 =
16.1g/mL). Source: FAN SHI LIU ZI Psidium guajava. Ref: 3826.
O
O
HO
O
O
O
OO
OH
O
O
OH
6281 3,4-Dimethoxyphenyl 1-O--D-[5-O-(3,4-dimethoxybenzoyl)]-apiofuranosyl-(16)--D-glucopyranoside

C28H36 O15 (612.59). Amorphous powder, []D22 = 72.0 (c = 1.89,
6285 l-O-3,4-Dimethoxy-phenylethyl-4-O-3,4-dimethoxy
MeOH). Pharm: NO production inhibitor (LPS-activated macrophage-like

J774.1 cells, IC50 = 75.9g/mL, control L-NMMA, IC50 = 27.4g/mL)
[4473]
cinnamoyl-6-O-cinnamoyl--D-glucopyranose
Source: BAN ZHEN ZHONG HUA SHU Tabebuia impetiginosa (bark),
C36H40O12 (664.71). Amorphous off-white powder. Pharm: Cytotoxic (EAC,
HE SE ZHONG HUA SHU Tabebuia avellanedae (inner bark). Ref: 3817,
T/C = 220%; P388, ED50 = 17.3g/mL). Source: FAN SHI LIU ZI Psidium
4473.
guajava. Ref: 3826.

O
O
O
O
O
O
O
OH OH
OO
OH
OH
OH
O
O
O
OO
O
OH
OH
185
6286 3,4-Dimethoxyphenyl 1-O--D-[5-O-(4-hydroxybenzoyl)]-apio-
6290 3,9-Dimethoxypterocarpan
furanosyl-(16)--D-glucopyranoside
Homopterocarpin; Baphinitone [606-91-7] C17H16O4 (284.31). Needles
(petroleum ether or EtOH), mp 88~89C, mp 83~85C, []D22 = 225
Pharm: NO production inhibitor (LPS-activated macrophage-like J774.1 cells,
(CHCl3). Pharm: Antineoplastic; antifungal; hepatoprotective (mus primary
IC50 = 44.1g/mL, control L-NMMA, IC50 = 27.4g/mL)
[4473]
. Source: BAN
cultured hepatocytes, antihepatotoxin induced by D-galactosamine (GalN),
ZHEN ZHONG HUA SHU Tabebuia impetiginosa (bark), HE SE ZHONG
100mol/L, InRt = (19.92.0)%, weak, control Silybin, 100mol/L, InRt =
HUA SHU Tabebuia avellanedae (inner bark). Ref: 3817, 4473.
(77.05.5)%)[4095]. Source: ZI TAN Pterocarpus indicus, CHAO XIAN HUAI

Maackia amurensis, GUANG BU DING GONG TENG Erycibe expansa, MA
DAO SI WO CI DOU Swartzia madagascariensis, ZA JIAO CHE ZHOU
OO
O
OH
OH OH
OH
CAO Trifolium hybridum, Pericopsis angolensis. Ref: 5, 658, 1521, 4095

O
OH
O
H
OH
H
6287 3,4-Dimethoxyphenyl 1-O--D-[5-O-(4-methoxybenzoyl)]-apio-
furanosyl-(16)--D-glucopyranoside
6291 9,10-Dimethoxy-pterocarpane-3-O--D-glucoside
Pharm: NO production inhibitor (LPS-activated macrophage-like J774.1 cells,
C23H28O10 (464.47). Source: HUANG QI Astragalus membranaceus, MENG
IC50 = 38.2g/mL, control L-NMMA, IC50 = 27.4g/mL)
[4473]
. Source: BAN
ZHEN ZHONG HUA SHU Tabebuia impetiginosa (bark), HE SE ZHONG

HUA SHU Tabebuia avellanedae (inner bark). Ref: 3817, 4473.
HO
OO
O
O
OH OH
OO
OH
OH
OH
OH
GU HUANG QI Astragalus mongholicus. Ref: 2, 660.
H
H
OH
6292 (E)-3,4'-Dimethoxystilbene
C16H16O2 (240.30). Source: GE ZHI HUA DI QIAN Corsinia coriandrina.
Ref: 3888.
OH
6288 (E)-3-(3,4-Dimethoxyphenyl)-2-propen-1-yl (Z)-2-[(Z)-2-methyl-
2-butenoyloxymethyl] butenoate
C21H26O6 (374.44). Pharm: Anti-inflammatory (NF-B inhibitor, hmn
monocytes, prevents LPS-induced cytokines (IL-1, IL-6, TNF, IL-8) release
6293 3,5-Dimethoxystilbene
and PGE2 synthesis: unstimulated control: PGE2 = 0.54pg/mL, IL-6 =
[78916-49-1] C16H16O2 (240.30). Source: HAI SONG ZI Pinus koraiensis. Ref: 6.
0.97pg/mL, IL-1= 0pg/mL, TNF- = 0.02pg/mL, IL-8 = 3.45pg/mL; LPS
(10ng/mL): PGE2 = 19.24pg/mL, IL-6 = 71.42pg/mL, IL-1 = 3.61pg/mL,

TNF- = 2.66pg/mL, IL-8 = 235.18pg/mL; LPS (10ng/mL +compound
1g/mL): PGE2 = 6.58pg/mL, IL-6 = 52.23pg/mL, IL-1 = 1.25pg/mL,
TNF- = 1.18pg/mL, IL-8 = 158.3pg/mL). Source: GUAN MU CHAI HU
6294 3,5-Dimethoxytoluene
Bupleurum fruticosum (aerial parts). Ref: 5033.
[4179-19-5] C9H12O2 (152.19). Source: XI XIN Asarum sieboldii, LIAO XI

XIN Asarum heterotropoides var. mandshuricum. Ref: 2, 660.
O
O
6289 (S)-()-7,8-Dimethoxyplatydesmine
6295 7,4'-Dimethoxy-8,3',5'-trihydroxy-6-O--D-glucopyranosyliso-
C17H21NO5 (319.36). Pharm: Cytotoxic (P388 cell line, ED50 = 7.5g/mL,
flavone
control Mithramycin, ED50 = 0.06g/mL; HT29, ED50 = 28.3g/mL,
C23H24O13 (508.44). Amorphous solid. Source: JUAN QIAO YUAN WEI Iris
Mithramycin, ED50 = 0.07g/mL; A549, ED 50= 1.9g/mL, Mithramycin,
potaninii (underground part). Ref: 4235.

OH
ED50 = 0.08g/mL). Source: SI ROU TUO GUO YE MI ZHU YU Melicope
semecarpifolia. Ref: 5405.

O
OH
O
O
OH
OO
HO
OH
OH
O
OH
O
OH
186
6296 3',4'-Dimethoxy-5,7,5'-trihydroxyl-flavone 3-O--L-rhamnopyra-
6301 2,8-Dimethyl-5-acetyl-bicyclo[5,3,0] decadiene-1,8
noside
C14H20O (204.31). Source: SAN QI Panax pseudo-ginseng var. notoginseng
3',4'-Dimethoxy-5,7,5'-trihydroxyl-flavone 3-O--L-rhamnopyranoside
[Syn. Panax notoginseng]. Ref: 2.
C23H24O12 (492.44). Source: SHAN HUANG PI Clausena excavata. Ref:

2135.
O
O
HO
OH
OH
OH
6302 ,-Dimethylacrylalkannin
O
O
C21H22O6 (370.41). mp 116~117C. Pharm: Antibacterial (Staphylococcus

aureus, Staphylococcus epidermidis and Mycobacterium tuberculosis H37Rv);
inhibits ejection of sperm (male toad, caused by injecting chorionic
OH OH
6297 4,9-Dimethoxy-1-vinyl--carboline
[88142-62-5] C15H14N2O2 (254.29). Source: KU SHU PI Picrasma
quassioides [Syn. Picrasma ailanthoides]. Ref: 12.
gonadotrophin); used in treatment of allergic purpura. Source: DIAN ZI CAO

Onosma paniculatum, OU ZI CAO Alkanna tinctoria (root: content scope =
0.46%~0.50%[5501]), XIN ZANG JIA ZI CAO Arnebia euchroma, ZI CAO
Lithospermum erythrorhizon. Ref: 2, 5, 658, 5501.
OH
OH
6298 4,4'-Dimethoxyvulpinic acid

C21H18O7 (382.37). Pharm: Antitubercular (Mycobacterium tuberculosis
6303 ,-Dimethylacrylshikonin
H37Ra, MIC = 25g/mL); anti-HSV-1 inactive; cytotoxic inactive (hmn
C21H22O6 (370.41). Sorrel lamellar crystals, mp 116~117C. Pharm:
lung cancer cells NCI-H187). Source: HUANG YING PI MA BO
Antibacterial (Staphylococcus aureus 209P, Staphylococcus aureus TPR27, S.
Scleroderma citrinum. Ref: 5406.
epidermidis TPR25, Sarcina lutea and Bacillus subtilis, MIC = 160g/mL);

antineoplastic (W256, in vitro and in vivo); contracts blood vessels (inhibits
OH
ACh-induced relaxation on intact thoracic aorta, IC 50 =

(1.4610.052)mol/L, 1,4-Naphthoquinone IC 50 = (1.5040.171)mol/L)
[4916]
. Source: DIAN ZI CAO Onosma paniculatum (root: content =
0.095%)[5508], JIA ZI CAO Arnebia guttata (root: content = 0.121%)[5508], XIN
O
O
6299 1,7-Dimethoxyxanthone
C15H12O4 (256.26). Source: YUAN ZHI Polygala tenuifolia (cortex). Ref:
ZANG JIA ZI CAO Arnebia euchroma (root: mean content of 3 origins =

0.879%)[5508], ZI CAO Lithospermum erythrorhizon (root: content =
0.137%[5508]). Ref: 661, 4916, 5501, 5508.
4507.
O
OH
OH
6300 5,8-Dimethoxyxanthyletin
Racemosin [68421-13-6] C16H16O5 (288.30). mp 179~180C. Source: SHI
6304 6(1,1-Dimethylallyl)-7,4'-dihydroxylflavan
JIAO CAO Boenninghausenia sessilicarpa, YAN JIAO CAO
C20H22O3 (310.40). Light yellow gum, []D = +3.5 (c = 0.14, MeOH). Source:
Boenninghausenia albiflora (root). Ref: 660, 1521, 2495.
TUO YUAN DUO TAN CAO Dorstenia elliptica (twig). Ref: 3754.
OH
O
O
HO
187
6305 8-(1,1-Dimethylallyl)genistein
6311 6-,-Dimethylallyltaxifolin 7-O--D-glucoside
C20H18O5 (338.36). Yellow prisms (CHCl3), mp 94~96C. Source: FEI LV
C26H30O12 (534.52). mp 170~172C, []D20 = 6.6 (c = 0.5, MeOH). Source:
BIN QIAN JIN BA Moghania philippinensis (root). Ref: 3500.
JIN LIAN MU Ochna integerrima (leaf). Ref: 5133.

OH
HO
OH
OO
HO
OH
OH
OH
OH
OH
OH
OH
6306 3-(1,1-Dimethyl allyl) herniarin

[20958-63-8] C15H16O3 (244.29). mp 126~128C. Source: CHOU CAO Ruta
graveolens. Ref: 6.
6312 3-(1,1-Dimethylallyl)-xanthyletin
C19H20O3 (296.37). mp 98~99C. Pharm: Phytogrowth inhibitor (100g/mL,
Amaranthus hypochondriacus, InRt = (74.91.5)%; E. crusgalli, InRt =
(83.71.9)%)[5253]. Source: YAN JIAO CAO Boenninghausenia albiflora,
Stauranthus perforatus (root). Ref: 2495, 5253.

6307 3'-(,-Dimethylallyl)-kievitone
3'-(3,3-Dimethylallyl)-kievitone C25H28O6 (424.50). Source: CU MAO GAN
CAO Glycyrrhiza aspera, GAN CAO Glycyrrhiza Uralensis, GUANG GUO
GAN CAO Glycyrrhiza glabra. Ref: 2431.
O
O
HO
OH
6313 Dimethylalpinumisoflavone
C22H20O5 (364.40). Source: CI TONG Erythrina variegata [Syn. Erythrina
OH
OH
indica] (stem cortex). Ref: 5220.

O
6308 3,3-Dimethylallyl-4-methoxy-2-quinolone
C18H23NO2 (285.39). Source: WU ZHU YU Evodia rutaecarpa. Ref: 877.

O
N
H
6314 4',7-Dimethylamentoflavone
C32H22O10 (566.53). Yellowish amorphous powder (MeOH), mp 317~319C,
6309 8-(,-Dimethylallyl)-pongamol
[]D17.6 = +15.92 (c = 0.26, C5H5N). Pharm: Tissue proteinase B inhibitor
C23H22O4 (362.43). Pharm: Cytotoxic (BST, LC50 = 2.69g/mL). Source:
(IC50 = 0.55mol/L); cytotoxic (A549, IC50 = 7.74mol/L, Bel7402, IC50 =
Lonchocarpus latifolius (root). Ref: 5108.
17.16mol/L, DU145, IC50 = 12.42mol/L, HT29, IC50 = 14.54mol/L).

Source: MO XI GE LUO YU SHAN Taxodium mucronatum (twig and leaf).
Ref: 4571.
6310 3,3-Dimethyl allyl-p-propenyl phenyl ether

C14H18O (202.30). Source: BA JIAO HUI XIANG Illicium verum. Ref: 6.
OH
O
O
HO
O
O
OH
OH
188
6315 5-O-(3'-Dimethylamino-3'-phenylpropionyl) taxinine M
6321 2,2-Dimethyl-2H-1-benzopyran-6-carboxylic acid methyl ester
C46H55NO15 (861.95). Colorless solid. Pharm: Cytotoxic (A549, ED50 =
2,2-Dimethyl-6-methoxycarbonyl-2H-benzopyran [34818-57-0] C13H14O3
(10.12.4)mol/L). Source: XI MA LA YA HONG DOU SHAN Taxus
(218.25). Source: BAI HUA LONG DAN Gentiana algida. Ref: 704.
wallichiana (needle leaf). Ref: 5225.

O
O O
O
O
O O
HO
O
O
6322 N20 ,N 20 -Dimethyl-N 3-benzoyl-3,20-diaminopregn-2-en-4-ol
Anticancer Alkaloid PMV70P691-001 C30H44N2O2 (464.70). Pharm:
Cytotoxic (estrone sulfatase assay). Source: YANG WO BAN DENG GUO
Pachysandra procumbens. Ref: 5038.
6316 N,N-Dimethylanomurine
+
Tetrahydrobenzylisoquinoline alkaloid C22H30NO4 (372.49). Colorless

amorphous powder, []D22 = 26.3 (c = 0.32, MeOH). Source: XIAO HUA
MU BAN SHU Xylopia parviflora (bark and root). Ref: 3794.
O
N
H
OH
O
N
6323 3-O-(2,3-Dimethylbutanoyl)-13-O-dodecanoyl-20-acetylingenol
C40H62O9 (686.93). Colorless gum, []D23 = 11.5 (c = 0.69, MeOH). Source:

GAN SUI Euphorbia kansui. Ref: 4368.
O
O
6317 Dimethyl azelate
Methyl azelate [1732-10-1] C11H20O4 (216.28). Source: DANG GUI Angelica
O
HO
sinensis. Ref: 2.
HO
O
O
O
O
6324 3-O-(2,3-Dimethylbutanoyl)-13-O-dodecanoyl-20-deoxyingenol
C38H60O7 (628.90). Colorless gum, []D23 = 4.4 (c = 0.73, MeOH). Source:
6318 1,2-Dimethylbenzene
GAN SUI Euphorbia kansui. Ref: 4368.
[95-47-6] C8H10 (106.17). Source: SHAN ZHA Crataegus pinnatifida. Ref: 2.

O
O
O
HO
HO
6319 ,-Dimethylbenzene methanol

[617-94-7] C9H12O (136.20). Source: SAN QI Panax pseudo-ginseng var.
OH
6325 3-O-(2,3-Dimethylbutanoyl)-13-O-dodecanoylingenol
C38H60O8 (644.90). Pharm: Induces cell cleavage arrest (Xenopus laevis
embryo cells at the blastular stage, at 10g/mL compound results in > 60%
cell cleavage arrest). Source: GAN SUI Euphorbia kansui. Ref: 4368.
6320 3,4-Dimethylbenzoic acid
3,4-Xylylic acid [619-04-5] C9H10O2 (150.18). mp 166C. Source: MU TIAN
LIAO Actinidia polygama. Ref: 6.

O
O
HO
O
OH
HO
HO
O
H
189
6326 20-O-(2,3-Dimethylbutanoyl)-13-O-dodecanoylingenol
6331 24,24-Dimethyl-5-cholesta-8-en-3-ol
C38H60O8 (644.90). Source: GAN SUI Euphorbia kansui. Ref: 4368.
C29H50 O (414.72). Source: JIAO GU LAN Gynostemma pentaphyllum.

Ref: 2.
O
O
O
HO
HO
H
H
HO
HO
6332 N,N-Dimethylconiine
C10H23N (157.30). Source: SA BA LU HUI Aloe sabaea. Ref: 728.
6327 1,2-Di-(a-methyl)-butanoyl-4-hydroxy-9-(-)furoyloxy-15acetoxy--dihydroagarofuran
C32H46O11 (606.72). Colorless gum, []D20 = +42 (c = 1.00, CHCl3). Pharm:

Cytotoxic (in vitro, Bel7402 liver carcinoma, IC50 = 38.26g/mL, control
Etoposide, IC50 = 7.00g/mL). Source: Euonymus nanoides (seed). Ref: 4962.
6333 7,7''-Di-O-methylcupressu-flavone
C32H22O10 (566.53). mp > 300C. Source: CE BAI YE Thuja orientalis [Syn.
O
O O
O O
Platycladus orientalis; Biota orientalis]. Ref: 6.

O
HO
OH
HO
OH
H
OH
6328 1S,6R-Di(2-)methylbutanoyloxy-4S-hydroxy-8S-benzoyloxy-9R-
(3-)furancarbonyloxy-13-acetyloxy--dihydroagarofuran
6334 1,4-Dimethyl-cis-cyclohexane
C39H50O13 (726.83). Yellow oil, []D = +39.4 (c = 6.3, CHCl3). Pharm:
[589-90-2] C8H16 (112.22). Source: SHAN ZHA Crataegus pinnatifida.
Cytotoxic (hmn Bel7402, IC50 = 6.9mol/L, hmn HL-60, IC50 = 51.4mol/L,
Ref: 2.
hmn A549, IC50 = 81.7mol/L, mouse, P388, IC50 = 51.2mol/L). Source:

Euonymus nanoides (seed: yield = 0.0053%dw). Ref: 1129.
6335 1,6-Dimethyl-cis-cyclohexane
[583-57-3] C8H16 (112.22). Source: SHAN ZHA Crataegus pinnatifida.

O
Ref: 2.
O
OH O
O
H H
6329 3,5-Dimethylbutylbenzene
6336 2,7-Dimethyl-1,4-dihydronaphthalene-5,8-diol 5-O--D-xylopyra-
C12H18 (162.27). Source: SHAN ZHA Crataegus pinnatifida. Ref: 2.
nosyl(16)--D-glucopyranoside
C23H32O11 (484.50). mp 215~217C, []D26 = 33.9 (c = 0.13, MeOH).
Source: RI BEN LU TI CAO Pyrola japonica (whole herb). Ref: 4294.
OH
6330 Dimethyl camphorate

C12H20O4 (228.29). Source: DANG GUI Angelica sinensis. Ref: 2.
OO
OO
OH
OH
OH
OH
OH
OH
190
6337 (+)-3,4-(6'',6''-Dimethyldihydropyrano)-4',5'-[2'''-(1-hydroxy-1-
6342 Dimethyl disulfide
methylethyl)-dihydrofurano]-2',3'''-dihydroxydihydrochalcone
2,3-Dithiabutane [624-92-0] C2H6S2 (94.20). mp 98C, bp 110C; 116~118C.
C25H30O6 (426.51). Yellow powder, mp 114~116C, []D25 = +414 (c = 0.013,
Source: DA SUAN Allium sativum, JIU CAI Allium tuberosum, YANG
MeOH). Source: Dorstenia barteri var. subtriangularis (twig). Ref: 3765.
CONG Allium cepa. Ref: 6.
HO
S
S
O
6343 4,6-Dimethyl dodecane

OH
C14H30 (198.40). Source: ROU CONG RONG Cistanche deserticola. Ref: 2.
OH
6338 4',7-Di-O-methyldihydroquercetin
5,3,3'-Trihydroxy-7,4'-dimethoxyflavanone C17H16O7 (332.31). Yellow
amorphous powder. Pharm: Cytotoxic (HeLa, IC50 = 22.4g/mL, control
Mitomycin C, IC50 = 1.7g/mL)[4092]. Source: JUAN QIAO YUAN WEI Iris
potaninii (underground part), TUAN JI AI NA XIANG Blumea glomerata.
6344 3,3'-Di-O-methylellagic acid
Ref: 4092, 4235.
C16H10O8 (330.25). Pharm: Antioxidant (in vitro, effect on conjugated diene

O
Punica granatum (seed: yield = 0.00063%). Ref: 4792.
formation of LDL or MDA level in rat brain). Source: SHI LIU ZHONG ZI
OH
OH
OH
OH
6339
4,4-Dimethyl-7,8-dihydroxy-3,5-dioxobicyclo[4.3.1]dec-1(10)-en-2-one
C10H14O5 (214.22). Colorless squama crystals, mp 175~177C. Source: MEI
LI JIN SI TAO Hypericum bellum. Ref: 2492.

OH
HO
6345 3,3'-Di-O-methylellagic acid 4-(5''-acetyl)--L-arabinofuranoside
HO
C23H20O13 (504.41). Off-white amorphous powder, []D28 = 180.0 (c = 0.13,

M2SO). Source: JI SU ZI Cornus capitata [Syn. Dendrobenthamia capitata]
(root). Ref: 5177.

O
O
6340 3,7-Dimethyl-1,8-dihydroxy-6-methoxy-isochroman
C12H16O4 (224.26). []D20 = 6.3 (c = 0.083, MeOH). Source: Penicillium
steckii. Ref: 3960.
O
OH
OH
OH
6346 4,4'-O-Dimethylellagic acid 3-(2'',3''-di-O-acetyl)--L-rhamnoside
O
OH
OH
C26H24O14 (560.47). Amor phous powder, []D = 21.6 (c = 0.1, MeOH).

Pharm: Cytotoxic (panel of hmn cancer cell lines, according to established
6341 (2S)-2-[(3aR*,4S*,7R*,7aS*)-3a,7a-Dimethyl-1,3-dioxo-4,7-epoxy-
protocols of Likitwitayawuid 1993 and Seo 2001, ED50 values of > 5mg/mL
octahydroisoindol-2-yl]-5-guanidino pentanoic acid
are regarded as inactive). Source: MA SI TE SI DU YING Elaeocarpus
C16H24N4O5 (352.39). Powder, mp 195.0~197.0C, []D = 21.1 (c = 2.2,
mastersii. Ref: 2020.
MeOH:H2O = 1:1). Source: BAN MAO Mylabris phalerata; Mylabris

cichorii. Ref: 4052.
O
OH
OH
O
N
O
O
OH
HN
NH
H2N
O
OO
O
O O
191
6347 3,4'-O-Dimethylellagic acid 4-O--L-rhamnopyranoside
6352 2,5-Dimethyl-3-O--D-glucopyranosylnaphthol
C22H20O12 (476.40). []D = 42.4 (c = 0.1, MeOH). Source: SHI LIU XIN
C18H22O6 (334.37). Yellowish oil. Source: DA MA JIN Hibiscus cannabinus
(bark). Ref: 5233.
O
OH
O
HO
O
O
OH
O
OH
OH
O
OH
6353 N,N-Dimethyl glycine methyl ester
OO
[7148-06-3] C5H11NO2 (117.15). Source: ROU CONG RONG Cistanche

deserticola. Ref: 2.
OH OH
6348 rel-(7R,8R,7'R,8'R)-3,4,3',4'-Dimethylenedioxy-5,5'-dimethoxy-
7,7'-epoxylignan
C22H24O7 (400.43). Pale yellow oil, []D21 = 10.1 (c = 0.01, MeOH). Pharm:
Antitrypanosomal (trypomastigote form of Trypanosoma cruzi (Y strain), IC50 =
3.47g/mL). Source: Piper solmsianum. Ref: 3450.
6354 (2E)-2,6-Dimethyl-2,5-heptadienoic acid

C9H14O2 (154.21). Colorless oil. Source: DA GUO XI FAN LIAN Passiflora
quadrangularis (fruit). Ref: 3900.
O
O
OH
6349 3,4-Dimethylenedioxypterocarpan
C17H12O6 (312.28). White crystals, mp 154~156C. Source: KEN NI YA HUI
YE Tephrosia aequilata. Ref: 1957.
O
O
6355 (2E)-2,6-Dimethyl-2,5-heptadienoic acid -D-glucopyranosyl ester

C15H24O7 (316.35). Colorless oil, []D25 = +12.6 (c = 0.78, MeOH). Source:
DA GUO XI FAN LIAN Passiflora quadrangularis (fruit). Ref: 3900.
O
H
O
H
6350 3,5-Dimethylene-1,4,4-trimethylcyclopentene
OO
HO
OH
C10H14 (134.22). Colorless oil. Source: Lavandula luisieri (essential oil). Ref:
OH
5301.
OH
6356 2,3-Dimethylheptane
[3074-71-3] C9 H20 (128.26). Source: SHAN ZHA Crataegus pinnatifida.
Ref: 2.
6351 Dimethyl ester of (1,2,3,4)-2,4-bis(3,4-dihydroxyphenyl)1,3-cyclobutanedicarboxylic acid
C20H20O8 (388.38). Colorless needles, []D = 0 (c = 0.47, MeOH). Pharm:
Antihistamine (inhibits histamine release, rat mast cell, induced by
antigen-antibody reaction, IC50 = 16.9g/mL, control Indomethacin, IC50 =
89.5g/mL); PGE2 production inhibitor (30g/mL, InRt = 76.5%). Source:
6357 4,4-Dimethyl-1,7-heptanedioic acid
XIAO HUA GUI ZHEN Bidens parviflora Ref: 3364.
C9H16O4 (188.23). White powder, easy dissolve in methanol and acetone, mp

104~107C. Source: CHAN YI TENG Securidaca inappendiculata. Ref:
HO
2183.
O
OH
HO
O
OH
HO
O
OH
192
6358 1-(1,5-Dimethyl-4-hexenyl)-4-methyl benzene
6364 1,3-Dimethylisoguaninium
C15H22 (202.34). Source: SHENG JIANG Zingiber officinale. Ref: 2.
C7H10N5O+ (180.19). Colorless needles (EtOH). Pharm: Inhibits specificly

basic fibroblast growth factor (bFGF)-induced proliferation of bovine aorta
endothelial cells (BAECs); reduces tube formation of BAECs in a
time-dependent manner. Source: Sponge Amphimedon paraviridis. Ref: 4351.
H
N
6359 3,5-Dimethyl-4-hydroxy-benzaldehyde
C9H10O2 (150.18). Source: LIU CHUAN YU Linaria vulgaris. Ref: 4237.
H
N
O
N
6365 Dimethyl lithospermate

HO
C29H26O12 (566.52). Pharm: Antioxidant (DPPH scavenger, IC50 =

0.1197mmol/L, control Propyl gallate, IC50 = 0.03mol/L; superoxide radical
6360 2,5-Dimethyl-7-hydroxy chromone
inhibitor, inactive, Propyl gallate, IC50 = 0.106mmol/L; iron chelating assay,
C11H10O3 (190.20). mp 220~222C. Source: HU ZHANG Polygonum
inactive, Propyl gallate, IC50 = 0.064mmol/L). Source: MING XIAN HUA
cuspidatum, REN SHEN Panax ginseng [Syn. Panax schinseng], TIAN
ZHU CHANG ZHU LIU LI CAO Lindelofia stylosa (aerial parts). Ref: 4533.
SHAN DA HUANG Rheum wittrocki. Ref: 2, 609.

HO
OH
OH
OH
O
O
6361 3,5-Dimethyl-8-hydroxy-7-methoxy-3,4-dihydroisocoumarin
C12H14O4 (222.24). Colorless needles. Pharm: Antifungal (Aspergillus niger,

MIC = 50g/mL control Nystatin, MIC = 12.5g/mL; Cladosporium
H
O
O
O
OH
O
OH
herbarum, MIC = 50g/mL, Nystatin, MIC = 12.5g/mL); antibacterial

(Bacillus subtilis, MIC = 25g/mL, control Chloramphenicol, MIC =
6366 6,8-Di-C-methylluteolin 7-methyl ether
3.13g/mL; Pseudomonas syringae,MIC = 100g/mL, control
C18H16O6 (328.32). Yellow needles (CHCl3MeOH), mp 288~290C. Pharm:
Chloramphenicol, MIC = 3.13g/mL). Source: Cytospora eucalypticola. Ref:
Antibacterial (oral pathogens: Streptococcus mutans, MIC > 500g/mL,
3367.
control Chlorhexidine gluconate, MIC = 1.25g/mL; Fusobacterium

nucleatum, MIC = 375g/mL, Chlorhexidine gluconate, MIC = 2.5g/mL).
Source: BAI MAO GEN(4) Hydrastis canadensis (root). Ref: 5418.
O
O
OH
OH
OH
6362 3,7-Dimethyl-8-hydroxy-6-methoxyisochroman
C12H16O3 (208.26). Source: Penicillium steckii. Ref: 3960.

OH
O
6367 Dimethylmatairesinol
O
C22H26O6 (386.45). Pharm: Cytotoxic (A549, ED50 = 1.9mol/L, ED50 = 5.0g/mL,

control Adriamycin, ED50 = 0.01mol/L, ED50 = 0.02g/mL; MCF7, ED50 =
OH
6363 (2E,6R)-2,6-Dimethyl-8-hydroxy-2-octenoic acid

8-O-[6'-O-(E)-p-coumaroyl]--D-glucopyranoside
Source: ZI YE Catalpa ovata (leaf, fallen leaf). Ref: 3536, 4290.
O
OH
1.8mol/L, ED50 = 4.7g/mL, Adriamycin, ED50 = 0.1mol/L, ED50 = 0.1g/mL;

HT29, ED50 = 1.4mol/L, ED50 = 3.5g/mL, Adriamycin, ED50 = 0.1mol/L, ED50
= 0.1g/mL)[5088]. Source: E SHEN Anthriscus sylvestris, TAI WAN SHAN
Taiwania cryptomerioides (heartwood). Ref: 5088, 5499.
O
O
O
O
O
O
O
HO
OH
O
OH
OH
193
6368 3,5-Dimethyl-4-methoxybenzoic acid
6374 7,8-Dimethyl-2-(1-methylethyl)phenanthren-3-ol
[21553-46-8] C10H12O3 (180.21). mp 145C. Source: JIAN YE FAN XIE YE
C19H20O (264.37). Yellowish gum. Source: XIU QIU SHU WEI CAO Salvia
Cassia acutifolia. Ref: 6, 660.
hydrangea (root). Ref: 5447.
OH
HO
O
6369 3,5-Dimethyl-8-methoxy-3,4-dihydroisocoumarin
C12H14O3 (206.24). Colorless needles. Source: Cytospora eucalypticola. Ref:
3367.
6375 2,4-Dimethyl-6-(3'-methyl-isobuten-5'-isopropyl)-phenyl-3,5hexanedione
C22H32O2 (328.50). Brick red oil. Source: XIAN MAI XUAN FU HUA Inula
nervosa. Ref: 795.
O
O
6370 N,N-Dimethyl-5-methoxy tryptamine
OH
5-Methoxy-N,N-dimethyl-tryptamine [1019-45-0] C13H18N2O (218.30). mp

47C. Pharm: Toxin (similar action with bufotenine). Source: WU ZHU YU
Evodia rutaecarpa, HONG MU JI CAO Desmodium gangeticum, PAI QIAN
CAO Desmodium pulchellum [Syn. Phyllodium pulchellum], YI CAO
6376 5,15-Dimethylmorindol
Phalaris arundinacea. Ref: 2, 6, 658.
C17H14O6 (314.30). Yellow amorphous powder. Source: HAI BA JI Morinda

citrifolia (fruit). Ref: 4542.
O
N
H
OH
6371 1,1-Dimethyl-2-(3-methyl-1,3-butadiene)cyclo-propane
C10H16 (136.24). Source: BAI ZHI Angelica dahurica [Syn. Angelica
HO
O
6377 3',5'-O-Dimethylmyricetin 3-O--D-2'',3''-diacetylglucopyranoside

C27H28O15 (592.52). Yellow amorphous powder, mp>250C. Source:
Warburgia stuhlmannii (leaf). Ref: 3398.
O
OH
6372 7,7-Dimethyl-2-methylenebicyclo[3.1.1]heptan-6-ol acetate

C12H18O2 (194.28). Colorless oil. Source: Psiadia anchusifolia (fresh leaf).
HO
Ref: 3787.
OH
O HO
O
O
O
OH
6378 2,6-Di-C-methyl-nicotinic acid 3,5-diethyl ester

6373 1,8-Dimethyl-4-(1-methylenyl)-spiro(4,5) dec-7-ene
C13H17NO4 (251.28). Colorless needles. Source: Viburnum tinus (leaf). Ref:
Isoacoradinene C15H24 (204.36). Source: DANG GUI Angelica sinensis, WU
5339.
WEI ZI Schisandra chinensis. Ref: 2, 660.

O
O
O
O
N
194
6379 2-(4',8'-Dimethylnona-3',7'-dienyl)-8-hydroxy-2-methyl-2H-chro-
6386 (3E)-3,7-Dimethyl-3-octene-1,2,6,7-tetrol
mene-6-carboxylic methyl ester
C 10 H 21 O 4 (204.27). Colorless oil. []D 25 = 11.9 (c = 0.67, MeOH).
C23H30O4 (370.49). Brown amorphous solid. Source: SAN XING HU JIAO Piper
Source: DA GUO XI FAN LIAN Passiflora quadrangularis (fruit). Ref:
umbellatum (branch), DUN YE HU JIAO Piper peltatum (branch). Ref: 5274.
3900.
OH
OH
OH
OH
OH
6380 (5E)-2,6-Dimethyl-5,7-octadiene-2,3-diol
6387 3,7-Dimethyloct-3(10)-ene-1,2,6,7-tetrol
C10H18O2 (170.25). Colorless oil. []D = 19.7 (c = 0.62, MeOH). Source:
C 10 H 20 O 4 (204.27). Source: BEI SHA SHEN Glehnia littoralis (fruit).
DA GUO XI FAN LIAN Passiflora quadrangularis (fruit). Ref: 3900.
Ref: 3525.
23
OH
OH
OH
OH
OH
OH
6381 4-O-[(2E,5E)-3,7-Dimethyl-2,5-octadiene-7-ol]-sinapyl alcohol

C21H30O5 (362.47). Source: LIAN YE TUO WU Ligularia nelumbifolia (root,
6388 (2S,6)-3,7-Dimethyloct-3(10)-ene-1,2,6,7-tetrol 1-O--D-gluco-
yield = 0.0013%dw). Ref: 4632.
pyranoside
Source: BEI SHA SHEN Glehnia littoralis (fruit). Ref: 3525.
O
OH
HO
HO
OH
HO
OH
6382 3,7-Dimethyl-2,6-octadien-1,6-olide
C10H14O2 (166.22). Source: Plagiochila rutilans. Ref: 5144.
OO
OH
OH
OH
6389 O-[3-(2,2-Dimethyl-3-oxo-2H-furan-5-yl)-3-hydroxybutyl]
O
bergaptol
C21H20O7 (384.39). Colorless needles (hexaneEtOAc), mp 168~169C, [] D
6383 3-(3',7'-Dimethyl-2',6'-octadienyl)-4-methoxybenzoic acid
= 5.0 (c = 0.12, MeOH). Source: TUO YUAN DUO TAN CAO Dorstenia
C18H24O3 (288.39). Amorphous solid. Source: GOU ZHUANG HU JIAO
elliptica (twig). Ref: 3754.
Piper aduncum. Ref: 2323.
OH
O
OH
6384 3,7-Dimethyl-1,5,7-octatrien-3-ol
C10H16O (152.24). Source: CHA YE Camellia sinensis [Syn. Thea sinensis].
Ref: 6.
6390 (E)-4-(1,5-Dimethyl-3-oxo-1,4-hexadienyl)benzoic acid
C15H16O3 (244.29). mp 156C. Pharm: Antifungal (TLC bioautography
method at very low concentration). Source: SI LI LAN KA TU MI SHU
OH
Bridelia retusa. Ref: 2021.
6385 3,7-Dimethyl-7-octenal
O
[141-26-4] C10H18O (154.25). Source: JU PI Citrus reticulata. Ref: 2.
HO
O
195
6391 (E)-4-(1,5-Dimethyl-3-oxo-1-hexenyl)benzoic acid
6397 8,8-Dimethyl-2-phenyl-10-prenyl-2,3-dihydro-8H-pyrano[3,2-g]
C15H18O3 (246.31). mp 122C. Pharm: Antifungal (TLC bioautography
chroman-4-one
method at very low concentration). Source: SI LI LAN KA TU MI SHU
C25H26O3 (374.48). Colorless needles (petroleum ether : CHCl3= 10:1), mp
Bridelia retusa. Ref: 2021.
121~122C. Source: GAN HUA DOU Fordia cauliflora (stem). Ref: 4564.
HO
O
O
6392 (R)-4-(1,5-Dimethyl-3-oxo-4-hexenyl)benzoic acid
C15H18O3 (246.31). mp 83~88C, []D25 = 68.1 (c = 0.34, CHCl3). Pharm:
6398 Dimethyl phthalate
Antifungal (TLC bioautography method at very low concentration). Source:
SI LI LAN KA TU MI SHU Bridelia retusa. Ref: 2021.
O
O
HO
6399 2,2-Dimethyl-8-prenyl-6-vinylchromene
6393 (R)-4-(1,5-Dimethyl-3-oxohexyl)benzoic acid
C15H20O3 (248.32). mp 62C, []D25 = 26.3 (c = 0.63, CHCl3). Pharm:
C18H22O (254.38). Colorless oil. Source: FENG JIAO Apis mellifera ligustica.
Ref: 4124.
Antifungal (TLC bioautography method at very low concentration). Source:

SI LI LAN KA TU MI SHU Bridelia retusa. Ref: 2021.
HO
6400 Dimethyl--propriothetin
[4337-33-1] C5H11O2S+ (135.11). Source: SHI CHUN Ulva lactuca. Ref: 6.

6394 N,N-Dimethylphenylalanine
C11H15NO2 (193.15). Colorless acicular crystals. Source: HUANG YING PI

MA BO Scleroderma citrinum. Ref: 2180.
OH
O
OH
6401 [6'',6''-Dimethylpyrano-(2'',3'':7,8)]-4'-methoxy-3-arylcoumarin
C21H18O5 (350.37). Source: Glycyrrhiza sp. Ref: 2431.
6395 (2'S,3'R)-5-(N,N-Dimethyl-3'-phenylisoseryl)-taxachitriene A
OH
C43H57NO15 (827.93). mp 93~95C, []D = +22.3 (CHCl3). Source: HONG

O
O
6402 3,3'-Dimethylquercetin
O
O
O
O
3,3'-Dimethoxyquercetin [4382-17-6] C17H14O7 (330.29). Yellowish acicular

O
crystals (methanol), mp 255C. Pharm: Antifungal; antiviral (epidemic type-1

N
poliomyelitis virus and Gesak-B4 virus, 0.01g/mL, InRt = 90%); cytotoxic (P388,
ED50 = 1.7g/mL); insect antifeedant (boll weevil); smooth muscle relaxant.
O
OH
O
Source: E BU SHI CAO Centipeda minima, GAN CAO Glycyrrhiza uralensis,

LU CAO Rhaponticum carthamoides. Ref: 171, 660, 900, 4006, 4007.
O
6396 3,4-Dimethyl-5-phenyloxazolidine
OH
C11H15NO (177.25). Source: MA HUANG Ephedra sinica. Ref: 2.

N
HO
O
OH
196
6403 (E)-3,7-Dimethyl-1-O-[-L-rhamnopyranosyl-(16)--D-gluco-
6409 (2S,2''S)-7,7''-Di-O-methyltetrahydroamentoflavone
pyranosyl-oct-2-en-7-ol
C32H26O10 (570.56). Yellow amorphous powder, []D = 25.4 (c = 0.024,
C22H40O11 (480.56). Viscous solid, []D24.3 = 57.0 (c = 0.383, MeOH).
Me2SO). Pharm: Antimalarial (Plasmodium falciparum W2, IC50 =
Source: YU YE GUI DENG QING Rodgersia pinnata (rhizome). Ref: 4570.
0.98g/mL, control Chloroquine. IC50 = 0.238g/mL; Plasmodium

falciparum D6, IC50 = 2.8g/mL, Chloroquine, IC50 = 0.026g/mL);
OH
OO
OO
cytotoxic inactive. Source: SHU ZHI YAN FU MU Rhus retinorrhoea (leaf).
OH
OH
Ref: 5201.
OH
OH
OH OH
OH
6404 E-Dimethyl rhoifolinate
OH
ED50 = 0.08g/mL)[5405]. Source: SI ROU TUO GUO YE MI ZHU YU

Melicope semecarpifolia. Ref: 5405.
OH
OH
6410 Di-O-methyltetrahydrofuriguaiacin B
C22H28O5 (372.47). Amorphous powder, []D = +43 (c = 0.5, CHCl3). Source:
SAN BAI CAO Saururus chinensis (underground part). Ref: 4122.
O
O
6405 Z-Dimethyl rhoifolinate

6411 7,7''-Di-O-methyltetrahydrohinokiflavone
1.45 (c = 1.0, MeOH). Source: NAN YIN DU SU TIE SHU GUO Cycas
beddomei (stem). Ref: 3929.
O
O
HO
O
O
O
OH
6406 Dimethyl sebacate

OH
6412 5,6-Dimethyl-3a,4,7,7a-tetrahydro-1,3-lsoben-zofurandione
C10H12O3 (180.21). Source: DU HUO Angelica pubescens f. biserrata [Syn.
Angelica pubescens]. Ref: 2.
O
O
6407 Dimethyl sulfide

[75-18-3] C2H6S (62.13). bp 37.5~38.0C. Source: DA SUAN Allium sativum,
SHUI SONG Codium fragile. Ref: 6.
6413 4,7-Dimethyl-1-tetralone
1,6-Dimethyl-4-keto-tetrahydronaphthalene [28449-86-7] C12H14O (174.24).
Oil, bp 118C/4mmHg, bp 146.5~147.0C/11.5mmHg, bp

145~152C/15mmHg, []D20 = +5.60 (c = 0.3035, chloroform). Pharm:
6408 Dimethyl sulfone
Antimalarial (in vitro, Plasmodium falciparum, EC50 = 86.2mol/L). Source:
Sulfonyl bis-methane [67-71-0] C2H6O2S (94.13). Source: MU ZEI Equisetum
XIANG FU Cyperus rotundus. Ref: 900, 1089.
hiemale. Ref: 2.
O
S
O
197
6414 Dimethyl tetrasulfide
6421 2,4-Dimethyl-undecane
[5756-24-1] C2H6S4 (158.33). Source: JIU CAI Allium tuberosum. Ref: 6.
S
S
6415 2,8-Dimethyl-2-[(3E,7E)-4,8,12-trimethyltrideca-3,7,11-trienyl]5-formyl-chroman-6-ol
C28H40O3 (424.63). Pale yellow oil, []D25 = 11.1 (c = 0.18, MeOH). Source:
DUO ZHI ZHI TENG HUANG Garcinia virgata (stem cortex). Ref: 3874.
6422 3,6-Dimethyl-undecane
C 13 H 28 (184.37). Source: ROU CONG RONG Cistanche deserticola.
Ref: 2.
HO
O
6416 2,8-Dimethyl-2-[(3E,7E)-4,8,12-trimethyltrideca-3,7,11-trienyl]7-formyl-chroman-6-ol
C28H40O3 (424.63). Source: DUO ZHI ZHI TENG HUANG Garcinia virgata
(stem cortex). Ref: 3874.
6423 Dineolignan
H
C36H30O4 (526.64). Yellow viscous oil. Source: TE LI NI DA HU JIAO Piper
aequale. Ref: 1910.
HO
6417 Dimethyl trisulfide

[3658-80-8] C2H6S3 (126.26). Source: DA SUAN Allium sativum. Ref: 2.
S
S
6418 N,N-Dimethyltryptamine
HO
[61-50-7] C12H16N2 (188.27). mp 48~49C. Pharm: Causes mental illness;

increases blood pressure; mydriatic. Source: CI YANG LI DOU Mucuna
6424 Dinochrome A
pruriens, LU ZHU GEN Arundo donax, HONG MU JI CAO Desmodium
(3S,5R,6R,3'S,5'R,8'R)-Epoxy-6,7-didehydro-5,6,5',8'-tetrahydro-,-c
gangeticum, PAI QIAN CAO Desmodium pulchellum [Syn. Phyllodium
arotene-3,5,3'-triol 3-O-acetate C 42 H 58 O 5 (642.93). Yellow crystal.
pulchellum]. Ref: 6, 658.
Pharm: Anti-carcinogenic (inhibits 50nmol/L 12-O-tetradecanoyl
phorbol 13-acetate (TPA)-stimulated
32
P-incorporation into the
phospholipids of HeLa cells, 25g/mL, InRt = 72.1%; inhibits the

proliferation of hmn malignant tumor cells, such as GOTO, OST and
N
H
6419 N,N-Dimethyltryptamine-methohydroxide
C13H20N2O (203.31). Source: LU ZHU GEN Arundo donax. Ref: 6.
HeLa cells). Source: ER JIAO DUO JIA ZAO Peridinium bipes. Ref:
4256.
OH
N
N
H
H O
6420 N,N-Dimethyltryptamine N-oxide
C12H16N2O (204.27). Pharm: Uterine stimulant. Source: CI YANG LI DOU
OH
Mucuna pruriens, HONG MU JI CAO Desmodium gangeticum, PAI QIAN

CAO Desmodium pulchellum [Syn. Phyllodium pulchellum]. Ref: 6.
+
O
N
H
198
6425 Dinochrome B
6428 (2S)-1,2-Di-O-[(9Z,12Z,15Z)-octadeca-9,12,15-trienoyl]-3-O--D-
(3S,5R,6R,3'S,5'R,8'S)-5',8'-Epoxy-6,7-didehydro-5,6,5',8'-tetrahydro-,-carot
galactopyranosyl glycerol
ene-3,5,3'-triol 3-O-acetate C42H58O5 (642.93). Yellow crystal. Pharm:
C45H74O10 (775.09). Colorless oil, []D26 = 3.0 (c = 0.4 CHCl3). Pharm:
Anti-carcinogenic (inhibits 50nmol/L 12-O-tetradecanoyl phorbol 13-acetate
Anti-inflammatory (inhibits chemotaxis of hmn peripheral blood neutrophils
32
(TPA)-stimulated P-incorporation into the phospholipids of HeLa cells,
in vitro, The inhibiting activity at 100, 50, 10, 1, and 0.1g/mL, InRt = 82%,
25g/mL, InRt = 35.0%). Source: ER JIAO DUO JIA ZAO Peridinium bipes.
77%, 62%, 64%, and 7%, respectively). Source: QUAN CHI QIANG WEI
Ref: 4256.
Rosa canina (fruit: yield = 0.025%dw). Ref: 4705.

OH
O
HO
HO
OH
O
OH
H
O
O
OH
6429 1,2-Di-O-(9Z,12Z,15Z-octadecatrienoyl)-3-O-[-D-glucose(16)O
-D-allose]-glycerol
C51H84O15 (937.23). Colorless gum, []D24 = +25.3 (c = 6.01, MeOH). Pharm:

Antibacterial (Bacillus subtilis, IZD = 13~15mm, control Chloramphenicol, IZD =
6426 (2S)-1,2-O-6,9,12,15-Dioctadecatetraenoyl-3-O-[-D-galactopyra-
16~20mm; Escherichia coli, IZD = 13~15mm, Chloramphenicol, IZD = 16~20mm;
nosyl-(1''''6''')-O--D-galactopyranosyl]-glycerol
Staphylococcus aureus, IZD = 10~12mm, Chloramphenicol, IZD = 16~20mm).
C51H80O15 (933.20). []D25 = +52 (c = 0.80, MeOH). Source: KA SHI QIAN
Source: YI BAO MA HUA TOU Serratula strangulata (root stem). Ref: 5244.
GOU ZAO Amphidinium carterae. Ref: 4448.

HO
OO
OH
OH
HO
O O HO
OO
OH
OH
HO
OH OH
H
OH
O
OH
OH
O
OH
O
O
HO
H
H
H
H
H
6427 1,2-Di-O-(9Z,12Z,15Z-octadecatrienoyl)-3-O-(6-amino-6-deoxy-D-glucosyl)-glycerol
C45H75NO9 (774.10). Colorless gum, []D24 = +25.5 (c = 3.01, MeOH).
6430 1,2-Di-O-(9Z,12Z,15Z-octadecatrienoyl)-3-O-(6-p-hydroxy-phenyl-
Pharm: Antibacterial (Bacillus subtilis, IZD = 10~12mm, control
propionamido-6-deoxy--D-glucosyl)-glycerol
Chloramphenicol, IZD = 16~20mm; Escherichia coli, IZD = 16~20mm,
C54H83NO11 (922.26). Colorless gum, []D24 = +25.8 (c = 2.7, MeOH). Pharm:
Chloramphenicol, IZD = 16~20mm; Staphylococcus aureus, IZD = 10~12mm,
Antibacterial (Bacillus subtilis, IZD = 13~15mm, control Chloramphenicol, IZD =
Chloramphenicol, IZD = 16~20mm); cytotoxic (SMMC-7721, IC50 =
16~20mm; Escherichia coli, IZD = 16~20mm, Chloramphenicol, IZD = 16~20mm;
(351.46.1)g/mL, control Vincristine, IC50 = (63.21.8)g/mL; B16, IC50 =
Staphylococcus aureus, IZD = 10~12mm, Chloramphenicol, IZD = 16~20mm);
(157.32.5)g/mL, Vincristine, IC50 = (70.72.8)g/mL; HeLa, IC50 =
cytotoxic (SMMC-7721, IC50 = (151.66.3)g/mL, control Vincristine, IC50 =
(168.21.9)g/mL, Vincristine, IC50 = (67.22.2)g/mL). Source: YI BAO
(63.21.8)g/mL; B16, IC50 = (70.32.2)g/mL, Vincristine, IC50 = (70.72.8)g/mL;
MA HUA TOU Serratula strangulata (root stem). Ref: 5244.
HeLa, IC50 = (121.93.1)g/mL, Vincristine, IC50 = (67.22.2)g/mL). Source: YI

BAO MA HUA TOU Serratula strangulata (root stem). Ref: 5244.
H2N
OH
H OH
H
H
O
OH
H
N
H
O
O
OH
H OH
HO
H
H
H
H
OH
H
H
O
O
OH
O
H
H
H
H
H
H
H
199
6431 :-Diolein
6436 Diosbulbin C
[98168-52-6] C39H72O5 (621.01). mp 21.5C, 25C. Source: MANG GUO HE
[20086-07-1] C19H22O7 (362.38). mp 247~250C (dec). Source: HUANG
Mangifera indica. Ref: 6.
YAO ZI Dioscorea bulbifera. Ref: 6, 641.
O
OH
HO
6432 :-Diolein
C39H72O5 (621.01). Source: MANG GUO HE Mangifera indica. Ref: 6.
H
O
OH
O
O
6437 Dioscin
HO
[19057-60-4] C45H72O16 (869.07). White amorphous powder, mp 288C,

[]D20 = 115 (c = 0.4, MeOH); []D25 = 108.0 (c = 0.07, pyridine).
6433 Dioncophyllinol B
Pharm: Antifungal (hmn pathogenic yeasts Candida albicans, MIC =
C23H25NO4 (379.46). Pharm: Antimalarial (Plasmodium falciparum K1, IC50
12.5g/mL; Candida glabrata, MIC = 12.5g/mL; Candida tropicalis,
= 34ng/mL, NF54, IC 50 = 43ng/mL, MIC > 200g/mL). Source:

SAN YE MU Triphyophyllum peltatum (leaf). Ref: 3962.
MIC = 25g/mL)[4931]; antifungal (Trichophyton mentagrophytes);

insecticidal; cytotoxic (HL-60); cytotoxic (in vitro: A375, IC50 =
(2.381.12)mol/L, control Mithramycin, IC 50 = (0.370.05)mol/L;
OH
L-929, IC50 = (2.671.38)mol/L, Mithramycin, IC 50 =

(0.310.03)mol/L; HeLa, IC50 = (3.061.95)mol/L, Mithramycin, IC 50
NH
OH
OH
= (0.190.03)mol/L)[5000] . Source: BAI YAO ZI Stephania cepharantha,

BI XIE Dioscorea hypoglauca [Syn. Dioscorea collettii var. hypoglauca],
CHUAN LONG SHU YU Dioscorea nipponica, CI JI LI Tribulus
terrestris, FU ZHOU SHU YU Dioscorea futschauensis, HUANG SHAN
YAO Dioscorea panthaica, LONG XUE SHU Dracaena draco (stem

cortex)[4696] , MIAN BI XIE Dioscorea spongiosa (Rhizome: yield =
6434 Diosbulbin A
0.0019%)[4692] , RI BEN SHU YU Dioscorea japonica, SHAN BI XIE
[20086-05-9] C20H24O7 (376.41). mp 265C. Source: HUANG YAO ZI
Dioscorea tokoro, SHAN YAO Dioscorea batatas [Syn. Dioscorea
Dioscorea bulbifera. Ref: 6, 641.
opposita], SHU KUI YE SHU YU Dioscorea althaeoides, XIAN XI SHU

YU Dioscorea gracillima, ZAO XIU Paris polyphylla, HU BEI HUANG
Costus sp., Trigonella sp. Ref: 4, 10, 658, 660, 2165, 4692, 4696, 4931,
5000, 5501.
HO
JING Polygonatum zanlanscianense, Dioscorea cayenensis (rhizome),
O
O
O
H
H
6435 Diosbulbin B
HO
[20086-06-0] C19H20O6 (344.37). mp 285C (dec). Source: HUANG YAO ZI

Dioscorea bulbifera. Ref: 6, 641.
OO
OH
OH
OO
OH
OO
O
OH OH
H
O
O
O
H
OH OH
H
H
200
6438 Dioscoreside C

O
pyridine). Source: HUANG SHAN YAO Dioscorea panthaica. Ref: 867, 2075.
O
H
H
H O
H
H
OO
HO
OH
OH
OO OH
OH OH
HO
H
O
H HO
6441 Diosgenin acetate
OH
OH
O
O
C29H44O4 (456.67). Source: FANG JI YE BA QIA Smilax menispermoidea, BI

XIE Dioscorea hypoglauca [Syn. Dioscorea collettii var. hypoglauca]. Ref:
OH
10, 660.
OH OH
6439 Dioscorine
[3329-91-7] C13H19NO2 (221.30). mp 55C. Pharm: Anticholinergic (gpg
ileum, in vitro); enhances action to boost blood pressure caused by adrenalin
H
O
(anesthetic cat); local anesthetic (gpg, local injection); similar action with
cocaine. Source: BAI SHU LANG Dioscorea hispida, CU MAO SHU YU
H
H
Dioscorea hirsuta. Ref: 6, 658.

N
6442 Diosgenin-3-di--O-glucopyranoside
Diosgenin-dioglucoside C39H62O13 (738.92). mp 271~273C. Source: SHAN

YAO Dioscorea batatas [Syn. Dioscorea opposita], DUN YE SHU YU
Dioscorea zingiberensis. Ref: 6, 10.
6440 Diosgenin
O
Dioscorea sapogenin [512-04-9] C27H42O3 (414.63). mp 205~206C;

189~192C; 196~198C; 204~205C; 199~202C; from moldy source plant,
both mp and content of sapogenin decreasing, mp 195~196C; 176~178C;
186~194C; 194~195C; 180~192C. Pharm: Estrogenic activity ;
antihypercholesterolemic (reduces the level of cholesterol in serum). Source:
HO
BAI SHU LANG Dioscorea hispida, BI XIE Dioscorea hypoglauca [Syn.
H
H
OO
OH
Dioscorea collettii var. hypoglauca] (dried rhizome: mean content of 3 batch
OO
HO
samples = 1.24%[5508]), CHA RUI SHU YU Dioscorea collettii, CHAI
OH
HUANG JIANG Dioscorea nipponica ssp. rosthornii, CHANG YAO GE
OH
CHONG LOU Paris polyphylla var. pseudothibetica (rhizome: content =
OH
OH
0.83%)[5508], CHUAN LONG SHU YU Dioscorea nipponica (dried rhizome:

content = 1.73%[5508]), DUN YE SHU YU Dioscorea zingiberensis (dried
6443 Diosgenin-3-O--D-glucopyranoside
rhizome: mean content = 2.39%[5508]), FANG JI YE BA QIA Smilax
Trillin C33H52O8 (576.78). mp 274C; 275~280C. Source: DUN YE SHU YU
menispermoidea, FU ZHOU SHU YU Dioscorea futschauensis, HU LU BA
Dioscorea zingiberensis, CHUAN LONG SHU YU Dioscorea nipponica, FU
Trigonella foenum-graecum (dried ripe seed: mean content of 3 origins =
ZHOU SHU YU Dioscorea futschauensis, YAN LING CAO Trillium
12.9%)[5508], HUANG SHAN YAO Dioscorea panthaica, LONG XUE SHU
tschonoskii, ZAO XIU Paris polyphylla. Ref: 6, 10, 660.
Dracaena draco (stem cortex)[4696], MAI DONG Ophiopogon japonicus

(dried tuberoid: mean content = 0.005%)[5508], MIAN BI XIE(I) Dioscorea
septemloba, QIU YAO GE CHONG LOU Paris fargesii (rhizome: content =

1.08%)[5508], SHAN YAO Dioscorea batatas [Syn. Dioscorea opposita]
O
H
(rhizome: content = 0.012%)[5508], SHU KUI YE SHU YU Dioscorea

althaeoides, XIA YE CHONG LOU Paris polyphylla var. stenophylla
(rhizome: content = 0.86%)[5508], XIAN XI SHU YU Dioscorea gracillima,

XIAO HUA DUN YE SHU YU Dioscorea parviflora, YUN NAN CHONG
OH
[5508]
LOU Paris polyphylla var. yunnanensis (rhizome: mean content = 0.94%)
ZAO XIU Paris polyphylla (rhizome: content = 0.90%)[5508], ZHANG LIU

TOU Costus speciosus, Paris sp., Trillium sp., Trigonella sp. Ref: 10, 658,
660, 4696, 5501, 5508.
OO
HO
OH
OH
H
H
201
6444 Diosgenin -3-O--D-glucopyranosyl (14) --L-rhamnopyranosyl
(14)--D-glucopyranosyl (14)--D-glucopyranoside
C51H82O22 (1047.21). White powder crystals, mp 229~233C (des), []D =
O
H
70.42 (c = 0.738, MeOH). Source: HU LU BA Trigonella foenum-graecum.

Ref: 4578.
H
O
H
H
OO
HO
OH
OH O O
O O OH
OH OH
OH OH
OO
HO
OO
OH OH
OH
OO
HO
OH
OH
OO
HO
6448 Diosgenin 3-O-[-L-rhamnopyranosyl (13)--L-rhamnopyranosyl (14)--L-rhamnopyranosyl (14)]--D-glucopyranoside
OO
OH
OH
C51H82O20 (1015.21). Colorless acicular crystals, mp 216~218C (dec.), [] D20

= 96.2 (c = 0.38, pyridine), easily solving in pyridine, solving in methanol,
OH
OH OH OH
ethanol and water. Source: CHUAN LONG SHU YU Dioscorea nipponica.
6445 Diosgenin palmitate
Ref: 2227.
C43H72 O4 (653.05). Source: CHA RUI SHU YU Dioscorea collettii, BI

XIE Dioscorea hypoglauca [Syn. Dioscorea collettii var. hypoglauca].
Ref: 10, 660.

O
H
H
O
H
O
HO
OO
OH
OH
OO
OO
OH
6446 Diosgenin-3-O--L-rhamnopyranosyl-(12)[-L-arabinofuranos-
OH
yl-(14)]--D-glucopyranoside
OO OH OH OH
C44H70O16 (855.04). mp 276~278C (dec). Source: ZAO XIU Paris polyphylla.

OH OH
Ref: 6.
O
6449 Diosgenin -3-O--L-rhamnopyranosyl (13)--L-rhamnopyranosyl (14)--D-glucopyranosyl (14)--D-glucopyranoside
O
H
H
HO
C51H82O21 (1031.21). White granular crystals, mp 196~197C (des), []D20 =
78.92 (c = 0.937, MeOH). Source: HU LU BA Trigonella foenum-graecum.
Ref: 4578.
OO
OH
HO
O
OH
O
OH
OO
OH
OH OH
H
H
6447 Diosgenin 3-O--L-rhamnopyranosyl-(14)--L-rhamnopyranos-
OH
yl-(14)-[-L-rhamnopyranosyl-(12)]--D-glucopyranoside
OH
[]D20 = 113 (c = 057, MeOH); mp 203~206C (dec). Pharm: Antifungal
OH
(hmn pathogenic yeasts Candida albicans, MIC = 100 g/mL; Candida
OO
[4931]
glabrata, MIC = 200g/mL; Candida tropicalis, MIC > 200g/mL)
cytotoxic (HSC-2 cells, LD50 = 2g/mL; HGF, LD50 = 2.8g/mL)[3023]; .
OO
HO
Diosgenin tetraglycoside C51H82O20 (1015.21). White amorphous powder,
OH
OO OH
Source: Dioscorea cayenensis (rhizome), YE XIANG SHU Cestrum

nocturnum (leaf: yield = 0.0024%fw), ZAO XIU Paris polyphylla. Ref: 4931,
6, 3023.
OO
HO
OH OH
OH
OH
H
H
202
6450 Diosindigo A
LIN SHENG XUAN SHEN Scrophularia nodosa, MI DIE XIANG
C24H20O6 (404.42). Deep blue needles (petrol ether-chloroform), Source:
Rosmarinus officinalis, NING MENG Citrus limon, NING MENG PI Citrus
Diospyros sylvatica (root). Ref: 3811.
limon, QIAN MA Urtica cannabina, RU DI JIN NIU Zanthoxylum nitidum,

YING BU BO Zanthoxylum avicennae. Ref: 6, 658, 660, 5501.
OH
OH
OH
OH
OO
OO
OH
6451 Dioslupecin A
C39H56O3 (572.88). Source: HAI SHI Diospyros maritima, XIAO HUA MU
OH
O
OH
OH OH
OH
LAN GUO Bruguiera parviflora. Ref: 1521, 2532.

6455 Diosphenol
[490-03-9] C10H16 O2 (168.24). Pharm: Diuretic. Source: MI HUA
XIANG MAO Cymbopogon densiflorus, YU XIANG CAO Mentha

H
rotundifolia. Ref: 658.
H
O
OH
HO
6452 Diosmetin
5,7,3'-Trihydroxy-4'-methoxyflavone [520-34-3] C16H12O6 (300.27). mp
253~255C. Pharm: Protects against shock. Source: BAI CI HUA Sophora
6456 Diospongin A
viciifolia, MENG GU SHAN LUO BO Scabiosa comosa, RONG MAO DAN
SHEN Salvia tomentosa, YAO YONG PU GONG YING Taraxacum officinale.
CHCl3). Pharm: Bone resorption inhibitor (bones were cultured with PTH
Ref: 6, 561, 602, 658, 660.
200mol/L, 45Ca release = (44.63.3)%, control 45Ca release = (15.41.3)%).

Source: HAI JIN BI XIE Dioscorea spongiosa (rhizome). Ref: 4921.
OH
HO
OH
O
OH
6453 Diosmetin 7-O--D-glucopyranoside

C22H22O11 (462.41). Pharm: Aldose reductase inhibitor (rat lens, IC50 =
23mol/L, control Epalrestat, IC50 = 0.072mol/L)
[4214]
. Source: YE JU HUA
Chrysanthemum indicum (flower: yield = 0.086%). Ref: 4214.

OH
O

CHCl3). Pharm: Bone resorption inhibitor (bones were cultured with PTH
200mol/L, 45Ca release = (30.50.4)%, contro 45Ca release = (15.41.3)%).
Source: HAI JIN BI XIE Dioscorea spongiosa (rhizome). Ref: 4921.
OO
HO
6457 Diospongin B
OH
OH
OH
OH
6454 Diosmin
[520-27-4] C28H32O15 (608.56). mp 278~280C. Pharm: Anti-inflammatory
(rat, ip, swollen foot model caused by carrageenan, ED50 = 100mg/kg); similar
action with vitamin C2 (gpg, enhances blood capillary resistance and reduces
loss of ascorbic acid in adrenal); similar action with vitamin P (rbt, reduces
blood capillary permeability); LD50 (mus, orl) = 10g/kg, (mus, ip) = 4g/kg.
Source: BA XIAN CAO Galium aparine, BAI CI HUA Sophora viciifolia,
BAI CI HUA YE Sophora viciifolia, FEI LONG ZHANG XUE Toddalia
asiatica [Syn. Toddalia aculeata; Paullinia asiatica], FO SHOU Citrus
medica var. sarcodactylis, GAO JIA SUO LAN PEN HUA Scabiosa
caucasica, JI CAI Capsella bursa-pastoris, JI CAI ZI Capsella bursa-pastoris,
OH
6458 Diospongin C
C19H24O4 (316.40). Light yellow oil, []D25 = 45.5 (c = 0.5, CHCl3). Pharm:
Bone resorption inhibitor (bones were cultured with PTH 200mol/L, 45Ca
release = (19.11.6)%, p<0.01, control 45Ca release = (15.41.3)%). Source:
HAI JIN BI XIE Dioscorea spongiosa (rhizome). Ref: 4921.
OH
OH
OH
OH
203
6459 Diospyrin
6464 ent-2,7-Dioxo-3-cleroden-15-oic acid
[28164-57-0] C22H14O6 (374.35). Pharm: Cytotoxic (EAC, high dose);
C20H30O4 (334.46). Colorless oil, [] D20 = 10 (c = 0.215, CHCl3). Pharm:
immunoenhancer (low dose). Source: Diospyros sp. Ref: 658.
Antimalarial (Plasmodium falciparum FcB1, IC50 = (8.00.2)g/mL, control
OH
Chloroquine, IC50 = (0.050.002)g/mL). Source: Nuxia sphaerocephala
O
OH
(leaf). Ref: 4419.
OH
O
6460 Diospyrol
C22H18O4 (346.39). Acicular crystals (methanol), mp 251~257C (dec). Pharm:
Anthelmintic (hookworm, dwarf tapeworm). Source: RUAN SHI Diospyros
mollis (the compound was isolated from the plant by K.Yoshihira, et al. in
6465 1-(1,6-Dioxo-2E,4E-decadienyl)piperidine
1969)[5505]. Ref: 661, 5505.
C15H23NO2 (249.36). Colorless oil. Source: HU JIAO Piper nigrum (root:
OH
OH
OH
yield = 0.00031%dw). Ref: 4753.
OH
6461 Diospyrosonaphthoside
4[-L-Rhamnosyl(12)--D-glucopyranosyloxy]-2-hydroxymethylene,5-hydroxy
naphthalene C23H30O12 (498.49). White amorphous powder, []D27 = 119.0 (c =
0.17, MeOH). Source: Diospyros angustifolia (stem cortex). Ref: 3835.
HO
6466 4,5-Dioxodehydroasimilobine
2-Hydroxy-1-methoxy-4H-dibenzo[de,g]quinoline-4,5-(6H)-dione
C17H11NO4 (293.28). Pharm: Platelet aggregation inhibitor (rbt platelets
OO
HO
OH
induced by thrombin, 50g/mL, add thrombin 0.1u/mL, AggRt =
HO
(86.61.6)%, control AggRt = (92.60.4)%; add AA, 100mol/L, 50g/mL,
OH
OO
OH OH
AggRt = (0.00.0)%, 2g/mL, control AggRt = (80.71.7)%, Aspirin

50g/mL, AggRt = (11.710.1)%; add collagen 10g/mL, 50g/mL, AggRt
OH
= (25.40.9)%, 2g/mL, AggRt = (81.50.0)%, control AggRt =

(89.30.5)%, Aspirin 100g/mL, AggRt = (81.30.5)%; add PAF 2ng/mL,
6462 Diospyrosooleanolide
2-Hydroxy-3-trans-p-coumaroyl-28,19-oleanolide C39H54O6 (618.86).
29
50g/mL, AggRt = (87.20.0)%, control AggRt = (93.00.6)%)[4938].
White amorphous powder, []D = 16.6 (c = 0.102, C5H5N). Source:
Source: MIAN MAO MA DOU LING Aristolochia mollissima (dried root
Diospyros angustifolia (stem cortex). Ref: 3835.
and stem: yield = 0.00037%dw), TAI WAN HU JIAO Piper taiwanense

(stem). Ref: 3026, 4938.
O
O
OH
O
HO
O
N
H
HO
6463 Diospyrososide
1[-L-Rhamnosyl(12)-(-D-glucopyranosyloxy)]-3,4,5-trimethoxy benzene
6467 3,12-Dioxo-15,16-epoxy-4-hydroxy-cleroda-13(16),14-diene
MeOH). Source: Diospyros angustifolia (stem cortex). Ref: 3835.

O
O
OO
HO
OH
OH
OO
OH
OH
OH
O
HO
204
6468 3,24-Dioxo-friedelan-29-oic acid
6474 3,11-Dioxo-labda-8(17),13(16),14-triene
[105249-56-7] C 30H46O4 (470.70). Colorless acicular crystals, mp 294C.
C20H28O2 (300.44). []D20 = +12.1 (c = 2.5, CHCl3). Source: YUAN YE TAI
Source: LEI GONG TENG Tripterygium wilfordii. Ref: 60.
Jamesoniella colorata. Ref: 3375.
O
O
OH
H
O
6475 3,11-Dioxo-olean-12-ene
6469 3,18-Dioxo-11-hydroxycona-1,4-diene
C30H46O2 (438.70). White lamellar crystals (acetone), easily soluble in CHCl3
C21H27NO3 (341.45). Orange rods (MeOH), mp 130~132C. Source: DUAN
and MeOH, mp 232~235C. Source: SI CHUAN QING FENG TENG Sabia
ROU MAO ZHI XIE MU Holarrhena pubescens (bark). Ref: 5231.
schumanniana (aerial parts). Ref: 4883.
H
N
HO
H
H
O
6470 3,8-Dioxo-7-hydroxy-7,9-cyclo-7,8-seco-24Z-tirucalladien-26-oic acid
6476 8,19-Dioxo-8,14-seco-chinan-14,11-olide
C30H46O5 (486.70). Colorless powder, mp 95~98C, []D = +255.1 (c = 1.0,
C20H30O4 (334.46). Colorless solid, mp 163~164C, []D27 = 101.5 (c = 0.47,
MeOH). Source: Juliania adstringens (bark). Ref: 3786.
CHCl3). Source: LONG BAI Juniperus chinensis var. kaizuka (leaf: yield =
0.00012%dw). Ref: 3050.
O
OH
H
H
O
OH
6471 7,11-Dioxo-3-hydroxy-8,24Z-tirucalladien-26-oic acid
C30H44O5 (484.68). Yellow powder, mp 94~95C, []D = 85.7 (c = 1.0,

MeOH). Source: Juliania adstringens (bark). Ref: 3786.
6477 3,22-Dioxo-20-taraxastene
C30H46O2 (438.70). Colorless solid, mp 245~248C, []D24 = +63.9 (c = 0.2,
CHCl3). Pharm: Cytotoxic inactive (HONE-1 cell, IC50 > 10mol/L; KB cell,
OH
IC50 > 10mol/L; HT29 cell, IC50 > 10mol/L). Source: RONG SHU Ficus
microcarpa (aerial root). Ref: 5254.
HO
6472 (2,5-Dioxo-4-imidazolidinyl)carbamic acid
C4H5O4N3 (159.10). Colorless block crystals, mp 244~246C. Source: ROU

CONG RONG Cistanche deserticola. Ref: 825.
O
HO
O
H
N
NH
N
H
6473 10,22-Dioxokopsan
6478 3,7-Dioxo-8,24Z-tirucalladien-26-oic acid

C30H44O4 (468.68). Colorless powder, mp 91~93C, []D = 27.7 (c = 1.0,
MeOH). Pharm: Cytotoxic (leukemia cells L1210, IC50 = 30g/mL). Source:
Juliania adstringens (bark). Ref: 3786.
C20H20N2O2 (320.39). Source: HONG HUA RUI MU Kopsia fruticosa (leaf).

Ref: 3830.
O
H
O
N
H
OH
205
6479 3,4-Dioxymethylene-5-methoxy-1-(1-oxopropyl)benzene
6484 Dipetaline
3,4-Methylendioxy -5-methoxy-1-(1-oxopropyl)benzene C11H12O4 (208.22).
[59701-36-9] C20H22O4 (326.40). Pharm: Cytotoxic (inhibits DNA
mp 87~88C, 91~92C. Source: SHA QIAN HU Ferula borealis. Ref: 6.
biosynthesis by blocking thymidine to go into HL-60 cells). Source: MEI

ZHOU HUA JIAO Zanthoxylum americanum [Syn. Xanthoxylum americanum]
Ref: 2176.
O
O
6480 (2S)-1,3-Di-(O-palmitoyl)-2-O-octadecanoyl glycerol

C53H102O6 (835.40). Source: XI NANG MA WEI ZAO Sargassum
parvivesiculosum. Ref: 2591.
6485 2,3-Diphenyl-2-cyclopropen-1-one
[886-38-4] C15H10O (206.25). Source: DU HUO Angelica pubescens f.
biserrata [Syn. Angelica pubescens]. Ref: 2.
O
O
O
6481 (2S)-1,2-Di-O-palmitoyl-3-O-(6-sulpho--D-quinovopyranosyl) glycerol

C41H78O12S (795.14). White powder. Source: XI NANG MA WEI ZAO
Sargassum parvivesiculosum. Ref: 2591.
6486 2,2'-Di-(2-phenylethyl)-8,6'-dihydroxy-5,5'-bichromone (AH11)

C34H26O6 (530.58). Light dark-yellow powder, mp 239~242C. Source:
CHEN XIANG Aquilaria agallocha. Ref: 13.
HO S
OH
OH
O
OH
HO
O
O
O
O
O
OH
6482 Dipentene
1,8-p-Menthadiene [138-86-3] C10H16 (136.24). bp 178C. Pharm: Antitussive
(dispels phlegm); sedative; sensitizer; irritant. Source: DA YE XIANG RU Mosla
6487 trans-1,7-Diphenyl-1-hepten-5-ol
trans-1,7-Diphenyl-5-hydroxy-1-heptene [87095-76-9] C19H22O (266.38).
dianthera, FENG XIANG SHU Liquidambar formosana [Syn. Liquidambar
White rhombic crystals (hexaneacetone), mp 47~49C, []D20 = +7 (c = 1.2,
taiwaniana], GANG SONG Baeckea frutescens, HAI SONG ZI Pinus koraiensis,
chloroform). Pharm: Anti-inflammatory (swollen foot model caused by
HU SUI ZI Coriandrum sativum, HUI XIANG Foeniculum vulgare, KUO YE XIE
carrageenan); nematocide (EC95 = 0.7g/mL). Source: CAO DOU KOU
CAO Valeriana officinalis var. latifolia, LU DOU LE HUA Pandanus tectorius,
Alpinia katsumadai. Ref: 978, 1069, 1151, 1152.
MO YAO Commiphora myrrha [Syn. Commiphora molmol], RU XIANG
HO
Boswellia carterii, YA ER QIN Cryptotaenia japonica. Ref: 6, 660.
6483 5,3'-Dipent-4-enoyloxy-3,6,7,4'-tetramethoxyflavone
6488 1,7-Diphenylhept-4-en-3-one
C19H20O (264.37). Colorless or yellow oleaginous liquid. Pharm:
5-Reductase inhibitor (rat prostate 5-Reductase, IC50 = (39030)mol/L,
control Curcumin, IC50 > 1000mol/L, Finasteride, IC50 = 0.01mol/L)[5345].
Source: GAO LIANG JIANG Alpinia officinarum. Ref: 435, 5345.
O
O
O
O
O
O
O
206
6489 1,3-Diphenylpropane-1,2-diol-3-one
6492 Diphylloside A
C15H14O3 (242.28). Source: LUO HUA SHENG Arachis hypogaea. Ref: 6.
Ikarisoside C [113558-11-5] C38H48O20 (824.79). Yellow powder, mp

204~206C. Source: CHUAN E YIN YANG HUO Epimedium fargesii, CU
MAO YIN YANG HUO Epimedium acuminatum, WAN SHAN YIN YANG
HUO Epimedium wanshanense, YIN YANG HUO Epimedium brevicornum.
Ref: 465, 565, 567, 624.
HO
OH
OH
OO
HO
OH
OH
6490 Diphyllin
OH
OH
OH O O
[22055-22-7] C21H16O7 (380.36). mp 291C. Pharm: Antineoplastic; cytotoxic
OH
OO
OH
HO
(hmn LoVo Cell Line, in Vitro, IC50 = (7.550.75)l/mL)[4206]; cytotoxic (in

vitro, 212, ED50 = 2.7g/mL, control cis-Platin, ED50 = 1.3g/mL; CaSki, no
OH
significant activity, control Actinomycin D, ED50 = 0.0019g/mL; Hep3B,

ED50 = 3.6g/mL, control 5-FU, ED50 = 0.0715g/mL; SiHa, no significant
activity, control Actinomycin D, ED50 = 0.00081g/mL; HepG2, ED50 =
0.4g/mL, control 5-FU, ED50 = 0.033g/mL; HT29, ED50 = 2.5g/mL,
control 5-FU, ED50 = 0.074g/mL; HCT116, ED50 = 0.8g/mL, control 5-FU,
ED50 = 0.48g/mL; MCF7, no significant activity; MCF7-ras, no significant
OH
6493 Diphylloside B
[118544-18-6] C38H48O19 (808.79). Yellow powder, mp 187~189C. Source:
WAN SHAN YIN YANG HUO Epimedium wanshanense, CU MAO YIN
YANG HUO Epimedium acuminatum. Ref: 465, 624.
OH
activity)[4612]; piscicide. Source: JUE CHUANG Rostellularia procumbens

[4612]
[Syn. Justicia procumbens] (whole herb: yield = 0.00024%dw)
, SHAN
Diphylleia sinensis (rhizome: content scope = 0.1%0.5%, mean content of 8
OO
HO
HE YE Diphylleia grayi (rhizome: content = 0.064%)[5508], WO ER QI
OH
OH
origins = 0.388% [5508]), Haplophyllum patavinum (shoot). Ref: 6, 279, 658,
OH
OH
OH
4206, 4612, 5508.

OH
OH O
O
O
O
OH OH
6494 Dipiperitylmagnolol
O
O
C38H50O2 (538.82). Source: DU HUO Angelica pubescens f. biserrata [Syn.

O
OH
OH HO
6491 Diphyllin acetylapioside

C28H26O12 (554.51). Pharm: Anti-inflammatory (5-lipoxygenase
inhibitor)[4415]. Source: XI BAN YA YUN XIANG CAO Haplophyllum
hispanicum. Ref: 4415.
6495 Dipotassium rabdosiin
O
C36H28K2O16 (794.81). Tan amorphous powder, []D22 = 113.4 (c = 0.91,
H2O). Pharm: Contraceptive. Source: XIN ZANG JIA ZI CAO Arnebia

euchroma. Ref: 2187.
O
O
O O
HO
HO
O
OH OH
O
H
OH
OH
OH
H
OH
OH
O
+
K
OH
207
6496 6,8-Diprenylgenistein
6500 5,3'-Dipropanoyloxy-3,6,7,4'-tetramethoxyflavone
5,7,4'-Trihydroxy-6,8-diprenylisoflavone C25H26O5 (406.48). Yellow
amorphous. Pharm: Antifungal (dermatophyte Trichophyton mentagrophytes,
250g/mL)[2347]. Source: KU TAN ZI Millettia pachycarpa, SAN XIAU YE
SHAN DOU GEN Euchresta japonica, PAN YUAN YU TENG Derris
scandens, Erythrina vogelii. Ref: 1521, 2347, 4421.

O
O
O
HO
O
O
OH
O
O
OH
6501 Dipropyl disulfide
6497 6,8-Diprenylnaringenin
4,5-Dithiaoctane [629-19-6] C6H14S2 (150.31). Colorless volatile oil with a
Lonchocarpol A C25H28O5 (408.50). Pharm: Cytotoxic (cyclooxygenase-2
strong odour of garlic. Pharm: Antifungal (plant pathogenic fungi
inhibitor, IC50 = 3.9g/mL)[5038]; cytotoxic (mouse mammary organ culture
Cladosporium sphaerospermum, MIC = 0.1g, control Nystatin, MIC = 1.0g;
assay, 86% at 10g/mL)[5038]. Source: PI JIU HUA Humulus lupulus (strobile),
Cladosporium cladosporioides, MIC = 1.0g, control Nystatin, MIC =
ZHEN YE XUE TONG Macaranga conifera. Ref: 4789, 5038.
1.0g)[5159]; antineoplastic (mechanism-based yeast bioassay for

OH
= 11g/mL, control Camptothecin, RS 52YK(rad 52Y), IC12 = 0.6g/mL)[5159];

flavorant. Source: SUAN CHOU MU JI CAO Petiveria alliacea (root, stem
HO
and leaf), DA SUAN Allium sativum, Allium sp. Ref: 2, 658, 5159.
OH
S S
6498 6,8-Diprenylumbelliferone
6502 Dipterocarpol
[471-69-2] C30H50O2 (442.73). Pharm: Induces growth of radial root nodule
500(mol ratio/32pmol TPA): EBV-EA-positive cells = (23.71.3)%
commensal Frankia. Source: RU DU XIANG Pistacia terebinthus, BING
PIAN Dryobalanops aromatica. Ref: 2, 658.
(viability = 60%), Curcumin, EBV-EA-positive cells = (22.81.8)%

(viability > 80%), compound IC50 = 216(mol ratio/32pmol TPA),
HO
-Carotene, IC50 = 400(mol ratio/32pmol TPA), Curcumin, IC50 = 341(mol
ratio/32pmol TPA)). Source: CHENG ZI Citrus junos. Ref: 5048.
H
O
HO
6503 cis-Diptoindonesin B
C42H32O9 (680.72). White amorphous powder, []D20 = 99 (c = 0.1, MeOH).
Source: JU YUAN YE LONG NAO XIANG Dryobalanops oblongifolia. Ref: 3422.
6499 2,6-Diprenyl-4-vinylphenol
HO
C18H24O (256.39). Amorphous powder. Source: FENG JIAO Apis mellifera

ligustica. Ref: 4124.
OH
HO
OH
HO OH
OH
O
HO
H
H
208
6504 trans-Diptoindonesin B
6508 1,2-Di-O-E-sinapoyl--gentiobiose
C42H32O9 (680.72). White amorphous powder, []D20 = 192 (c = 0.1,
C34H42 O19 (754.70). Source: OU ZHOU YOU CAI Brassica napus (seed).
MeOH). Source: JU YUAN YE LONG NAO XIANG Dryobalanops
Ref: 5289.
oblongifolia. Ref: 3422.

HO
OO
HO
OH
OH
OH
HO
OO
OH
O
OH
OH
OH
OH
O
HO
OH
H
HO
6509 1,2-Di-O-E-sinapoyl--glucopyranose
H
C28H32O14 (592.56). Source: OU ZHOU YOU CAI Brassica napus (seed). Ref: 5289.
OH
OO
HO
OH
6505 Discarine M
OH
C26H37N3O5 (455.60). White amorphous powder, []D20 = 176.7 (c = 0.2,

MeOH:CHCl3 = 1:1). Source: Discaria americana (bark). Ref: 3793.
OH
OH
H
O
OO
H
H N H N
O
H
H
N
H H
6510 1,6-Di-O-sinapoylglucose
1,6-Di-O-E-sinapoyl--glucopyranose C28H32O14 (592.56). Source: OU
ZHOU YOU CAI Brassica napus (seed). Ref: 5289.
O
O
O
6506 Discarine N
C32H33N3O5 (539.64). White powder, mp 233~235C, []D20 = +98.1 (c =
OH
C34H42O19 (754.7). Yellow prisms, mp 133~135 (MeOH). Source: CHOU
H N H N
O
H
OH
O
O
6511 3',6-Disinapoylsucrose
H
H
OO
OO
OH
HO
0.092, MeOH:CHCl3 = 1:1). Source: Discaria americana (bark). Ref: 3793.
OH
CAO Ruta graveolens (dried aerial parts). Ref: 3073.
N H
HO
HO
HO
HO
HO
HO
O
O
O
OH
OH
O
HO
6507 Disenecionyl cis-khellactone

C24H26 O7 (426.47). Pharm: Antispasmodic; coronary vasodilator. Source:
HUI BAI XIE HAO Seseli incanum, LI BA NEN XIE HAO Seseli
libanotis. Ref: 658.
6512 Disinomenine
[596-58-7] C38H44N2O8 (656.78). mp 222C. Source: BIAN FU GE
Menispermum dauricum, QING FENG TENG Sinomenium acutum. Ref: 6.
O
O
O
OH
HO
O
O
O
O
H
O
O
N
O
N
O
209
6513 Dispardiol B
6517 Dispegatrine
5,7-Dihydroxy-8-(2,3-dihydroxy-3-methylbutyl)-6-(2-methyl-1-oxobutyl)-4-p
[102488-56-2] C40H48N4O42+ (648.85). Colorless square crystals, mp > 280C
henyl-2H-[1]benzopyran-2-one C25H28O7 (440.50). []D25 = 0 (c = 0.08,
(dec), []D23 = +230 (c = 0.1, methanol). Pharm: Adrenergic -receptor
CHCl3). Source: BU DENG HONG HOU KE Calophyllum dispar (fruit and
blocker. Source: HAI NAN LUO FU MU Rauvolfia verticillata var.
stem cortex). Ref: 5196.
hainanensis. Ref: 46.

H
H H
N
OH
HO
O
OH
H H
H H
HO
HO
HO
N
H H
HO
OH
6514 Disparinol B
6518 Dissectol A
C25H26O6 (422.48). Pharm: Cytotoxic (KB, EC50 = 7g/mL). Source: BU
C16H26O7 (330.38). Syrup, []D26 = +125.0 (c = 2.0, MeOH). Pharm:
DENG HONG HOU KE Calophyllum dispar (fruit and stem cortex). Ref:
Antitubercular (Mycobacterium tuberculosis, showed modest activity when
5196.
compared to rifampicin in an agar diffusion assay). Source: SHEN LIE YE

JIAO HAO Incarvillea dissectifoliola. Ref: 5403.
O
OH
OH
HO
OH H
HO
HO
OH
6515 Disparinol D
5,7-Dihydroxy-8-(2-hydroxy-3-methylbut-3-enyl)-6-(2-methyl-1-oxopropyl)-
6519 (2S)-1,2-Distearoyl-3-O-(6-sulpho--D-quinovopyranosyl)-glycerol
4-phenyl-2H-[1]benzopyran-2-one C24H24O6 (408.46). []D25 = 0 (c = 0.16,
C45H85O12S (850.24). Source: KA SHI QIAN GOU ZAO Amphidinium
CHCl3). Pharm: Cytotoxic (KB, EC50 = 21g/mL). Source: BU DENG HONG
carterae. Ref: 4448.
HOU KE Calophyllum dispar (fruit and stem cortex). Ref: 5196.
O
O
OH
OO
O
HO
OH
O
OH
OH
HO
O
O
6516 Disparpropylinol B
5,7-Dihydroxy-8-(2-hydroxy-3-methylbut-3-enyl)-6-(2-methyl-1-oxobutyl)-4propyl-2H-[1]benzopyran-2-one C22H28O6 (388.46). Yellow crystals, mp
111~112C (n-hexane:EtOAc = 9:1), []D25 = 0 (c = 0.6, CHCl3). Pharm:
6520 Diterp-Complex-RA
C42H60O13 (772.94). mp 213~215C, []D = 46.5 (c = 0.16, MeOH). Source:
XIA YE XIANG CHA CAI Isodon angustifolia. Ref: 4067.
Cytotoxic (KB, EC50 = 4g/mL). Source: BU DENG HONG HOU KE

Calophyllum dispar (fruit and stem cortex). Ref: 5196.
H
O
OH
H
H
H
O
HO
HO
H
O
O
OH
OH
OH
210
6521 Diterpenoid EF-D
6527 Diuranthoside G
C27H38O7 (474.60). Pharm: Irritant (to skin). Source: NONG DA JI Euphorbia
C62H100O33 (1373.47). White powder. Source: NAN CHUAN LU SI CAO
fortissima. Ref: 658.
Diuranthera inarticulata. Ref: 2122.
O
O
O
H
H
OH
O
OH
O
HO
OH
6522 2,6-Ditertbutyl-4-methyl phenol
HO
OH
[128-37-0] C15H24O (220.36). Source: REN SHEN Panax ginseng [Syn.

Panax schinseng], SAN QI Panax pseudo-ginseng var. notoginseng [Syn.
OH
HO
OO
OH
OH
OH
OO
HO
O
HO
O O
O
O
O
OH
OH
OH
OH
OH
Panax notoginseng], XI YANG SHEN Panax quinquefolium. Ref: 2.
OH
OH
6528 Diuvaretin
OH
C30H28O6 (484.55). Colorless crystals, mp 127~131C (CHCl3). Pharm:

Cytotoxic (hmn promyelocytic leukemia HL-60 cells, IC50 = 6.1mol/L).
Source: JIAN ZI YU PAN Uvaria acuminata (root). Ref: 4261.
HO
6523 Ditertbutyl phthalate

C16H22O4 (278.35). Source: SAN QI Panax pseudo-ginseng var. notoginseng
HO

O
OH
OH
6529 Divaricatol
C17H18O7 (334.33). White crystalline powder, mp 168~171C, []589nm = 30.
Pharm: Analgesic (mus writhing method, orl, 1 mg/kg). Source: FANG FENG
6524 Dithiocyclopentene
Saposhnikovia divaricata [Syn. Ledebouriella seseloides]. Ref: 3508.
C3H4S2 (104.19). Source: DA SUAN Allium sativum. Ref: 2.
OH
OH
6525 L-3,6-Ditigloyloxytropane
6530 Divaricoside
[23517-33-1] C18H27NO4 (321.42). Source: MAO MAN TUO LUO GEN
Sarmentogenin 3-O--oleandroside C30H46O8 (534.70). mp 220~223C.
Datura innoxia. Ref: 6, 660.
Pharm: Cardiotonic (one of main components in divasides). Source: YANG
JIAO AO ZI Strophanthus divaricatus. Ref: 4, 6, 658.
6526 Diuranthoside F
HO
C62H100O33 (1373.47). White powder. Source: NAN CHUAN LU SI CAO
Diuranthera inarticulata. Ref: 2122.
H
O
OH
OO
OH
HO
HO
OH
OH
OH
OH
O
OH
OH
HO
HO
O O
OO
O
O
OH
OH
O
O
HO
OH
OH
OH
6531 Divinyl sulfide

H
Vinyl sulfide [627-51-0] C4H6S (86.16). Source: DA SUAN Allium sativum.

Ref: 2.
OH
S
OH
211
6532 Divostroside
6537 Docosanoic acid
Sarmentogenin 3-O--L-diginoside C30H46O8 (534.70). mp 225~231C.
[112-85-6] C22H44O2 (340.59). Source: BU GU ZHI Psoralea corylifolia,
Pharm: Toxin (vertebrate). Source: YANG JIAO AO ZI Strophanthus
GAN DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa f.
divaricatus. Ref: 6, 658.
huechingensis], GUANG JING QIAN CAO Rubia wallichiana (stem),

O
QIANG HUO Notopterygium incisum, WU SE MEI Lantana camara (aerial

parts). Ref: 2, 4309, 4369.
HO
H
H
OO
OH
HO
HO
O
6538 (4E,6E,2S,3R)-2-N-Docosanoyl-4,6-tetradecasphingadienine
6533 L-Djenkolic acid

C7H14N2O4S2 (254.33). Pharm: Toxin. Source: YU ZHUANG HE HUAN
Albizzia lophantha, Mimosa sp., Acacia sp. Ref: 658.
O
H2N
O
HO
OH
C36H69NO3 (563.96). White powder; mp 71.8C, []D20 = 3.6 (c = 0.176,

CHCl3). Pharm: Neurotrophic (neurite outgrowth promoter, measuring neurite
length of PC12 cell, 10mol/L, activity greater than that of 50ng/mL NGF).
Source: BAI JIANG CAN Bombyx mori. Ref: 4684.
S
S
NH2
6534 Docosane
[629-97-0] C22H46 (310.61). Source: DANG SHEN Codonopsis pilosula,
HN
SAN QI Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng].
HO
Ref: 2.
OH
6539 Docosyl caffeate

C31H52O4 (488.76). mp 115C. Source: SHAN DOU GEN Sophora
subprostrata [Syn. Sophora tonkinensis], ZI CAO Lithospermum
erythrorhizon. Ref: 6, 408, 2193.
6535 Docosanedioic acid
[505-56-6] C22H42O4 (370.58). mp 124.2~124.4C. Source: LIN BEI ZI

Toxicodendron succedaneum [Syn. Rhus succedanea], QI ZI Rhus verniciflua
[Syn. Toxicadendron verniciflum]. Ref: 6.
HO
HO
OH
O
6540 -Dodecalactone
[2305-05-7] C12H22O2 (198.31). Source: XING REN Prunus armeniaca. Ref: 2.
OH
O
6536
1,22-Docosanediol
[22513-81-1] C22H46O2 (342.61). Source: MU JIN PI Hibiscus syriacus.
6541 Dodecane
Ref: 519.
[112-40-3] C12H26 (170.34). Source: REN SHEN Panax ginseng [Syn. Panax
schinseng], XI YANG SHEN Panax quinquefolium, LANG DU Stellera
chamaejasme. Ref: 2, 660.
HO
HO
212
6542 Dodecanol
6548 ()-Dolabella-3,7,18-triene
[112-53-8] C12H26O (186.34). Source: DANG GUI Angelica sinensis. Ref: 2.
C20H32 (272.48). Source: KAN MAI NIANG ZHUANG SHA CAO Cyperus
OH
alopecuroides (essential oil). Ref: 5129.
6543 cis-4-Dodecenoic acid
6549 Dolabeserpenoic acid A
Linderic acid [2430-94-6] C12H22O2 (198.31). mp 1.0~1.3C, bp
(3E,7Z)-Dollabella-3,7,12-trien-17-oic acid C20H30O2 (302.46). Amorphous
170~172C/13mmHg. Source: ZHEN CAI Litsea pungens. Ref: 6.
powder. []D = 32.1 (c = 1.5, CHCl3). Pharm: Antifungal. Source: PU FU

QIANG DAO YAO Hypoestes serpens. Ref: 2063.
O
OH
HO
6544 Dodecenoic acid

C12H22O2 (198.31). bp 165~168C/8mmHg. Source: BING LANG Areca
catechu, FU LING Poria cocos, YANG RU Capra hircus; Ovis aries. Ref: 2, 6.
O
OH
6550 Dolichodial
[5951-57-5] C10H14O2 (166.22). Pharm: Anthelmintic; lacrimator. Source: MA
SHI XIANG KE KE Teucrium marum. Ref: 658.
H
O
H
O
6545 n-Dodecyl acetate

[112-66-3] C14H28O2 (228.38). bp 150.5~151.5C/15mmHg. Source: HEI MA
6551 Dolineone
YI Formica fusca. Ref: 6.
[10065-28-8] C19H12O6 (336.30). mp 233~235C. Pharm: Antiviral (HSV-1,

O
O
50g/mL, InRt = 15.4%; HSV-2, 50g/mL, InRt = 24.4%). Source: DI GUA

ZI Pachyrhizus erosus, DOU SHU Pachyrrhizus erosus (seed). Ref: 6, 4180.
O
H
O
H
O
O
6552 Domesticine
6546 Dodecyl isopropyl ether
[476-71-1] C19H19NO4 (325.37). mp 115~117C. Pharm: Convulsant (high
C15H32O (228.42). Source: DU HUO Angelica pubescens f. biserrata [Syn.
dose, warm-blooded animal such as dog); inhibits CNS with activity similar
to that of morphine (poikilotherm such as frog); inhibits heart (rbt and frog,
in vitro); reduces intestinal vessel tension (gpg, in vitro); mild anesthetic (low
dose, warm-blooded animal such as mus or dog); paralyses striated muscle;

paralyses uterus (high dose, rbt, in vitro); uterine stimulant (low dose, rbt, in
vitro); rises intestinal vessel tension (gpg, in vivo). Source: GE CAI KE SHI
ZI JIN Corydalis gortschakovii, JIAN JU ZI JIN Corydalis suaveolens [Syn.
6547 Doederleinic acid
Corydalis sheareri], NAN TIAN ZHU GEN Nandina domestica, NAN TIAN
7()-Oxa-bicyclo-[4,1,0]-hept-3-ene-3-carboxylic acid-5()-hydroxy C7H8O4
ZHU GENG Nandina domestica, NAN TIAN ZHU ZI Nandina domestica.
(156.14). White granular powder, mp 185~186C, []D10 = 13.8 (c = 0.2,
Ref: 4, 6, 658.
EtOH). Source: DA YE CAI Selaginella doederleinii. Ref: 484.
O
OH
HO
O
OH
O
O
213
6553 Dongnoside A
6556 Dongnoside D
3-O-[-L-Rhamnopyranosyl-(14)--D-glucopyranosyl-(12)-[-D-xylopyr
3-O-[-D-Glucopyranosyl-(13)-[-D-xylopyranosyl-(13)--D-xylopyran
anosyl-(13)--D-glucopyranosyl-(13)]--D-glucopyranosyl-(14)--D-g
osyl-(12)]--D-glucopyranosyl-(14)--D-galactopyranoside]
alactopyranoside] [149664-94-8] C62H102O31 (1343.49). mp 265~270C, []D
[125288-52-0] C55H90O26 (1167.31). Source: DONG YI HAO JIAN MA
= 51.5. Source: DONG YI HAO JIAN MA Agave east-one. Ref: 2503.
Agave east-one. Ref: 10.
O
O
O
H
HO
O
O
OH
OH
OH
OH
OO
OH
HO
OO
HO
HO
OH
HO
OO
OH
OH
OH
OH O O
OH
OH
OO
OH
OH
HO
OO
HO
OH
OH
O
OH
OO
OH
O
OH
OH
OH
OH
OH OH
6554 Dongnoside B
3-O-[-L-Rhamnopyranosyl-(14)--D-glucopyranosyl-(12)-[-D-glucopy
6557 Dongnoside E
ranosyl-(13)]--D-glucopyranosyl-(14)--D-galactopyranoside]
3-O-[-D-Glucopyranosyl-(13)-[-D-xylopyranosyl-(12)]--D-
[149664-93-7] C57H94O27 (1211.37). mp 275~277C, []D = 50.8. Source:
glucopyranosyl-(14)--D-galactopyranoside] [125265-72-7]
DONG YI HAO JIAN MA Agave east-one. Ref: 2503.
C 50 H 82 O 22 (1035.20). Source: DONG YI HAO JIAN MA Agave

O
east-one. Ref: 10.
O
H
HO
HO
OO
HO
OO
OH
H
O
OH
O
O
HO
OH OH
OH
OO
OH
OH
HO
OH
OH
OH
OO
OH
O
OH
HO
OO
HO
OH
OO
H
H
OH
OH OH
OH
OH OH
OH
6555 Dongnoside C
3-O-[-L-Rhamnopyranosyl-(14)--D-xylopyranosyl-(12)-[-D-glucopyr
6558 Dopa
anosyl-(13)]--D-glucopyranosyl-(14)--D-galactopyranoside]
L-3,4-Dihydroxyphenylalanine [59-92-7] C9H11NO4 (197.19). mp () 283C,
[125265-73-8] C56H92O26 (1181.34). Source: DONG YI HAO JIAN MA
() 271~272C (dec). Pharm: Precursor to biosynthesis of arterenol and
Agave east-one. Ref: 10.
dopamine; LD50 (mus, orl) = 3650mg/kg, (rat, orl) 4000mg/kg, (rbt, orl) =
609mg/kg. Source: CAN DOU Vicia faba, MAO DOU Mucuna
O
O
H
HO
O
OH
OH
OH
HO
OO
HO
OH
OH
OO
OO
OH
O
OO
OH
OH
H
H
cochinchinensis, CHANG CHUN YOU MA TENG Mucuna sempervirens,

BAI HUA YOU MA TENG Mucuna birdwoodiana, LI DOU Stizolobium
capitatum, CAN DOU YE Vicia faba, CAN DOU JIA KE Vicia faba, MA
CHI XIAN Portulaca oleracea, XU SUI ZI JING ZHONG BAI ZHI
Euphorbia lathyris, Lupinus sp. Ref: 6, 658.
H2N
OH
H O
OH
OH OH
OH
OH
214
6559 Dopamine
6564 Dorsmanin D
4-(2-Aminoethyl)pyrocatechol [51-61-6] C8H11NO2 (153.18). Pharm:
C26H28O7 (452.51). Source: MAN NI DUO TAN CAO Dorstenia mannii
Enhances myocardial contractility and increases blood flow; improves
peripheral circulation and markedly increases amount of urine;

neurotransmitter (in adrenal medulla and brain); Precursor to biosynthesis of
adrenalin. Source: AN LU LONG SHE LAN Lophophora williamsii, JIN
OH
QUE ER Cytisus scoparius [Syn. Spartium scoparium], MA CHI XIAN
HO
Portulaca oleracea, SHAN YAO Dioscorea batatas [Syn. Dioscorea
opposita], XIANG JIAO Musa paradisiaca var. sapientum [Syn. Musa
OH
sapientum]. Ref: 2, 6, 658.
OH
OH
6565 Dorsmanin E
OH

H2 N
OH
OH
6560 Doradexanthin
4-Ketolutein [29125-77-7] C40H54O3 (582.87). Source: LI YU PI Cyprinus
carpio, JIN YU Carassius auratus. Ref: 6, 660.

OH
HO
6566 Dorsmanin Fa
2''-Epidorsmanin Fa C25H28O7 (440.50). Beige plates (CH2Cl2), mp
6561 Dorsmanin A
168~170C. Source: MAN NI DUO TAN CAO Dorstenia mannii (aerial
parts). Ref: 5116.

HO
OH
OH
O
OH
6562 Dorsmanin B
OH

OH
6567 Dorsmanin Fb
2''-Epidorsmanin Fb C25H28O7 (440.50). Beige plates (CH2Cl2), mp
168~170C. Source: MAN NI DUO TAN CAO Dorstenia mannii (aerial
parts). Ref: 5116.
HO
OH
OH
6563 Dorsmanin C
OH
OH
6568 Dorsmanin Ga
2''-Epidorsmanin Ga C25H28O7 (440.50). Colorless powder, mp 148~150C.
OH
OH
Source: MAN NI DUO TAN CAO Dorstenia mannii (aerial parts). Ref: 5116.
OH
OH
OH
O
HO
OH
OH
215
6569 Dorsmanin Gb
6575 Dotriacontanic acid
2''-Epidorsmanin Gb C25H28O7 (440.50). Colorless powder, mp 148~150C.
[3625-52-3] C32H64O2 (480.87). Source: HUI BAO HAO Artemisia
Source: MAN NI DUO TAN CAO Dorstenia mannii (aerial parts). Ref: 5116.
roxbugiana. Ref: 503.
OH
O
OH
OH
HO
O
OH
6576 DraconinA
6570 Dorsmanin H
(23S,24S)-Spirosta-5,25(27)-diene-1,3,23,24-tetrol-O-{O-(2,3,4-tri-O-acety
l--L-rhamnopyranosyl)-(12)--L-arabinopyranosyl} C44H64O17 (864.99).
Amorphous solid, []D20 = 70 (c = 1.5, ethanol). Pharm: Cytotoxic (in vitro,

HL-60, IC50 = 9.7mol/L). Source: LONG XUE SHU Dracaena draco (stem
OH
HO
HO
cortex: yield = 0.00034%). Ref: 4696.
OH
OH
OH
6571 Dorsmanin I
OH
OH
O
O
6,7-(2,2-Dimethylpyrano)-8-prenyl-5,3',4'-trihydroxyflavanone C25H26O6
(422.48). Yellow plates (hexane-EtOAc), mp 172~174C, []D = 27 (c =
0.12, MeOH). Source: MAN NI DUO TAN CAO Dorstenia mannii (aerial
parts). Ref: 5116.
HO
HO
O
6577 DraconinB
(23S,24S)-Spirosta-5,25(27)-diene-1,3,23,24-tetrol 1-O-{O-(2,3-di-O-acetOH
O
yl--L-rhamnopyranosyl)-(12)--L-arabinopyranosyl} C42H62O16 (822.95).

Amorphous solid, []D20 = 100 (c = 2.6, ethanol). Pharm: Cytotoxic (in vitro,
OH
HL-60, IC50 = 39mol/L). Source: LONG XUE SHU Dracaena draco (stem
cortex: yield = 0.0017%). Ref: 4696.
OH
6572 Dorsmanin J
HO
C25H28O6 (424.50). Brown gum, []D = 17 (c = 0.17, MeOH). Source: MAN

NI DUO TAN CAO Dorstenia mannii (aerial parts). Ref: 5116.
HO
OH
O
O
H
OH
OH
O
O
OH
6,7-(2,2-Dimethyldihydropyrano)-8-prenyl-5,3',4'-trihydroxyflavanone
HO
O
OH
6578 DraconinC
OH
(23S,24S)-Spirosta-5,25(27)-diene-1,3,23,24-tetrol 1-O-{O-(2-O-acetyl-
6573 Doryanine
-L-rhamnopyranosyl)-(12)--L-arabinopyranosyl} C40H60O15 (780.92).
C11H9NO3 (203.20). Source: HOU KE GUI Cryptocarya chinensis (wood). Ref: 3092.
Amorphous solid, []D20 = 85 (c = 11.5, ethanol). Pharm: Cytotoxic inactive

(in vitro, HL-60, IC50 > 100mol/L). Source: LONG XUE SHU Dracaena
O
O
draco (stem cortex: yield = 0.0039%). Ref: 4696.
6574 Doryphornine
OH
C11H11NO3 (205.22). Source: BIAN FU GE GEN Menispermum dauricum,
HO
Doryphora sassafras (bark). Ref: 1521, 3792.
O
HO
O
OH
O
O
OH
HO
O
OH
OH
216
6579 Dracorubin
6584 Dracunculifoside E
[6219-63-2] C32H24O5 (488.55). Source: LONG XUE SHU Dracaena draco.
Ref: 658.
Source: XIAO LONG YE KUO BAO JU Baccharis dracunculifolia (aerial

parts). Ref: 4137.
O HO
HO
O
O
OH
HO
OH
OH
6585 Dracunculifoside F
6580 Dracunculifoside A
C28H41O11 (552.62). Amorphous powder, []D = 24.4 (c = 0.75, MeOH).
parts). Ref: 4137.
parts). Ref: 4137.
26
O
OH
HO
HO
OH OH
OH
HO
HO
OH
OH
OH
HO
OH
6586 Dracunculifoside G
OH
6581 Dracunculifoside B

parts). Ref: 4137.
O
parts). Ref: 4137.
HO
O
HO
O
HO
OH
OO
O
OH
HO
OH
OH OH
OO
OH
OH
HO
OH
6587 Dracunculifoside H
OH
6582 Dracunculifoside C
parts). Ref: 4137.
HO
HO
parts). Ref: 4137.

O
HO
O
O
OH
OO
O
OH
HO
OH OH
OO
OH
OH
OH
HO
OH
6588 Dracunculifoside I
OH
6583 Dracunculifoside D

parts). Ref: 4137.
O
parts). Ref: 4137.

O
O
HO
HO
OO
O
OH
OH
O
HO
HO
O
HO
OH
OH OH
OH
OH
OH
217
6589 Dracunculifoside J
6594 Dracunculifoside O
parts). Ref: 4137.
parts). Ref: 4184.
HO
OH
O
HO
OH
OH OH
OH
OH
OH
OO
OH
OH
HO
6590 Dracunculifoside K
OH

6595 Dracunculifoside P
parts). Ref: 4184.

O
O
HO

parts). Ref: 4184.
HO
OO
HO
OH
OH
OH
OH OH
OH
6591 Dracunculifoside L
OO
O
OH
OH
HO
OH

parts). Ref: 4184.
6596 Dracunculifoside Q
HO
OH
O O
HO O
O
O
parts). Ref: 4184.
O
OH
HO
OH
6592 Dracunculifoside M
OO
OH
OH OH
OH
OH
OH
22
C30H44O11 (580.68). Amorphous powder, []D = 35 (c = 0.35, MeOH).

parts). Ref: 4184.
HO
OH
O
HO
6597 Dracunculifoside R
OH
HO
OH

OH
HO
OH
parts). Ref: 4184.

O
6593 Dracunculifoside N
OH
22

O
H
O
HO
O
HO
parts). Ref: 4184.
OH
O
OO
HO
OH OH
OH
OH
OH
OO
HO
OH
OH
O
O
OH
218
6598 Drazepinone
6602 Drevogenin I
3,5,12a-Trimethyl-2,5,5a,12a-tetrahydro-1H-naphtho[2',3':4,5]furo[2,3-b]azep
cis-5-H,3,8,14,17-Tetrahydroxy-12-O-isovaleryl-20-O-isovaleryl-pr
in-2-one C19H19NO2 (293.37). []D25 = +7.1 (c = 0.2). Pharm: Herbicide.
egnane [125310-02-3] C31 H52O8 (552.76). Prismatic crystals, mp
Source: Drechslera siccans. Ref: 5268.
235~238C, []D25 = +34.5 (c = 0.15, MeOH). Source: KU SHENG Dregea

sinensis. Ref: 134.
O
N
O
OH
OH
H
6599 Dregeoside B
HO
OH
12,20-Di-O-isovaleryl-tomentogenin-3-O--L-oleandropyranosyl-(14)-O-L-oleandropyrano-side [133086-69-8] C 45H76O13 (825.10). White powder, mp

123~126C, []D20 = +38.5 (c = 0.25, methanol). Source: KU SHENG
6603 Drevogenin II
Dregea sinensis. Ref: 165.
cis-5-H,3,14,17-Trihydroxy-12-O-acetyl-20-O-benzoyl-pregnane
[125472-06-2] C30H42O7 (514.67). Prismatic crystals, mp 235~237C, []D25 =
+36.5 (c = 0.52, MeOH). Source: KU SHENG Dregea sinensis. Ref: 134.
OH
O
O
OH
OH O O
OO
O
O
OH
H
H
HO
OH
6600 Dresigenin B
20-O-(2-Methylbutyryl)tomentogenin C26H44O6 (452.64). Colorless acicular
crystals, mp 232~235C. Source: KU SHENG Dregea sinensis. Ref: 363.
6604 Driportlandin
(5',9',10')-7-O-(3-Methoxy-8'(12')-drimen-11'-yl)-scopoletin C26H34O5
(426.56). White amorphous solid, []D25 = +30.1 (c = 0.40, CHCl3). Pharm:
OH
OH
P-glucoprotein inhibitor (hmn MDR1 gene transfected mouse lymphoma cells,

reverses multidrug resistance (MDR), more active than positive control
Verapamil). Source: BO TE LAN DA JI Euphorbia portlandica (whole herb).
H
H
HO
Ref: 5019.
OH
6601 Dresioside I
O
Dihydrosarcostin 3-O--D-thevetopyranosyl-(14)--D-oleandropyranosyl-
(14)--D-cymaropyranoside C42H72O16 (833.03). White amorphous powder,

mp 151~154C. Source: KU SHENG Dregea sinensis. Ref: 363.
O
OH
OH
OH
H
OO
6605 Droserone
3,5-Dihydroxy-2-methyl-1,4-naphthoquinone [478-40-0] C11H8O4 (204.18).
mp 181C. Pharm: Antibacterial (hmn Mycobacterium tuberculosis H37RV, in
vitro, MIC = 25g/mL). Source: DUN ZHUANG MAO GAO CAI Drosera
peltata, HUI TE KE MAO GAO CAI Drosera whittakeri, MAO GAO CAI
Drosera peltata var. lunata. Ref: 6, 621, 658.
OO
O
OH
OH
OO
O
OH
OH
OH
OH
219
6606 Drummondin A
6611 Dryocrassin
[119171-76-5] C26H30O8 (470.52). Pharm: Antimicrobial; cytotoxic (P388, KB).
[12777-70-78] C43H48O16 (820.85). Yellow crystals (acetone), mp 209~214C;
Source: DE LA MENG DE JIN SI TAO Hypericum drummondii. Ref: 658.
yellowish powder crystals, mp 210~214C. Pharm: Schistosomacide

(Bilharzia japonica). Source: GUAN ZHONG Dryopteris crassirhizoma
(dried rhizome: content scope = 2.15%~6.95%, mean content = 4.37%[5508]).
OH
Ref: 658, 5508.
HO
OH HO
HO
HO
HO
6607 Drummondol
HO
OH
OH
O
OH
OH
OH
OH
O
O
C12H18O5 (242.27). Source: HONG HAI JIAO Capsicum annuum (stem and
6612 Dryocrassyl formate
root: yield = 0.00021%dw). Ref: 4779.
C31H52O2 (456.76). mp 67C, []D = +21.3 (c = 0.2, CHCl3). Source: BING

YE SUO LUO Yathea podophylla (fresh frond). Ref: 4401.
OH
H
O
OH
H
H
6608 Drupacine
[49686-57-9] C18H21NO5 (331.37). Source: HAI NAN CU FEI Cephalotaxus
6613 Drypearmoracein A
hainanensis [Syn. Cephalotaxus mannii], SAN JIAN SHAN Cephalotaxus
(E)-4,5,6,7-Tetrahydroxy-2-benzylhept-2-enoic acid C14H18O6 (282.30).
[4675]
fortunei (drupe: yield = 0.10%)
Colorless crystals, mp 250C, []D = +27 (c = 0.750, MeOH). Source: LA
, ZHONG GUO CU FEI ZHI YE
Cephalotaxus sinensis [Syn. Cephalotaxus harringtonia var. sinensis]. Ref: 2,
GEN HE GUO MU Drypetes armoracia. Ref: 3389.

OH
OH
660, 4675.
OH
O
O
OH
OH
6614 Drypearmoracein B
2,3-Dihydroxy-9,10-tetrahydroanthra-1,4-quinone C14H10O4 (242.23). White crystals,
HO
mp 160C. Source: LA GEN HE GUO MU Drypetes armoracia. Ref: 3389.
6609 Drymaritin
OH
25
C15H10N2O2 (250.26). Pale yellow amorphous solid, mp 181~183C, []D =

0 (c = 0.02, CHCl3). Pharm: Anti-HIV (H9 lymphocytes, EC50 = 0.699g/mL,
OH
TI = 20.6). Source: ER RUI HE LIAN DOU Drymaria diandra [Syn.

Drymaria cordata ssp. diandra] (whole herb: yield = 0.0011%dw). Ref: 4758.
6615 Drypemolundein A
C15H14O4 (258.28). White crystals, mp 148~150C, []D25 = 137.0 (c = 1.01,
CHCl3). Source: Drypetes molunduana (stem). Ref: 3989.
O
HO
6610 Dryobalanone
6616 Drypemolundein B
20,21-Dihydroxydammar-24-en-3-one [17939-10-5] C30H50O3 (458.73).
Source: BING PIAN Dryobalanops aromatica. Ref: 2.
CHCl3). Source: Drypetes molunduana (stem). Ref: 3989.
OH
HO
H
H
O
H
O
220
6617 Dubiin
OH
C22H30O6 (390.48). Pharm: Cytotoxic (L1210 in tissue culture, IC50 = 50~60g/mL).

Source: XI YE YI MU CAO Leonurus sibiricus (aerial parts). Ref: 4328.
O
H
H
HO
OH
O
O
6622 Dulcinone
H
6,8-Dihydroxy-2,7-dimethyl-4H-chromen-4-one C11H10O4 (206.20). Yellow
solid. Pharm: Antioxidant inactive (DPPH scavenger, 10mol/L, ScRt = 3%;

O
control BHT, 10mol/L, ScRt = 43%, IC50 = 19.00mol/L). Source: TIAN

SHAN ZHU ZI Garcinia dulcis (flower). Ref: 4422.
6618 Dubinidine
[22964-77-8] C15H17NO4 (275.31). mp 132~133C; hydrochloride: mp

195~196C; nitrate: mp 176~177C. Pharm: Anti-diuretic (2000mg/kg);
sedative (mus and rat, 100mg/kg orl); antipyretic (mus and rat, 100mg/kg orl).
HO
Source: DA YE YUN XIANG CAO Haplophyllum perforatum. Ref: 658.
OH
6623 Dulcinoside
5,7,4'-Trihydroxyflavone 6-C-[-rhamnopyranosyl-(l6)]--glucopyranoside
C27H30O14 (578.53). Yellow solid, mp 200~202C. Pharm: Antioxidant (DPPH
OH
scavenger, 10mol/L, ScRt = 22%, control BHT, 10mol/L, ScRt = 43%).

Source: TIAN SHAN ZHU ZI Garcinia dulcis (fruit). Ref: 5319.
HO
6619 Ducheside A
OH
3'-O-Methyl-ellagic acid-4-O--D-xylopyranoside C20H16O12 (448.34).

18
Yellowish powder, mp > 360C, []D = 11.3 (c = 0.035, methanol). Source:

SHE MEI Duchesnea indica. Ref: 368.
HO
OH OO
O
OH
OH
OH OH
HO
OH
O
O
OH
OH
OH
3,5,6,7,8,3',4'-Heptahydroxyflavan C15H14O8 (322.27). Light brown solid, mp

240~242C, []D29 = 72.0 (c = 0.012, CH3OH). Pharm: Antioxidant (DPPH
OH
scavenger, 10mol/L, ScRt = 87%, control BHT, 10mol/L, ScRt = 43%).
6620 Ducheside B
3'-O-Methyl-ellagic acid 4-O--L-arabinofuranoside C20H16O12 (448.34).
Source: TIAN SHAN ZHU ZI Garcinia dulcis (fruit). Ref: 5319.

OH
Yellowish powder, mp > 360C, []D19 = 126.5 (c = 0.027, methanol).

O
HO
OH
OH
Source: SHE MEI Duchesnea indica. Ref: 368.

O
OH
HO
HO
O
O
OH
6624 Dulcisflavan
O
O
HO
OH
OH
OH
OH
6625 Dulcisisoflavone
7-Hydroxy-2'',2''-dimethylchromano[5,6:6'',5'']-2''',2'''-dimethylchromano[3',4'
:5''',6''']isoflavone C25H26O5 (406.48). Yellow solid, mp 178~180C. Pharm:
6621 Dulcidiol
25
C27H38O4 (426.6). Gum, []D = 33.5 (c = 0.50, CHCl3). Pharm: Cytotoxic

(in vitro, SCL, ED50 = 45.3mol/L; SCL-6, ED50 = 46mol/L; SCL-37'6, ED50
= 42.6mol/L; SCL-9, ED50 = 41.6mol/L; Kato3, ED50 = 29mol/L;
NUGC-4, ED50 = 105.1mol/L; control Vinblastine Sulfate: SCL, ED50 =
5.9mol/L; SCL-6, ED50 = 6.1mol/L; SCL-37'6, ED50 = 5.3mol/L; SCL-9,
Antioxidant (DPPH scavenger, 10mol/L, ScRt = 15%, control BHT,

10mol/L, ScRt = 43%). Source: TIAN SHAN ZHU ZI Garcinia dulcis (fruit).
Ref: 5319.
O
HO
ED50 = 5.3mol/L; Kato3, ED50 = 6.1mol/L; NuGc-4, ED50 = 5.3mol/L).

Source: YE GAN CAO Scoparia dulcis (aerial parts: yield = 0.00231%dw).
Ref: 4703.
221
6626 Dulcisxanthone A
6630 Dulcisxanthone E
1,3-Dihydroxy-2,6-bis(3-methyl-2-butenyl)-2,2-dimethylchromeno(5''',6''':8,7)
1,3,6,7-Tetrahydroxy-2-(3,7-dimethyl-2,6-octadienyl)-5-(3-methyl-2-butenyl)
xanthone C28H30O5 (446.55). Yellow solid, mp 119~120C. Pharm:
xanthone C28H32O6 (464.56). Yellow solid. Pharm: Antioxidant inactive
Antioxidant (DPPH scavenger, 10mol/L, ScRt = 2%, control BHT, 10mol/L,
(DPPH scavenger, 10mol/L, ScRt = 15%; control BHT, 10mol/L, ScRt =
ScRt = 43%); antibacterial (Staphylococcus aureus ATCC 25923, MIC >
43%, IC50 = 19.00mol/L). Source: TIAN SHAN ZHU ZI Garcinia dulcis
128g/mL, control Vancomycin, MIC = 2g/mL; Staphylococcus aureus
(flower). Ref: 4422.
MRSA SK1, MIC > 128g/mL, Vancomycin, MIC = 2g/mL). Source: TIAN
SHAN ZHU ZI Garcinia dulcis (fruit). Ref: 5319.
HO
OH
OH
HO
OH
O
OH
6631 Dulcisxanthone F
1,6-Dihydroxy-2-(3-methyl-2-butenyl)-3-methoxy-2'',2''-dimethylchromeno-(5'
',6'':8,7)-xanthone C24H24O6 (408.46). Yellow solid. Pharm: Antioxidant
6627 Dulcisxanthone B
inactive (DPPH scavenger, 10mol/L, ScRt = 2%; control BHT, 10mol/L,
1,6,7-Trihydroxy-3-methoxy-2,8-bis(3-methyl-2-butenyl)xanthone C24H26O6
ScRt = 43%, IC50 = 19.00mol/L). Source: TIAN SHAN ZHU ZI Garcinia
(410.47). Yellow solid, mp 170~172C. Pharm: Antioxidant (DPPH scavenger,
dulcis (flower). Ref: 4422.
10mol/L, ScRt = 18%, control BHT, 10mol/L, ScRt = 43%). Source: TIAN
O
HO
O
OH
SHAN ZHU ZI Garcinia dulcis (fruit). Ref: 5319.
6632 Dulcitol
OH
Galactitol [608-66-2] C6H14O6 (182.17). mp 188.5C, bp 275~280C/1mmHg;
HO
mp 110~111C (anhydrate); mp 188~190C, bp 275~280C/1mmHg. Pharm:

HO
Sweetener (sugar substitute); laxative (veterinary). Source: A LA BO PO PO
NA Veronica persica (aerial parts), DOU SHU Pachyrrhizus erosus (seed),

6628 Dulcisxanthone C
DU ZHONG Eucommia ulmoides, FU FANG TENG Euonymus fortunei, GUI
1-Hydroxy-2,3,4,6-tetramethoxyxanthone C17H16O7 (322.31). Yellow solid,
JIAN YU Euonymus alatus, HAI HONG DOU Adenanthera pavonina, JI CAI
mp 125~128C. Pharm: Antioxidant inactive (DPPH scavenger, 10mol/L,
Capsella bursa-pastoris, LEI GONG TENG Tripterygium wilfordii, OU
ScRt = 2%; control BHT, 10mol/L, ScRt = 43%, IC50 = 19.00mol/L).
ZHOU HUA QIU Sorbus aucuparia, PI PA YE Eriobotrya japonica, SHI LIU
Source: TIAN SHAN ZHU ZI Garcinia dulcis (flower). Ref: 4422.
GEN Punica granatum, SHUI ZHI Gardenia jasminoides var. grandiflora,

SHUI ZHI YE Gardenia jasminoides var. grandiflora, SI MIAN MU
Euonymus bungeanus, SUO LA MU Salacia prinoides [Syn. Salacia
OH
O
O
O
O
chinensis], WU YE TENG Cassytha filiformis, YE ZI RANG Cocos nucifera,

YUAN CAN ZI Bombyx mori, ZI GUO WEI MAO Euonymus atropurpureus.
Ref: 2, 6, 587, 658, 1521, 4180, 4211.
OH
6629 Dulcisxanthone D
Tovophyllin B; 1,6-Dihydroxy-5-(3-methyl-2-butenyl)-2',2'-dimethylchromeno(5',6':2,3)-2''',2'''-dimethylchromeno(5''',6''':8,7)xanthone C28H28O6
(460.53). Orange solid, mp 218~220C. Pharm: Antioxidant inactive (DPPH
HO
scavenger, 10mol/L, ScRt = 16%; control BHT, 10mol/L, ScRt = 43%, IC50
= 19.00mol/L)
[4422]
; antitubercular (Mycobacterium tuberculosis,MIC =
25g/mL)[4358]. Source: DAO NIAN ZI Garcinia mangostana (fruit, fruit hull),

TIAN SHAN ZHU ZI Garcinia dulcis (flower). Ref: 3066, 4358, 4422.
OH
HO
6633 Dulxanthone E
5,9,10,12-Tetramethoxy-2,2-dimethyl-2H-pyrano[5,6-b]xanthen-6-one
C22H22O7 (398.42). Yellow cubes, mp 191~192C. Source: TIAN SHAN ZHU
OH
ZI Garcinia dulcis. Ref: 2399.
O
HO
OH
HO
O
O
O
O
222
6634 4,6-Dumortadien-3-one
6638 Dunniana acid B
[240417-19-0] C15H22O (218.34). Oil. Source: MAO DI QIAN Dumortiera
hirsuta. Ref: 2283.
HEI GUO HUANG PI Clausena dunniana (aerial parts: yield =

0.00075%dw). Ref: 4615.
H
O
6635 Dumosaol
3-(4-Hydroxy-3-methoxy-benzyl)-5-[2-(4-hydroxy-3-methoxy-phenyl)-3-hydr
OH
oxymethyl-7-methoxy-2,3-dihydro-benzofuran-5-yl]-4-hydroxymetyl-dihydro
-furan-2-one C30H32O10 (552.58). Amorphous powder, mp 70~72C, []D27 =
6639 Dunnisinin
+30.44 (c = 0.77, MeOH). Source: YUN NAN TIE SHAN Tsuga dumosa
C11H14 O5 (226.23). Colorless acicular crystals, mp 178~179C, []D25 =
+213.5 (c = 0.2, MeOH). Source: XIU QIU QIAN CAO Dunnia sinensis.
Ref: 764.
O
O
O
HO
OH
O
OH
HO
O
6640 Dunnisinoside
C 26 H 30 O 13 (550.52). Colorless prisms, mp 221~223C, [] D 25 = +28.4
OH
(c = 0.25, MeOH). Source: XIU QIU QIAN CAO Dunnia sinensis. Ref:
764.
6636 Dumoside
(20S)-3,16-dihydroxy pregn-5-ene-22-carboxylic acid
(22,16)-lactone-3-O--chacotrioside C40H62O16 (798.93). white amorphous,
25
mp 185.5~187C, []D = 13.38 (c = 0.36, MeOH). Source: GUAN MU

TIAN MEN DONG Asparagus dumosus, HAI JIN BI XIE Dioscorea
spongiosa (Rhizome: yield = 0.00013%)[4692]. Ref: 1908, 4692.
OH
HO
OH
O
H
H
HO
HO
OH
OH
OO
6641 Durupcoside C
OH
Hederagenin 3-O--D-glucopyranosyl(13)--D-glucopyranosyl(13)-
OH O O
OH O O
-L-arabinopyranoside C47H76O18 (929.12). Amorphous powder (MeOH),

[]D27 = +35.7 (c = 0.28, MeOH). Source: LIAO DONG CONG MU YE
OH OH
Aralia elata. Ref: 4471.
OH OH
6637 Dunniana acid A

HEI GUO HUANG PI Clausena dunniana (aerial parts: yield = 0.00035%dw).

Ref: 4615.
OH
O
HO
H
OH
OO
HO
O O
HO
O O
OH
OH
OH
OH
OH
OH
H
OH
O
OH
223
6642 Dutadrupine
6647 Dymacrin C
C30H46O3 (454.70). []D = +16 (c = 1, CHCl3). Pharm: Cytotoxic (KB cells,
IC50 = 5.0g/mL)[2407]. Source: DA HUA JIAN MU Dysoxylum macranthum.
Ref: 2407.

O
6643 -4,8,13-Duvatriene-1,3-diol
HO
(1S,2E,4R,6R,7E,11E)-2,7,11-Cembratriene-4,6-diol [57605-81-9] C20H34O2

(306.49). mp 127.0~127.5C (hexane), []D25 = +162 (chloroform). Pharm:
Antineoplastic (tumor caused by TPA, mus skin cancer caused by DMBA);
anti-inflammatory; prostaglandin biosynthesis inhibitor (IC50 = 0.39mmol/L);
plant growth inhibitor; aldose reductase inhibitor; pesticide (kills aphids, LC50
6648 Dymacrin D
C30H46O2 (438.70). []D = 36 (c = 1, CHCl3). Source: DA HUA JIAN MU
Dysoxylum macranthum. Ref: 2407.
= 15.7g/aphid). Source: YAN CAO Nicotiana tabacum. Ref: 900.

OH
OH
6644 -3,8,13-Duvatriene-1,5-diol
C20H34O2 (306.49). Crystals (Et2O), mp 150~152C, []D25 = +40. Source:
YAN CAO Nicotiana tabacum. Ref: 1521.
6649 Dymacrin E
C30H46O3 (454.70). []D = +4 (c = 1, CHCl3). Source: DA HUA JIAN MU
OH

OH
H
H
H
6645 Dymacrin A
C30H46O4 (470.70). []D = +31 (c = 1, CHCl3). Source: DA HUA JIAN MU

HO
H
OH
H
6650 Dymacrin F
O
HO

H
6646 Dymacrin B
C30H46O3 (454.70). []D = 17 (c = 1, CHCl3). Pharm: Cytotoxic (KB cells, IC50 =
5.6g/mL). Source: DA HUA JIAN MU Dysoxylum macranthum. Ref: 2407.

H
H
H
HO
O
HO
O
OH
OH
224
6651 Dymacrin G
6655 Dymacrin K
OH
H OH
OH
OH
O
O
6656 Dysobinin
6652 Dymacrin H
[62655-03-2] C30H38O6 (494.63). mp 185~187C, []D = +150 (chloroform).
Pharm: Anti-inflammatory; CNS depressant. Source: HONG GUO JIAN MU
IC50 = 8.3g/mL)
[2407]
. Source: DA HUA JIAN MU Dysoxylum macranthum.
Dysoxylum binectariferum. Ref: 661.
Ref: 2407.
O
O
H
OH
O
H
O
6653 Dymacrin I
H
O
H
OH
O
OH
6654 Dymacrin J
IC50 = 1.0g/mL)[2407]. Source: DA HUA JIAN MU Dysoxylum macranthum.
Ref: 2407.
H
O
H
O
O
OH
OH
O
O
OH
225
E
6657 Ebeienine
C27H43NO2 (413.65). mp 274.5~278.5C, []D = 2.9 (c = 0.5, MeOH).
Source: XI BEI MU Fritillaria imperialis (bulb), ZI HUA E BEI BEI MU
Fritillaria ebeiensis var. purpurea. Ref: 1521, 2201, 4217.
6661 Ebeinone
[125409-58-7] C27H41NO2 (411.63). mp 108~110C, []D = 54.9 (c = 0.47,
MeOH). Source: E BEI BEI MU Fritillaria ebeiensis, XI BEI MU Fritillaria
imperialis (bulb), ZI HUA E BEI BEI MU Fritillaria ebeiensis var. purpurea,
ZHE BEI MU Fritillaria verticillata var. thunbergii [Syn. Fritillaria
thunbergii]. Ref: 2201, 4217.
N
N
HO
HO
6662 Ebelin lactone
OH
[3649-76-1] C30H46O3 (454.70). mp 182~185C. Source: SUAN ZAO REN
6658 Ebeiensine
C27H41NO3 (427.63). mp 228~230C, []D = 38 (c = 0.16, CHCl3). Source:
Ziziphus jujuba var. spinosa. Ref: 2.
E BEI BEI MU Fritillaria ebeiensis, AN HUI BEI MU Fritillaria anhuiensis,

ZHE BEI MU Fritillaria verticillata var. thunbergii [Syn. Fritillaria
thunbergii]. Ref: 2201.
H
H
HO
O
H
H
HO
6663 Ebracteatoside A
H

Source: XIAO HUA LAO SHU LE Acanthus ebracteatus (aerial parts). Ref:
5211.
6659 Ebeietinone
OH
C27H43NO3 (429.65). mp 199~203C, []D = 53.3 (c = 0.24, CHCl3). Source:
OH
ZI HUA E BEI BEI MU Fritillaria ebeiensis var. purpurea. Ref: 2201.

OO
HO
OH
H
OH
HO
H
H
HO
OH OH
OH
O
6664 Ebracteatoside B
6660 Ebeinine
(3R)-1-Octen-3-ol-3-O--D-xylopyranosyl-(1'''6')-O-[-D-glucopyranosyl-
C27H45NO2 (415.67). mp 114~115C, []D = 45.0 (c = 0.70, MeOH). Source:
(1''2')]-O--D-glucopyranoside C25H44O15 (584.62). Amorphous powder,
E BEI BEI MU Fritillaria ebeiensis, ZI HUA E BEI BEI MU Fritillaria
[]D22 = 45.0 (c = 2.11, MeOH). Source: XIAO HUA LAO SHU LE
ebeiensis var. purpurea. Ref: 2201.
Acanthus ebracteatus (aerial parts). Ref: 5211.
N
H
H
H
HO
H
H
OO
O
OH
OH
OH
OH
OH
OO
HO
OH
OH
OH
OH
226
6665 Ebracteatoside C
6669 Ebracteolatanolide A
(6R)-7-Octene-1,6-diol 6-O--D-glucopyranosyl-(12)-O--D-glucopyra-
C20H28O4 (332.44). White acicular crystals, mp 210C. Source: YUE XIAN
noside C20H36O12 (468.50). Amorphous powder, []D22 = 19.8 (c = 2.62,
DA JI Euphorbia ebracteolata. Ref: 404.
MeOH). Source: XIAO HUA LAO SHU LE Acanthus ebracteatus (aerial

O
parts). Ref: 5211.

O
HO
H
HO
HO
OH
H
OH
OO
HO
6670 Ebracteolatanolide B
OH
C20H30O5 (350.46). White acicular crystals, mp 218C. Source: YUE XIAN
OH
OH
DA JI Euphorbia ebracteolata. Ref: 404.

O
6666 Ebracteatoside D
(6R)-7-Octene-1,6-diol 6-O--D-xylopyranosyl-(16)-O--D-glucopyra-
HO
noside C19H34O11 (438.48). Amorphous powder, []D22 = 57.7 (c = 0.35,
MeOH). Source: XIAO HUA LAO SHU LE Acanthus ebracteatus (aerial
OH
OH
parts). Ref: 5211.

H
HO
OO
6671 Ebracteolatinoside A
OH
OH
OH
C18H19NO11 (425.35). Sallow powder, mp 160C. Source: YUE XIAN DA JI
OH
OH
Euphorbia ebracteolata. Ref: 820.
OH
6667 Ebractelatinoside B
HO
3,3'-Diacetyl-4,4'-dimethoxy-2,2',6,6'-tetrahydroxy diphenyl methane-6'-O-D-glusopyranoside C25H30O13 (538.51). Yellowish amorphous powder, mp
OO
OH
OH
260~261C. Source: YUE XIAN DA JI Euphorbia ebracteolata. Ref: 678.
N
H
HO
OH
OH
OH HO
6672 Eburical
C31H50O2 (454.74). Source: A LI HONG Fomes officinalis. Ref: 6.
HO
OH
OO
OH
OH
OH
6668 Ebractelatinoside C
2,4-Dihydroxy-6-methoxy-3-methyl acetophenone 4-O--D-xylopyranosyl-
HO
(16)--D-glucopyranoside C21H30O13 (490.47). White amorphous powder,

mp 198C. Source: YUE XIAN DA JI Euphorbia ebracteolata. Ref: 678.
6673 Eburicodiol
C31H52O2 (456.76). Source: A LI HONG Fomes officinalis. Ref: 6.
O
OH
HO
OO
OO
OH
OH
OH
OH
OH
OH
HO
227
6674 Eburicoic acid
6679 Ecdysterone
C31H50O3 (470.74). mp 292~293C. Source: A LI HONG Fomes officinalis,
-Ecdysone C 27 H 44 O 7 (480.65). mp 237.5~239.5C. Pharm: Insect
FU LING Poria cocos. Ref: 2.
ecdysone; low toxin. Source: BAI MAO XIA KU CAO Ajuga
O
HO
decumbens, CANG BAI CHENG GOU FENG Diploclisia glaucescens,

CHUAN NIU XI Cyathula officinalis (root: content = 0.057%) [5508],
DUN YE TU NIU XI Achyranthes aspera var. indica (root: content =

0.018%) [5508], JI MAO SONG Podocarpus imbricatus, LOU LU
Rhaponticum uniflorum (dried root: mean content of 3 origins =
HO
0.3993% [5508] ) , LUO HAN SONG YE Podocarpus macrophyllus, LUO
YAN CAO Lemmaphyllum microphyllum, MA NIU XI Cyathula
6675 Eburicol
[6890-88-6] C31H52O (440.76). mp 158~159C. Source: A LI HONG Fomes
officinalis. Ref: 6.
capitata (root: content = 0.046%) [5508], NIU XI Achyranthes bidentata

(root: mean content of 13 origins = 0.06% [5508] ), SANG YE Morus alba,
SHUI LONG GU Polypodium niponicum, TU NIU XI Achyranthes
aspera, WA WEI Lepisorus thunbergianus, XIAO YE GUAN ZHONG
Matteuccia struthiopteris, YAN LING CAO Trillium tschonoskii, ZI QI
Osmunda japonica, ZI SHAN Taxus cuspidata. Ref: 2, 6, 194, 580, 582,

658, 660, 5501, 5508.
HO
OH
OH
6676 Eburicyl acetate
OH
C33H54O2 (482.80). mp 142~143C. Source: A LI HONG Fomes officinalis. Ref: 6.

HO
H
HO
OH
O
O
6680 20-Ecdysterone 2-O--D-glucopyranoside
C33H54O12 (642.79). White solid. Source: JIANG XI QING NIU DAN
6677 Eburnamonine
Tinospora craveniana (root). Ref: 4557.
[4880-88-0] C19H22N2O (294.40). Pharm: Vasodilator. Source: MAN CHANG

CHUN HUA Vinca minor. Ref: 658.
OH
OH
H N
OH
N
OO
HO
OH
OH
6678 Ecdysone
OH
HO
OH
-Ecdysone [3604-87-3] C27H44O6 (464.65). mp 242C. Pharm: Insect ecdysone
(badly inhibits growth of ovary in juvenile female fly). Source: BAI JIANG CAN
Bombyx mori (in 1954, the compound was first isolated from the animal by
6681 Ecdysterone-3-O--D-glucopyranoside
A.Butenandt, et al.)[5505], DA HUA JIAN QIU LUO Lychnis fulgens, DUO ZU JUE
C33H54O12 (642.79). White powder. Source: LOU LU Rhaponticum uniflorum.
Polypodium vulgare, LUO YAN CAO Lemmaphyllum microphyllum, OU ZHOU
Ref: 444.
JUE Pteridium aquilinum, SHUI LONG GU Polypodium niponicum, XIAO WU

MAO JUE Blechnum minus, XIAO YE GUAN ZHONG Matteuccia struthiopteris,
OH
OH
YUAN CAN E Bombyx mori, ZI QI Osmunda japonica. Ref: 6, 658, 5505.
OH
H
OH
HO
HO
H
HO
HO
OH
OH
OO
OH
OH
OH
OH
228
6682 Ecdysterone-22-O--D-glucopyranoside
6687 Echinatine N-oxide
C33H54O12 (642.79). White powder, mp 240~242C. Source: MAO JIAN QIU
Heliotridine viridiflorate N-oxide [20267-93-0] C15H25NO6 (315.37). Source:
LUO Lychnis coronaria. Ref: 2189.
YAO YONG DAO TI HU Cynoglossum officinale. Ref: 6.
HO
O
OH
HO
N
OH
HO
OH
6688 Echinenone
OH
H
HO
O
OH
OH OH
HO
[432-68-8] C40H54O (550.88). mp 192~193C. Source: HAI XIA Penaeus

orientalis. Ref: 6.
6683 Ecgonine
[481-37-8] C9H15NO3 (185.22). Pharm: Local anesthetic; supertoxic agent.
Source: GU KE Erythroxylum coca. Ref: 658.
O
OH
6689 Echinocystic acid
OH
Echinaystic acid C30H48O4 (472.71). Pharm: Cytotoxic inactive (HL-60, IC50 >
100mol/L, control Taxol, IC50 = (4.1E-41.1E-4)mol/L; MCF7, IC50 >

100mol/L, Taxol, IC50 = (15.32.6)mol/L; Bel7402, IC50 > 100mol/L, Taxol,
6684 Echimidine
IC50 = (0.30.1)mol/L; BGC823, IC50 > 100mol/L; HeLa, IC50 > 100mol/L,
[520-68-3] C20H31NO7 (397.47). Gum, []D = +6.6 (c = 0.3, CHCl3). Pharm:
Taxol, IC50 = (33.06.1)mol/L; KB, > 100mol/L, Taxol, IC50 > 100mol/L)[5015];
Mutagen (drosophila); toxin (exhibits hepatic toxicity). Source: CHE QIAN
apoptosis inducer inactive (HL-60 cells, 15mol/L, sub-G1 population =
YE LAN JI Echium plantagineum, DONG FANG XI MEN FEI CAO
(8.74.7)%, control sub-G1 population = (5.43.2)%, positive control Taxol,
Symphytum orientale, KUAI JING XI MEN FEI CAO Symphytum tuberosum,
sub-G1 population = (40.50.2)%)[5015]. Source: HUA NAN ZAO JIA Gleditsia
XI MEN FEI CAO Symphytum officinale (root: yield = 0.00038%dw)[3039],
fera (fruit: content = 0.0224%)[5508], ZAO JIA Gleditsia sinensis [Syn. Gleditsia
XIN FEI CAO Symphytum caucasicum. Ref: 658, 3039.
horrida] (fruit: mean content = 0.1168%[5508]). Ref: 5015, 5508.
O HO H
O
O
HO
OH
HO
6685 Echinatin
OH
OH
H
H
C16H14O4 (270.29). Source: JI GAN CAO Glycyrrhiza echinata (cultured

6690 Echinoisoflavanone
cells). Ref: 2431.
C22H24O7 (400.43). Pharm: Anti-inflammatory (NO production inhibitor)[4415].

OH
Source: Echinosophora koreensis (root). Ref: 1521, 4415.
HO
OH
Indicine [480-83-1] C15H25NO5 (299.37). mp 109~110C, 97~98C. Pharm:

Ganglionic blocker; enhances blood pressure increase caused by
adrenaline; toxin (low toxicity in mus with single iv dose, but continuous
injection causes liver denaturation). Source: DA WEI YAO Heliotropium
indicum, GOU SHI HUA Cynoglossum amabile, YAO YONG DAO TI HU
Cynoglossum officinale, XIN FEI CAO Symphytum caucasicum. Ref: 6, 658.
H
HO
6686 Echinatine
6691 Echinopsine
[83-54-5] C10H9NO (159.19). mp () 152C, () 135C. Pharm: Enhances
myocardial contractility and reduces scope of contraction (frog heart in vitro,
narcosis cat, in vivo); enhances tension of intestinal canal (cat, in vitro, but inhibits
the tension in rbt); antihypertensive (narcosis cat); similar action with strychnine;
vasodilator (rbt ear, in vitro). Source: XIN JIANG LAN CI TOU Echinops ritro,
WU ZHU YU Evodia rutaecarpa (fruit). Ref: 4, 6, 658, 660, 5031.
O
HO
O
OH
HO
OH
229
6692 Echinorine
6696 Echioidinin-5-O--D-glucopyranoside
[18095-64-2] C11H12NO+ (174.22). Source: XIN JIANG LAN CI TOU
C22H22O10 (446.41). Pale yellow solid (MeOH), mp 245~246C, []D28 = 70.1 (c
Echinops ritro. Ref: 6, 660.
= 0.2, C5H5N). Source: Andrographis neesiana (whole herb). Ref: 4357.
OH
6693 Echinosophoroside A1
nosyl kudzusapogenol A 22-O--L-arabinopyranoside C52H84O23 (1077.24). Source:
OH
OH
CHAO XIAN LANG YA CI Sophora koreensis (root). Ref: 4056.
C20H30O11 (446.46). White powder, mp 108~110C. Source: ZI HUA SONG
OH
GUO JU Echinacea purpurea. Ref: 2219.
H
OH
O
OO
OH
OH
OO
OH
OH
OH OH
OH
OH
6698 Echitamidine
OO
OH
OH
OH
OO
HO
OH
OH
OH
OH
6697 Echipuroside A
OH
HO
OO
HO
3-O--L-Rhamnopyranosyl(12)--L-arabinopyranosyl(12)--D-glucuronopyra
[38681-90-2] C20H24N2O3 (340.43). mp 244C (dec). Source: PEN JIA SHU

Winchia calophylla, XIANG PI MU Alstonia scholaris. Ref: 270, 1521.
OO
N
OH
OH OH
N
H
6694 Echinosophoroside B
H
O
3-O--L-Rhamnopyranosyl(12)--L-arabinopyranosyl-(12)--D-glucuronopyr
anosyl abrisapogenol C 22-O--L-arabinopyranoside C52H84O22 (1061.24). Source:
6699 Echitamine
CHAO XIAN LANG YA CI Sophora koreensis (root). Ref: 4056.
C22H29N2O4 (385.49). Hydrate: (C22H30N2O5), white crystals, mp 206C, []D20 =

29 (ethanol); chloride: long acicular crystals (water), mp 295C, []D15 = 58.
OH
Pharm: Ganglionic blocker (curariform action); diuretic; antihypertensive (high
OH
dose). Source: DAO ZHUANG JI GU CHANG SHAN Alstonia spatulata, GAN
H
OH
HO
OO
OH
OH
ZHUANG GUAN JI GU CHANG SHAN Alstonia spectabilis. Ref: 6, 661.

HO
OO
O
N
OO
OH
OH
OH
OH
HO
LAO JI GU CHANG SHAN Alstonia boonei, XIANG PI MU Alstonia scholaris,
N
H
HO
OO
6700 Eckol
[88798-74-7] C18H12O9 (372.29). Colorless flake crystals (acetonewater), mp
OH OH
6695 Echioidinin-2'-O--D-glucopyranoside
C22H22O10 (446.41). Yellow needles (MeOH), mp 276~278C (dec). Source:
Andrographis rothii (whole herb). Ref: 4311.
243~244C; Amorphous powder. Pharm: Antifibrinolysis (2-macroglobulin,

IC50 = 2.5g/mL, 2-fibrinolysin, IC50 = 1.6g/mL); antithrombotic;
tyrosinase inhibitor; antioxidant (DPPH scavenger, IC50 = 11.5mol/L, control
Ascorbic acid, IC50 = 10.3mol/L)[4376]. Source: HEI KUN BU Ecklonia
kurome, Brown alga Ecklonia stolonifera. Ref: 1019, 4376.
OH
OH
OH
OH
O
O
OH
OH
OH
HO
O
OH
O
HO
OH
230
6701 Eckstolonol
6704 Eclalbasaponin XIII
C18H10O9 (370.27). Off-white powder, []D20 = 0 (c = 0.008, MeOH). Pharm:
Echinocystic acid 3-O-(6'-O-methyl)--D-glucuronopyranoside C37H58O10
Antioxidant (DPPH scavenger, IC50 = 8.8mol/L, control Ascorbic acid, IC50
(662.87). White powdery crystals, mp 195~198C. Source: MO HAN LIAN
= 10.3mol/L). Source: Brown alga Ecklonia stolonifera. Ref: 4376.
Eclipta prostrata [Syn. Eclipta alba]. Ref: 2266.
OH
HO
O
HO
O
OO
OH
OH
OH
OH
OH
OH
OH
6702 Eclalbasaponin XI
6705 Ecliptasaponin A
3-O-[-D-Glucopyranosyl(12)--D-glucopyranosyl]-16-ethoxy-olean-12-e
3,16-Dihydroxyolean-12-ene-28-oic acid 3-O--D-glucopyranoside
ne-28-oic acid 28-O--D-glucopyranoside C50H82O19 (987.20). White crystals
C36H58O9 (634.86). White acicular crystals, mp 237~238C (methanol).
mp 231~233C. Source: MO HAN LIAN Eclipta prostrata [Syn. Eclipta
Source: MO HAN LIAN Eclipta prostrata [Syn. Eclipta alba]. Ref: 349.
alba]. Ref: 2124.
H
H
OH
OH
HO
HO
OO
OH
OH
OH
OO
OH
OH
O
HO
H
HO
OH
OH
OH
OO
6706 Ecliptasaponin B
OH
3-O-(-D-Glucopyranosyl-(14)--D-glucopyranosyl-16-hydroxyolean-12
OH
-ene-28-oic acid-28-O--D-glucopyranoside C48H78O19 (959.15). White
OH
acicular crystals, mp 220~221C (methanol). Source: MO HAN LIAN Eclipta

prostrata [Syn. Eclipta alba]. Ref: 349.
6703 Eclalbasaponin XII

3-O-[(2-O-Sulfuryl--D-glucopyranosyl)(12)--D-glucopyranosyl]-echinoc
ystic acid 28-O--D-glucopyranoside C48H78O22S (1039.21). White
amorphous powder, mp 130~131C. Pharm: Induces distortion of mycelial
(mold of rice blast). Source: MO HAN LIAN Eclipta prostrata [Syn. Eclipta
alba]. Ref: 2124.
HO
HO
O O
OH
OH
O
OH
H
HO
OO
OH
OH
HO
OO
H
HO
OO
OH
OH
OH
6707 Ecliptasaponin D
C36H58O9 (634.86). White powder, mp 240~243C. Source: MO HAN LIAN
Eclipta prostrata [Syn. Eclipta alba]. Ref: 392.
OH
O
S
HO
OH
OH
OO
H
OH
OH
OH
OH
OH
O
O
OH
OH
OH
OO
HO
OH
OH
OH
OH
231
6708 Edulinine
6712 Effusanin C
[27495-36-9] C16H21NO4 (291.35). mp 140~142C. Pharm: Analgesic; CNS
C22H30O7 (406.48). mp 243~245C, []D21 = 54.0 (c = 0.46, C5H5N). Source:
depressant; anti-epilepsy (rat, brain hippocampus section CA1, eximine-induced
KAI ZHAN XIANG CHA CAI Isodon effusa. Ref: 4067.
epilepsy); cytotoxic (P388 cell line, ED50 = 27.1g/mL, control Mithramycin, ED50 =
0.06g/mL; HT29, ED50 = 43.6g/mL, Mithramycin, ED50 = 0.07g/mL; A549,
OH
ED50= 25.5g/mL, Mithramycin, ED50 = 0.08g/mL)[5405]. Source: CHOU CAO

O
Ruta graveolens, SI ROU TUO GUO YE MI ZHU YU Melicope semecarpifolia.

O
Ref: 6, 1625, 1626, 5405.
H
O
O
OH
OH
H
OH
6713 Effusanin D
C24H32O8 (448.52). mp 188~190C, []D21 = 28.2 (c = 0.41, CHCl3). Source:
OH

6709 Edultin
Cnidimine [15591-75-0] C21H22O7 (386.41). Pharm: Reversing MDR of
KBV200 cells (obviously)[2787]. Source: SHE CHUANG ZI Cnidium monnieri
(ripe seed: mean content of 6 origins = 0.652%[5508]). Ref: 6, 2787, 5508.

O
O
H
O
O
OH
OH
H
H
O
O
6714 Effusanin E
C20H28O6 (364.44). Colorless prisms (EtOH), mp 231~235C, mp 240~242C,
[]D23 = 28.2 (c = 0.06, EtOH); []D = 81.3 (c = 0.28, C5H5N); mp
6710 Effusanin A
250~252C, []D21 = 81.3 (c = 0.20, C5H5N). Pharm: Cytotoxic
C20H28O5 (348.44). Colorless needles (EtOH), mp 252~256C, []D23 = 53.8
(DNA-damaging activity, mutant yeast strain RAD 52Y, IC12 = 95g/mL,
(c = 0.4, EtOH); mp 262~265C, []D = 76.0 (c = 0.05, EtOH); mp
control Streptonigrin, IC12 = 0.4g/mL; wild type yeast strain RAD+, IC12 >
266~268C, []D20 = 79.7 (c = 0.35, C5H5N). Pharm: Cytotoxic
100g/mL, Streptonigrin, IC12 = 1.0g/mL) [5348]. Source: KAI ZHAN
(DNA-damaging activity, mutant yeast strain RAD 52Y, IC12 = 20g/mL,
XIANG CHA CAI Isodon effusa, SHAN DI XIANG CHA CAI Isodon
control Streptonigrin, IC12 = 0.4g/mL; wild type yeast strain RAD+, IC12 =
oresbia (aerial parts), ZHOU YE XIANG CHA CAI Isodon rugosus [Syn.
50g/mL, Streptonigrin, IC12 = 1.0g/mL)
[5348]
. Source: KAI ZHAN XIANG
Rabdosia rugosa]. Ref: 3808, 4067, 5348.
CHA CAI Isodon effusa, ZHOU YE XIANG CHA CAI Isodon rugosus [Syn.
HO
Rabdosia rugosa]. Ref: 4067, 5348.

OH
H
O
OH
H
O
O
OH
O
OH
OH
6715 Effusin
OH
6711 Effusanin B
C22H28O6 (388.46). mp 211~213C, []D35 = +21 (c = 1.12, C5H5N). Source:
C22H30O6 (390.48). Colorless prisms (acetonehexane), mp 254~256C, [] D23
= 60 (c = 0.1, MeOH); mp 258~260C, []D = 66.7 (c = 0.027, EtOH); mp

264~267C, []D20 = 61 (CHCl3). Pharm: Cytotoxic (DNA-damaging
activity, mutant yeast strain RAD 52Y, IC12 = 12g/mL, control
Streptonigrin, IC12 = 0.4g/mL; wild type yeast strain RAD+, IC12 =
35g/mL, Streptonigrin, IC12 = 1.0g/mL)[5348]. Source: KAI ZHAN XIANG
CHA CAI Isodon effusa, ZHOU YE XIANG CHA CAI Isodon rugosus [Syn.
6716 Egomaketone
Rabdosia rugosa]. Ref: 4067, 5348.
[59204-74-9] C10H12O2 (164.21). bp 124~126C/20mmHg. Source: BAI SU

ZI Perilla frutescens, ZI SU GENG Perilla frutescens var. arguta. Ref: 6, 660.
O
O
H
O
H
OH
O
OH
232
6717 Egonol glucoside
6722 Eicosanol
C26H30O9 (486.52). Viscous yellowish oil, []D25 = 15.2 (c = 0.6, MeOH).
1-Eicosanol [629-96-9] C20H42O (298.56). mp 65.5C, bp 220C/3mmHg.
Source: RI BEN AN XI XIANG JING PI Styrax japonica. Ref: 2546.
Source: KU CAO Vallisneria spiralis, ZI CAO Lithospermum erythrorhizon.

Ref: 6, 660.
OH
HO
O
OH
OH
O
O
OH
6723 (4E,6E,2S,3R)-2-N-Eicosanoyl-4,6-tetradecasphingadienine
6718 Ehrenoside
23
[106323-63-1] C34H44O19 (756.72). Amorphous powder, []D = 58 (c =
CHCl3). Pharm: Neurotrophic (neurite outgrowth promoter, measuring neurite
0.16, MeOH). Pharm: Antioxidant (DPPH scavenger, 0.5mmol/L, InRt = 50%,
length of PC12 cell, 10mol/L, activity greater than that of 50ng/mL NGF).
control BHA, 0.5mmol/L, InRt = 30%)[4191]. Source: SHU CHI PO PO NA
Source: BAI JIANG CAN Bombyx mori. Ref: 4684.
Veronica pectinata var. glandulosa (aerial parts). Ref: 4191.

OH
OH
OH
OO
HO
O
O
OH
O OH O O
OH
OH
HN
OH
HO
OH
OH
OH
6724 (4E,2S,3R)-2-N-Eicosanoyl-4-tetradecasphingenine
6719 Eicosandioic acid
[2424-92-2] C20H38O4 (342.52). mp 122~123C. Source: LIN BEI ZI
CHCl3). Source: BAI JIANG CAN Bombyx mori. Ref: 4684.
Toxicodendron succedaneum [Syn. Rhus succedanea], QI ZI Rhus verniciflua

[Syn. Toxicadendron verniciflum]. Ref: 6.
O
OH
OH
O
HN
OH
HO
6720 Eicosane
n-Eicosane [112-95-8] C20H42 (282.56). Source: DONG CHONG XIA CAO
Cordyceps sinensis, REN SHEN Panax ginseng [Syn. Panax schinseng],
ROU CONG RONG Cistanche deserticola, SAN QI Panax pseudo-ginseng
6725 11-Eicosenoic acid

[5561-99-9] C20H38O2 (310.52). Source: QIANG HUO Notopterygium
incisum. Ref: 2.
O
var. notoginseng [Syn. Panax notoginseng]. Ref: 2.
OH
6726 Eicosyl caffeate

C29H48O4 (460.70). Source: ZI CAO Lithospermum erythrorhizon. Ref: 2193.
6721 Eicosanetetraenoic acid
HO
C20H32O2 (304.48). mp 49.5C. Source: NIU GAN Bos taurus domesticus;

Bubalus bubalis, ZI CAI Porphyra tenera. Ref: 6.
HO
O
O
O
OH
233
6727 3-O-14,15-Eicosylenoyl-1-cyano-2-methyl-1,2-propene
6732 Elanine
C25H43NO2 (389.63). Colorless wax. Source: LUAN SHU Koelreuteria
C41H56N2O11 (752.91). Source: HEI SHUI CUI QUE HUA BIAN ZHONG
Delphinium potaninii var. jiufengshanense (root). Ref: 4227.

H
OH
OH
6728
3-O-14,15-Eicosylenoyl-4-O-stearoyl-1-cyano-2-oxymethyl-1,2-propene
C43H77NO4 (672.10). Colorless wax. Source: LUAN SHU Koelreuteria
6733 Elaterin
Cucurbitacin [18444-66-1] C32H44O8 (556.70). mp 234C. Source: GUA DI
Cucumis melo, SI GUA ZI Luffa cylindrica. Ref: 6.
O
O
O
HO
O
HO
6729 Eicosyl ferulate

C30H50O4 (474.73). Source: YA MA ZI Linum usitatissimum. Ref: 6.
O
OH
O
O
6734 Elatine
[26000-16-8] C38H50N2O10 (694.83). mp 233~235C. Pharm: Ganglionic

blocker; muscle relaxant (competitive); toxin. Source: FEI YAN CAO
Consolida ajacis [Syn. Delphinium ajacis], GAO FEI YAN CAO Delphinium
OH
elatum. Ref: 6, 658.

H
6730 Elaeocarpusin
C47H34O32 (1110.78). Source: AN MO LE Phyllanthus emblica (fruit juice).

N
Ref: 3094.
O
H
OH
OH HO
HO
O
OH
HO
O
OH
O
O
O
O
OH
O
O
OH
6735 Elatol
O
O
O
OH
OO
HO
O
O
C15H22BrClO (333.70). Oil, []D24 = +75.3 (c = 0.318, MeOH). Pharm:
OH
Antibacterial (Clostridium cellobioparum, MIC = 5g/disc; Proteus mirabilis,

MIC = 5g/disc; Flavobacterium helmiphilum, MIC = 10g/disc;
OH
Chromobacterium violaceum, Clostridium fallax, Clostridium novyi,

Clostridium sordellii, Escherichia coli, Enterobacter aerogenes, Shigella
OH
flexneri, Vibrio cholerae, Vibrio parahaemolyticus, Vibrio vulnificus, MIC =
OH
15~30g/disc)[5183]. Source: GAO AO DING ZAO Laurencia elata (the

compound was isolated from the plant by J.J.Sions, et al. in 1974)[5505], LUE
6731 Elaidic acid

trans-9-Octadecenoic acid [112-79-8] C18H34O2 (282.47). mp 44.5C. Source:
DA AO DING ZAO Laurencia majuscula. Ref: 5183, 5505.
DENG LONG CAO Physalis peruviana, HU TAO YE Juglans regia. Ref: 6.

HO
H
H
Br
OH
Cl
234
6736 Eleagnine
HONG CHAI HU Bupleurum scorzonerifolium, HUANG HUA HAO Artemisia
Tetrahydroharman [525-40-6] C12H14N2 (186.26). mp 180.0~181.5C;
annua, HUO XIANG Agastache rugosus, JING JIE Schizonepeta tenuifolia [Syn.
178~180C. Source: LU ZHU GEN Arundo donax, SHA ZAO SHU PI
Nepeta tenuifolia], MU XIANG Saussurea lappa [Syn. Aucklandia lappa], REN
Elaeagnus angustifolia. Ref: 6.
SHEN Panax ginseng [Syn. Panax schinseng], SAN QI Panax pseudo-ginseng var.
notoginseng [Syn. Panax notoginseng], SHANG ZUO JIAN YE GUANG E TAI
Porella acutifolia ssp. Tosana, SHENG JIANG Zingiber officinale, WU WEI ZI
NH
Schisandra chinensis, YIN CHEN HAO Artemisia capillaris. Ref: 2, 5, 660, 3932,
N
H
5501.
6737 Eleganin
[57498-84-7] C22H26O9 (434.45). mp 142~143C, []D22 = 108. Pharm:
Antineoplastic; cytotoxic. Source: HUA LI SHE BIAN JU Liatris elegans,

CU CAO SHE BIAN JUJU Liatris scabra. Ref: 658.
6742 -Elemene
[30824-67-0] C15H24 (204.36). Source: HUANG HUA HAO Artemisia annua,
REN SHEN Panax ginseng [Syn. Panax schinseng], SAN QI Panax
O
O
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng], SHENG JIANG
Zingiber officinale. Ref: 2, 660.
O
O
HO
O
6738 Elegansamine
6743 -Elemene
[120090-58-6] C29H36N2O6 (508.62). mp 172~173C. Source: GOU WEN
[20307-84-0] C15H24 (204.36). bp 107C/10mmHg. Source: REN SHEN
Gelsemium elegans. Ref: 13.
Panax ginseng [Syn. Panax schinseng]. Ref: 2.
O
O
N
N
OH
6744 cis--Elemene diastereomer

C15H24 (204.36). Colorless oil. Source: BO BAN HE YE TAI Scapania
6739 Elema-1,3-dien-7-ol
undulata (essential oil). Ref: 3752.
(+)-(1R,3R,4R)-4-Ethenyl-4-methyl-3-(1-methylethenyl)-1-(1-methylethyl)-cy
clohexanol C15H26O (222.37). Colorless oil. Source: YING ZHI YE TAI
Lepidozia vitrea (essential oil). Ref: 5209.

OH
6745 Elemicin
[487-11-6] C12H16O3 (208.26). bp 144~147C/10mmHg. Pharm: Anesthetic (mus,
rbt, cat, and dog, iv); platelet aggregation inhibitor (rbt). Source: BAN KE HU
JIAO Piper banksii, CHANG XIANG MAO Cymbopogon procerus, DU HENG

Asarum forbesii, GAO DA HU JIAO Macropiper excelsum, HAI FENG TENG
6740 ()-cis--Elemene
Piper kadsura [Syn. Piper futokadsura], HUI HUI SU GENG Perilla frutescens
C15H24 (204.36). Colorless oil. Source: BO BAN HE YE TAI Scapania
var. crispa, JIAN ZI SU Perilla frutescens var. acuta [Syn. Perilla frutescens var.
undulata (essential oil). Ref: 3752.
purpurascens], JIAN ZI SU YE Perilla frutescens var. acuta [Syn. Perilla

frutescens var. purpurascens], LIAO XI XIN Asarum heterotropoides var.
mandshuricum (whole herb: content scope = 0.011%~0.069%)[5501], NAN HE SHI
Daucus carota, SHAN ZHU YU Cornus officinalis [Syn. Macrocarpium officinale],

SHUANG YE XI XIN Asarum caulescens, SI JING JIE BA DOU Croton
6741 -Elemene
C15H24 (204.36). bp 117~124C/15.5mmHg. Pharm: Cytotoxic (leukemia cell, IC50
= 33.5g/mL); antineoplastic (animal model, EAC ascites tumour, ARS ascites
nepetaefolius, XI XIN Asarum sieboldii, YE XIANG MAO Cymbopogon goeringii,

YUN NAN ZHANG Cinnamomum glanduliferum, ZHAO WA GAN LAN
Canarium commune. Ref: 2, 658, 660, 2537, 5501.
tumour, YAS ascites tumour, S180 ascites tumour). Source: BING PIAN
Dryobalanops aromatica, CANG ZHU Atractylodes lancea, DONG LING CAO
Rabdosia rubescens, DU HUO Angelica pubescens f. biserrata [Syn. Angelica
pubescens], GUANG HUO XIANG Pogostemon cablin [Syn. Mentha cablin],
O
O
O
235
6746 Elemol
6751 Elephantopin
[32142-08-8] C15H26O (222.37). mp 52.5~53.5C. Source: BEI CANG ZHU
[13017-11-3] C19H20O7 (360.37). mp 262~264C, []D25 = 398. Pharm:
Atractylodes chinensis, CANG ZHU Atractylodes lancea, HOU PO Magnolia
Antineoplastic (rat, W256, 50~100mg/kg; mus, P388); cytotoxic (KB, ED50 =
officinalis, MU XIANG Saussurea lappa [Syn. Aucklandia lappa], SHENG
0.28~2.00g/mL). Source: GAO DI DAN CAO Elephantopus elatus. Ref: 661.
JIANG Zingiber officinale. Ref: 2, 660.
O
O
O
O
O
O
OH
6752 Eleutherin
6747 Elenolide
[478-36-4] C16H16O4 (272.30). Orange crystals, mp 173~175C, []D34 =
[24582-91-0] C11H12O5 (224.22). Acicular crystals (hot ethanol), mp 155.2C,
345.6 (chloroform). Pharm: Antibacterial (Staphylococcus aureus,
[]D20 = +360 (chloroform). Pharm: Antihypertensive. Source: YOU GAN

LAN Olea europaea. Ref: 661.
Mycobacterium smegmatis); increases coronary flow. Source: XIAO HONG

SUAN Eleutherine americana. Ref: 661.
O
O
O
O
O
6753 Eleutherol
[480-00-2] C14H12O4 (244.25). Pharm: Increases coronary flow. Source:
6748 -Eleostearic acid
XIAO HONG SUAN Eleutherine americana. Ref: 658.
[506-23-0] C18H30O2 (278.44). Source: TONG YOU Aleurites cordata [Syn.
OH
Aleurites fordii]. Ref: 658.
O
O
O
OH
6754 Eleutheroside B1
7-Hydroxy-6,8-dimethoxycoumarin glucoside [16845-16-2] C17H20O10
(384.34). mp 218C. Pharm: Increases the weight and RNA content of both prostate
6749 -Eleostearin
and testis (male mus, orl, 5~7mg/(kgd)). Source: WU JIA PI Acanthopanax
C57H92O6 (873.37). Source: TONG YOU Aleurites cordata [Syn. Aleurites
gracilistylus. Ref: 6, 658.
fordii]. Ref: 6.
O
HO
O OH
OH
O
OH
6755 Eleutheroside I
Mubenin B; Raddeanin B [35790-94-4] C41H66O11 (734.98). mp 234~235C

6750 Elephantin
(dec), mp 237~240C, []D24 = +12 (c = 0.5, MeOH). Pharm: Hemolytic.
[21899-50-3] C20H22O7 (374.39). mp 242~244C, []D27 = 380. Pharm:
Source: CI WU JIA YE Acanthopanax senticosus [Syn. Eleutherococcus
Antineoplastic (rat, W256, 50~100mg/kg; mus, P388); cytotoxic (KB, ED50 =
senticosus], DUO BEI YIN LIAN HUA Anemone raddeana (root: yield =
0.28~2.00g/mL); plant growth regulator. Source: GAO DI DAN CAO
0.0043%), NA TENG GUO Stauntonia hexaphylla. Ref: 6, 660, 900, 1312.
Elephantopus elatus. Ref: 661.

O
O
O
O
OH
O O
OH
O
O
OH
OH OH
OH
236
6756 Eleutheroside K
6758 Ellagic acid-4-O--D-xylopyranoside
-Hederin; Oleanolic acid 3-O--L-rhamnopyranosyl (12)--L-arabinopyra-
C19H14O12 (434.12). Pink. Pharm: Antibacterial (Erwinia carotovora, IZD =
noside [35790-95-5] C41H66O11 (734.98). White needles, mp 221~223C;
12mm/100g, control Quercetin sulfate, IZD = 21mm/10g; Staphylococcus
White amorphous powder, []D23 = +10.9 (c = 0.55, MeOH). Pharm:
aureus, IZD = 0mm/100g, Quercetin sulfate, IZD = 14mm/10g;
Cytotoxic (hmn gastric carcinoma cells BGC823, hmn myelocytic leukemia
Corynebacterium accolens, IZD = 0mm/100g, Quercetin sulfate, IZD =
cell K562, obvious effect)[4812]; hemolytic. Source: CI WU JIA Acanthopanax
28mm/10g); antifungal (Candida albicans, IZD = 0mm/100g, control
senticosus [Syn. Eleutherococcus senticosus] (seed), CI WU JIA YE
Nystatin, IZD = 11mm/20g); xanthine oxidase inhibitor (IC50 = 2.1g/mL,
Acanthopanax senticosus [Syn. Eleutherococcus senticosus], DUO BEI YIN
IC50 = 4.7mol/L; control Quercetin, IC50 = 3.4g/mL, IC50 = 10 mol/L).
LIAN HUA Anemone raddeana, HUANG HUA BAI JIANG Patrinia
Source: DA YE KU NUO NI Cunonia macrophylla (leaf). Ref: 5250.
scabiosaefolia, YANG CHANG CHUN TENG Hedera helix. Ref: 6, 658, 660,
HO
2240, 4812, 4904.
O
HO
O
O
O
OH
H
OH
OO
OH
O
OO
OH
OH
OH
OH
OH
OO
6759 Ellipticine
OH OH
[519-23-3] C17H14N2 (246.31). Yellowish acicular crystals (ethyl acetate), mp
6757 Ellagic acid
311~315C (dec). Pharm: cytotoxic (in vitro, Lu1, IC50 = 0.02g/mL
2,3,7,8-Tetrahydroxy[1]benzopyrano[5,4,3-cde][1]benzopyran-5,7-dione
(0.08mol/L), LNCaP, IC50 = 0.8g/mL (3.25mol/L), Col2, IC50 = 0.3g/mL
[476-66-4] C14H6O8 (302.20). Yellow, mp > 360C. Pharm: Hemostatic;
(1.22mol/L), HUVEC, IC50 = 0.09g/mL (0.37mol/L), KB, IC50 =
uterine stimulant; antimutagenic (caused by aromatic hydrocarbons);
0.04g/mL (0.16mol/L), HOG.R5, IC50 = 0.02g/mL (0.08mol/L))[3009];
antiplasmodial[5361]; ACE inhibitor (IC50 = 400mol/L, control Lisinopril,
cytotoxic (in vitro, Lu1, ED50 = 0.02g/mL; Col2, ED50 = 0.3g/mL; KB,
IC50 = 1 nmol/L); NEP inhibitor (IC50 > 500mol/L, control Phosphoramidon,
ED50 = 0.04g/mL; LNCaP, ED50 = 0.8g/mL; KB in absence of 1g/mL
IC50 = 9 nmol/L); APN inhibitor inactive; antibacterial (Erwinia carotovora,
vinblastine, ED50 = 0.3g/mL; KB in presence of 1g/mL vinblastine, ED50 =
IZD = 15mm/100g, control Quercetin sulfate, IZD = 21mm/10g;
0.2g/mL; BC-1, ED50 = 0.5g/mL)[3479]; cytotoxic (BC, IC50 = 0.3g/mL;
Staphylococcus aureus, IZD = 0mm/100g, Quercetin sulfate, IZD =
KB, IC50 = 0.3g/mL)[3858]; cytotoxic (Vero cells, IC50 = (0.40.1)g/mL,
14mm/10g; Corynebacterium accolens, IZD = 12mm/100g, Quercetin
colorimetric method (P. Skehan, et al., J Natl Cancer Inst 1990, 82,
sulfate, IZD = 28mm/10g)
[5250]
; antifungal (Candida albicans, IZD =
10mm/100g, control Nystatin, IZD = 11mm/20g)[5250]; xanthine oxidase
1107-1112))[4078]; cytotoxic (A549, IC50 = 0.8mol/L; Col2, IC50 = 1.6mol/L;

SNU638, IC50 = 1.6mol/L; HT1080, IC50 = 1.2mol/L)[4081]; cytotoxic (hmn
inhibitor (IC50 = 2.8g/mL, IC50 = 9.3mol/L; control Quercetin, IC50 =
small cell lung cancer NCI-H187 cell line, IC50 = (0.350.15)g/mL)[5061];
3.4g/mL, IC50 = 10mol/L)[5250]. Source: DA FEI YANG CAO Euphorbia
cytotoxic (NCI-H187, IC50 = 0.2~0.3g/mL; KB, IC50 = 0.2~0.3g/mL;
hirta, DA YE KU NUO NI Cunonia macrophylla (leaf), HE ZI Terminalia

chebula, HONG KUAI ZI Chamaenerion angustifolium [Syn. Epilobium
angustifolium], HUA XIANG SHU YE Platycarya strobilacea, MANG GUO
Mangifera indica, NING MENG AN YE Eucalyptus citriodora, QIAN QU
BC-1, IC50 = 0.2~0.3g/mL; Vero cell, IC50 = 0.2~0.3g/mL)[5062];

cytotoxic (KB, ED50 = 0.10g/mL)[5075]; cytotoxic (KB, EC50 = 0.3g/mL; BC,
EC50 = 0.3g/mL)[5092]; cytotoxic (Col2, IC50 = 0.3g/mL; P388, IC50 =
0.1g/mL)[5400]; cytotoxic (KB cells, IC50 = (0.30.1)g/mL; BC, IC50 =
CAI Lythrum salicaria, SHU ZHANG LAO GUAN CAO Geranium
(0.30.1)g/mL)[5435]; cytotoxic (P388, ED50 = 0.61g/mL; KB, ED50 =
sibiricum, XIAN HE CAO Agrimonia pilosa var. japonica, Tristaniopsis
0.54g/mL; Col2, ED50 = 0.60g/mL; Lu1, ED50 = 0.61g/mL; BCA-1, ED50 =
calobuxus (bark), YUN NAN FENG CHE ZI Combretum yunnanensis

(branch)[4693], occurs in many plants (widely distributed in higher plants:
0.52g/mL)[5478]; antineoplastic (L1210, EAC cells, liver cancer in rat, P388,

S180)[661]; antitrypanosomal (Trypanosoma cruzi)[661]; hemolytic (animal
found by Bate-Smith in 75 genera of dicotyledons and in only one
model)[661]. Source: GU CHENG MEI GUI SHU Ochrosia elliptica, WEI BAI
monocotyledonous sp. Hypoxis filiformis in family Amaryllidaceae). Ref: 6,
BAI JIAN MU Aspidosperma subincanum. Ref: 661, 3009, 3479, 3858, 4078,
71, 658, 1521, 4693, 5034, 5250, 5361.
4081, 5061, 5062, 5075, 5092, 5400, 5435, 5478, 5507.
O
OH
OH
HO
HO
O
O
N
H
237
6760 Elliptifoline
6765 Elymoclavine
C36H40N2O8 (628.73). White powder, mp 184~185C, []D22 = 88.9 (c = 0.6,
[548-43-6] C16H18N2O (254.33). mp 250~252C. Pharm: Inhibits release of
CHCl3). Pharm: Cytotoxic (A549, ED50 = 18.9g/mL; HL-60, ED50 >
galactin; CNS stimulant. Source: MAI JIAO Claviceps purpurea, QIAN NIU
50g/mL; HT29, ED50 > 50g/mL; KB, ED50 > 50g/mL; P388, ED50 =
ZI Pharbitis nil. Ref: 6, 658.
3.41g/mL). Source: DA YE SHU LAN Aglaia elliptifolia (leaf: yield =

0.00071%dw). Ref: 3031.
O
HO
O
H
N
N
OH
HO
N
H
6766 Emarginatine
C38H46N2O17 (802.79). Pharm: Cytotoxic (KB ED50 = 1.7mg/L, Colon205
ED50 = 4.1mg/L). Source: NAN SHE TENG GEN Celastrus orbiculatus [Syn.
Celastrus articulatus]. Ref: 2511.
6761 Elliptinol
C18H24N2O3 (316.4). White powder, mp 162~163C, []D22 = +38.6 (c = 0.05,
CHCl3). Pharm: Cytotoxic (A549, ED50 > 50g/mL; HL-60, ED50 =
32.1g/mL; HT29, ED50 > 50g/mL; KB, ED50 >50g/mL; P388, ED50 =
N
O
3.62g/mL). Source: DA YE SHU LAN Aglaia elliptifolia (leaf: yield =

0.00005%dw). Ref: 3031.
O
H
N
H
O
OH
OH
H
HN
OH OH
O
O
HO
O
O
O
O
6762 Elliptone
C20H16O6 (352.35). Pharm: Anti-tumor promotor (in vivo, mouse skin tumor,
inhibits TPA-induced EBV-EA activation, 100 mol ratio/32pmol TPA,
EBV-EA positive cells = 76.8% viability, positive control -Carotene,
EBV-EA positive cells = 82.7% viability). Source: YU TENG Derris trifoliata
(stem). Ref: 4982.
O
2,5-Dihydroxy-3-undecyl-2,5-cyclohexadiene-1,4-dione [550-24-3] C17H26O4

(294.39). Orange crystals (MeOH or hexaneEtOH), mp 145~146C, mp
143C. Pharm: Analgesic; anti-fertility agent (rat); anti-inflammatory;
antipyretic; anthelmintic (teniafuge); DPPH free radical scavenger (IC50 =
(23.30.5)mol/L, control Trolox, IC50 = (25.40.8)mol/L)[4244];
antineoplastic (rat, autochthoneous fibrosarcomas induced by
6767 Embelin
methylcholanthrene, prolonged the survival time of the animals)[5369];
cytotoxic (in vitro, fibrosarcoma cell line, concentration-dependent decrease

H
O
O
in thymidine uptake and glutathione levels of the tumor cells)[5369]. Source:

AI ZI JIN NIU Ardisia humilis, BA BEI SUAN TENG ZI Embelia barbeyana,
CHI YE TIE ZI Myrsine semiserrata, CU YE MAI MI HUA SHU Rapanea
6763 Elsholtzia ketone
neurophylla, CU ZHUANG SUAN TENG ZI Embelia robusta, LA ZHU
[488-05-1] C10H14O2 (166.22). bp 210C. Source: BAN BIAN SU Elsholtzia
GUO Aegiceras corniculatum, MA GUI HUA Embelia oblongifolia, SAN
ciliata. Ref: 6.
HUA MI HUA SHU Rapanea umbellata, TIE ZI Myrsine africana, WEI

LING XIAN Clematis chinensis, XIAN SUAN QIANG Embelia ribes, XIAO
TOU TIE ZI Myrsine capitellata, YOU SE ZI JIN NIU Ardisia colorata
(fruit), ZHU SHA GEN Ardisia crenata, ZI JIN NIU Ardisia japonica,
6764 Elsholtzidiol
[28666-20-8] C10H16O3 (184.24). mp 58~59C. Source: XIANG RU
Connarus ritchiei, Embelia kilimandscharica, Embelia tsjersium-cottam,

Rapanea sp. Ref: 6, 658, 1521, 4244, 5369.
Elsholtzia splendens. Ref: 6.

OH
O
HO
O
OH
OH
O
238
6768 Embelinone
6772 Emetine
3,16-dioxo-13 17-methyleneoxyoleanane C30H46O3 (454.70). Clear needles,
Cephaeline methylether [483-18-1] C29H40N2O4 (480.65). White powder, mp
mp 257~259C []D25 = 4 (c = 0.6, CHCl3). Source: KEN NI YA XIAN
74C, turning yellow if exposed or heated, []D20 = 50 (c = 2, chloroform),
SUAN QIANG Embelia schimperi. Ref: 2058.
easily soluble in ethanol, acetic ester, chloroform, ether, insoluble in

water.[5507] Pharm: Antiamebic; antineoplastic; antiviral; antitussive (dispels
phlegm); emetic; LD (hmn) = 10~20mg/kg. Source: TU GEN Cephaelis
ipecacuanha (root: content scope = 2%4%)[5507], YANG CHANG CHUN
TENG Hedera helix. Ref: 658, 661, 5507.
H
O
H
O
6769 Embinin
H
H
[52589-13-6] C29H34O14 (606.59). mp 181C. Pharm: Xanthinoxidase
HN
inhibitor (50g/mL, InRt = 22.8 %); aldose reductase inhibitor (rat eye lens,
10mol/L InRt = 12.7%). Source: HU DIE HUA Iris japonica, YUAN WEI
Iris tectorum. Ref: 6, 1632, 1631.
6773 Emindole PA
C33H47NO2 (489.75). Colorless amorphous powder. Source: ZI LUO KE BAO
Emericella purpurea. Ref: 1101.
O
O
HO
O
OH
OH
N
H
OH
OH
OO
OH
6774 Emindole PB
C33H47NO2 (489.75). Colorless amorphous powder. Source: ZI LUO KE BAO
OH OH
Emericella purpurea. Ref: 1101.

6770 Ememodin
C20H26O6 (362.43). mp 237~239C, []D17 = 131 (c = 0.0498, EtOH).
Source: MAO GUO XIANG CHA CAI Isodon trichocarpa. Ref: 4067.
H
H
OH
6775 Emindole PC
O
C33H47NO2 (489.75). Colorless crystalline powder (ether), mp 238~240C.
Source: ZI LUO KE BAO Emericella purpurea. Ref: 1101.
O
HO
O
N
H
6771 Ememogin
C20H26O7 (378.43). mp > 300C, []D
24
= 145.8 (c = 0.20, C5H5N). Source:
MAO GUO XIANG CHA CAI Isodon trichocarpa. Ref: 4067.
OH
6776 Emodin
Orange red prismatic crystals, mp 250~257C. Pharm: Antibacterial
H
O
HO
1,3,8-Trihydroxy-6-methylanthraquinone [518-82-1] C15H10O5 (270.24).
HO
O
O O
(Staphylococcus aureus, Bacillus coli, Bacillus pyocyaneus, Bacillus

dysenteriae, Bacillus influenzae, Bacillus diphtheriae, Bacillus subtilis,
Bacillus paratyphosus, Coccus catarrhal, and -Streptococcus); antineoplastic
(mus, B16 melanoma BL, 50mg/(kgd), InRt = 76%, mus, mammary cancer
OH
and EAC); antifungal (Trichophyton interdigitali, Microsporum sp.);

antispasmodic; antispirochetic; antitussive; cytotoxic (Walker sarcoma, P388);
239
diuretic; antihypertensive; inhibits coronal wart growth in potato flower tray;
6778 Emodin-1-O--D-glucopyranoside
antitrypanosomal (Trypanosoma brucei, IC50 = (18.14.2)g/mL, control
C21H20O10 (432.39). Pharm: Inhibits sperm movement (hmn); antioxidant
Melarsoprol, IC50 = (0.00150.0009)g/mL; Trypanosoma cruzi, IC 50 =
inactive (DPPH radical scavenger); cytotoxic inactive (MCF, HM02, HEPG2).
(19.82.4)g/mL, control Benznidazole, IC50 = (0.390.15)g/mL)[5008];
Source: DA HUANG Rheum officinale, HU ZHANG Polygonum cuspidatum,
antileishmanial (Leishmania donovani, IC50 = (20.50.5)g/mL, control
NIU XI XI Rumex patientia, OU SHU LI Rhamnus frangula [Syn. Frangula
Miltefosine, IC50 = (0.230.03)g/mL)[5008]; antimalarial (Plasmodium
alnus], TANG GU TE DA HUANG Rheum tanguticum, ZHANG YE DA
falciparum, IC50 = (9.71.2)g/mL, control Chloroquine, IC50 =
HUANG Rheum palmatum. Ref: 2, 658, 660, 5232.
(0.0550.02)g/mL, control Artemisinin, IC50 = (0.00110.0006)g/mL)[5008];

cytotoxic (L6, IC50 = (20.32.6)g/mL, control Podophyllotoxin, IC50 =
0.0075g/mL)[5008]; cytotoxic (in vitro, Calu1, IC50 = (6.252.9)mol/L; HeLa,
HO
IC50 = (15.64.2)mol/L; K562, IC50 > 100mol/L; Raji, IC50 =

(43.87.3)mol/L; Vero, IC50 = (401.7)mol/L; Wish, IC50 =
(28.81.9)mol/L, 1,3,8-trihydroxy for anthraquinone plays a significant role
in the cytotoxic activity)
[3057]
; cytotoxic inactive (MCF, HM02, HEPG2)
[5232]
antioxidant inactive (DPPH radical scavenger assay)[5232]; antioxidant inactive
HO
OO
OH
OH
OH
OH
(DPPH radical scavenger, IC50 > 100g/mL; control Ascorbic acid, IC50 =
3.9g/mL)[4711]. Source: BAI HE Lilium brownii var. viridulum [Syn. Lilium
brownii var. colchesteri], CHAO XIAN YIN YANG HUO Epimedium
koreanum, CHI MA Boehmeria platanifolia [Syn. Boehmeria tricuspis], DA
HUANG Rheum officinale, DONG FANG WEI SI MU Vismia orientalis (stem
cortex), DUN YE JUE MING Cassia obtusifolia (ripe seed: mean content =
0.011%)
[5508]
6779 Emodin-3-O--D-glucopyranoside
C21H20O10 (432.39). Amorphous. Pharm: Antioxidant inactive (DPPH radical
scavenger assay)[5232]; cytotoxic inactive (MCF, HM02, HEPG2)[5232]. Source:
JUE MING ZI Cassia tora, NIU XI XI Rumex patientia. Ref: 2, 5232.
, GANG BAN GUI GEN Polygonum perfoliatum, HE SHOU
WU Polygonum multiflorum (dried tuberoid (raw): content scope of 9 batch
OH
OH
samples = 0.0026%~0.132%, mean content = 0.044%)[5508], HE SHOU WU

Polygonum multiflorum (dried tuberoid (preparing): content scope of 8 batch
samples = 0.0020%~0.168%, mean content = 0.042%)[5508], HU ZHANG
[5508]
Polygonum cuspidatum (rhizome: mean content = 1.40%
HO
), HUANG HAO
OH
Artemisia scoparia [Syn. Artemisia capillaris var. scoparia], JUE MING ZI
OH
OH
Cassia tora, MAO GUO YI HE GUO Ventilago calyculata, NI BO ER YANG

TI Rumex nepalensis, NIU ER DA HUANG Rumex crispus, NIU SHE CAO
Rumex dentatus (root: mean content = 0.0805%[5508]), NIU XI XI Rumex
6780 Enaimeone A
patientia (root: mean content = 0.1159%)[5508], OU SHU LI Rhamnus frangula
C21H39O5 (362.47). Pharm: Antioxidant inactive (PMN cellular
[Syn. Frangula alnus], SHU LI Rhamnus davurica, SUAN MO Rumex
chemiluminescence assay, FMLP-induced and OZ-induced oxidative burst).
acetosa (root: mean content = 0.3025%)[5508], TANG GU TE DA HUANG
Source: Hypericum papuanum Ref: 5371.
Rheum tanguticum, TIAN SHAN DA HUANG Rheum wittrocki, TIE ZI

Myrsine africana, WANG JIANG NAN Cassia occidentalis, WANG JIANG
NAN ZI Cassia occidentalis (ripe seed: content = 0.0016%)[5508], YANG TI
Rumex japonicus (root: mean content = 0.0881%)[5508], YI HE GUO Ventilago
O
OH
leiocarpa (stem)[3057], ZANG BIAN DA HUANG Rheum emodi [Syn. Rheum

australe] (stem and rhizome: content = 1.38%[5508]; yield = 0.53%dw[4711]),
O
ZHANG YE DA HUANG Rheum palmatum (stem and rhizome: content =
OH
0.42%)[5508], occurs in many plants. Ref: 2, 4, 458, 511, 608, 658, 660, 3057,
4711, 5008, 5232, 5501, 5508.
OH
OH
6781 Enaimeone B
OH
6777 Emodin anthrone

[491-60-1] C15H12O4 (256.26). mp 236C. Source: JUE MING ZI Cassia tora. Ref: 2, 6.
OH
OH
OH
O
OH
OH
240
6782 Enaimeone C
6787 Enanderianin G
Source: ZI MAO XIANG CHA CAI Isodon enanderianus. Ref: 1948.
OH
O
O
OH
22
= 76.9 (c = 0.52, MeOH). Source:
ZI MAO XIANG CHA CAI Isodon enanderianus. Ref: 4067.
O
H
OH
O
H
H
O
C22H30O7 (406.48). Colorless cubic crystals (MeOH), mp 235~237C, []D20

= 33.3 (c = 0.20, MeOH). Pharm: Cytotoxic (hmn tumor K562 cells, IC50 =

ZI MAO XIANG CHA CAI Isodon enanderianus. Ref: 4067.
0.67g/mL, control cis-Platin, IC 50 = 0.52g/mL). Source: ZI MAO

XIANG CHA CAI Isodon enanderianus (aerial parts). Ref: 5475.
O
H
O
OH
1,7,13-Trihydroxy-11-acetoxy-7,20-epoxy-ent-kaur-16-en-15-one
6784 Enanderianin B
O
OH
6789 Enanderianin K
O
OH
OH
HO
OH
OH
Source: ZI MAO XIANG CHA CAI Isodon enanderianus. Ref: 1948.
C24H32O9 (464.52). mp 225~227C, []D
O
OH
OH
6783 Enanderianin A
6788 Enanderianin H
O
OH
O
OH
O
OH
OH
H
O
OH
O
OH
6785 Enanderianin C
Xerophilusin H [247939-40-8] C22H30O7 (406.48). Colorless acicular crystals,
23
[]D = 149.4 (c = 0.43, pyridine), mp 238~240C, mp 262~264C. Pharm:
6790 Enanderianin L
7,13-Dihydroxy-1-acetoxy-7,20-epoxy-ent-kaur-16-en-15-one
Cytotoxic (K562, IC50 = 1.17g/mL, control Mitoxantrone, IC50 = 0.29g/mL;
HL-60, IC50 = 0.87g/mL, Mitoxantrone, IC50 = 0.29g/mL; HCT, IC50 =
89.8 (c = 0.25, MeOH). Pharm: Cytotoxic (hmn tumor K562 cells, IC50 =
52.78g/mL, Mitoxantrone, IC50 = 1.54g/mL; MKN28, IC50 = 1.86g/mL,
0.16g/mL, control cis-Platin, IC 50 = 0.52g/mL). Source: ZI MAO
[5182]
Mitoxantrone, IC50 = 0.02g/mL)
. Source: HAN SHENG XIANG CHA
XIANG CHA CAI Isodon enanderianus (aerial parts). Ref: 5475.
CAI Isodon xerophilus (leaf), ZI MAO XIANG CHA CAI Isodon

enanderianus. Ref: 894, 4067, 5182.
OH
OH
H
O
H
O
O
O
OH
OH
O
OH
6791 Enanderianin M
6786 Enanderianin F
7,13,15-Trihydroxy-1-acetoxy-7,20-epoxy-ent-kaur-16-ene C22H32O6
(392.50). Colorless needles (Me2CO), mp 253~255C, []D20 = +25.0 (c =
MeOH). Source: ZI MAO XIANG CHA CAI Isodon enanderianus. Ref:
0.08, MeOH). Pharm: Cytotoxic (hmn tumor K562 cells, very weak). Source:
1948.
ZI MAO XIANG CHA CAI Isodon enanderianus (aerial parts). Ref: 5475.
O
H
O
OH
H
O
O
H
OH
OH
241
6792 Enanderianin N
6797 Encecalinol
7,14,15-Trihydroxy-1-acetoxy-7,20-epoxy-ent-kaur-16-ene C22H32O6
Encecalol C14H18O3 (234.30). Pharm: Antifungal (Trichophyton
(392.50). Colorless needles (Me2CO), mp 216~218C, []D20 = +5.7 (c = 0.26,
mentagrophytes ATCC28185, MIC = 12.5g/mL, control Miconazole, MIC =
MeOH). Pharm: Cytotoxic (hmn tumor K562 cells, very weak). Source: ZI
8g/mL; Trichophyton rubrum ATCC28188, MIC = 12.5g/mL, Miconazole,
MAO XIANG CHA CAI Isodon enanderianus (aerial parts). Ref: 5475.
MIC = 8g/mL; Candida albicans ATCC10231, MIC = 100g/mL, Nistatin,
MIC = 16g/mL)[5472]. Source: FU CHUI FE LAO JU Flourensia cernua,
MIC = 8g/mL; Candida niger ATCC10335, MIC = 200g/mL, Miconazole,

O
Eupatorium aschenbornianum. Ref: 1521, 5472.
OH
OH
OH
O
H
6793 Enanderianin O
7,14,15-Trihydroxy-1-acetoxy-7,20-epoxy-ent-kaurane C22H34O6
HO
(394.51). Colorless cubes (Me2CO), mp 196~198C, []D20 = 38.5 (c = 0.13,
MeOH). Source: ZI MAO XIANG CHA CAI Isodon enanderianus (aerial

parts). Ref: 5475.
6798 5-Ene-methyl-7,12-didehydroxy-cholate-3-O--D-glucopyranoside
C31H50O8 (550.74). White lamellar crystals, mp 201~205C, soluable in
methanol. Source: SAN LENG Sparganium stoloniferum. Ref: 497.
H
OH
OH
OH
O
H
O
O
H
H
6794 Enanderianin P
3,14,17-Trihydroxy-18-alent-abieta-7(8),15(16)-diene C20H30O4 (334.46).
Colorless cubes (Me2CO), mp 187~189C, []D24 = 0.7 (c = 5.00, MeOH).
H
HO
OH
Pharm: Cytotoxic (hmn tumor K562 cells, IC50 = 0.59g/mL, control

cis-Platin, IC50 = 0.52g/mL). Source: ZI MAO XIANG CHA CAI Isodon
OO
OH
OH
enanderianus (aerial parts). Ref: 5475.
6799 5-Ene-methyl-7,12-didehydroxy-cholate-3-O--L-rhamnopyranosOH
yl-(14)--D-glucuronopyranoside
C37H58O13 (710.8). White amorphous powder, mp 215~219C, soluble in
OH
H
HO
methanol. Source: SAN LENG Sparganium stoloniferum. Ref: 497.
6795 Enanthic acid

Heptanoic acid [111-14-8] C7H14O2 (130.19). Source: DANG SHEN
Codonopsis pilosula, CHAI HU Bupleurum chinense, SAN QI Panax
OH
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng], XI YANG SHEN
OO
Panax quinquefolium. Ref: 2, 6.
OH
OH
OO
OH
OH
O
OH OH
6800 3-Ene-nonanone-2
6796 Encecalin
C14H16O3 (232.28). Pharm: Pesticide; phytotoxic (yeast and bacteria). Source:
[14309-57-0] C9H16O (140.23). Source: SAN QI Panax pseudo-ginseng var.

XIAN ZE LAN Eupatorium glandulosum. Ref: 658.

O
O
O
O
242
6801 Engelhardione
6806 Enmelol
C19H20O4 (312.37). Colorless needles (CH2Cl2MeOH), mp 73~75C. Pharm:
C20H30O5 (350.45). mp 263~265C, []D35 = 48 (c = 0.0863, EtOH). Source:
Antitubercular (Mycobacterium tuberculosis 90-221387, MIC =
MAO GUO XIANG CHA CAI Isodon trichocarpa, SHAN DI XIANG CHA
3.125g/mL; Mycobacterium tuberculosis H37Rv, MIC = 0.2g/mL).
CAI Isodon oresbia (aerial parts). Ref: 4067, 3808.
Source: HUANG QI II Engelhardia roxburghiana (root). Ref: 5059.

HO
OH
OH
OH
OH
OH
6802 Enhydrin
6807 Enmenin monoacetate
[33880-85-2] C23H28O10 (464.47). Pharm: Antihypertensive. Source: ZHAO
C26H36O8 (476.57). Source: SHAN DI XIANG CHA CAI Isodon oresbia
JU Enhydra fluctuans. Ref: 658.

O
O
O
H
O
H
O
O
O
6803 Enmedol
C22H30O6 (390.48). mp 297~299C, []D
27.5
= 45 (c = 0.1147, MeOH).
Source: MAO GUO XIANG CHA CAI Isodon trichocarpa. Ref: 4067.
6808 Enmenol
C20H30O6 (366.46). mp 255~257C. Source: LU SHAN XIANG CHA CAI
Isodon rubescens var. lushanensis (leaf), MAO GUO XIANG CHA CAI
OH
Isodon trichocarpa. Ref: 4067, 4353.
O
H
O
OH
O
O
OH
OH
6804 Enmein
H
OH
OH
[3776-39-4] C20H26O6 (362.43). Colorless short columnar crystals, mp
10
297~299C (dec), []D = 156 (acetone), []D = 131.3 (c = 1.0, C5H5N).
OH
OH
Pharm: Antineoplastic (male mus, EAC, 10~15mg/kg ip, biotic prolonged rate
= (39~66)%). Source: MAO YE XIANG CHA CAI Isodon japonica [Syn.
6809 Entadamide A
Rabdosia japonica] (the compound was isolated from the plant in 1965)[5505],
C6H11NO2S (161.22). Pale yellow oil. Pharm: Antitubercular inactive
MAO GUO XIANG CHA CAI Isodon trichocarpa, SHAN DI XIANG CHA
(Mycobacterium tuberculosis H37Ra); antimalarial inactive (Plasmodium
CAI Isodon oresbia (aerial parts). Ref: 661, 4067, 5505, 3808, 4067.
falciparum, EC50 > 20g/mL). Source: TAI GUO NIU XU HUA
Clinacanthus siamensis (leaf). Ref: 4410.
H
N
OH
O
S
HO
6805 Enmein-3-acetate
C22H28O7 (404.46). mp 267~271(dec)C, []D17 = 112 (c = 1.0, C5H5N).
Source: MAO YE XIANG CHA CAI Isodon japonica [Syn. Rabdosia
japonica]. Ref: 4067.
O
O
6810 Entadamide C
C6H11NO3S (177.22). Colorless needles (acetone), mp 141~142C. Pharm:
Antitubercular inactive (Mycobacterium tuberculosis H37Ra); antimalarial
inactive (Plasmodium falciparum, EC50 > 20g/mL). Source: TAI GUO NIU
XU HUA Clinacanthus siamensis (leaf). Ref: 4410.
H
N
O
O
O
OH
OH
O
S
OH
243
6811 Entagenic acid
Source: BAN XIA Pinellia ternata (dried tuber: content = 0.0020%)[5501 5508],
[5951-41-7] C30H48O5 (488.71). mp 310~315C. Source: KE TENG ZI Entada
BAN ZI MA HUANG Ephedra lepidosperma (herbaceous twigs: content =
phaseoloides [Syn. Lens phaseoloides]. Ref: 6.
0.024%)[5508], DAN ZI MA HUANG Ephedra monosperma (herbaceous twigs:

content = 1.247%)[5508], HUANG HUA REN Sida acuta, LI JIANG MA
HUANG Ephedra likiangensis (herbaceous twigs: mean content of 3 origins =
0.727%)[5508], MA HUANG Ephedra sinica (herbaceous twigs: content scope
OH
HO
MA HUANG Ephedra przewalskii (herbaceous twigs: mean content of 2
O
OH
OH
= 0.272%~0.889%[5501], mean content of 5 origins = 0.654%)[5508], MO GUO

origins = 0.027%)[5508], MU ZEI MA HUANG Ephedra equisetina
(herbaceous twigs: content scope = 1.113%~1.409%[5501], mean content of 2

origins = 1.256%[5508]), SHAN LING MA HUANG Ephedra gerardiana
6812 Enterolactone
[78473-71-9] C18H18O4 (298.34). Pharm: Cancer-preventing activity. Source:
family Brassicaceae spp. Ref: 1521, 1582.
OH
HO
(herbaceous twigs: content = 0.696%[5508]), SHU ZHUANG MA HUANG

Ephedra procera (herbaceous twigs: content = 0.06%)[5508], SHUANG SUI
MA HUANG Ephedra distachya (herbaceous twigs: content = 0.19%)[5508],
XI ZANG ZHONG MA HUANG Ephedra intermedia var. tibetica
(herbaceous twigs: content = 1.060%)[5508], XI ZI MA HUANG Ephedra
regeliana (herbaceous twigs: content = 0.054%)[5508], YI ZHU AI MA
HUANG Ephedra minuta var. dioeca (herbaceous twigs: mean content of 2

origins = 0.567%)[5508], ZANG MA HUANG Ephedra saxatilis (herbaceous
6813 Ephedradine B
twigs: content =0.601%)[5508], ZHONG MA HUANG Ephedra intermedia
[71327-57-6] C29H38N4O5 (522.65). Crystals without free alkali,
(herbaceous twigs:), ZHONG MA HUANG Ephedra intermedia (herbaceous
dihydrobromide: (C29H38N4O52HBrH2O) mp 219~221C, []D = 101.5
twigs: content scope = 0.125%~0.47%[5501], mean content of 3 origins =
(water). Pharm: Antihypertensive. Source: Ephedra sp. Ref: 661.
0.266%[5508]), Ephedra tweediana (herbaceous twigs: content = 0.0028%)[5508].

Ref: 4, 658, 660, 5501, 5507, 5508.
O
OH
O
H
H
O
HN
N
H
N
H
HO
H
N
H
H
6814 Ephedradine C
6816 (4S,5R) Ephedroxane
[73276-37-6] C30H40N4O5 (536.68). Crystals without free alkali,
[16251-46-0] C11H13NO2 (191.23). Pharm: Anti-inflammatory. Source: AI
dihydrobromide: (C30H40N4O52HBrH2O) mp 224~225C, []D = 100.7
MA HUANG Ephedra minuta, MA HUANG Ephedra sinica, MU ZEI MA
(water). Pharm: Antihypertensive. Source: Ephedra sp. Ref: 661.
HUANG Ephedra equisetina, SHAN LING MA HUANG Ephedra

gerardiana, SHUANG SUI MA HUANG Ephedra distachya, ZHONG MA
HUANG Ephedra intermedia. Ref: 2, 658, 660.
O
O
O
H
HN
N
H
O
N
H
N
H
6817 4-Epi-abietic acid

C20H30O2 (302.46). White amorphous powder. Source: JIA DI FENG PI
Illicium jiadifengpi (bark). Ref: 4560.
6815 Ephedrine
Ephedine; 1-Phenyl-2-methylaminopropanol [299-42-3] C10H15NO (165.24).
mp 38.1C, bp 225C, []D20 = 6.3 (ethanol), []D21 = 41 (1mol HCl),
easily soluble in water, ethanol, soluble in chloroform, benzene, ether.[5507]
Pharm: Antiasthmatic (bronchial smooth muscle relaxant); contracts

peripheral blood vessels; increases blood pressure; adrenergic - and
-receptor agonist to produce sympathomimetic action; CNS stimulant.
H
O
OH
244
6818 6-Epi-8-O-acetylharpagide
6822 ent-Epiafzelechin-(2O7,48)-epiafzelechin
C17H26O11 (406.39). White amorphous powder, []D = 36 (c = 0.0035,
Mahuangnin A C30H24O10 (544.52). Amorphous powder, mp > 300C.
MeOH). Source: ZA JIAO YOU(2) Caryopteris clandonensis. Ref: 3988.
Source: MA HUANG GEN Ephedra sinica, XING REN Prunus armeniaca.

Ref: 1230, 1896.
OH
HO
OH
O
HO
HO
H
OO
OH
OH
O
O
OH
OH
OH
O
OH
6819 ()-Epiafzelechin
[24808-04-6] C15H14O5 (274.28). White crystals, mp 248~250C, []D =
OH
HO
59 (c = 0.1, MeOH). Pharm: Antioxidant (DPPH free radical scavenger,

IC50 = 7.5g/mL)[3028]. Source: AN MO LE Phyllanthus emblica (branch
and leaf)[3094] , NAN SHE TENG YECelastrus orbiculatus [Syn. Celastrus
articulatus], NAN SHE TENG Celastrus orbiculatus [Syn. Celastrus
articulatus] (aerial parts: yield = 0.0025%dw)[3028], OU ZHOU CI BAI
6823 ()-Epiafzelechin-4-(2-hydroxyethyl)thio ether

C17H18O6S (350.39). Red amorphous powder, []D = +208.5 (c = 0.4, MeOH).
Source: XIAO GUO YE JIAO Musa acuminata (fruit). Ref: 3913.
Juniperus communis, XI BO JUE MING Cassia sieberiana. Ref: 713,

3028, 3094.
OH
O
HO
OH
HO
OH
O
OH
OH
OH
OH
6824 4-Epiaglain A
6820 ent-Epiafzelechin-(2O7, 48)-(+)-afzelechin
C38H44N2O9 (672.78). Amorphous powder, []D20 = 1.0 (c = 0.97, CHCl3).
C30H24O10 (544.52). Amorphous powder, mp > 300C. Source: XING REN
Source: TUE YUAN MI ZI LAN Aglaia elliptica (leaf). Ref: 4127.
Prunus armeniaca. Ref: 1896.
OH
HO
H
O
O O
O
OH
OH
HO
OH
OH
OH H
H
N
6821 ent-Epiafzelechin-(2O7,48)-()-afzelechin
6825 Epi--amyrin
C30H24O10 (544.52). Amorphous powder, mp > 300C. Source: XING REN
[5937-48-4] C30H50O (426.73). Source: MI DIE XIANG Rosmarinus
Prunus armeniaca. Ref: 1896.
OH
HO
O
OH
OH
H
HO
O
HO
OH
OH
245
6826 6-Epiangustifolin
6829 8-Epiapodantheroside
C21H28 O6 (376.45). Colorless needles (MeOH), mp 240~242C, []D17 =
94.7 (c = 0.41, MeOH). Pharm: Cytotoxic (in vitro, K562, IC50 =
MeOH). Source: ZHI ZI YE Gardenia jasminoides [Syn. Gardenia florida].
0.87g/mL; control cis-Platin, IC 50 = 0.52g/mL)[4732]. Source: LU
Ref: 4408.
SHI DONG LING CAO Isodon rubescens var. lushiensis (leaf: yield =
0.0004%dw)[4732], ZI MAO XIANG CHA CAI Isodon enanderianus. Ref:
2030, 4732.
HO
H
O
HO
HO
O
O
OO
OH
OH
OH
6827 34-Epiannomolon A
C35H62 O7 (594.88). White powder, mp 82.1~82.7C, []D23 = 5.0 (c =
6830 (+)-8,8'-Epi-aristoligone
0.02, CH2Cl2). Pharm: The data are from mixture of annomolon A and
(7'R,8R,8'S)-8,8'-Dimethyl-3',4',4,5-tetramethoxy-2,7'-cyclolignan-7-one
34-epi-annomolon A: cytotoxic (BST, LC50 = 0.375g/mL); cytotoxic (in
C22H26O5 (370.45). Yellow crystals, mp 146.5~149.3C, []D25 = 30.0 (c =
vitro, A549, ED50 = 1.26g/mL; MCF7, ED50 = 0.303g/mL; HT29, ED50
1.33, CHCl3). Source: Holostylis reniformis (root). Ref: 3784.
= 0.193g/mL; A498, ED50 = 0.93g/mL; PC3, ED50 = 0.198g/mL;

MIA-PaCa-2, ED50 = 0.00312g/mL; control Adriamycin: A549, ED50 =
0.00113g/mL; MCF7, ED50 = 0.0182g/mL; HT29, ED 50 =
0.0128g/mL; A498, ED50 = 0.00226g/mL; PC3, ED50 = 0.0502g/mL;
O
O
O
MIA-PaCa-2, ED50 = 0.00262g/mL). Source: MAO YE FAN LI ZHI

Annona cherimolia (seed). Ref: 4731.
O
O
OH
O
O
OH
OH
6831 ()-8,8'-Epi-aristoligone
(7'R,8S,8'S)-8,8'-Dimethyl-3',4',4,5-tetramethoxy-2,7'-cyclolignan-7-one
C22H26O5 (370.45). Yellow crystals, mp 130.0~132.0C, []D25 = 64.3 (c =

6828 34-Epiannomolon B
C35H62 O8 (610.88). White powder, mp 86.3~87.2C, []D23 = +6.0 (c =
O
O
0.02, CH2Cl2). Pharm: The data are from mixtures of annomolon B and
34-epi-annomolon B: cytotoxic (BST, LC50 = 0.07g/mL); cytotoxic (in
vitro, A549, ED50 = 1.37g/mL; MCF7, ED50 = 0.047g/mL; HT29, ED50

= 0.0719g/mL; A498, ED50 = 0.377g/mL; PC3, ED50 = 0.0553g/mL;
MIA-PaCa-2, ED50 = 0.00748g/mL; control Adriamycin: A549, ED50 =
0.00113g/mL; MCF7, ED50 = 0.0182g/mL; HT29, ED 50 =

0.0128g/mL; A498, ED50 = 0.00226g/mL; PC3, ED50 = 0.0502g/mL;
MIA-PaCa-2, ED50 = 0.00262g/mL). Source: MAO YE FAN LI ZHI
6832 Epiaschantin
Annona cherimolia (seed). Ref: 4731.
C22H24O7 (400.43). []D20 = +95 (c = 0.2, CHCl3). Source: LIAN YE TONG

Hernandia Sonora [Syn. Hernandia ovigera] (seed). Ref: 5030.
OH
O
OH
OH
O
OH
H
O
H
O
O
O
246
6833 10-Epiatractyloside A
6837 3-Epibetulinic acid 28-O--L-rhamnopyranosyl-(14)--D-gluco-
C21H36O10 (448.52). Amorphous powder, []D22 = +14 (c = 1.2, MeOH).
pyranosyl(16)--D-glucopyranoside
Source: CANG ZHU Atractylodes lancea, GUAN CANG ZHU Atractylodes
C48H78O17 (927.15). White powder, mp 208~210 C []D20 = 38.7 (c = 0.4,
japonica (fresh rhizome). Ref: 4310, 4348.
MeOH). Source: DONG BEI CI REN SHEN Oplopanax elatus. Ref: 467,
1521.
OH
OH
H
O
HO
H
OO
HO
HO
HO
OH
OH
OH
OH
6834 Epi-baiyecrystal C
Source: BAI YE XIANG CHA CAI Isodon leucophyllus. Ref: 4067.
OH
OH
OH
6838 (+)-4-Epi--bisabolol
C15H26O (222.37). Source: FEN CHA DANG GUI Angelica furcijuga
HO
O
H
O
H
OO
O
O
OH
OH OH
C26H38O9 (494.59). mp 224~225.5C, []D22.3 = 5.68 (c = 0.26, MeOH).
OO
OO
OH
O
OH
OH
6839 Epi-bisdehydrotuberostemonine J
C22H29NO4 (371.48). mp 186~188C, []D20 = 16.1 (c = 0.1, MeOH). Pharm:
6835 Epiberberine
Antitussive inactive (guinea pig cough model)[5463]. Source: BAI BU Stemona
C20H18NO4 (336.37). Pharm: Cytotoxic (topoisomerase I inhibitor in
tuberosa. Ref: 5463.
vitro)[5369]. Source: DUO HUA XIAO BO Berberis floribunda, HUANG

LIAN Coptis chinensis (rhizome: mean content = 1.29%[5508]), NAN TIAN
[5508]
(rhizome: mean content = 0.54%)
, SAN YE HUANG LIAN Coptis
ZHU YE Nandina domestica, SAN JIAO YE HUANG LIAN Coptis deltoidea
H
N H
trifolia. Ref: 1521, 5369, 5508.
6840 ()-(1S*,5S*,6S*,7S*,10S*)-7-Epi-bourbon-3-en-5,11-oxide
C15H22O (218.34). Colorless oil. Source: XIAO E TAI Mylia taylorii

(essential oil), LUO XIAO E TAI Mylia nuda (essential oil). Ref: 3840.
H
O
O
6836 3-Epi-betulinic acid acetate

C32H50O4 (498.75). []D26 = +75.1 (c = 0.21, EtOH). Source: HUANG QI II
Engelhardia roxburghiana (root). Ref: 5059.
6841 Epibueropyridinium A
C18H19NO5 (329.36). Colorless hyaloid oil. Source: XUAN SHEN
Scrophularia ningpoensis. Ref: 8.
O
OH
O
OH
O
O
HO
OH
247
6842 Epibuphanisine
6846 Epicalyxin I
C17H19NO3 (285.35). Pharm: AChE inhibitor (IC50 = (5475)mol/L,
C42H38O9 (686.77). Light yellow amorphous solid, []D25 = +28.3 (c =
control Galanthamine, IC50 = (1.90.2)mol/L) . Source: Crinum
0.025, MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 12.1mol/L;
moorei. Ref: 4952.
HT1080, ED50 = 5.88mol/L; control Curcumin, Colon26-L5, ED50 =

23.2mol/L; HT1080, ED50 = 23.4mol/L)[3035]. Source: YUN NAN CAO
KOU Alpinia blepharocalyx (seed: yield = 0.000040%[3035]; yield =
0.000040%dw[3048]). Ref: 3035, 3048.
O
O
HO
N
OH
O
6843 Epicalyxin B
C35H34O8 (582.66). Source: ZHU SUI SHAN JIANG Alpinia pinnanensis
HO
O
O
HO
OH
OH
OH
6847 Epicalyxin J
H
OH
OH
C42H38O9 (686.77). Light yellow amorphous solid. Pharm: Cytotoxic
(mixture of calyxin J and epicalyxin J (1:1): Colon26-L5, ED50 =

13.7mol/L; HT1080, ED50 = 0.32mol/L; control Curcumin, Colon26-L5,
OH
OH
ED50 = 23.2mol/L; HT1080, ED50 = 23.4mol/L). Source: YUN NAN

CAO KOU Alpinia blepharocalyx (seed: yield = 0.000056%). Ref: 3035.
6844 Epicalyxin F
HO
C35H34O8 (582.66). Light yellow amorphous solid, []D25 = +103.1 (c = 0.05,
OH
MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 0.89mol/L; HT1080, ED50

= 1.71mol/L; control Curcumin, Colon26-L5, ED50 = 23.2mol/L; HT1080,
ED50 = 23.4mol/L). Source: YUN NAN CAO KOU Alpinia blepharocalyx
O
HO
(seed: 0.000043%). Ref: 3035.
OH
O
OH
HO
O
HO
OH
OH
6848 Epicalyxin K
O
C35H34O8 (582.66). Pale yellow amorphous solid, []D25 = 17.0 (c = 0.085,
MeOH). Pharm: Cytotoxic (Colon26-L5, ED50 = 33.0mol/L; HT1080,

ED50 = 4.75mol/L; control Curcumin, Colon26-L5, ED50 = 23.2mol/L;
HT1080, ED50 = 23.4mol/L). Source: YUN NAN CAO KOU Alpinia
6845 Epicalyxin H
C35H34O7 (566.66). Source: ZHU SUI SHAN JIANG Alpinia pinnanensis

OH
HO
O
HO
OH
OH
H
OH
HO
OH
O
O
OH
248
6849 Epicalyxin M
inhibits cancer cell invasion (MM1 cells, in vitro, 10g/mL, InRt = 20.3%)[4329];
C35H34O8 (582.66). Yellow amorphous solid (An epimeric mixture of calyxin M
bone marrow cell proliferation promotor (1~100mg/mL, promotes proliferation of
and epicalyxin M). Pharm: Cytotoxic (mixture of calyxin M and epicalyxin M (3:2):
cultured bone marrow cells, stimulates formation of myeloid colonies and
Colon26-L5, ED50 = 42.1mol/L; HT1080, ED50 = 10.1mol/L; control Curcumin,
enhances the effect of IL-3 to increase the number of colony forming-units in
Colon26-L5, ED50 = 23.2mol/L; HT1080, ED50 = 23.4mol/L). Source: YUN
culture (CFU-c))[5390]; bone marrow cell proliferation promoter (ex vivo, model
NAN CAO KOU Alpinia blepharocalyx (seed). Ref: 3035.
mouse of decreasing bone marrow functions, orally 100mg/(kgd), stimulates

IL-3-induced CFU-c formation of bone marrow cells)[5390]; antioxidant (DPPH
OH
HO
free radical scavenger, 10mol/L, ScRt = 82%, control BHT, 10mol/L, ScRt =
43%)[5319]; antioxidant (DPPH free radical scavenger, IC50 = 8.5g/mL)[3028].
HO
OH
Source: A LA BO JIAO JIN HE HUAN Acacia nilotica, AN MO LE

Phyllanthus emblica (branch and leaf)[3094], BAI GUO Ginkgo biloba, BI LU
GOU TENG Uncaria tomentosa, CAO YUAN LAO GUAN CAO Geranium
pratense, CHA YE Camellia sinensis [Syn. Thea sinensis], DAN ZI SHAN ZHA
Crataegus monogyna, DAO NIAN ZI Garcinia mangostana (fruit hull)[3066], E
6850 5-Epicanadense
O
O
rhynchophylla [Syn. Nauclea rhynchophylla], GUAN YE LIAN QIAO
Hypericum perforatum, HAI ER CHA Acacia catechu (dried decocted extract of

OH
OH
H
gambir (dried decocted extract of trunk: content scope of 10 origins =

1.57%3.84%; mean content = 2.45%)[5508], GOU TENG Uncaria
RONG WEI LING CAI Potentilla anserina, ER CHA GOU TENG Uncaria
trunk: content scope of 8 origins = 7.56%14.20%; mean content = 11.3%[5508]),

HEI ZI LI GUO JI SHENG Scurrura atropurpurea, HONG QI YE SHU
Aesculus carnea, JIA ZHOU QI YE SHU Aesculus californica, JIAN PU ZHAI
GU KE Erythroxylum cambodianum (aerial parts), LING LAN Convallaria
keiskei [Syn. Convallaria majalis], MAO GUO QI Acer nikoense (stem cortex),
MEI LI TENG HUANG Garcinia speciosa (trunk bark and stems), NAN SHE
6851 7-Epicandicandiol
TENG Celastrus orbiculatus [Syn. Celastrus articulatus] (aerial parts: yield =
C20H32O2 (304.48). Colorless needles (CHCl3). Source: Sideritis ozturkii
0.050%dw)[3028], QUAN SHEN Polygonum bistorta, SHA ZAO Elaeagnus
angustifolia, SHAN CHA Camellia japonica, SUO LA MU Salacia prinoides

[Syn. Salacia chinensis] (stem), TIAN SHAN ZHU ZI Garcinia dulcis (fruit),
TUO YUAN GOU TENG Uncaria elliptica, YUE JU YE Vaccinium vitis-idaea,
ZHU BAI Myrica nagi [Syn. Podocarpus nagi], Pterocarpus sp., occurs in many
plants. Ref: 6, 658, 661, 1521, 3028, 3066, 3094, 4304, 4329, 4378, 4461, 5319,
OH
OH
5341, 5375, 5390, 5491, 5508.

OH
6852 24-Epicastasterone
C28H48O5 (464.69). Source: YANG JIAN QIU LUO Lychnis viscaria. Ref: 2418.
HO
OH
OH
OH
OH
OH
HO
6854 Epicatechin
Epicatechol C15H14O6 (290.28). mp (+) 245C (dec), () 245C (dec), (+/~)
224~226C (dec). Pharm: antioxidant (DPPH radical scavenger, IC50 = 1.7g/mL;
HO
O
control Ascorbic acid, IC50 = 3.9g/mL)[4711]. Source: BAI GUO YE Ginkgo

biloba, DA HUANG Rheum officinale, HAI ER CHA Acacia catechu, SHAN LI
6853 ()-Epicatechin
HONG Crataegus pinnatifida var. major, SHAN ZHA Crataegus pinnatifida,
5,7,3',4',-Tetrahydroxyflavanol C15H14O6 (290.28). mp 242C, []D = 68.2
TANG GU TE DA HUANG Rheum tanguticum, YE SHAN ZHA Crataegus
(96% ethanol). Pharm: Antiallergic; antibacterial; anti-inflammatory;
cuneata, ZANG BIAN DA HUANG Rheum emodi [Syn. Rheum australe] (root:
antimutagenic; inhibits lactic acid bacteria; antioxidant (inhibits free-radical
yield = 0.033%dw)[4711], ZHAI YE BAN FENG HE Pterospermum lanceaefolium,
induced lysis of rat red blood cells and exhibits strong and dose-dependent
ZHANG YE DA HUANG Rheum palmatum. Ref: 2, 6, 433, 660, 4711, 5375.
protection of cell membrane)[5341]; cholinesterase inhibitor; antihypercholesterolemic (reduces the level of cholesterol in serum); antioxidant (DPPH free
radical scavenger, for 40mol/L DPPH radical, SC50 = 4.1mol/L)[4378]; DPPH
OH
HO
scavenger (IC50 = 8.5g/mL); -hexosaminidase inhibiter inactive (RBL-2H3

cells, inhibits release of -hexosaminidase, 100mol/L, InRt = (3.91.2)%)[4304];
OH
OH
OH
249
6855 Epicatechin-(2O7,46)-catechin
6858 Epicatechin-(2O7,48)-ent-epicatechin
C30H24O12 (576.52). Colorless needles (H2O), mp 271~273C (dec), []D =
C30H24O12 (576.52). White crystalline powder (H2O), mp 260C (dec). Pharm:
+10.12 (c = 1.05, acetone). Pharm: Hyaluronidase inhibitor. Source: LUO
Hyaluronidase inhibitor. Source: LUO HUA SHENG Arachis hypogaea. Ref: 2284.
OH
HUA SHENG Arachis hypogaea. Ref: 2284.

O
HO
OH
OH
OH
OH
HO
OH
OH
OH
HO
OH
HO
OH
HO
6859 Epicatechin-(46,2O7)-ent-epicatechin
OH
C30H24O12 (576.52). White amorphous powder (H2O/MeOH); mp 280C (dec).
OH
OH
Pharm: Hyaluronidase inhibitor. Source: LUO HUA SHENG Arachis

hypogaea. Ref: 2284.
6856 Epicatechin-(2O7,46)-ent-catechin
OH
C30H24O12 (576.52). White amorphous powder (H2O); mp 262C (dec). Pharm:

Hyaluronidase inhibitor. Source: LUO HUA SHENG Arachis hypogaea. Ref: 2284.
HO
OH
OH
O
HO
OH
OH
OH
OH
HO
O
OH
OH
HO
OH
OH
6860 Epicatechin-(2O7,46)-[epicatechin-(48)]-catechin
OH
C45H36O18 (864.78). Off-white amorphous powder, mp 272C (dec), [] D =
OH
+86.2 (c = 0.3, acetone). Pharm: Antioxidant (DPPH scavenger, IC50 =
OH
(1.210.11)mol/L; control EGG, IC50 = (1.130.08)mol/L). Source: LUO
6857 [Epicatechin-(48)] 5-epicatechin
HUA SHENG Arachis hypogaea (seed). Ref: 3848.
C90H74O36 (1731.57). Pharm: Tanning agent. Source: ROU GUI Cinnamomum
OH
cassia [Syn. Cinnamomum aromaticum]. Ref: 658.

O
HO
O
OH
OH
O
HO
OH
HO
OH
OH
OH
HO
OH
OH
OH
OH
OH
6861 Epicatechin-(2O7,48)epicatechin-(48)-catechin-
OH
(48)-epicatechin
OH
C60H48O24 (1153.04). Off-white amorphous powder, mp 260C (dec), [] D =
OH
OH
HO
OH
OH
OH
HO
OH
OH
OH
OH
OH
(1.320.16)mol/L; control EGG, IC50 = (1.130.08)mol/L). Source: LUO
OH
OH
OH
HO
+27.6 (c = 0.3, acetone). Pharm: Antioxidant (DPPH scavenger, IC50 =
OH
HUA SHENG Arachis hypogaea (seed). Ref: 3848.

OH
OH
HO
OH
OH
OH
OH
OH
OH
O
OH
OH
OH
OH
O
OH
OH
OH
HO
O
OH
OH
OH
OH
HO
HO
OH
OH
HO
HO
OH
250
6862 Epicatechin-(2O7,46)-epicatechin-(2O7,48)-
6866 ()-Epicatechin 4-(2-hydroxyethyl)thio ether
epicatechin
C17H18O7S (366.39). Source: XIAO GUO YE JIAO Musa acuminata (fruit).
C45H34O18 (862.76). Pale yellow amorphous powder, []D21 = +184.9 (c = 1.08,
Ref: 3913.
OH
MeOH). Source: CHANG JIE ZHU Parameria laevigata (bark). Ref: 3523.
HO
OH
O
HO
OH
OH
O
OH
OH
OH
6867 ()-Epicatechin-pentaacetate
OH
OH
OH
HO
HO
OH
OH
C25H24O11 (500.46). Source: BAI GUO Ginkgo biloba. Ref: 2.
HO
OH
HO
6863 Epicatechin-8-C--D-galactopyranoside
C21H24O11 (452.42). Light-brown amorphous powder, []D = 25.8 (c = 0.9,
MeOH). Pharm: Antioxidant (inhibits NADPH -dependent lipid peroxidation
in microsomes and autoxidation of linoleic acid); antioxidant (DPPH

scavenger, effective). Source: KE KE Theobroma cacao. Ref: 2023.
6868 7-Epicephalomannine
C45H53NO14 (831.92). mp 210C, .[]D = 7.32 (MeOH). Source: ZA JIAO
OH
HO
O
HO
HO
HO
HO
OH
O O
OH
OH
O
O
OH
OH O
OH
6864 ()-Epicatechin-3-O-gallate
H
O
O
Galloylepicatechin C22H18O10 (442.38). mp 253C. Pharm: Inhibits cancer cell

invasion (MM1 cells, in vitro, 10g/mL, InRt = 59.9%)[4329]; bone marrow cell
proliferation promotor (100mg/mL, stimulates formation of myeloid colonies) [5390].
6869 6-O-Epiacetylscandoside
Source: CHA YE Camellia sinensis [Syn. Thea sinensis], DA HUANG Rheum
officinale, HEI ZI LI GUO JI SHENG Scurrura atropurpurea, ZHANG YE DA
MeOH). Source: MA LAI BAN DAO RAN MU SHU Saprosma scortechinii
HUANG Rheum palmatum, TANG GU TE DA HUANG Rheum tanguticum, TAO
(stem and leaf). Ref: 4219.
GEN Prunus persica. Ref: 2, 6, 660, 4329, 5390.
OH
HO
OH
O
OH
HO
HO
OH
OH
OH
OH
OH
OH
OH
6865 ()-Epicatechin-5-O--D-glucopyranosyl-3-benzoate
6870 8'-Epi-cleomiscosin A
C28H28O12 (556.53). Bright pink needles (CH2Cl2:MeOH =1:1), mp 191~192C;
C20H18O8 (386.36). Amorphous powder, []D25 = +15.5 (c = 0.1, C 5D5N).
[]D25 = 95 (c = 0.3, MeOH). Pharm: Antioxidant (DPPH scavenger, IC50 =
Pharm: Tyrosinase inhibitor (IC50 = (1.331.06)mol/L, control Kojic acid,
[3028]
25g/mL)
. Source: NAN SHE TENG Celastrus orbiculatus [Syn. Celastrus
articulatus] (aerial parts: yield = 0.0026%dw). Ref: 3028.
IC50 = (16.670.52)mol/L, L-Mimosine, IC 50 = (3.680.02)mol/L) .

Source: A FU HAN DU JUAN HUA Rhododendron collettianum. Ref: 2544.
OH
HO
OH
O
HO
HO
HO
OO
OH
O
O
O
O
HO
OH
251
6871 6''-Epi-calyflorenone B
6875 4-Epicurcumenol
C36H38O11 (646.70). Pale amorphous solid, mp 110~112C (Et2Opetrol),
C15H22O2 (234.34). Colorless oil, []D26 = +120.1 (c = 1.8, CHCl3). Pharm:
[]D20 = 30.05 (c = 0.183). Source: E CHI TENG Calycopteris floribunda
NO production inhibitor (mus peritoneal macrophages, induced by LPS,
(green part). Ref: 3779.
100mol/L, InRt = (40.11.4)%, control L-NMMA, 100mol/L, InRt =

(79.20.9)%, p<0.01). Source: PING E SHU Curcuma zedoaria [Syn.
Curcuma aeruginosa]. Ref: 4150.
O
OH
OH
O
O
O
6876 Epicurzerenone
C15H18O2 (230.31). Source: PING E SHU Curcuma zedoaria [Syn. Curcuma
6872 6''-Epi-calyflorenone C
aeruginosa]. Ref: 6.
C35H36O11 (632.67). Pale amorphous solid, mp 117~119C (Et2Opetrol),

[]D20 = 21.86 (c = 0.183). Source: E CHI TENG Calycopteris floribunda
O
(green part). Ref: 3779.
O
O
6877 Epidanshenspiroketallactone
O
O
OH
C17H16O3 (268.32). Source: DAN SHEN Salvia miltiorrhiza, GAN XI SHU

WEI CAO Salvia przewalskii. Ref: 1521, 4538.
O
O
OH
O
O
6873 3-Epiconamine
C 22H36N2 (328.55). mp 95~100C. Source: ZHI XIE MU PI
Holarrhena antidysenterica. Ref: 6.

6878 16-Epideacetylakuammiline
C21H24 N2O3 (352.44). Source: HONG HUA RUI MU Kopsia fruticosa
N
H
(leaf). Ref: 3830.
H
H
O
H
HO
H2N
6874 (+)-14-Epicorynoline
[51151-82-7] C21H21NO5 (367.41). Source: ZI HUA YU DENG CAO
6879 16-Epideacetylakuammiline N(4)-oxide
Corydalis incisa. Ref: 6.
C21H24N2O4 (368.44). []D = 66 (c = 0.15, CHCl3). Source: MA LAI XI YA

O
RUI MU Kopsia griffithii. Ref: 1854.
OH
O
N
OH
O
H
O
O
N
H
252
6880 13-Epi-10-deacetylbaccatin III
6885 20-Epi-16'-decarbomethoxy-conoduramine
C29H36O10 (544.60). Source: JIANG GUO ZI SHAN Taxus baccata. Ref: 662.
C41H54N4O3 (650.91). Source: YAO YONG GOU YA HUA Ervatamia
OH O
HO
OH
OH O
N H
H
H
N
O
6881 7-Epi-9,10-deacetylbaccatin VI
N
H
OH OH
6886 1-Epidechloroacutumine
OH
C19H25NO6 (363.41). []D25 = 45 (c = 0.2, MeOH). Source: BIAN FU GE

O

O
OH
OH
O
6882 1-Epideacetylbowdensine
C17H21NO5 (319.36). Source: GUAN MU WEN SHU LAN Crinum

O
macowanii (bulb). Ref: 4000.
O
O
OH
HO
6887 4-Epidehydroabietic acid

[5155-70-4] C20H28O2 (300.44). White amorphous powder. Source: JIA DI
O
H
O
FENG PI Illicium jiadifengpi (bark). Ref: 4560.
6883 1-Epideacetylbowdensine
C17H21NO5 (319.36). Source: Crinum moorei. Ref: 4952.
OH
HO
OH
O
H
O
6888 12-Epi-11-dehydroklaineanone
C20H26O6 (362.43). Colorless glassy resin, []D25 = 11.2 (c = 0.1, MeOH).
Pharm: Plant growth inhibitor (Cucumber seedling, root growth, IC50 >
6884 7-Epi-10-deacetyltaxuyunnanine A
200mol/L, shoot growth, IC50 > 200mol/L; Rice seedling, root growth, IC50
7-Epi-10-deacetyltaxol; Taxuspinanane E C44H55NO13 (805.93). []D = 22.9
> 200mol/L, shoot growth, IC50 > 200mol/L)[5215]. Source: CHANG YE
(MeOH). Source: YUN NAN HONG DOU SHAN Taxus yunnanensis, ZI
KUAN MU Eurycoma longifolia (leaf). Ref: 5215.
SHAN Taxus cuspidata. Ref: 662.

OH
OH O
O
N
O
OH
OH
O
O
H
O
OH
OH O
H
O
O
253
6889 3-Epidehydrotumulosic acid
6894 5-Epidilatanolide A
C31H48O4 (484.73). Pharm: Antineoplastic (EBV-EA induced by TPA, mol
C15H22O2 (234.34). Colorless solid, mp 106~107C, []D = 21.5 (c = 0.40,
ratio/TPA = 1000, relative percentage of EBV-EA = 0% (positive control
CHCl3). Source: BA XI ER YE TAI Frullania brasiliensis. Ref: 1981.
value 32pmol, 20ng TPA =100%), viability of Raji cells = 70%; reference
compound -Carotene, relative percentage = 8.6%). Source: FU LING Poria
cocos (sclerotium: yield = 0.00029%dw). Ref: 4616.
O
HO
6895 5-Epidilatanolide B
OH
C15H20O2 (232.33). Colorless oil, []D = +50.8 (c = 0.27, CHCl3). Source: BA

XI ER YE TAI Frullania brasiliensis. Ref: 1981.
HO
6890 17-Epi-12-dehydroxyheudebolin
C32H40O9 (568.67). White crystals (hexaneEtOAc), mp 122~124C, []D20 =

190.1 (c = 1.3, CHCl3). Source: Turreanthus africanus (seed). Ref: 3884.
6896 1-Epi-dioncophylline B
C23H25NO3 (363.46). Pharm: Antimalarial (Plasmodium falciparum K1, IC50
O H
= 155ng/mL, NF54, IC 50 = 273ng/mL, MIC > 200g/mL). Source:

SAN YE MU Triphyophyllum peltatum (leaf). Ref: 3962.
O
O
O
O
O
NH
O
OH
OH
6891 Epideoxyarteannuin B
Deoxyisoartemisinin B C15H20O2 (232.33). Source: HUANG HUA HAO
Artemisia annua. Ref: 660, 5224.

6897 9,13-Epi-dioxiabiet-8(14)-en-18-ol
C20H32O3 (320.48). Colorless oil, []D = 51.8 (c = 1.0, CHCl3). Pharm:

O
5g/mL; T98G, IC50 > 5g/mL; SKBR3, IC50 > 5g/mL). Source: BEI FEI
XUE SONG Cedrus atlantica (cone). Ref: 5248.
6892 4-Epi-4-deoxyphorbol 12,13-bis(isobutyrate)
O
O
[250258-02-7] C28H40O7 (488.63). Oil, []D = +3 (c = 0.7, CHCl3). Source:

DUN YE DA JI Euphorbia obtusifolia var. obtusifolia. Ref: 2365.
O
O
OH
O
H
6898 5,9-Epidioxy-8,14-epoxy-(22E)-ergosta-6,22-dien-3-ol
OH
CHCl3). Source: HOU SHU SHAN GU Panellus serotinus, Pleurotus eryngii.

Ref: 4183.
O H
OH
6893 20-Epi-19,20-dihydro-decarbomethoxy vobasine

H
C19H24N2O (296.42). Source: YAO YONG GOU YA HUA Ervatamia

O
N
H
HO
H
254
6899 5,9-Epidioxy-(22E)-ergosta-7,22-diene-3,6-diol
6903 5,8-Epidioxyergosta-6,9(11),22-trien-3-ol
C28H44O4 (444.66). Amorphous powder, []D23 = 8.8 (c = 0.1, CHCl3).
C28H42O3 (426.65). Source: JIA LIAN QIAO Duranta repens (whole herb).
Source: HOU SHU SHAN GU Panellus serotinus. Ref: 3526.
Ref: 4179.
O
HO
HO
OH
6900 5,9-Epidioxy-(22E)-ergosta-7,22-diene-3,6-diol
6904 5,8-Epidioxyergosta-6,9(11),22-trien-3-ol
9(11)-Dehydroergosterol peroxide C28H42O3 (426.65). White needles (EtOAc).
Source: ZI DING XIANG MO Lepista nuda, HOU SHU SHAN GU Panellus
Source: AI LI SI DUO KONG JUN Polyporus ellisii, JIA LIAN QIAO
serotinus, SONG XUN Tricholoma matsutake [Syn. Armillaria matsutake],
Duranta repens (whole herb). Ref: 2435, 4179.
Pleurotus eryngii. Ref: 3526, 4183.
O
HO
HO
OH
6901 5,8-Epidioxyergosta-6,22-dien-3-yl stearate

C 46 H 78 O 4 (695.18). White amorphous powder, [] D
25
= +13 (c = 0.2,
6905 5,9-Epidioxy-3-hydroxy-(22E)-ergosta-7,22-dien-6-one
C28H42O4 (442.64). Source: Pleurotus eryngii. Ref: 4183.
CH 2 Cl 2 ). Pharm: Antitubercular (Mycobacterium tuberculosis growth

inhibitor, MIC = 4g/mL). Source: Ruprechtia triflora (aerial parts).
Ref: 5416.
H
HO
O
O
6906 5,8-Epidioxy-24(R)-methylcholesta-6,22-diene-3-ol
Ergosterol peroxide C28H44O3 (428.66). Colorless needles, mp 180~182C,
6902 (22E,24R)-5,8-Epidioxyergosta-6,9,22-triene-3-ol 3-O--D-
[]D = 33.3 (c = 0.3, CHCl3). Pharm: DNA Topoisomerase I Inhibitor
glucopyranoside
(inhibits the relaxation of supercoiled DNA (pBR322) induced by DNA
topoisomerase I); cytotoxic (marginal activity, selective cytotoxic activity
Source: Chlorophyllum molybdites. Ref: 4112.
against hmn colon tumor cells, Colon205 ED50 = 8.56g/mL). Source:

Penicillium oxalicum. Ref: 5046.
O
O
OO
HO
OH
OH
HO
O
OH
255
6907 5,8-Epidioxy-24(R)-methylcholesta-6,22-dien-3-D-glucopy-
6912 ()-10-Epi--eudesmol
ranoside
[140447-22-9] C34H54O8 (590.80). Pharm: Antiproliferative (K562, Jurkat,

WM-1341, HL-60 and RPMI-8226 tumor cell lines, 10g/mL, greater inhibitor
by 10% to 40% than 5, 8-Epidioxy-24(R)-methylcholesta-6, 22-dien-3-ol).
Source: DONG CHONG XIA CAO Cordyceps sinensis. Ref: 2322.
OH
H
6913 10-Epieupatoroxin
O
O
[20071-54-9] C20H24O8 (392.41). mp 230~232C, []D26 = 109 (c = 0.33,
OO
HO
methanol). Pharm: Cytotoxic (KB, ED50 = 2.6g/mL). Source: YUAN YE ZE
OH
OH
LAN Eupatorium rotundifolium. Ref: 661.

OH
OH
6908 Epi-eriocalyxin A
C20H24O5 (344.41). Source: MAO E XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.
O
HO
O
O
6909 5-Epi-eudesm-4(15)-ene-1,6-diol
6914 3-Epifagomine
C15H26O2 (238.37). Colorless monoclinic crystals (petroleum etherEtOAc),
C6H13NO3 (147.18). Pharm: Lactace inhibitor (isomaltose enzyme
[]D20 = 88 (c = 0.6, CHCl3); white powder, []D20 = +36.5 (c = 0.32, CHCl3).
inhibitor)[2513]. Source: SANG BAI PI Morus alba. Ref: 2513.
Pharm: Anti-HIV (MT-2 cell infected by HIV-IIIB virus, 10g/mL, weak

activity)[4786]; anti-HIV-1 (HIV-1 replication inhibitor in vitro, HOG.R5, IC50 =
17.4g/mL (73.1mol/L), cytotoxic, 20g/mL, inactive)[4688]. Source: DIE DA
LAO Litsea verticillata (leaf and twig: yield = 0.00011%dw), ZHONG JIAN
JIN JI ER Caragana intermedia (aerial parts). Ref: 4688, 4786.
H
N
HO
HO
OH H
OH
6915 6-Epiforesticine
H
C24H39NO6 (437.58). White amorphous powder. Source: GUA YE WU TOU
OH
Aconitum hemsleyanum. Ref: 2208.

6910 7-Epieudesm-4(15)-ene-1,6-diol
C15H26O2 (238.37). White powder, []D20 = 35.3 (c = 0.05, CHCl3). Pharm:
Anti-HIV-1 inactive (in vitro, HOG.R5)[4688]. Source: DIE DA LAO Litsea

O
verticillata (leaf and twig: yield = 0.00015%dw). Ref: 4688.

OH
N
H
O
OH
OH
OH
6911 7-Epi-eudesm-4(15)-ene-1,6-diol
20
C15H26O2 (238.37). White powder, []D = 16.0 (c = 0.03, CHCl3). Pharm:
6916 3-Epifortuneine
C20H25NO3 (327.43). Source: SAN JIAN SHAN Cephalotaxus fortunei. Ref: 2.
Anti-HIV-1 inactive (in vitro, HOG.R5). Source: DIE DA LAO Litsea

verticillata (leaf and twig: yield = 0.00008%dw). Ref: 4688.
O
OH
OH
OH
256
6917 2''-Epiframeroside
6921 L-Epigallocatechin
C27H38O15 (602.59). Colorless amorphous powder, []D24 = 116 (c = 0.22,
()-Epigallocatechin [970-74-1] C15H14O7 (306.27). mp 227C. Pharm:
MeOH). Source: A FU HAN DING XIANG Syringa afghanica. Ref: 2006.
Angiotensin I-converting enzyme inhibitor; platelet aggregation inhibitor (rbt,
OH
O
H
stronger than aspirin, weaker than persantin); antibacterial (Bacillus typhosus,

OO
O
OH
Bacillus paratyphosus, Staphylococcus hemolyticus flavus, Staphylococcus

aureus); cytotoxic (HeLa, in vitro); antispasmodic (rat); lipoxidase inhibitor
(soy, IC50 = 10~20mol/L); inhibits cancer cell invasion (MM1 cells, in vitro,
O
HO
OO
10g/mL, InRt = 27.8%)[4329]; antioxidant (DPPH free radical scavenger, for

40mol/L DPPH radical, SC50 = 2.5mol/L)[4378]; bone marrow cell
proliferation promotor (100mg/mL, stimulates formation of myeloid
OH
colonies)[5390]; inhibits degranulation and release of -hexosaminidase
OH
OH
(RBL-2H3 cells, 100mol/L, InRt = (12.64.2)%, control Curcumin,
6918 Epifriedelanol
100mol/L, InRt = (62.61.0)%, did not affect the enzyme activity of
Friedelan-3-ol; Friedelinol [16844-71-6] C30H52O (428.75). Colorless
-hexosaminidase)[4163]. Source: A LA BO JIAO JIN HE HUAN Acacia
acicular crystals, mp 283.5~285.0C; mp 263~265C. Pharm: NFAT
nilotica, AN MO LE Phyllanthus emblica (branch and leaf)[3094], CHA YE
transcription factor inhibitor inactive (IC50 > 50mol/L, positive control
Camellia sinensis [Syn. Thea sinensis], KUN MING SHAN HAI TANG
Cyclosporin A, IC50 = (0.310.01)mol/L)[4511]. Source: CHAO XIAN LUO
Tripterygium hypoglaucum, SUO LA MU Salacia prinoides [Syn. Salacia
WAN Gymnaster koraiensis (leaf), DONG FENG CAI Doellingeria scaber
chinensis] (stem), YANG MEI SHU PI Myrica rubra (bark: yield =
[Syn. Aster scaber], DUO SUI SHI KE YE Lithocarpus polystachyus, GUI
0.0066%)[4163]. Ref: 6, 612, 1564, 1565, 1566, 1567, 1568, 1569, 3094, 4163,
JIAN YU Euonymus alatus, HUO XIANG Agastache rugosus, HUO YANG
4329, 4378, 5375, 5390.
LE Euphorbia antiquorum, KU DI DAN Elephantopus scaber, KU HAO

Conyza blinii, LIANG YE YAN DOU TENG Millettia nitida, LONG YAN
OH
YE Euphoria longan [Syn. Dimocarpus longan], NAN ZHU ZI Vaccinium

bracteatum, QIU FENG MU Bischofia javanica [Syn. Bischofia trifoliata],
TIAO JING CAO Euonymus japonicus, XI YUAN TENG Pericampylus
OH
HO
glaucus, XUAN FU HUA Inula britannica, YU DAI GEN Pedilanthus
OH
OH
tithymaloides, ZI WAN Aster tataricus. Ref: 6, 505, 596, 660, 4511.
OH
6922 Epigallocatechin-(48)-epicatechin-3-O-gallate ester

H
C37H30O17 (746.64). Pharm: Tanning agent. Source: CHA YE Camellia

sinensis [Syn. Thea sinensis]. Ref: 658.
HO
OH
6919 Epifriedelinol acetate

C32H54O2 (470.79). mp 282~285C. Source: QIU FENG MU Bischofia
javanica [Syn. Bischofia trifoliata], YU DAI GEN Pedilanthus tithymaloides.
OH
HO
Ref: 6.
OH
OH
OH
HO
OH
OH
O
OH
OH
OH
OH
6920 2-Epigalanthamine
[1668-85-5] C17H21NO3 (287.36). mp 190C. Source: SHI SUAN Lycoris
radiata [Syn. Amaryllis radiata]. Ref: 6.
6923 Epigallocatechin 3-gallate (EGCG)

()-Epigallocatechin-3-O-gallate [989-51-5] C22H18O11 (458.38). mp
OH
215~216C; []D25 = 121.2 (c = 0.99, acetone). Pharm: Special spicery of tea;

inhibits cancer cell invasion (MM1 cells, in vitro, 10g/mL, InRt = 72.8%,
O
5g/mL, InRt = 59.7%)[4329]; bone marrow cell proliferation promotor

(100mg/mL, stimulates formation of myeloid colonies) [5390]; 5-reductase
inhibitor inactive (IC50 > 1mmol/L; control Finasteride, IC 50 =
(0.380.06)mol/L; -Linolenic acid, IC50 = (160.324.6)mol/L)[5398];
257
inhibits cell proliferation of PBMC (activated by phytohemagglutinin (PHA),
6926 Epigomisin O
IC50 = 28.9mol/L, inhibitory mechanism may involve the blocking of IL-2
[73036-31-4] C23H28O7 (416.48). Source: WU WEI ZI Schisandra chinensis. Ref: 2.
and IFN- production)[4100]; TNF- release inhibitor (BALB/3T3 cells,

okadaic acid-stimulated, mean IC50 = 26mol/L)[4416]; anti-inflammatory
(NF-B pathway)[4415]; anti-inflammatory (NO production inhibitor)[4415];
anti-inflammatory (modulator of cytokine network: leukocyte elastase
MMP-2/9 inhibitor)[4416]; antioxidant (DPPH scavenger, IC50 =
(1.130.08)mol/L)[3848]; antioxidant (hydroxyl radical scavenger, IC50 =
O
O
O
O
OH
0.43mol/L)[4499]; antioxidant (superoxide anion radical scavenger, IC50 =

0.53mol/L)[4499]. Source: CHA YE Camellia sinensis [Syn. Thea sinensis],
HEI ZI LI GUO JI SHENG Scurrura atropurpurea, MEI ZHOU JIN LV MEI
Hamamelis virginiana, YOU GAN YE Phyllanthus emblica (branch and leaf),
YANG PU TAO YE Syzygium samarangense, MAO GUO QI Acer nikoense,
6927 8-Epi-grandifloric acid

Source: TAI GUO SHAN QIAN NIU Thunbergia laurifolia. Ref: 1968.
H
MAO YANG MEI Myrica esculent, YE WU TONG Mallotus japonicus. Ref:

6, 658, 1521, 3848, 4100, 4205, 4329, 4415, 4416, 4499, 5390, 5398.
HO
O
O
OH
H
HO
OH
OH
O
OH
OH
HO
O
OH
OH
6928 Epiguaipyridine
OH
OH
Guaipyridine [41447-48-7] C15H21N (215.34). Source: GUANG HUO

XIANG Pogostemon cablin [Syn. Mentha cablin]. Ref: 2, 6, 660.
OH
6924 ()-Epigallocatechin 4-(2-hydroxyethyl)thio ether

C17H18O8S (382.39). Source: XIAO GUO YE JIAO Musa acuminata (fruit).
Ref: 3913.
6929 4-Epihenryine
OH
Henryine A; Amethystoidin A C20H28O5 (348.44). mp 264~267C, []D25 = +30.8
OH
O
HO
(c = 4.5, C5H5N). Source: E XI XIANG CHA CAI Isodon henryi. Ref: 4067.
O
OH
OH
OH
OH
O
OH
OH
HO
6930 ()-Epihernandulcin
6925 Epigeoside
Catechin-3-O--L-rhamnopyranosyl-(14)--D-glucopyranosyl-(16)--D-
C15H24O2 (236.36). Source: TIAN SHE CAO Lippia dulcis (aerial parts). Ref: 4508.
O
glucopyranoside C33H44O20 (760.71). Colorless powder, mp 165~168C,
OH
20
[]D = 32.5 (c = 1.05, methanol). Source: SI MAO TENG Epigynum
auritum. Ref: 208.
6931 Epiheteroconessine
OH
OH
HO
[In DNP] C25H44N2 (372.64). mp 148~150C. Source: ZHI XIE MU PI

Holarrhena antidysenterica. Ref: 6.
H
OH
OO
HO
OH
OH
OO
OH OH
OH
OH
OH
OH
H
N
258
6932 ()8,8'R-Epi-holostylone
6936 11-Epi-23-hydroxytoonacilide
(7'R,8S,8'R)-8,8'-Dimethyl-4-hydroxy-3',4',5-trimethoxy-2,7'-cyclolignan-7-o
C31H38O11 (586.64). White crystals, mp 139~142C. Source: XIAO YE DU
ne C21H24O5 (356.42). Amorphous yellow solid, []D25 = 171.6 (c = 0.32,
LIAN Turraea parvifolia. Ref: 2052.
CHCl3). Source: Holostylis reniformis (root). Ref: 3784.

OH
O
O
O
O
HO
O
O
6937 4-Epiisocembrol
6933 ()8,8'S-Epi-holostylone
C20H34O (290.49). Source: HAI SONG ZI Pinus koraiensis. Ref: 6.
(7'R,8S,8'S)-8,8'-Dimethyl-4-hydroxy-3',4',5-trimethoxy-2,7'-cyclolignan-7-on
e C21H24O5 (356.42). Yellow crystals, mp 169.0~172.0C, []D25 = 40.6 (c =
OH

O
O
HO
6938 3-Epi-isomasticadienolalic acid

C30H46O5 (486.70). []D25 = +23.6 (c = 0.5, CHCl3). Pharm:
O
Anti-inflammatory (chronic inflammation model, in the form of eczema,
provoked by repeated administration of TPA to the ears of mouse, swelling

reduction = 39%, control Dexamethasone, swelling reduction = 85%;
6934 7-Epi-19-hydroxybaccatin III

C31H38O12 (602.64). Source: HONG DOU SHAN Taxus chinensis. Ref: 662.
reduces leukocyte infiltration, measured as tissue peroxidase activity, InRt =

57%, Dexamethasone, InRt = 55%); toxic (rat peritoneal
polymorphonuclear leukocytes, 100mol/L). Source: ROU MAO XIAO RU
XIANG Schinus molle (fruit). Ref: 5459.
O
OH
OH
O O
OH
O
HO
OH O
OH
O
O
O
HO
6935 11-Epi-21-hydroxytoonacilide
6939 Epi-kansenone
C31H38O11 (586.64). White crystals, mp 124~126C. Source: XIAO YE DU
Tirucalla-8,24-diene-3-ol-7-one C30H48O2 (440.72). Colorless gum, []D23
LIAN Turraea parvifolia. Ref: 2052.
= 10.2 (c = 0.43, MeOH). Pharm: Cell division arrester (cultured

individual Xenopus laevis cells at blastular stage, 10g/mL, >50% cleavage
arrest). Source: GAN SUI Euphorbia kansui (dried root: yield = 0.00008%).
Ref: 4690.
O
O
O
O
OH
HO
O
259
6940 3-Epikatonic acid
6945 15-Epileoheteronone E
[76035-62-6] C30H48O3 (456.72). Colorless acicular crystals, mp 284~286C
C22H34O6 (394.51). White amorphous powder. Source: YI MU CAO Leonurus
(MeOH). Pharm: Spermaticidal (mus, 0.125mg/mL). Source: LEI GONG
heterophyllus [Syn. Leonurus artemisia] (aerial parts). Ref: 4534.
TENG Tripterygium wilfordii. Ref: 2, 60, 670, 1572.
OH
O
OH
O
H
H
HO
6946 15-Epileopersin B
6941 16-Epikopsinine
persicus, YI MU CAO Leonurus heterophyllus [Syn. Leonurus artemisia]
C21H26N2O2 (338.45). Source: HONG HUA RUI MU Kopsia fruticosa (leaf).
(aerial parts). Ref: 2499, 4534.

OH
Ref: 3830.
N
O
N
H
O
O
6942 4-Epi-larreatricin
6947 15-Epileopersin C
8'-Epi-larreatricin C18H20O3 (284.36). Pharm: Antioxidant (Takamatsu DCFH
C20H32O5 (352.48). Oil liquid. Source: YI MU CAO Leonurus heterophyllus
method, myelomonocytic HL-60 cells, IC50 = (18.02.5)g/mL; control
[Syn. Leonurus artemisia] (aerial parts), BO SI YI MU CAO Leonurus
NDGA, IC50 = (0.70.3)g/mL, Vitamin C, IC50 = (1.90.7)g/mL, Trolox,
persicus. Ref: 4534, 2499.
IC50 = (1.40.5)g/mL)[3850]; cytotoxic (XTT assay, HL-60 cells, IC50 >

50.0g/mL; control NDGA, IC50 = (2.60.2)g/mL, Vitamin C, IC50 >
OH
10.0g/mL, Trolox, IC50 > 10.0g/mL)[3850]. Source: SAN CHI LA RUI A
Larrea tridentata (leaf). Ref: 1521, 3850.

O
H
OH
HO
OH
O
6943 15-Epileoheteronone B
6948 15-Epi-leopersin J
C20H32O5 (352.48). Oil liquid. Source: BO SI YI MU CAO Leonurus persicus.

Ref: 2499.
OH
OH
O
O
OH
6944 15-Epileoheteronone D
O
6949 15-Epi-leopersin O
Ref: 2499.
OH
OH
O
O
HO
H
OH
O
260
6950 15-Epi-leopersin Q
6955 Epilupinine
Isolupinine [486-71-5] C10H19NO (169.27). mp 77~78C. Source: Lupinus
Ref: 2499.
varius. Ref: 1521.

OH
OH
HO
6956 12-Epilycodoline
OH
C16H25NO2 (263.38). []D25 = 44 (MeOH). Source: DONG BEI SHI SHAN
6951 Epilippidulcine A
C15H24O3 (252.36). Colorless oil, []D31 = 118.4 (c = 0.5, CHCl3). Source:
Huperzia miyoshiana. Ref: 5412.
TIAN SHE CAO Lippia dulcis (aerial parts). Ref: 4508.

H
O
OH
OH
OH
6952 8-Epiloganic acid
6957 ()-4-Epi-maaliol
C15H26O (222.37). Colorless oil. Source: TIE JIAO JUE YU TAI Plagiochila
parts), GAN DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa f.
asplenioides (essential oil). Ref: 5257.
huechingensis], ROU CONG RONG Cistanche deserticola. Ref: 2, 502, 628,

3954.
HO
O
OH
H
HO
6958 Epi-maoecrystal P
H
OO
HO
OH

MAO E XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.
OH
OH
O
6953 8-Epiloganin
racemosa] (leaf, flower and twig: yield = 0.0003%dw)[4723], TIAN SHE CAO
Lippia dulcis (aerial parts). Ref: 4508, 4723.

O
C17H26O10 (390.39). Source: JI ZI MU Sinoadina Racemosa [Syn. Adina
O
OH
OH
6959 Epimedin A
4'-Methoxy-5-hydroxy-8-3,3-dimethylallyl-flavone-3-glucosyl-(12)rhamno
HO
O
H
O
HO
side-7-glucoside [110623-72-8] C39H50O20 (838.82). Source: CHAO XIAN

YIN YANG HUO Epimedium koreanum (aerial parts: content = 0.345%[5508]),
YIN YANG HUO Epimedium brevicornum. Ref: 2,660, 1521, 5508.
OH
OH
OH
6954 3-Epilupeol
C30H50O (426.73). Pharm: Cytotoxic (hmn fibrosarcoma cells HT1080, ED50

> 100g/mL; control Adriamycin, ED50 = 0.1g/mL)[4437]. Source: LIE WEI
LIE LAN Bursera graveolens (stem), RI BEN HUANG BAI Phellodendron
japonicum (leaf). Ref: 4437, 4502.
HO
OO
OH
OH
OH
OH
OH
HO
H
H
HO
OH O
O
OH
OH
OH
261
6960 Epimedin B
6962 Epimedokoreanoside I
4'-Methoxy-5-hydroxy-8-3,3-dimethyl allylflavone-3-xyloxyl-(12)rham-
[130756-11-5] C44H56O22 (936.92). Source: YIN YANG HUO Epimedium
noside-7-glucoside [110623-73-9] C38H48O19 (808.79). Source: CHAO XIAN
brevicornum. Ref: 2.
YIN YANG HUO Epimedium koreanum (aerial parts: content scope =

0.39%1.24%, mean content = 0.82%[5508]), CHUAN E YIN YANG HUO
Epimedium fargesii, JIAN YE YIN YANG HUO Epimedium sagittatum

HO
(aerial parts: mean content of 3 origins = 0.552%)[5508], ROU MAO YIN

YANG HUO Epimedium pubescens (aerial parts: content = 0.739%)
[5508]
WU
SHAN YIN YANG HUO Epimedium wushanense (aerial parts: mean content
of 2 origins = 0.349%)
[5508]
OO
OH
OH
O
OH
, YIN YANG HUO Epimedium brevicornum (aerial
OH
O
OH
O
parts: mean content of 2 origins = 1.09%[5508]), Epimedium spp. Ref: 2, 567,
660, 1521, 5508.
OH
OH
OH
O
HO
OO
6963 Epimedokoreanoside II
OH
OH
OH
OH
OH
brevicornum. Ref: 2.
O
O
OH
OO
OH
OH
HO
OH
O
OH
6961 Epimedin C
O
OH
O
4'-Methoxy-5-hydroxy-8-3,3-dimethyl allylflavone-3-rhamnosyl-(12)rham-
HO
noside-7-glucoside [110642-44-9] C39H50O19 (822.82). Yellow powder, mp

240~245C, soluble in methanol. Pharm: Immunoenhancer (enhances
OH
OH
multiplication of lymphocyte, recovers to produce interleukin-2). Source:
O
O
OH
CHAO XIAN YIN YANG HUO Epimedium koreanum (aerial parts: content
scope = 0.19%0.89%, mean content = 0.61%[5508]), CHUAN DIAN YIN
6964 Epimedoside C
YANG HUO Epimedium davidii, CHUAN E YIN YANG HUO Epimedium
fargesii, CU MAO YIN YANG HUO Epimedium acuminatum (aerial parts:
brevicornum. Ref: 2, 112.
content = 2.18%[5508]), JIAN YE YIN YANG HUO Epimedium sagittatum

(aerial parts: content scope = 0.39%1.60%, mean content = 1.09%)[5508],
QIAN LING YIN YANG HUO Epimedium leptorrhizum (aerial parts: content
OH
= 1.56%)[5508], ROU MAO YIN YANG HUO Epimedium pubescens (aerial

parts: content scope = 1.14%1.36%, mean content = 1.25%)[5508], TIAN
PING SHAN YIN YANG HUO Epimedium myrianthum (aerial parts: content
= 2.22%)[5508], WU SHAN YIN YANG HUO Epimedium wushanense (aerial
O
O
HO
OH
OH
OH
OH
OH
parts: content scope = 1.63%3.11%, mean content = 2.37%[5508]), YIN

YANG HUO Epimedium brevicornum (aerial parts: mean content of 2 origins
= 1.141%[5508]). Ref: 2, 114, 540, 567, 623, 624, 660, 1521, 1784, 5508.
6965 Epimeredinoside A
2-(3-Methoxy-4-hydroxy) phenyl ethanol 1-O--L-[(13)-rhamnopyranosyl6-O-feruloyl] glucoside C31H40O15 (652.66). Yellowish amorphous powder,
O
HO
OO
mp 140~141C (MeOH). Source: GUANG FANG FENG Anisomeles indica

[Syn. Epimeredi indica] (whole herb). Ref: 4592.
OH
OH
OH
OH
OH
OH
OH OH O
O
OO
O
OH
O OH
O
OH OH
OH
OH OH
O
OH
262
6966 23-Epimeric 3,23-dihydroxycycloart-24-en-26-oic acid

C30H48O4 (472.71). Shining crystals (CHCl3MeOH), mp 240~242C. Source:
H
O
MANG GUO Mangifera indica. Ref: 1868.

O
OH
OH
O
OH
6972 22-Epimolvizarin
C35H62O7 (594.88). White solid, mp 104~105C, []D = +19.3 (c = 0.064,
HO
MeOH). Source: FAN LI ZHI Annona squamosa. Ref: 886.
6967 12-Epi-methyl-barbascoate
OH
C19H22O5 (330.38). Source: WU LU BA DOU Croton urucurana. Ref: 4552.
6973 17-Epinaucleidinal
O
[77513-46-3] C20H20N2O3 (336.39). []D = +97.7 (c = 0.085, EtOH). Pharm:

Antibacterial (in vitro: Staphylococcus aureus, Bacillus subtilis, Bacillus coli,
Bacillus diphtheriae, Streptococcus sp., Streptobacillus sp., Salmonella sp.,
6968 Epi-6-methylcryptoacetalide
C19H24O3 (300.40). Source: AI JI SHU WEI CAO Salvia aegyptiaca. Ref: 1919.
O
OH
OH
Bacillus proteus, Bacillus lactis, Klebsiella pneumoniae); antileishmanial;

antifungal (Aspergillus niger). Source: KUAN YE WU TAN Nauclea latifolia.
Ref: 2178.
O
O
N
H H
6969 3-Epimethylschelhammericine B
C20H27NO3 (329.44). Source: SAN JIAN SHAN Cephalotaxus fortunei. Ref: 2, 27.
O
6974 3-Epineoruscogenin
Spirost-5,25(27)-dien-1,3r-diol C27H40O4 (428.62). Colorless prisms, []D24 =

61.7 (c = 1.67, CHCl3). Source: KAI KOU JIAN Tupistra chinensis
6970 3-Epi-O-Methyl-scilliphaeosidin
O
C25H34O5 (414.55). Amorphous powder. []D28 = +49.9 (c = 0.66, MeOH).
OH
Source: HAI CONG Urginea maritima (bulb). Ref: 3513.
O
O
HO
OH
6975 Epinodosin
C20H26O6 (362.43). mp 245~248C, []D27 = 200 (c = 0.027, C5H5N).
H
H
OH
Source: LU SHAN XIANG CHA CAI Isodon rubescens var. lushanensis

(leaf), MAO YE XIANG CHA CAI Isodon japonica [Syn. Rabdosia
O
H
japonica]. Ref: 4067, 4067, 4353.
6971 12a-Epimillettosin
O
C22H18O7 (394.38). Pharm: Antimalarial (antiplasmodial, chloroquine-resistant W2 strain of Plasmodium falciparum, IC50 = 22.2mol/L, control
Chloroquine, IC50 = 0.094mol/L, control Quinine, IC50 = 0.209mol/L;

chloroquine-sensitive D6 strain of Plasmodium falciparum, IC50 =
19.4mol/L, control Chloroquine, IC50 = 0.009mol/L, control Quinine, IC50
= 0.044mol/L). Source: Millettia usaramensis ssp. usaramensis. Ref: 3454.
O
H
OH
OH
263
6976 Epinodosinol
6981 3-Epi-oleanolic acid-28-O--L-rhamnopyranosyl-(14)--D-glu-
C20H28O6 (364.44). mp 236~238C. Source: MAO YE XIANG CHA CAI
copyranosyl-(16)--D-glucopyranoside
Isodon japonica [Syn. Rabdosia japonica]. Ref: 4067.
3-Hydroxyolean-12-en-28-oic acid O--L-rhamnopyranosyl-(14)O--D-glucopyranosyl-(16)--D-glucopyranosyl ester C48H78O17
(927.15). White powder, mp 207~209C, []D20 = 15 (c = 0.4, methanol).
OH
Source: DONG BEI CI REN SHEN Oplopanax elatus, SAN YE MU

TONG Akebia trifoliata (stem). Ref: 370, 660, 4545.
H
O
H
OH
OH
H
H
HO
6977 4-Epi-11-nor-aristola-1(10),11-diene
C14H20 (188.32). Colorless oil. Source: RI BEN BIAN TAI Bazzania japonica.
OO
HO
OH
OH O O
Ref: 3399.
OO
OH
OH
OH
OH
OH OH
6982 Epioritin-(46)-epioritin-(46)-epioritin-4-ol
C45H44O16 (840.84). Source: Acacia galpinii (heartwood), Acacia caffra
6978 4-Epi-11-nor-aristola-9,11-diene
OH
OH
Ref: 3399.
HO
HO
OH
OH
OH
HO
OH
HO
OH HO
6979 4-Epi-11-nor-aristola-1,9,11-triene
Ref: 3399.
OH
6983 Epioritin-(46)-epioritin-(46)-epioritin-4-ol nona-O-methylether tetra-acetate

C62H64O20 (1129.19). Source: Acacia galpinii (heartwood). Ref: 3753.
6980 3-Epioleanolic acid
[25499-90-5] C30H48O3 (456.72). Pharm: Gastroprotective (30 mg/kg, Gp =
(88.85.1)%; control Carbenoxolone, Gp = (88.45.4)%, p<0.05)
[5461]
. Source:
SHOU LIAN LIANG YI MU Amphipterygium adstringens (stem cortex), SU
O
O
O
O
O
O
O
O
O
O
O
OH
H
H
HE XIANG Liquidambar orientalis. Ref: 6, 5461.
HO
O
O
264
6984 Epioritin-4-ol-(66)-epioritin-4-ol
6988 13-Epi-2-oxo-kolavelool
C20H32O2 (304.48). Colorless amorphous solid, mp 158~159C (hexane),
[]D25 = 25.0 (c = 0.10, CHCl3). Source: BA XI MA DOU LING

Aristolochia chamissonis. Ref: 1904.
OH
OH
HO
OH
OH
HO
OH
O
OH
OH
OH
HO
6985 Epioritin-4-ol-(66)-epioritin-4-ol hepta-O-methylether

triacetate
6989 Epipachysamine A
[2309-42-4] C26H46N2O (402.67). mp 203~205C. Source: XUE SHAN LIN

O
O
O
N
O
O
O
O
O
H
H
N
H
H
6986 Epioritin-(46)-oritin-(46)-epioritin-4-ol
6990 Epipachysamine AII

C26H46N2O (402.67). Colorless flake crystals (dichloromethaneacetone), mp
OH
OH
HO
HO
201~203C, []D25 = 17 (c = 1.24). Pharm: Antiulcerative (inhibits secretion

hydrochloric acid in gastric juice); LD50 (mus, ip) = 47.2mg/kg, CD50 (mus, ip)
= 32.5mg/kg. Source: XUE SHAN LIN Pachysandra terminalis. Ref: 941,
OH
1141, 1197, 1200.
OH
OH
HO
OH
HO
OH HO
H
H
H
OH
6987 Epioritin-(46)-oritin-(46)-epioritin-4-ol nona-O-methylether tetra-acetate

O
O
O
O
O
O
O
O
O
O
O

6991 Epipachysamine B
H
N
H
N
O
265
6992 Epipachysamine C
6997 7-Epiphlomiol
[4215-74-1] C25H46N2 (374.66). Source: XUE SHAN LIN Pachysandra
[139757-58-7] C17H26O13 (438.39). Source: MENG GU CAO SU Phlomis
terminalis. Ref: 6.
mongolica. Ref: 561.

O
OHOH
H
HO
H
H
N
HO
H
HO
OO
OH
OH
6993 Epipachysamine D
OH
6998 3-Epiphlomurin
C18H28O11 (420.42). []D21 = 22.2 (c = 0.7, MeOH). Source: JIN HUANG

CAO SU Phlomis aurea (leaf) Ref: 5093.
H
O
H
N
H
HO
OO
HO
OH
6994 Epipachysamine E
OH
OH

6999 Epiphyllic acid

C18H14O8 (358.31). Source: QIU YUAN YE TAI Jamesoniella autumnalis, XI
TAI Pellia epiphylla. Ref: 1521, 4549.

O
H
HO
H
O
H
N
H
OH
OH
HO
H
HO
6995 Epipachysamine F
OH
[5141-99-1] C23H42N2 (346.60). mp 250~253C. Source: XUE SHAN LIN

7000 (+)-Epipinoresinol
[24404-50-5] C20H22O6 (358.39). Source: DU ZHONG Eucommia ulmoides.
Ref: 2.
NH2
OH
H
H
N
O
HO
6996 Epipachysandrine A
C30H46N2O2 (466.71). mp > 295C. Source: XUE SHAN LIN Pachysandra
terminalis. Ref: 6.
7001 3-Epipomolic acid

C30H48O4 (472.71). Source: DUO SUI PO BU MU Cordia multispicata (leaf).
Ref: 4106.
HO
OH
H
N
H
H
OH
H
HO
266
7002 Epiporphyroxine
7007 Epirhododendrin
C19H19NO6 (357.37). Source: HUO XIANG YE LV RONG HAO Meconopsis
C16H24O7 (328.37). Source: MAO GUO QI Acer nikoense (stem cortex). Ref: 4304.
betonicifolia, Papaver spp. Ref: 1521.

HO
O O
OH
OH
HO
NH
H
H
O
OH
HO
7008 12-Epirockogenin
HO
O
[545-77-7] C27H44O4 (432.65). mp 218C. Source: FAN MA Agave americana,

JIAN MA Agave sisalana, TAN XIANG Santalum album. Ref: 6, 10.
7003 Epiquinidine
[572-59-8] C20H24N2O2 (324.43). mp 113C. Source: JIN JI LE Cinchona
OH
ledgeriana. Ref: 6.
H
HO
H
H
HO
H
H
7009 3-Epiruscogenin
7004 Epiquinine
(25R)-Spirost-5-en-1,3-diol C27H42O4 (430.63). White amorphous powder,
[572-60-1] C20 H24 N2O2 (324.43). Source: JIN JI LE Cinchona ledgeriana.
[]D24 = 63.8 (c = 1.28, CHCl3). Source: KAI KOU JIAN Tupistra chinensis
Ref: 6.

H
OH
H
H
HO
HO
7010 4-Epi-sandaracopimaric acid
7005 22-Epirhodeasapogenin-3-O--D-glucopyranoside
C20H30O2 (302.46). White amorphous powder. Source: JIA DI FENG PI
C33H54O9 (594.79). Source: WAN NIAN QING GEN Rohdea japonica [Syn.
Illicium jiadifengpi (bark). Ref: 4560.
Orontium japonicum]. Ref: 660.

H
O
O
OH
H
H
HO
OO
OH
7011 3-Episapeline A
OH
OH
H
O
OH
OH
7006 22-Epirhodeasapogenin-1-O--L-rhamnopyranosyl(12)--D-
OH
H
H
xylopyranoside
C38H62O12 (710.91). Source: WAN NIAN QING GEN Rohdea japonica [Syn.
Orontium japonicum]. Ref: 660.
HO
O
O
OH
OH OH
C19H22N2O2 (310.40). Acicular crystals, mp 300C (dec), []D30 = +34.7 (c = 0.085,

ethanol). Source: DIAN JI GU CHANG SHAN Alstonia yunnanensis. Ref: 42.
OH
OH O O
OH
7012 16-Episarpagine
HO
N
H H
OH
267
7013 Epi-sarsasapogenin
7017 21-Episerratenediol
Serratendiol [1449-06-5] C30H50O2 (442.73). Colorless powder, mp
CHA RUI SHU YU Dioscorea collettii. Ref: 10, 24, 660.
303~308C, mp 303-304C (MeOH), []D26 = -19.6 (c = 0.3, CHCl3). Source:

PU DI WU GONG Lycopodium cernuum (root, stem and leaf: yield =
0.0027%dw)[4633], QIAN CENG TA Huperzia serrata [Syn. Lycopodium
serratum]. Ref: 6, 109, 4633.

OH
HO
HO
7014 3-Epischelhammericine
7018 21-Episerratriol
[24204-36-2] C19H23NO3 (313.40). Source: HAI NAN CU FEI Cephalotaxus
C30H50O3 (458.73). mp 330~333C. Source: PU DI WU GONG Lycopodium
hainanensis [Syn. Cephalotaxus mannii], SAN JIAN SHAN Cephalotaxus
cernuum. Ref: 6.
OH
fortunei. Ref: 2, 27, 660.
O
O
HO
HO
7019 Epishyobunone
[39020-72-9] C15H24O (220.36). Source: BAI CHANG Acorus calamus.
7015 13-Epi-sclareol
Ref: 6.
C20H36O2 (308.51). Pharm: Antibacterial (gram-positive bacteria, showing a

bactericidal and lytic action, inhibits oxygen consumption of intact
gram-positive cells, but not with gram-negative bacteria, NADH oxidase
inhibitor, cytochrome C reductase inhibitor). Source: Pseudognaphalium
cheiranthifolium, Pseudognaphalium heterotrichium Ref: 4075.
OH
7020 15-Epi-sibiricinone D
C21H34O5 (366.5). Source: XI YE YI MU CAO Leonurus sibiricus (aerial
parts). Ref: 4744.
OH
7016 4-Episcopadulcic acid B
25
C27H34O5 (438.57). Gum, []D = +3.0 (c = 0.50, CHCl3). Pharm: Cytotoxic

(in vitro, SCL, ED50 = 37mol/L; SCL-6, ED50 = 136.9mol/L; SCL-37'6,
ED50 = 59.3mol/L; SCL-9, ED50 = 48.3mol/L; Kato3, ED50 = 124.3mol/L;
H
OH
NuGc-4, ED50 = 109.9mol/L; control Vinblastine Sulfate: SCL, ED50 =

5.9mol/L; SCL-6, ED50 = 6.1mol/L; SCL-37'6, ED50 = 5.3mol/L; SCL-9,
7021 15-Epi-sibiricinone E
ED50 = 5.3mol/L; Kato3, ED50 = 6.1mol/L; NUGC-4, ED50 = 5.3mol/L).
C21H34O5 (366.5). Source: XI YE YI MU CAO Leonurus sibiricus (aerial
Source: YE GAN CAO Scoparia dulcis (aerial parts: 0.00185%dw).
parts). Ref: 4744.
Ref: 4703.
H
O
H
O
O
O
OH
O
O
OH
268
7022 Epismilagenin
7026 Epitaxifolin
C27H44 O3 (416.65). Source: QIAN JIN TENG Stephania japonica. Ref:
C15H12O7 (304.26). Pharm: Cytotoxic (cyclooxygenase-1 inhibitor). Source:
10, 24.
PU
(2)
TAO Vitis vinifera (cell culture). Ref: 5038.
OH
OH
HO
OH
HO
OH
7023 3-epi-spathodic acid

C30H48O5 (488.71). Pharm: Quinone reductase inducer inactive (mouse
7027 7-Epitaxol
Hepa lclc7 hepatoma cells, CD > 10g/mL). Source: Coussarea brevicaulis.
[In DNP] C47H51NO14 (853.93). mp 168~171C, []D = 32.3 (MeOH).
Ref: 3434.
Pharm: Cytotoxic (KB, ED50 = 3.010-5g/mL). Source: DUAN YE HONG

DOU SHAN Taxus brevifolia. Ref: 662, 1831.
HO
H
O
OH
H
HO
O
N
O O
OH
OH
OH O
OH
H
O
O
7024 Epistephanine
[549-08-6] C37H38N2O6 (606.73). mp 202C. Pharm: Adrenergic antagonist
(blocks adrenergic nerve markedly). Source: BI XIE Dioscorea hypoglauca
[Syn. Dioscorea collettii var. hypoglauca], CHA RUI SHU YU Dioscorea
collettii, CHUAN LONG SHU YU Dioscorea nipponica, DUN YE SHU YU
Dioscorea zingiberensis, FU ZHOU SHU YU Dioscorea futschauensis, MU
FANG JI Cocculus trilobus [Syn. Cocculus sarmentosus], QIAN JIN TENG
7028 7-Epitaxuyunnanine A
C46H57NO14 (847.97). []D = 47.3 (CHCl3). Source: YUN NAN HONG
DOU SHAN Taxus yunnanensis. Ref: 662.
Stephania japonica, RU LAN Stephania hernandifolia, SHU KUI YE SHU

O
YU Dioscorea althaeoides. Ref: 6, 658, 660.
O O
O
O
OH
OH
OH O
H
O
O
O
O
7025 Epitaraxerol
7029 2-Epitripdiolide
C30H50O (426.73). Pharm: Cytotoxic inactive (A2780 ovarian cancer cell line,
C20H24O7 (376.41). Yellowish needles, mp 224~226C. Source: LEI GONG
IC50 = 18.8mg/mL)
[5379]
. Source: SHANG LU Phytolacca esculenta [Syn.
TENG Tripterygium wilfordii (root cortex). Ref: 4871.
Phytolacca acinosa] (berry), MU SHU DI SHANG BU FEN Manihot

esculenta. Ref: 4714, 5379.
O
O
HO
O
O
H
HO
OH
269
7030 Epitulipinolide
7034 5-Epi-vibsanin E
[24164-13-4] C17H22O4 (290.36). mp 91~92C, []D25 = +76 (c = 3.2,
C25H36O5 (416.56). []D21 = 34.7 (c = 0.21, CHCl3). Source: RI BEN JIA MI
chloroform). Pharm: Cytotoxic (KB, ED50 = 2.1g/mL); antineoplastic.
Viburnum awabuki (leaf). Ref: 4168.
Source: BAI CI GUO TUN CAO Ambrosia dumosa, BEI MEI E ZHANG
QIU Liriodendron tulipifera, CHA MI SEN TUN CAO Ambrosia chamissonis.
Ref: 658, 661.
O
O
O
7035 5-Epivibsanin G
C25H36O6 (432.56). Colorless amorphous solid, []D26 = +5 (c = 3.4, CHCl3).
Pharm: Cytotoxic (in vitro, NUGC-3, weak activity). Source: XIANG QI JIA
MI Viburnum odoratissimum (leaf and flower: yield = 0.00016%dw). Ref:

O
3004.
OH
O
O
7031 Epitulipinolide diepoxide

[39815-40-2] C17H22O6 (322.36). mp 214~215C (ethanolether), [] D25 =
OH
55.7 (c = 0.525, chloroform). Pharm: Cytotoxic (KB, ED50 = 0.34g/mL);

O
antineoplastic; insect antifeedant. Source: BEI MEI E ZHANG QIU
Liriodendron tulipifera. Ref: 658, 661.
7036 5-Epi-vibsanin H
C25H36O6 (432.56). []D21 = +49.2 (c = 0.41, CHCl3). Pharm: Cytotoxic (KB
cells, IC50 = 45.5mol/L)[4168]. Source: RI BEN JIA MI Viburnum awabuki
(leaf), XIANG QI JIA MI Viburnum odoratissimum (leaf and flower: yield =
0.00036%dw)[3004]. Ref: 3004, 4168.
H
O
O
OH
O
O
OH
7032 Epivernodalol
C20H24O8 (392.41). mp 132C, []D25 = +92.5 (c = 0.5, CHCl3). Pharm:
7037 5-Epi-vibsanin K
Cytotoxic (in vitro, hmn colon carcinoma cell lines HCT15, IC50 =
C25H36O7 (448.56). []D21 = +52.4 (c = 0.20, CHCl3). Source: RI BEN JIA MI
(39.31.8)mol/L, control 5-FU, IC 50 = 66mol/L; colon carcinoma HT29,
Viburnum awabuki (leaf). Ref: 4168.
IC50 = (21.90.8)mol/L, 5-FU, IC 50 = 49mol/L; breast carcinoma T47D,
IC50 = (22.50.7)mol/L, control Adriamycin, IC 50 = 0.075mol/L; cervix

carcinoma SiHa, IC50 = (43.41.8)mol/L, 5-FU, IC 50 = 0.034mol/L).
O
O
Source: Vernonia lasiopus. Ref: 5359.
C16H17NO3 (271.32). Pharm: AChE inhibitor (IC50 = (2399)mol/L, control
O OH
7038 Epivittatine
OH
OH
Galanthamine, IC50 = (1.90.2)mol/L). Source: Crinum moorei. Ref: 4952.

OH
OH
O
H
O
7039 16-Epi-voacarpine
7033 5-Epi-vibsanin C
24
C25H36O5 (416.56). []D = +38.6 (c = 0.59, CHCl3). Pharm: Cytotoxic (KB

cells, IC50 = 10.7mol/L). Source: RI BEN JIA MI Viburnum awabuki (leaf).
[114027-38-2] C21H24N2O4 (368.44). mp 162~165C (dec), []D = +42.3.

O
Ref: 4168.
O
O
O
O
O
OH
OH
N
H
N
HO
270
7040 Epivogeloside
7044 3-Epizaluzanin C
Isozaluzanin C C15H18O3 (246.31). Pharm: Cytotoxic (in vitro, HepG2, CD50 =
racemosa] (leaf, flower and twig: yield = 0.0016%dw)[4723], LIU QIU SHE
15g/mL; HeLa, CD50 = 13.5g/mL; OVCAR-3, CD50 = 7.5g/mL; control
GEN CAO Ophiorrhiza liukiuensis (whole herb). Ref: 4527, 4723.
Cisplatin, HepG2, CD50 = 2.8g/mL; HeLa, CD50 = 5.2g/mL; OVCAR-3,

CD50 = 3g/mL; without significant antibacterial effect)[4720]. Source: MU
XIANG Saussurea lappa [Syn. Aucklandia lappa] (root: yield =
0.0003%dw)[4720]. Ref: 2, 4720.
H
H
HO
HO
OO
OH
OH
OH
7045 13,14-Epoxide 9,11,12-trihydroxytriptolide

C20H26O7 (378.43). Colorless filiform crystals, mp 268~270C. Source: LEI
7041 Epiwilsonine
GONG TENG Tripterygium wilfordii. Ref: 256.
C20H25NO4 (343.43). Pharm: Cytotoxic (KB oral epidermoid carcinoma, ED50
OH
= 1.94g/mL)[4253]. Source: SAN JIAN SHAN Cephalotaxus fortunei, TAI
HO
WAN CU FEI Cephalotaxus wilsoniana (twig), ZHONG GUO CU FEI ZHI
YE Cephalotaxus sinensis [Syn. Cephalotaxus harringtonia var. sinensis]. Ref:
OH
2, 660, 4253.
7046 10,15-Epoxy-11(151)-abeo-10-deacetylbaccatin III

O
C29H34O9 (526.59). []D = 18 (CH2Cl2). Source: XI MA LA YA HONG
DOU SHAN Taxus wallichiana. Ref: 662.
OH
O
HO
O
7042 C-3-Epiwilsonine
O
O
C20H25NO4 (343.43). Source: TAI WAN CU FEI Cephalotaxus wilsoniana
(leaf: yield = 0.00048%dw). Ref: 4759.
7047 13,14-Epoxyabiet-7-en-19,6-olide
C20H28O3 (316.44). Oil, []D25 = 8.8 (c = 0.12, CHCl3). Source: LONG BAI
Juniperus chinensis var. kaizuka (leaf: yield = 0.000017%dw). Ref: 3050.
O
O
O
H
7043 C-3-Epiwilsonione
1,2-Didehydro-6,7-epoxy-3,16,17-trimethoxyerythrinan-8-one C20H23NO5
(357.41). Colorless powder, []D28 = +11 (c = 0.104, CHCl3). Pharm:
Cytotoxic (in vitro, HepG2, IC50 = 52g/mL; MCF7, IC50 = 42g/mL; Hep3B,
IC50 = 52g/mL; HT29, IC50 = 24.4g/mL). Source: TAI WAN CU FEI
Cephalotaxus wilsoniana (leaf: yield = 0.00067%dw). Ref: 4759.
7048 (E)-1,10-Epoxy-3-acetoxy-6-hydroxygermacra-4,11(13)-dien12,8-olide
C17H22O6 (322.36). Amorphous solid, []D25 = +54 (c = 0.35, CHCl3). Source:
Anthemis carpatica (aerial parts). Ref: 3974.
O
O
O
O
O
HO
271
7049 15,16-Epoxy-12(R)-acetoxy-8(17),13(16),14-ent-labdatrien-19-oic acid
7053 (2''S,3''S)-Epoxyangeloyldecursinol
C22H30O5 (374.48). Yellow oil, []D25 = 10.8 (c = 0.93, CHCl3). Pharm:
C19H20O6 (344.37). Colorless needles (MeOH), mp 140~142C, []D = +91
Angicidal (inhibits growth of alga Raphidocelis subcapitata, 72h IC50 =
(c = 0.5, CHCl3). Pharm: Neuroprotective (primary cultures of rat cortical
107.8mol/L). Source: BI CHI YAN ZI CAI Potamogeton pectinatus (whole
cells, control, cell viability = 100%, injured by glutamate, cell viability =
herb). Ref: 3488.
0%, 0.1mol/L, cell viability = (70.06.0)%, p<0.001, 1mol/L, cell

viability = (52.54.4)%, p<0.01, 10mol/L, cell viability = (49.03.0)%,
p<0.01). Source: CHAO XIAN DANG GUI Angelica gigas (root: yield =
0.00015%dw). Ref: 4796.
O
O
HO
7050 13,17-Epoxyalisol A
C30H50O6 (506.73). Colorless powder. Source: ZE XIE Alisma orientale [Syn.

Alisma plantago-aquatica var. orientale]. Ref: 2213.
7054 (3'R,4'R)-3'-Epoxyangeloyloxy-4'-acetoxy-3',4'-dihydroseselin
C21H22O8 (402.40). Pharm: Antiallergic. Source: SHI SHI DANG GUI
Angelica shkiokiana. Ref: 658.
OH
O
HO
OH
OH
O
7051 13,17-Epoxyalisol A 24-acetate

C32H52O7 (548.77). Colorless needles, mp 262~263C. Source: ZE XIE
7055 Epoxyarteannuinic acid
Alisma orientale [Syn. Alisma plantago-aquatica var. orientale]. Ref: 2213.
C15H22O3 (250.34). Source: HUANG HUA HAO Artemisia annua. Ref: 2.
H
O
O
HO
OH
O
OH
OH
O
H
O
7056 cis-1',2'-Epoxyasarone
1,2,4-Trimethoxy-5-(E-3'-methyloxiranyl) benzene C12H16O4 (224.26).
7052 (2''R,3''R)-Epoxyangeloyldecursinol
Colorless oil. Source: SHI CHANG PU Acorus tatarinowii. Ref: 8, 660.
C19H20O6 (344.37). Colorless needles (MeOH), mp141~143C, []D = +24 (c = 0.5,

CHCl3). Pharm: Neuroprotective (primary cultures of rat cortical cells, control, cell
viability = 100%, injured by glutamate, cell viability = 0%, 0.1mol/L, cell viability
O
O
= (47.54.0)%, p<0.01, 1mol/L, cell viability = (61.15.0)%, p<0.01, 10mol/L,

cell viability = (56.72.8)%, p<0.01). Source: CHAO XIAN DANG GUI Angelica
gigas (root: yield = 0.0003%dw). Ref: 4796.
7057 6,7-Epoxybisabola-2,11-diene
(2,6-Dimethyl-2-(4-methylpent-4-enyl)-1-oxaspiro[2.5]oct-5-ene) C15H24O
(220.36). Colorless oil. Source: NING BIAN E TAI Radula perrottetii
(essential oil). Ref: 5272.
O
H
O
O
O
O
O
O
272
7058 (3R,4R,6S)-3,4-Epoxybisabola-7(14),10-dien-2-one
7064 Epoxycyperene
C15H24O (220.36). Source: KAN MAI NIANG ZHUANG SHA CAO Cyperus
KUAN DONG HUA Tussilago farfara (flower bud). Ref: 3531.
7059 1,8-Epoxy-1(6),2,4,7,10-bisabolapentaen-4-ol
7065 20R,24R-Epoxy-25-dammaren-3-one
C15H18O2 (230.31). Colorless oil. Source: RI BEN LIU SHAN Cryptomeria
C30H48O2 (440.72). Colorless acicular crystals (MeOH), mp 225C, []D21.5 =
japonica (black heartwood). Ref: 4279.
+57 (c = 1.0, CHCl3). Source: XIANG GANG JIAN MU Dysoxylum

hongkongense. Ref: 422.
OH
O
7060 2,3-Epoxycalealactone A
0.001, CHCl3). Pharm: Cytotoxic (U937, IC50 > 5mol/L; control

Parthenolide, IC50 = 1.9mol/L). Source: YOU KA MEI JU Calea urticifolia
(leaf). Ref: 3887.
7066 1,10-Epoxydehydroleucodin
C15H16O4 (260.29). Source: YI KUA Artemisia myriantha (aerial parts). Ref: 4618.
H
O
OH
O
O
H
O
7061 4,5-Epoxy--caryophyllene
C15H24O (220.36). Source: Stauranthus perforatus (root). Ref: 5253.
7067 22,23-Epoxy-10-deoxy-21-hydroxyiridal
C30H50O4 (474.73). Source: SHI GUAN YUAN WEI Iris cristata. Ref: 2417.
OH
O
HO
7062 8,9-Epoxycoleon U-quinone
C20H24O6 (360.41). Pharm: Cytotoxic (in vitro, K562, IC50 = 13.9g/mL;

control Mitoxanthrone, IC50 = 2g/mL). Source: HUANG QIAO RUI HUA
Coleus xanthanthus (aerial parts: yield = 0.00047%dw). Ref: 4625.
7068 (3S*,6R*)-4,7-Epoxy-6-deoxypseudoanisatin
C15H22O5 (282.34). []D23 = +42.6 (c = 0.96, MeOH). Source: MIN WAN BA
OH
O
JIAO Illicium minwanense (pericarp: 0.00011%dw). Ref: 4697.

O
O
OH
7063 Epoxycollinin
OH
H
HO
7069 -Epoxy-dihydroartemisinic acid
sp. Ref: 2176.
C15H24O3 (252.36). Source: HUANG HUA HAO Artemisia annua (seed). Ref: 3435.
O
O
O
O
HO
273
7070 7,8-Epoxy-8-dihydrogeniposide
7075 2,5-Epoxy-5,10-dihydroxy-6-angeloyloxy-9-(2R-methylbutyryl-
oxy)-germacran-8,12-olide
MeOH). Source: ZHI ZI Gardenia jasminoides [Syn. Gardenia florida]
Ineupatolide [75102-66-8] C25H36O9 (480.56). Source: ZE LAN YANG ER
(leaf). Ref: 4408.
JU Inula eupatorioides. Ref: 1521.
OH
H
O
O
HO
HO
HO
OO
OH
OH
OH
7076 2,5-Epoxy-5,10-dihydroxy-6-angeloyloxy-9-(3-methylbutyryloxy)-
7071 (Z)-6,7-Epoxy-6,7-dihydroligustilide
germacran-8,12-olide
[247017-80-7] C25H36O9 (480.56). White crystals, mp 160~164C, []D25 =
+1.13 (c = 1.0, MeOH). Source: DONG BEI AN HUA JIN WA ER

Carpesium triste var. manshuricum. Ref: 2349.
OH
H
O
O
O
HO
O
O
O
O
O
7077 6,15-Epoxy-1,4-dihydroxyeudesmane
7072 Epoxydihydrolinalool
C15H26O3 (254.37). Source: ZHOU YE MU LAN Magnolia praecocissima
[60047-17-8] C10H18O2 (170.25). Source: XING ZI Prunus armeniaca. Ref: 6.
(seed). Ref: 4181.

OH
HO
HO
7078 ent-8S,12S-Epoxy-7R,16-dihydroxyhalima-5(10),13-dien-15,16- olide

7073 Epoxydihydro-oleanolic acid
C20H28O5 (348.44). White amorphous powder, []D = 110 (CHCl3, c 0.05).
C30H48O4 (472.71). Source: NAN HE SHI Daucus carota. Ref: 6.
Pharm: Cytotoxic (Lu1, ED50 = 15.4g/mL, control Ellipticine, ED50 =

0.02g/mL; Col2, ED50 = 14.8g/mL, Ellipticine, ED50 = 0.3g/mL; KB,
ED50 = 16.9g/mL, Ellipticine, ED50 = 0.04g/mL; LNCaP, ED50 =
O
OH
H
O
H
HO
13.7g/mL, Ellipticine, ED50 = 0.8g/mL). Source: Alomia myriadenia (aerial

parts). Ref: 3479.
HO
7074 2,5-Epoxy-5,10-dihydroxy-6-angeloyloxy-9-(2-methylbutyryloxy)germacran-8,12-olide
OH
[247050-76-6] C25H36O9 (480.56). White crystals, mp 190~193C, []D25 =

4.3 (c = 1.0, MeOH). Source: DONG BEI AN HUA JIN WA ER Carpesium
7079 (3S,5R,6S,7E,9R)-5,6-Epoxy-3,9-dihydroxy-7-megastigmene
triste var. manshuricum. Ref: 2349.

OH
H
O
O
O
HO
HO H
O
O
HO
274
7080 12,16-Epoxy-11,14-dihydroxy-6-methoxy-17(15-16)-abeo-abieta-
7083 (23S)-17,23-Epoxy-28,29-dihydroxy-3-[(O--L-rhamnopyranos-
5,8,11,13,15-pentaene-3,7-dione
yl-(12)-O--D-glucopyranosyl-(12)--L-arabinopyranosyl-(16)--
C21H22O6 (370.41). mp 248.0C, []D20 = +50.0 (c = 0.5, CHCl3). Pharm:
D-glucopyranosyl)oxy]-27-norlanost-8-en-24-one
Antiproliferative (in vitro, MTT assay, CEM, IC50 = 24.2mol/L, control
C52H84O23 (1077.24). Pharm: Cytotoxic (Hmn oral squamous cell carcinoma
Doxorubicin, IC50 = 0.036mol/L, HeLa, IC50 = 12.7mol/L, Doxorubicin,
cells HSC-2, IC50 = 19g/mL, control Etoposide, IC50 = 24g/mL). Source:
IC50 = 0.027mol/L, HCT8, IC50 > 72.2mol/L, Doxorubicin, IC50 =
XUE GUANG HUA Chionodoxa luciliae (fresh bulb). Ref: 4308.
0.024mol/L, MCF7, IC50 > 72.2mol/L, Doxorubicin, IC50 = 0.183mol/L,

O
B-16, IC50 > 72.2mol/L, Doxorubicin, IC50 = 0.056mol/L). Source:

Aegiphila lhotzkyana (root). Ref: 4940.
O
O
HO
OH
OH
O
OH
H
OH
OH
OH
HO
OO
OO
OH
OH
OO
OH
7081 (22S,23R)-16,23-Epoxy-18,23-dihydroxy-22-(2-methyl-1-propen-
OH
OH
OO
yl)-24-norchol-5-en-3-yl O--L-rhamnopyranosyl-(12)--D-glucopyranoside
OH OH

Pharm: Cytotoxic (HL-60 cells, IC50 > 10mol/L, control Etoposide, IC50 =
0.025mol/L). Source: XIA FENG XIN ZI Galtonia candicans (bulb). Ref:
4116.
7084 24,25-Epoxy-3,23-dihydroxy-7-tirucallene
C30H50O3 (458.73). Prisms (Me2CO), mp 155~157C. Source: HAI NAN
JIAN MU Dysoxylum hainanense (bark). Ref: 3987.
O
H
OH
HO
OH
O
H
HO
OO
HO
OH
7085 6,7-Epoxy-4-dumorten-3-one
OH
OH
OO
C15H22 O2 (234.34). Oil. Source: MAO DI QIAN Dumortiera hirsuta. Ref:

2283.
H
OH OH
O
7082 6,7-Epoxy-5,20-dihydroxy-1-oxowitha-2,24-dienolide
C28H38O6 (470.61). Pharm: BChE inhibitor (IC50 = (502)mol/L, control

Galanthamine IC50 = (0.500.001)mol/L, Eserine IC50 =
[2563]
(0.040.0001)mol/L); AChE inhibitor inactive

SHUI QIE Withania somnifera. Ref: 2563.
. Source: CUI MIAN
7086 Epoxyeleganolactone
1,2-Epoxy-13-hydroxy-6,10,14-phytatrien-20,1-olide [165133-76-6] C20H30O4
(334.46). Oil, []D25 = 0.9 (c = 2.8, CH2Cl2). Source: SHUANG CHA ZAO
Bifurcaria bifurcata. Ref: 2405.
OH
H
O
H
H
OH
H
O
HO
O
O
275
7087 (20R)-3,10-Epoxy-9-epi-cucurbita-24-ene
7092 8,9-Epoxy-10-epi-ryanodine
[259657-91-5] C30H50O (426.73). Oil. Source: Senecio selloi. Ref: 2416.


parts). Ref: 5139.
H
O
OH
OH
HO OH
H
OH
N
H
7088 (20S)-3,10-Epoxy-9-epi-cucurbita-24-ene
OH
[259657-93-7] C30H50O (426.73). Oil. Source: Senecio selloi. Ref: 2416.
7093 6,9-Epoxy-ergosta-7,22-dien-3-ol
H
C28H44O2 (412.66). White acicular crystals, mp 229~230C. Source: SHI HU

XIAO GU Mycena dendrobii. Ref: 851.
H
H
O
H
O
7089 4,5-Epoxy-8-epiinnunolide
HO
C15H20O3 (248.32). Source: SHANG ZUO JIAN YE GUANG E TAI Porella
7094 21R,23R-Epoxy,21-ethoxy,24S,25-dihydroxyapotirucalla-7-en-
acutifolia ssp. tosana. Ref: 3932.
3-one
C32H52O5 (516.77). White crystals. Source: MA LA BA JIAN MU Dysoxylum
malabaricum (leaf). Ref: 5130.

H
OH
OH
7090 7,8-Epoxy-8-epi-loganic acid

O
OH
O
H
7095 (+)-6,11-Epoxy-eudesmane
HO
C15H26O (222.37). Colorless oil. Source: Tritomaria polita (essential oil).
H
OO
OH
Ref: 3446.
OH
OH
H
7091 8,9-Epoxy-10-epi-ryanodine

7096 4,15-Epoxyeudesmane-1,6-diol
C15H26O3 (254.37). Source: YI NIAN PENG Erigeron annuus (aerial parts),
SU MEN BAI JIU CAO Erigeron sumatrensis (aerial parts). Ref: 4338.
parts). Ref: 5139.

HO
OH
N
H
O
O
OH
OH
OH
H
O
OH
OH
OH
276
7097 6,14-Epoxyeudesm-4(15)-en-1-ol
7103 3(15)-Epoxygymnomitrane
C15H24O (220.36). Oil, []D21 = 4.8 (c= 0.83). Source: JIE XING YE TAI
CHCl3). Source: FEI CHENG FEI PENG Erigeron philadelphicus (aerial
Jungermannia truncata. Ref: 4201.
parts). Ref: 4338.
OH
O
H
7104 (9R,10S)-Epoxyheptadecan-4,6-diyn-3-one
7098 8,9-Epoxy-ferutinin
C17H24O2 (260.38). Light yellow oil, []D25 = 70.0 (c = 1.0, CHCl3). Pharm:
C22H30O5 (374.48). Source: YI LANG A WEI Ferula kuhistanica (stem). Ref:
DGAT inhibitor (IC50 = 9g/mL, control Evocarpine, IC50 = 8.1g/mL).
3977.
Source: REN SHEN Panax ginseng [Syn. Panax schinseng]. Ref: 4943.
O
O
OH
HO
O
O
7099 3,4-Epoxyfilicane
7105 (2R,3R,5R)-2,3-Epoxy-6,9-humuladien-5-ol-8-one
[23983-65-5] C30H50O (426.73). mp 229~231C. Source: ZHU ZONG CAO
C15H22O3 (250.34). Pharm: CYP3A4 inhibitor (IC50 = 42.6mol/L, control
Adiantum capillus-veneris. Ref: 6.
Ketoconazole, IC50 = 0.245mol/L); CYP2D6 inhibitor inactive (IC50 >

100mol/L, control Quinidine, IC50 = 0.078mol/L). Source: FANG XIANG
JIANG Zingiber aromaticum (rhizome: 0.00060%dw). Ref: 4669.
OH
O
7100 rel-1S,2S-Epoxy-4R-furanogermacr-10(15)-en-6-one
C15H18O3 (246.31). Colorless oil, []D = 160.0 (c = 2.5, CHCl3). Pharm:
7106 (2R,3S,5R)-2,3-Epoxy-6,9-humuladien-5-ol-8-one
Cytotoxic (in vitro, MCF7, IC50 = 40mol/L, weak activity). Source: MO
YAO Commiphora myrrha [Syn. Commiphora molmol]. Ref: 3093.
Ketoconazole, IC50 = 0.245mol/L); CYP2D6 inhibitor inactive (IC50 >

100mol/L, control Quinidine, IC50 = 0.078mol/L). Source: FANG XIANG
JIANG Zingiber aromaticum (rhizome: 0.00050%dw). Ref: 4669.

O
OH
7101 ()-1,10-Epoxy-guaia-11-ene
O

O
7107 1,2-Epoxy-10-hydroperoxy-3,4,8-trihydroxyguaia-11(13)en-12,6-olide
C15H20O8 (328.32). Colorless gum, []D20 = +24 (c = 0.10, MeOH). Pharm:
Antifungal (Candida albicans, MIC = 20g/mL). Source: GUAN MU YA JU
7102 Epoxyguaine
Ajania fruticulosa (aerial parts). Ref: 5222.

OH
C15H24O (220.36). bp 102~104C/1mmHg. Source: XIANG FU Cyperus

rotundus. Ref: 6.
OH
HO
O
HO
O
O
277
7108 4,5-Epoxy-6-hydroxy amorphan-12-oic acid
7113 8,9-Epoxy-21-hydroxy-10-epi-ryanodine
EP-1 C25H33NO11 (523.54). Crystals (CHCl3:Me2CO = 3:1), mp 193C, []D =

Ref: 5139.
HO OH
OH
OH
OH
OH
OH
N
H
OH
7109 4,5-Epoxy-6-hydroxy amorphan-12-ol
OH
C15H26O3 (254.37). Colorless oil. Source: HUANG HUA HAO Artemisia
7114 (1,2,5,810)-1,10-Epoxy-2-hydroxy-3,7(11)-guaiadien-12,8-
annua (seed). Ref: 3435.
olide
C15H18O4 (262.31). Yellow oil, []D25 = +61.0 (c = 0.4, CHCl3). Pharm:
CYP3A4 inhibitor and CYP2D6 inhibitor (in vitro, CYP3A4, IC50 =

98.2mol/L; CYP2D6, IC50 > 100mol/L; control Ketoconazole, CYP3A4,
IC50 = 0.72mol/L; control Quinidine, CYP2D6, IC50 = 0.082mol/L). Source:
OH
BI CHENG QIE Piper cubeba (fruit: yield = 0.00023%dw). Ref: 4797.

OH
7110 (1S*,3R*,4R*,6S*,11S*)-3,4-Epoxy-6-hydroxy-dolabella-7E,12-
HO
dien-14-one
C20H30O3 (318.46). Clear film, []D20 = 77.3 (c = 0.21, CHCl3). Source:

H
fungus Stachybotrys chartarum. Ref: 5104.
7115 5H-2,4-Epoxy-3-hydroxy-guaia-1(10),11(13)-dien-6,12-olide
C15H18O4 (262.31). Colorless gum, []D20 = +12.9 (c = 0.1, EtOH). Pharm:
Cytotoxic (KB ATCC CCL17, IC50 = 3.6g/mL). Source: Warionia saharae.
HO
7111 (13S)-8,9-Epoxy-18-hydroxy-10-epi-ryanodine
Ref: 5399.
HO

(c = 0.2). Source: QU CHONG CAO Spigelia anthelmia (aerial parts). Ref:
O
O
5139.
7116 7-11-Epoxy-5-hydroxy-9-guaiaen-8-one
OH
OH
OH
H
N
H
C15H22O3 (250.34). Pharm: NO production inhibitor (mus peritoneal
HO OH
OH
OH
7112 8,9-Epoxy-20-hydroxy-10-epi-ryanodine
O
O
OH
(c = 0.1). Source: QU CHONG CAO Spigelia anthelmia (aerial parts). Ref:

5139.
7117 1,4-Epoxy-16-hydroxyheneicos-1,3,12,14,18-pentaene
C21H32O2 (316.49). Viscous oil. Source: YA LUO CHUN Cipadessa baccifera.
OH
N
H
OH
OH
Ref: 745.
O
OH
OH
O
HO
OH
OH
278
7118 1,4-Epoxy-16-hydroxyheneicos-1,3,12,14-tetraene
7124 12(S)-15,16-Epoxy-19-hydroxy-neo-cleroda-13(16),14-dien-18,6:
C21H34O2 (318.50). Viscous oil. Source: YA LUO CHUN Cipadessa baccifera.
20,12-diolide
Ref: 745.
C20H24O6 (360.41). White powder, []D25 = +26.0 (c = 0.001, MeOH). Source:

SHI CAN XIANG KE KE Teucrium chamaedrys. Ref: 3431.
OH
7119 1,5-Epoxy-3-hydroxy-1-(4-hydroxy-3,5-dimethoxyphenyl)-7-(4-
O
O
hydroxy-3-methoxyphenyl)heptane
C22H28O7 (404.46). Colorless oil, []D16 = 24 (c = 0.19, EtOH). Source:
O
OH
HO
7125 14,15-Epoxy-3-hydroxy-9-oxo-11(108)-abeolanosta-22-cis,
OH
24-trans-dien-26-oic acid
C30H44O5 (484.68). White needles (MeOH), mp 210C (dec). Pharm: Cytotoxic
(in vitro, MCF7, GI50 = 69.6mol/L; NCI-H460, GI50 = 70.3mol/L; SF268,
OH
GI50 = 95.7mol/L; control Doxorubicin, GI50 = 0.043mol/L; NCI-H460,
7120 22,23-Epoxy-21-hydroxyiridal
GI50 = 0.094mol/L; SF268, GI50 = 0.093mol/L). Source: MEI LI TENG

HUANG Garcinia speciosa (bark). Ref: 4790.
OH
O
HO
OH
OH
O
7121 ent-15,16-Epoxy-3-hydroxy-kauran-2-one
C20H30O3 (318.46). Colorless needle crystals, mp 123C, []D24 = 5 (c = 0.13,
HO
MeOH). Pharm: Antibacterial (inhibits colony formation of X. campestris pv.

oryzae, 200mg/L, InRt = 30%). Source: DAO CAO Oryza sativa (leaf). Ref: 3814.
7126 14,15-Epoxy-3-hydroxy-9-oxo-11(108)-abeolanosta-24-transen-26-oic acid

C30H46O5 (486.7). White needles (MeOH), mp 205~207C. Pharm: Cytotoxic
O
O
H
HO
(in vitro, MCF7, GI50 = 63.8mol/L; NCI-H460, GI50 = 68.6mol/L; SF268,

GI50 = 86.4mol/L; control Doxorubicin, GI50 = 0.043mol/L; NCI-H460,
GI50 = 0.094mol/L; SF268, GI50 = 0.093mol/L). Source: MEI LI TENG
7122 12,17-Epoxy-17-hydroxylabda-13(E)-ene
HUANG Garcinia speciosa (bark). Ref: 4790.
20
C20H34O2 (306.49). mp 150~152C, []D = 8.526 (c = 1.08, CHCl3).

Pharm: Cytotoxic inactive (in vitro, BT474, CHAGO, HepG2, Kato3,
OH
SW620: > 10g/mL). Source: GUANG YE BA DOU Croton oblongifolius
[Syn. Croton laevigatus]. Ref: 5363.
HO
O
OH
7127 14,15-Epoxy-3-hydroxy-9-oxo-11(108)-abeolanost-24-transen-26-oic acid

C30H46O5 (486.7). Yellowish gum. Source: MEI LI TENG HUANG Garcinia
7123 (3S,5R,6S,7E)-5,6-Epoxy-3-hydroxy-7-megastigmen-9-one
speciosa (bark). Ref: 4790.
OH
O
O
HO
HO
279
7128 5,6-Epoxy-4-hydroxy-1-oxowitha-2,14,24-trienolide
H
O
C28H36O5 (452.60). Pharm: BChE inhibitor (IC50 = (124.01.1)mol/L,

O
control Galanthamine IC50 = (0.500.001)mol/L, Eserine IC50 =

(0.040.0001)mol/L); AChE inhibitor (IC50 = (62.52.0)mol/L, control
HO
HO
HO
Source: CUI MIAN SHUI QIE Withania somnifera. Ref: 2563.
OH
O
HO
Galanthamine IC50 = (8.20.01)mol/L, Eserine IC50 = (0.850.0001)mol/L).
O O
HO
HO
OH
H
OH
HO
H
O
HO
OH
7132 (23S)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl-
(12)-O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)--D
O
OH
-glucopyranosyl)oxy]-27-norlanost-8-en-24-one
C52H84O22 (1061.24). Pharm: Cytotoxic (in vitro, HSC-2, IC50 = 32mol/L;
7129 5,6-Epoxy-4-hydroxy-1-oxo-witha-2,16,24-trienolide
30
C28H36O5 (452.60). mp 268C, []D = +92.60 (c = 0.25, CHCl3). Source:
control Etoposide, IC50 = 41mol/L). Source: QI YI PU TAO FENG XIN ZI

Muscari paradoxum (bulb: yield = 0.001%fw). Ref: 4793.

H
O
O
H
O
OH
O
HO
HO
HO
HO
O
HO
HO
O
O
OH
O
OH
H
OH
HO
HO
OH
7130 (23R)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl(12)-O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)--
7133 (23S,25R)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranos-
D-glucopyranosyl)oxy]-27-norlanost-8-ene-15,24-dione
yl-(12)-O-[O--D-glucopyranosyl-(12)--D-glucopyranosyl-(13)]-O-
-D-glucopyranosyl-(12)--L-arabinopyranosyl-(16)--D-glucopyran
Pharm: Cytotoxic inactive (in vitro, HSC-2, 100mol/L; control Etoposide,
osyl)oxy]lanost-8-en-23,26-olide
IC50 = 41mol/L). Source: QI YI PU TAO FENG XIN ZI Muscari paradoxum
(bulb: yield = 0.00054%fw). Ref: 4793.
28

H
O
O
O
OH
O
HO
HO
HO
HO
O O
O
HO
HO
O
O
OH
H
OH
OH
HO
HO
OO
OO
OH
OH
OH
HO
OH
HO
7131 (23S)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl(12)-O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)-D-glucopyranosyl)oxy]-27-norlanost-8-ene-15,24-dione
C52H82O23 (1075.22). Pharm: Cytotoxic (in vitro, HSC-2, IC50 = 63mol/L;
control Etoposide, IC50 = 41mol/L). Source: QI YI PU TAO FENG XIN ZI
Muscari paradoxum (bulb: yield = 0.0034%fw). Ref: 4793.
O
OH
HO
HO
OO
OO
O
OH
OH
O
O
OH
OH
OH
OH OH
H
OH
OH
280
7134 (23S)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl(12)-O-[-D-glucopyranosyl-(13)]-O--D-glucopyranosyl-(12)--L-arabi
nopyranosyl-(16)--D-glucopyranosyl)oxy]-27-norlanost-8-en- 24-one

OH
OO
OO
OH
OH
OH
HO
O
HO
OO
H
OH
OH
O
OH
OH
O
OH
O
OO
HO
HO
OH
OH
OO
OO
OH
OH
H
OH
HO
OH
(12)-O-[O--D-glucopyranosyl-(12)--D-glucopyranosyl-(13)]-O-
O
OH
OH
OO
OH
OH
HO
OH OH
OH
-D-glucopyranosyl-(12)--L-arabinopyranosyl-(16)--D-glucopy-
OH
OH
ranosyl)oxy]-27-norlanost-8-ene-15,24-dione
O
O
OH
Pharm: Cytotoxic (Hmn oral squamous cell carcinoma cells HSC-2, IC50 >
OH OH
50g/mL, control Etoposide, IC50 = 24g/mL). Source: XUE GUANG HUA

Chionodoxa luciliae (fresh bulb). Ref: 4308.
7135 (23R)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl-
(12)-O-[O--D-glucopyranosyl-(12)--D-glucopyranosyl-(13)]-OO
-D-glucopyranosyl-(12)--L-arabinopyranosyl-(16)--D-glucopy-
ranosyl)oxy]-27-norlanost-8-en-24-one
OH

cells HSC-2, IC50 > 50g/mL, control Etoposide, IC50 = 24g/mL). Source:
O
OO
HO
HO
O
OH
HO
OO
OO
OH
OH
OH
OH
OH
OH O O
HO
OH
OH OH
OH
7138 (23R)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl(12)-O-[O--D-xylopyranosyl-(12)--L-arabinopyranosyl-(13)]O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)--D-glucopyranosyl)oxy]-27-norlanost-8-ene-15,24-dione
Pharm: Cytotoxic inactive (in vitro, HSC-2, 100mol/L; control Etoposide,
OH
OH
OH
H
OH
OO
HO
H
OH
OH
OH O O
OO
OH
OH
OH
OH
HO
OH
OO
HO
HO
OO
OO
OH
OH OH
OH
IC50 = 41mol/L). Source: QI YI PU TAO FENG XIN ZI Muscari paradoxum

(bulb: yield = 0.00094%fw). Ref: 4793.
H
O
7136 (23S)-17-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosylO--D-glucopyranosyl-(12)--L-arabinopyranosyl-(16)--D-gluC64H104O32 (1385.52). Pharm: Cytotoxic (Hmn oral squamous cell carcinoma
OH
O
HO
(12)-O-[O--D-glucopyranosyl-(12)--D-glucopyranosyl-(13)]copyranosyl)oxy]-27-norlanost-8-en-24-one
OH
HO
HO
HO
HO
O HO
O
O O
HO
OH
O O HO
HO
O
O
OH
OH
OH
H
OH
281
7143 14,15-Epoxy-3-hydroxyserratan-21-ol
(12)-O-[O--D-xylopyranosyl-(12)--L-arabinopyranosyl-(13)]-O-
C30H50O3 (458.73). Colorless needles (CHCl3CH3OH), mp 280~283C,
-D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)--D-glucopy-
[]D20 = +0.2 (c = 0.44, C5H5N). Source: QIAN CENG TA Huperzia serrata
ranosyl)oxy]-27-norlanost-8-ene-15,24-dione
[Syn. Lycopodium serratum]. Ref: 5349.
28
OH
Pharm: Cytotoxic (in vitro, HSC-2, IC50 = 19mol/L; control Etoposide, IC50
= 41mol/L). Source: QI YI PU TAO FENG XIN ZI Muscari paradoxum
(bulb: yield = 0.0051%fw). Ref: 4793.

H
HO
OH
HO
O O
HO
HO
HO
OH
O
HO
HO
O HO
O
HO
7144 14,15-Epoxy-3-hydroxy-serratan-21-ol
O O HO
HO
O O
OH
C30H50O3 (458.73). Colorless prisms (CHCl3CH3OH), mp 272~274C, []D20

= 19.7 (c = 0.57, CHCl3). Source: QIAN CENG TA Huperzia serrata [Syn.
H
OH
O
HO
OH
OH
7140 (23S)-17,23-Epoxy-29-hydroxy-3-[(O--L-rhamnopyranosyl(12)-O-[O--D-xylopyranosyl-(12)--L-arabinopyranosyl-(13)]O--D-glucopyranosyl-(12)-O--L-arabinopyranosyl-(16)--D-glu
HO
copyranosyl)oxy]-27-norlanost-8-en-24-one
7145 14,15-Epoxy-21-hydroxyserratan-3-one
Pharm: Cytotoxic (in vitro, HSC-2, IC50 = 7.3mol/L; control Etoposide, IC50
C30H48O3 (456.72). Needles, mp 310~312C (MeOHCHCl3), []D = 14.5 (c
= 41mol/L). Source: QI YI PU TAO FENG XIN ZI Muscari paradoxum
= 0.52). Source: RI BEN YU LIN SONG Picea jezoensis (cuticle). Ref: 3076.
OH
(bulb: yield = 0.00033%fw). Ref: 4793.

H
OH
HO
HO
HO
OH
O
HO
HO
O HOO
O O HO
HO
O
O
O
O
OH
O O
OH
H
OH
HO
HO
7146 8,10-Epoxy-9-hydroxy thymol 3-O-tiglate

C15H18O4 (262.31). []D23 = 32.0 (c = 1.1, CHCl3). Source: PEI LAN
Eupatorium fortunei (aerial parts). Ref: 3077.
OH
7141 5,20-Epoxy-20-hydroxy-ros-15-ene

O
OH
7147 1,4-Epoxy-5-hydroxy-10H-xantha-11(13)-en-12,8-olide
H
H
O

CHANG YE TIAN MING JING Carpesium longifolium (aerial parts: yield =
OH
0.0009%dw). Ref: 4736.

O
7142 14,15-Epoxy-3-hydroxyserratan-21-ol-3-O-acetate
O
HO
+12.9 (c = 1.00, CHCl3). Source: QIAN CENG TA Huperzia serrata [Syn.
7148 22,23-Epoxyiridal

OH
O
O
O
HO
OH
O
282
7149 2',3'-Epoxyisocapnolactone
7155 ent-16,17-Epoxy-kaurane
C19H18O6 (342.35). White needles, mp 103~105C. Source: JI XIAO XIAO
C20H32O (288.48). mp 174.0~176.5C, []D17 = 45.9 (c = 0.18, CHCl3).
YUN XIANG MU Micromelum minutum (leaf). Ref: 3467.
Source: ZHE BEI MU Fritillaria verticillata var. thunbergii [Syn. Fritillaria

thunbergii]. Ref: 2182.
O
O
7150 (+)-6,11-Epoxy-isodaucane

H
Ref: 3446.
7156 ()-16,17-Epoxykauran-19-oic acid

C20H30O3 (318.46). White solid, mp 154~156C, []D20 = 98.4 (c = 1,
CHCl3). Pharm: Na+,K+-ATP inhibitor (crude enzyme Na+,K+-ATPase from
rat brain, IC50 = 480mol/L). Source: GUANG YE BA DOU Croton

oblongifolius [Syn. Croton laevigatus] (semi-synthetic derivative). Ref:
7151 Epoxyisolinearol
C22H34O5 (378.51). Colorless needles (CHCl3). Source: Sideritis ozturkii
5404.
O
H
HO
OH
OH
O
7152 2,3-Epoxy-jaeschkeanadiol p-methoxybenzoate

C23H32O5 (388.51). Source: YI LANG A WEI Ferula kuhistanica (stem). Ref: 3977.
7157 ent-15,16-Epoxy-kauran-17-ol
C20H32O2 (304.48). mp 160C, []D20 = +9.4 (c = 1.5, CHCl3). Source: ZHE
BEI MU Fritillaria verticillata var. thunbergii [Syn. Fritillaria thunbergii].
Ref: 2182.
OH
HO
O
O
7153 2,3-Epoxyjuanislamin
C23H28O9 (448.47). White powder, []D20 = +154.0 (c = 0.001, CHCl3).

Pharm: Cytotoxic (U937, IC50 = 1.8mol/L; control Parthenolide, IC50 =
1.9mol/L). Source: YOU KA MEI JU Calea urticifolia (leaf). Ref: 3887.
7158 ent-16,17-Epoxykauran-15-one
C20H30O2 (302.46). Oil, []D23 = 109.0 (c = 0.28). Source: JIE XING YE
TAI Jungermannia truncata. Ref: 4201.
O
O
O
OH
O
O
7154 ent-15,16-Epoxy-kauran-2,3-dione
Oryzadione C20H28O3 (316.44). Colorless needle crystals, mp 138C, []D24 =
7159 12,15-Epoxy-8(17),13-labdadien-18-oic acid
13 (c = 0.21, MeOH). Pharm: Antibacterial (inhibits colony formation of X.
C20H30O3 (318.46). Amorphous, []D27 = +37.6 (c = 0.19, CHCl3). Source:
campestris pv. oryzae, 200mg/L, InRt = 40%). Source: DAO CAO Oryza
TAI WAN SHAN MU Cunninghamia konishii (wood). Ref: 4176.
sativa (leaf). Ref: 3814.

O
O
H
O
O
H
O
OH
283
7160 12,15-Epoxylabda-8(17),12,14-trien-16-al
7166 13,14-Epoxy-3-methoxyserratan-21-ol
C20H28O2 (300.44). Orange oil, []D20 = +50.5 (c = 0.42, CHCl3). Source:
C31H52O3 (472.76). Prisms, mp 242~244C (MeOHCHCl3), []D = +31 (c =
Turreanthus africanus (seed). Ref: 3884.
0.38). Source: RI BEN YU LIN SONG Picea jezoensis (cuticle). Ref: 3076.
OH
O
O
7167 13,l4-Epoxy-3-methoxyserratan-21-ol
7161 15,16-Epoxy-8(17),13(16),14-ent-labdatrien-19-oic acid
C31H52O3 (472.76). Colorless prisms, mp 264~267C, []D23.5 = +4.7 (c =
Daniellic acid C20H28O3 (316.44). Pharm: Angicidal (inhibits growth of alga
0.11, CHCl3). Pharm: Antineoplastic promoter (mouse skin carcinogenesis,
Raphidocelis subcapitata, 72h IC50 = 17.2mol/L). Source: AO SHI DAN NI
TPA-induced EBV-EA activation assay, compound concentration (mol
SU MU Daniellia oliveri, BI CHI YAN ZI CAI Potamogeton pectinatus
ratio/32 pmol TPA) = 500, EBV-EA viability = 25.7%, IC50(mol ratio/32
pmol TPA) = 288; control Oleanolic acid, compound concentration (mol

ratio/32 pmol TPA) = 500, EBV-EA viability = 30.0%, IC50(mol ratio/32
O
pmol TPA) = 360). Source: YU LIN YUN SHAN Picea jezoensis var.
jezoensis (stem cortex). Ref: 5477.
HO
OH
H
7162 (E)-8,17-Epoxylabd-12-ene-15,16-dial
7168 14,15-Epoxy-3-methoxyserratan-21-ol
O
O

OH
7163 1,10-Epoxylepidozenal
C15H22O2 (234.34). Source: MIAN MAO MA DOU LING Aristolochia
mollissima (dried root and stem: yield = 0.00031%dw). Ref: 3026.

O
O
H
7169 13,14-Epoxy-21-methoxyserratan-3-one
H
C31H50O3 (470.74). Prisms, mp 219~222C (MeOHCHCl3), []D = 98 (c =
0.83). Source: RI BEN YU LIN SONG Picea jezoensis (cuticle). Ref: 3076.
7164 1,10-Epoxy-8-methoxyeremophil-7(11)-en-12,8-olide
C16H22O4 (278.35). Colorless crystals, mp 102~103C (hexane), []D = 87.5 (c =
1, CHCl3). Source: HUANG SE QIAN LI GUANG Senecio flavus. Ref: 2409.

O
O
O
O
7170 8-Epoxymethylacrylyloxyambrosin
7165 5,20-Epoxy-20-methoxy-ros-15-ene
[219319-63-8] C19H22O6 (346.38). Source: YIN JIAO JU Parthenium

hysterophorus. Ref: 2393.
O
H
O
H
O
O
O
284
7171 8-Epoxymethylacrylyloxy-11,13-dihydroparthenin
7177 Epoxynepapakistamine A
[219319-61-6] C19H24O7 (364.40). Non-crystalline. Source: YIN JIAO JU
(20S)-20-(N-Methylamino)-3-(tigloylamino)-5-pregna-16,17-epoxy-2,4
Parthenium hysterophorus. Ref: 2393.
-di-O-acetate C31H48N2O6 (544.74). Colorless crystalline solid (CHCl3), mp
119~120C, []D25 = +14 (c = 0.07, CHCl3). Pharm: BChE inhibitor (horse
OH
serum BChE, IC50 = (77.40.024)mol/L, control Eserine IC50 =
(0.8570.008)mol/L); AChE inhibitor (electric eel AChE, IC50 > 200mol/L,
H
O
control Eserine IC50 = (0.0410.001)mol/L). Source: YUN NAN YE SHAN
HUA Sarcococca coriacea [Syn. Sarcococca wallichii] (leaf). Ref: 4241.

O
H H
N
7172 8-Epoxymethylacrylyloxyparthenin
[219319-59-2] C19H22O7 (362.38). Non-crystalline. Source: YIN JIAO JU

Parthenium hysterophorus. Ref: 2393.
O
OH
O
H
N
H
H
O
O
H
H
7178 22,29-Epoxy-30-norhopane-13-ol
C29H48O2 (428.70). Colorless solid, mp 264~266C, [] D25 = +15.10 (c =
7173 5,6-Epoxy-24(R)-methylcholesta-7,22-dien-3-ol
0.25, CHCl3). Pharm: Antibacterial (Salmonella typhimurium, 100g/disk,
[23637-31-2] C28H44O2 (412.66). Source: DONG CHONG XIA CAO
IZD = 9mm, control Kanamycin, 30g/disk, IZD = 14mm; Bacillus subtilis,
Cordyceps sinensis. Ref: 2322.
100g/disk, IZD = 8mm, Kanamycin, 30g/disk, IZD = 31mm). Source: BAN

YUE XING TIE XIAN JUE Adiantum lunulatum. Ref: 5124.
OH
O
HO
7174 ent-15,16-Epoxy-3-myristoyloxy-kauran-2-one
Antibacterial (inhibits colony formation of X. campestris pv. oryzae, 500mg/L,
InRt = 30%). Source: DAO CAO Oryza sativa (leaf). Ref: 3814.
7179 (+)-1,5-Epoxy-nor-ketoguaia-11-ene
C14H20O2 (220.31). Source: CHEN XIANG Aquilaria agallocha. Ref: 13.
O
O
7175 1,10-Epoxy-nardosin-7,11-diene
C15H22O (218.34). []D20 = +195 (c = 0.61, CHCl3). Source: Gackstroemia
O
7180 ()-12,13-Epoxyoleic acid

C18H32O3 (296.45). []D20 = 0 (c = 0.5, CHCl3). Pharm: COX-1 inhibitor
(100g/mL, InRt = 30%, control trans-Resveratrol, IC50 = 0.25g/mL);
COX-2 inhibitor (100g/mL, InRt = 58%, control trans-Resveratrol, IC50 =
0.30g/mL). Source: LIAN YE TONG Hernandia Sonora [Syn. Hernandia
7176 15,16-Epoxy-neo-clerodan-1,3,13(16),14-tetraen-18,19-olide
ovigera] (seed). Ref: 5030.

O
O
OH
285
7181 ent-15,16-Epoxy-3-oxa-kauran-2-one
7186 ent-15,16-Epoxy-3-palmitoyloxy-kauran-2-one
C19H28O3 (304.43). Colorless needle crystals, mp 183C, []D24 = 54 (c =
C36H60O4 (556.88). Amorphous, []D24 = 17 (c = 0.14, MeOH). Source:
0.05, MeOH). Pharm: Antibacterial (inhibits colony formation of X.
DAO CAO Oryza sativa (leaf). Ref: 3814.
campestris pv. oryzae, 210mg/L, InRt = 45%). Source: DAO CAO Oryza
sativa (leaf). Ref: 3814.
O
O
H
O
7182 5H-3,4-Epoxy-14-oxo-guaia-1(10),11(13)-dien-6,12-olide
C15H16O4 (260.29). Colorless gum, []D20 = +9.4 (c = 0.1, EtOH). Pharm:
Cytotoxic (KB ATCC CCL17, IC50 = 3.5g/mL). Source: Warionia saharae.
7187 5,6-Epoxyphysalin B
C28H30O10 (526.55). Source: TIAN PAO ZI Physalis minima. Ref: 6.
H
Ref: 5399.
O
HO
H
O
O
7183 15,16-Epoxy-12-oxo-8(17),13(16),14-ent-labdatrien-20,19-olide
7188 3,4-Epoxy-5-pipermethystine
C20H24O4 (328.41). Colorless oil, [] D = +22.5 (c = 0.43, CHCl3). Source:
C16H17NO5 (303.32). Colorless needles (hexane), mp 59C, []D22 = 98.8 (c
FU YE YAN ZI CAI Potamogeton natans. Ref: 5184.
= 0.5, Me2CO). Source: KA WA HU JIAO Piper methysticum. Ref: 3373.
25
O
O
O
O
7184 15,16-Epoxy-12-oxo-8(17),13(16),14-ent-labdatrien-19,20-olide
25
C20H24O4 (328.41). Colorless oil, [] D = +65.3 (c = 0.04, CHCl3). Source:

FU YE YAN ZI CAI Potamogeton natans. Ref: 5184.
7189 2,3-Epoxyplumbagin
C11H8O4 (204.18). Pale yellow needles (hexane), mp 92~93C, 95~96C,
[]D28 = 4.51 (c = 2.41, CHCl3). Pharm: Ichthyotoxin (MLC = 3.0mg/L,
control Juglone, MLC = 0.2mg/L). Source: HAI SHI Diospyros maritima
(fruit). Ref: 4185.

O
O
O
O
OH
7185 ent-15,16-Epoxy-2-palmitoyloxy-kauran-2-one
Antibacterial (inhibits colony formation of X. campestris pv. oryzae, 500mg/L,
InRt = 45%). Source: DAO CAO Oryza sativa (leaf). Ref: 3814.
7190 20R,21-Epoxyresibufogenin 3-formate

C25H32O6 (428.53). Colorless needles, mp 147~150C, []D19 = 11.5 (c = 0.1,
CHCl3). Pharm: Cytotoxic (in vitro, KB, IC50 > 25g/mL; MH-60, IC50 >
25g/mL). Source: CHAN SU Bufo bufo gargarizans; Bufo melanostictus
(dried secretion of skin glands: yield = 0.00082%dw). Ref: 4634.
O
O
O
O
H
O
O
O
H
H
H
O
286
7191 20S,21-Epoxyresibufogenin 3-formate
7195 3,4-Epoxyrupicolin C
C25H32O6 (428.53). Colorless needles, mp 180~182C, []D19 = +17.2 (c = 0.1,
8-Angeloyloxy-1-hydroxy-3,4-epoxy-5,7H-10(14),11(13)-guaiadien-12
CHCl3). Pharm: Cytotoxic (in vitro, KB, IC50 > 25g/mL; MH-60, IC50 >
,6-olide C20H24O6 (360.41). White amorphous powder, mp 88~89C, []D25 =
25g/mL). Source: CHAN SU Bufo bufo gargarizans; Bufo melanostictus
5.83 (c = 0.03, MeOH). Pharm: Anti-inflammatory (RAW264.7 cells,
LPS-induced: NF-B inhibitor, IC50 = (0.890.02)mol/L, control PTN, IC50

= (3.420.08)mol/L; NO production inhibitor, IC50 = (2.340.05)mol/L,
PTN, IC50 = (2.410.06)mol/L, AG, IC50 = (34.180.98)mol/L; TNF-

production inhibitor, IC50 = (7.580.22)mol/L, PTN, IC50 =
(2.680.11)mol/L). Source: LIN DI HAO Artemisia sylvatica (aerial parts).

O
H
Ref: 3837.
O
O
O
O
HO
7192 20R,21-Epoxyresibufogenin
C24H32O5 (400.52). Colorless needles, mp 90~94C, []D19 = 17.0 (c = 0.1,
CHCl3). Pharm: Cytotoxic (in vitro, KB, IC50 = 8.09g/mL; MH-60, IC50 =
1.8g/mL). Source: CHAN SU Bufo bufo gargarizans; Bufo melanostictus
H O
7196 3,4-Epoxyrupicolin D
8-Methybutyryloxy-1-hydroxy-3,4-epoxy-5,7H-10(14),11(13)-guaiadi
LPS-induced: NF-B inhibitor, IC50 = (2.730.01)mol/L, control PTN, IC50
O
HO
en-12,6-olide C20H26O6 (362.43). White needles, mp 118~119C, []D25 =

Ref: 3837.
7193 20S,21-Epoxyresibufogenin
C24H32O5 (400.52). Colorless plates, mp 184~186C, []D18 = +18.2 (c = 0.1,
CHCl3). Pharm: Cytotoxic (in vitro, KB, IC50 = 10.88g/mL; MH-60, IC50 =
1.82g/mL). Source: CHAN SU Bufo bufo gargarizans; Bufo melanostictus
O
O
H
H
HO
O
HO
H O
7197 3,4-Epoxyrupicolin E
8-Sovaleryloxy-1-hydroxy-3,4-epoxy-5,7H-10(14),11(13)-guaiadien-1
2,6-olide C20H26O6 (362.43). White needles, mp 117~118C, []D25 =

LPS-induced: NF-kB inhibitor, IC50 = (2.680.06)mol/L, control PTN, IC50
7194 (3R,15R)-ent-15,16-Epoxy-1(10)-rosen-3-ol
C20H32O2 (304.48). []D20 = 4.9 (c = 0.78, CHCl3). Source: Heteroscyphus
billardierii, Plagiochila deltoidea. Ref: 4284.

Ref: 3837.
O
O
HO
HO
H
H O
O
287
7198 Epoxysarcovagenine D
7203 Epoxysuberosin
(20S)-20-(N-Methylamino)-3-(tigloylamino)-5-pregna-2-en-16,17-epoxy
-4-one C27H40N2O3 (440.63). Yellowish amorphous solid (CHCl3), mp
119~120 C, []D25 = +24 (c = 0.116, CHCl3). Source: YUN NAN YE SHAN
HUA Sarcococca coriacea [Syn. Sarcococca wallichii] (leaf). Ref: 4241.

H H
N
O
H
O
H
N
H
Source: Citrus tamurana. Ref: 5048.

H
O
O
7199 15,16-Epoxy-5,10-seco-clerodan-1(10),2,4,13(16),14-pentaen-18,19-
7204 1,2-Epoxytagitinin C
olide
C19H24O7 (364.4). Pharm: Cytotoxic (antiproliferative, Col2 cells, IC50 =

1.7g/mL); cytotoxic (cellular differentiation inducer, hmn promyelocytic

leukemia HL-60 cells, 4g/mL, activity denotes percentage of cells
differentiated < 10%); cytotoxic (MMOC model, inhibits DMBA-induced
preneoplastic lesion formation, 10g/mL, rel-InRt = 44.4%, control DMBA,
rel-InRt =100%). Source: ZHONG BIN JU Tithonia diversifolia (aerial parts:

yield = 0.0013%dw). Ref: 4622.
OH
7200 2,3-Epoxysesamone
C15H14O5 (274.28). Pale yellow crystals (MeOH), mp 85~86C, []D25 = 43
(c = 0.34, CHCl3). Pharm: Antifungal (Cladosporium fulvum, 10g/spot)[5234].

Source: HU MA GEN Sesamum indicum. Ref: 5234.
7205 20,21-Epoxy-taraxastane-3,22-diol
C30H50O3 (458.73). Colorless crystals, mp 223~224C (CHCl3MeOH), []D25 =
OH
+121 (c = 0.56, CHCl3). Pharm: Cytotoxic (SMMC-7721, IC50 =
(113.64.3)g/mL, control Vincristine, IC50 = (63.21.8)g/mL; B16, IC50 =

(51.43.7)g/mL, Vincristine, IC50 = (70.72.8)g/mL; HeLa, IC50 =
(88.76.0)g/mL, Vincristine, IC50 = (67.22.2)g/mL); antibacterial (Bacillus

OH
subtilis, IZD = (13.90.8)mm, control Chloramphenicol, IZD = (14.51.1)mm;

Escherichia coli, IZD = (14.12.9)mm, Chloramphenicol, IZD = (14.91.3)mm;
7201 Epoxyshikoccin
C22H30O6 (390.48). mp 124~126C, []D = 6.3 (c = 0.35, MeOH).
Staphylococcus aureus, IZD = (10.52.1)mm, Chloramphenicol, IZD =
Source: XI SI GUO XIANG CHA CAI Isodon shikokiana var. occidentalis.
(15.11.2)mm). Source: Saussurea petrovii (whole herb). Ref: 5219.
25
Ref: 4067.
O
O
O
O
OH
7202 16,17-Epoxyshikokianal acetate

C26H34O10 (506.55). mp 205.0~206.5C, []D20 = +66 (c = 0.32, CHCl3).
Source: SI GUO XIANG CHA CAI Rabdosia shikokiana. Ref: 4067.
H
HO
7206 1,2-Epoxy-3,4,8,10-tetrahydroxyguaia-11(13)-en-12,6-olide
Antifungal (Candida albicans, MIC = 20g/mL)[5222]. Source: GUAN MU YA
OH
O
H
OH
HO
HO
OH
JU Ajania fruticulosa (aerial parts). Ref: 5222.
18
O
O
288
7207 1,2-Epoxy-3,4,9,10-tetrahydroxyguaia-11(13)-en-12,6-olide
7211 6,7-Epoxy-3,5,17-trihydroxy-1-oxo-witha-24-enolide
C28H40O7 (488.63). mp 258C, []D30 = +66.00 (c = 0.25, MeOH). Source:
Antifungal (Candida albicans, MIC = 20g/mL). Source: GUAN MU YA JU
Ajania fruticulosa (aerial parts). Ref: 5222.

OH OH
H
OH
HO
H
HO
7208 22,23-Epoxy-tirucalla-7-ene-3,24,25-triol
C30H50O4 (474.73). Colorless needles (Me2CO), mp 118~120C, []D26 = 4.7
(c = 0.95, CH3OH). Source: HAI NAN JIAN MU Dysoxylum hainanense
(bark). Ref: 3987.
HO
O
OH
7212 (20S,22R)-3,6-Epoxy-4,5,27-trihydroxy-1-oxowitha-24-enolide
MeOH). Pharm: Neurite outgrowth activity (hmn neuroblastoma
SH-SY5Y cell line, 1mol/L). Source: CUI MIAN SHUI QIE Withania
somnifera (root). Ref: 4198.
OH
OH
OH
H
O
H
O
HO
7209 4(R),23-Epoxy-2,3,19-trihydroxy-24-norurs-12-en-28-oic acid

25
H
H
H
H
OH
OH
C29H44O6 (488.67). White powder, mp 232~234C, []D = +33.4 (c = 0.05,

MeOH). Source: YANG TI Rumex japonicus (stem). Ref: 4541.
7213 6,7-Epoxy-3,5,20-trihydroxy-1-oxowitha-24-enolide
C28H40O7 (488.63). White amorphous powder, []D25 = 196 (c = 0.006,
HO
MeOH). Pharm: AChE inhibitor inactive; BChE inhibitor inactive. Source:

CUI MIAN SHUI QIE Withania somnifera. Ref: 2563.
O
HO
OH
H
HO
O
OH
H
O
H
H
7210 5,6-Epoxy-4,17,27-trihydroxy-1-oxowitha-2,24-dienolide
HO
17-Hydroxy withaferin C28H38O7 (486.61). White amorphous powder, []D25 =
OH
H
H
+12 (c = 0.11, CH2Cl2). Pharm: BChE inhibitor (IC50 = (161.51.1)mol/L,

control Galanthamine, IC50 = (0.500.001)mol/L, Eserine IC50 =
7214 (20S,22R)-5,6-epoxy-4,14,15-trihydroxy-1-oxowith-2,24-di-
(0.040.00)mol/L) [2563]; AChE inhibitor inactive[2563]. Source: CUI MIAN
enolide
SHUI QIE Withania somnifera, CUI MIAN SHUI QIE Withania somnifera
C28H38O7 (486.61). Colorless needles, []D = +68 (c = 0.2,MeOH). Source:
(leaf). Ref: 2563, 5329.
DENG LONG CAO Physalis peruviana. Ref: 1915.

OH
H
OH O
H
O
H
OH
O
OH
H
OH
OH
289
7215 ent-12,16-Epoxy-2,15,19-trihydroxypimar-8-ene
7220 14S*,15-Epoxyvibsanin C
MeOH). Source: XI XIAN Siegesbeckia orientalis (aerial parts: yield =
XIANG QI JIA MI Viburnum odoratissimum (leaf). Ref: 3512.
0.00033%). Ref: 4764.

O
O
O
OH
OH
O
O
HO
H
O
H
OH
7221 Equisetin
7216 ent-12,16-Epoxy-2,15,19-trihydroxypimar-8(14)-ene
[57749-43-6] C22H31NO4 (373.50). Amorphous powder, mp 65~66C. Pharm:
Antibacterial (gram-positive bacteria). Source: Fusarium equiseta. Ref: 2094.
MeOH). Source: XI XIAN Siegesbeckia orientalis (aerial parts: yield =

OH
0.00083%). Ref: 4764.

O
HO
OH
HO
H
H
OH
7222 Equisetrin
7217 3,6-Epoxy-5,3',4'-trihydroxy-12',13',20'-trinor-,-caroten-19,11-olide
C27H30O16 (610.53). mp 195~196C. Source: WEN JING Equisetum arvense.
C37H48O6 (588.79). Reddish solid. Source: MU LI (Oyster) Crassostrea gigas.
Ref: 6, 1521.
Ref: 4515.
OH
O
OH
OH
O
O
OH
HO
OO
OH
OH
OH
7218 (9S,10S)-ent-9,10-Epoxyverticillol
C20H34O2 (306.49). Colorless crystals (n-hexane), mp 157~158C, [] D18 =
114.2 (c = 1.81). Source: ZHAO WA JIA KE TAI Jackiella javanica. Ref:
OO
OH
OH
OH
OH
OH
7223 Erectquione A
2,6-Dihydroxyl-3-geranyl-5-isoprenyl-2,5-dihexadiene-1,4-dione C21H28O4
(344.45). Red oil. Source: XIAO LIAN QIAO Hypericum erectum. Ref: 1990.
5303.
O
OH
HO
OH
O
H
7224 Erectquione B
7219 14R*,15-Epoxyvibsanin C
2,6-Diisobutyryloxy-3-geranyl-5-isoprenyl-2,5-dihexadiene-1,4-dione
C29H40O6 (484.64). Yellow oil. Source: XIAO LIAN QIAO Hypericum
XIANG QI JIA MI Viburnum odoratissimum (leaf). Ref: 3512.
erectum. Ref: 1990.
OH
H
O
290
7225 Erectquione C
7231 Ergochrysin
C25H34O6 (430.55). Yellow oil, []D25 = 10 (c = 0.10, CHCl3). Source: XIAO
C31H28O14 (624.56). mp 285C (dec). Source: MAI JIAO Claviceps purpurea.
LIAN QIAO Hypericum erectum. Ref: 1990.
Ref: 6.
HO
O
O
OH
O
O
O
OH
OH
OH
OH
OH
7226 Eremanthin
Vanillosmin [37936-58-6] C15H18O2 (230.31). Pharm: Schistosomacide.
7232 Ergocornine
Source: Vernonia sp. Ref: 658.
[564-36-3] C31H39N5O5 (561.69). mp 181~184C (dec). Pharm: Antineoplastic

(rat, mammary cancer caused by DMBA); inhibits release of galactin; uterine
stimulant; contracts blood vessels. Source: MAI JIAO Claviceps purpurea,

WU ZHAO LONG Ipomoea cairica [Syn. Ipomoea palmata]. Ref: 5, 6, 658.
O
O
7227 Eremofukinone
N
O
OH
C15H24O (220.36). bp 75~100C/0.15mmHg. Source: FENG DOU CAI
N
H
Petasites japonicus. Ref: 6.
N
H
H
7233 Ergocorninine
[564-37-4] C31H41N5O5 (563.70). mp 228C (dec). Source: MAI JIAO
Claviceps purpurea. Ref: 6.
7228 8H-Eremophil-3,7(11)-diene-12,8(14,6)-diolide
C15H16O4 (260.29). Colorless plates, mp 230~231C, []D20 = +28.0 (c = 0.20,
CHCl3). Source: DONG E LUO DU WU Ligularia tongolensis (root). Ref:
4523.
N
O
OH
N
H
O
O
N
H
O
O
7229 Eremophilene
C15H24 (204.36). bp 129.5C/13mmHg. Source: DU HUO Angelica pubescens
f. biserrata [Syn. Angelica pubescens], FENG DOU CAI Petasites japonicus,
XIE CAO Valeriana officinalis. Ref: 2.
7234 Ergocristine
[511-08-0] C35H39N5O5 (609.73). mp 165~170C (dec). Pharm: Contracts
blood vessels (similar physiological activity with ergot); inhibits release of
galactin. Source: MAI JIAO Claviceps purpurea. Ref: 6, 658.
7230 Eremophilenolide
C15H22O2 (234.34). Pharm: Antispasmodic. Source: Petasites sp. Ref: 658.
H
N
O
OH
O
N
H
O
N
O
O
291
7235 Ergocristinine
7239 Ergolide
[54999-07-4] C17H22O5 (306.36). White acicular crystals, mp 169~170C, []D
= +133 (c = 1.26, CH2Cl2). Pharm: Anti-inflammatory (NF-B pathway)[4415];

anti-inflammatory (NO production inhibitor)[4415]. Source: SHUI CHAO
YANG Inula helianthus-aquatica. Ref: 430, 4415.
O
O
N
N
H
O
OH
O
N
O
H
O
H
7240 Ergometrine
Ergobasine; Ergonovine; Ergostetrine; Ergoklinine; Ergotrate; Syntometrine

[60-79-7] C19H23N3O2 (325.41). Tetrahedral crystals (acetic ester), acicular
7236 Ergocryptine
Ergokryptine [511-09-1] C32H41N5O5 (575.71). Combining with solvent,
prismatic crystals (acetone or benzene or methanol); recrystallization in
methanol, mp 212C (dec), []D20 = 120 (pyridine); []D20 = 198
(chloroform). Pharm: Antineoplastic; galactin inhibitor (female sheep); toxin.
Source: MAI JIAO Claviceps purpurea. Ref: 5, 6, 658.
crystals (benzene), mp 162C, [] D20 = 16 (c = 1, peridine), []D20 = 44

(chloroform), []D20 = +42 (ethanol), easily soluble in methanol, ethanol,
acetic ester, acetone, slightly soluble in chloroform.[5507] Pharm: Inhibits
release of galactin; similar action with arterenol to nerve system; uterine
stimulant; used in treatment of post-partum uterus bleeding. Source: MAI
JIAO Claviceps purpurea, YIN YE SHU Ipomoea argyrophylla MO XI GE
XUAN HUA River corymbosa (the compound was isolated from the plant by
A.Hofmann, et al. in 1961)[5505]. Ref: 4, 658, 5505, 5507.
O
N
N
H
O
OH
HO
N
H H
NH
N
H
7241 Ergometrinine
7237 Ergoflavine
[479-00-5] C19H23N3O2 (325.41). mp (+) 195~197C (dec). Source: MAI
C30H26O14 (610.53). mp 350C (dec). Source: MAI JIAO Claviceps purpurea.
JIAO Claviceps purpurea. Ref: 6.
Ref: 6.
HO
OH
O
OH
OH
O OH
NH
O
OH
O
OH
NH
7238 -Ergokryptinine
[511-10-4] C32H41N5O5 (575.71). mp 240~242C (dec). Source: MAI JIAO
7242 Ergosecalinine
C24H28N4O4 (436.52). mp 217C (dec). Source: MAI JIAO Claviceps
purpurea. Ref: 6.
O
N
N
O
OH
N
H
N
H
NH
O
N
H
H
N
O
N
H
292
7243 Ergosine
7248 (24S)-Ergost-5-en-3,7-diol
[561-94-4] C30H37N5O5 (547.66). mp 228C (dec). Pharm: Anti-fertility agent
C28H48O2 (416.69). Colorless crystals, mp 211~213C, [] D28 = 64.1 (c =
(rat, sc); anti-inflammatory (rat, swollen foot model caused by 5-HT and
0.05, CHCl3). Source: Lobophytum sp. Ref: 4432.
carrageenan); 5-HT receptor blocker (gpg uterus in vitro); adrenergic -receptor

blocker (gpg testis in vitro); contracts blood vessels and Increases blood pressure
(cat, iv); inhibits release of galactin; oxytocic (rbt uterus iv, in vivo); similar
action with ergotamine. Source: MAI JIAO Claviceps purpurea. Ref: 6, 658.
N
HO
O
N
H
HN
HO
7249 Ergost-7-en-3-one
5,8-Epi-dioxyergost-6-en-3-ol C28H46O (398.68). Source: MU TI CENG
KONG JUN Fomes fomentarius [Syn. Pyropolyporus fomentarius; Boletus
fomentarius; Polyporus fomentarius]. Ref: 3972.
OH
7244 Ergosinine

O
N
H
O
HN
H
H
O
OH
N
7250 Ergosterol
O
(22E)-Ergosta-5,7,22-trien-3-ol [57-87-4] C28H44O (396.66). mp 163C. Pharm:

Transforms into vitamin D2 under ultraviolet ray. Source: A LI HONG Fomes
officinalis, BAI JIANG CAN Bombyx mori, BAI QU CAI Chelidonium majus,
7245 22E,24R-Ergosta-7,22-diene-3,5,6,9-tetraol
C28H46O4 (446.68). White powder. Source: DUO ZHI RU GU Lactarius
DONG CHONG XIA CAO Cordyceps sinensis (dried fungal stroma growing on
larva of a caterpillar: content = 0.213%[5508]), FU LING Poria cocos, JI ZONG
Collybia albuminosa, LING ZHI Ganoderma lucidum, MA BO Lasiosphaera
rolemus. Ref: 752.
fenzlii, MAI JIAO Claviceps purpurea, MU ER Auricularia auricula, NIU

HUANG Bos taurus domesticus; Bubalus bubalis, REN GONG YONG
H
CHONG CAO Cordyceps militaris cv. (sclerotium and stroma: content =

0.210%)[5508], SANG HUANG Phellinus igniarius, SHUANG BAO MO GU
Agaricus bisporus, SONG XUN Tricholoma matsutake [Syn. Armillaria
OH
HO
OH
OH
matsutake], XIANG XUN Lentinus edodes, YONG CHONG CAO Cordyceps

militaris (sclerotium and stroma: content = 0.226%)[5508], YUAN CAN SHA
Bombyx mori, ZHEN MO Armillariella mellea, ZHU LING Polyporus
7246 Ergosta-7,22-dien-3-yl pentadecanoate
umbellatus, ZI ZHI Ganoderma japonicum [Syn. Ganoderma sinense], occurs in
C43H74O2 (623.07). White powder, mp 113~115C. Source: LING ZHI
many plants. Ref: 2, 6, 587, 660, 1407, 5508.
Ganoderma lucidum (sporocarp). Ref: 4810.
HO
7251 Ergosterol peroxide

O
5,8-Epidioxyergosta-6,22-dien-3-ol [2061-64-5] C28H44O3 (428.66). Colorless
7247 Ergosta-4,6,8(14),22-tetraen-3-one
acicular crystals, mp 182~184C, mp 165~169C, []D25 = 34 (c = 0.6, CHCl3).
[19254-69-4] C28H40O (392.63). mp 114~115C. Source: A LI HONG Fomes
Pharm: Anti-HIV-1 (weakly). Source: LING ZHI Ganoderma lucidum (dried
officinalis, LING Trapa bispinosa, ZHU LING Polyporus umbellatus. Ref: 2, 6.
sporocarp: yield = 0.003%)[4603], ZI DING XIANG MO Lepista nuda, Pleurotus

eryngii, Antrodia camphorata (fruit: yield = 0.060%dw). Ref: 2169, 3003, 4183, 4603.
H
H
O
O
HO
293
7252 Ergotamine
7256 Erigerenone B
[113-15-5] C33H35N5O5 (581.68). mp 212~214C (dec). Pharm: Adrenergic
receptor blocker (large dose, to turn over boost pressure action due to
FEI CHENG FEI PENG Erigeron philadelphicus, YI NIAN PENG Erigeron
adrenalin); smooth muscle stimulant (peripheral blood vessel in vitro);
annuus, SU MEN BAI JIU CAO Erigeron sumatrensis (aerial parts). Ref:
relieves headache (recovers normal for over-dilation and excess beat of
4366.
cerebral arteries); uterine stimulant; toxin (damages vascular endothelial cells

in high dose). Source: MAI JIAO Claviceps purpurea. Ref: 4, 658.
O
O
O
O
N
NH
O
OH
7257 Erigerenone C
H

FEI CHENG FEI PENG Erigeron philadelphicus (aerial parts). Ref: 4366.
N
H
7253 Ergotaminine
7258 Erigerol
C25H40O6 (436.59). Source: FEI CHENG FEI PENG Erigeron philadelphicus
O
N
O
N
H
O
OH

N
HO H
7254 Ergothioneine
N
H
O
H
OH
[497-30-3] C9H15N3O2S (229.30). mp 290C (dec). Source: MAI JIAO

7259 Erinacerin A
C27H31NO4 (433.55). Colorless oil, []D21 = +0 (c = 0.4, MeOH). Source:
O
O
+
HOU TOU JUN Hericium erinaceus [Syn. Hydnum erinaceus]. Ref: 4513.
H
N
N
SH
N
O
7255 Erigerenone A
FEI CHENG FEI PENG Erigeron philadelphicus (aerial parts). Ref: 4366.
7260 Erinacerin B
C19H24O5 (332.40). Amorphous powder, []D24 = +12.7 (c = 0.2, MeOH). Source:
HOU TOU JUN Hericium erinaceus [Syn. Hydnum erinaceus]. Ref: 4513.
OH
OH
O
O
O
O
O
O
294
7261 Erinacine A
7265 Erinacine G
Erinacin A [156101-08-5] C25H36O6 (432.56). White crystals mp 74~76C,
Erinacin G [182927-59-9] C25H36O8 (464.56). []D25 = 13 (c = 0.25,
[]D = +216 (c = 0.28, methanol). Pharm: Stimulates synthesis of NGF (mus
methanol). Source: HOU TOU JUN Hericium erinaceus [Syn. Hydnum
neuroglia astrocytes in vitro, 1.0 mmol/L, NGF = 250.1pg/mL, comparing
erinaceus]. Ref: 1521.

H
with adrenaline NGF = 69.2pg/mL) Source: HOU TOU JUN Hericium
O
OH
erinaceus [Syn. Hydnum erinaceus]. Ref: 948, 1174.
OH
H
O
OH
OH
7266 Erinoside
C16H20O11 (388.33). Amorphous solid. Source: Erinus alpinus (frozen whole
OO
O
herb). Ref: 5291.
OH
OH
OH
OH
O
HO
7262 Erinacine B
O HO
OO
OH
Erinacin B [156101-10-9] C25H36O6 (432.56). White crystals mp 125~127C,

[]D = 34.9 (c = 0.18, methanol). Pharm: Stimulates synthesis of NGF (rat
OH
spider neuroglia cell in vitro, 1.0 mmol/L, NGF = 129pg/mL, comparing with
OH
adrenaline NGF = 69pg/mL) Source: HOU TOU JUN Hericium erinaceus
7267 Eriocalysin A
[Syn. Hydnum erinaceus]. Ref: 948, 1174.
C20H24O5 (344.41). mp 242~244C, []D18.5 = +157.2 (c = 0.127, CHCl3).

Source: MAO E XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.
O
OH
OH
7268 Eriocalysin B
Rabdosianone C20H24O5 (344.41). mp 216~218C, []D18.5 = 185.2 (c = 0.108,
7263 Erinacine C
Erinacin C [156101-09-6] C25H38O6 (434.58). White crystals mp 115~118C,
CHCl3). Source: MAO E XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.
O
[]D = 72.5 (c = 0.73, methanol). Pharm: Stimulates synthesis of NGF (mus
spider neuroglia cell in vitro, 1.0 mmol/L, NGF = 299pg/mL, comparing with
adrenaline NGF = 69.2pg/mL) Source: HOU TOU JUN Hericium erinaceus

H
[Syn. Hydnum erinaceus]. Ref: 948, 1174.
O
OH
OH
7269 Eriocalysin C
C22H28O7 (404.46). mp 191.5~192.5C, []D22 = 67.1 (c = 0.26, MeOH).
OH

O
OH
OH
O
7264 Erinacine E
Erinacin E [178232-25-2] C25H36O6 (432.56). mp 161~163C, []D25 = 114
(c = 0.50, methanol). Pharm: Stimulates synthesis of NGF (rat spider
neuroglia cell in vitro, 5.0 mmol/L, NGF = 105pg/mL) Source: HOU TOU
JUN Hericium erinaceus [Syn. Hydnum erinaceus]. Ref: 1175.
H
O
OH
O
H
H
OH
OH
7270 Eriocalysin D
MAO E XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.
OH
H
O
OH
OH
O
OH
O
295
7271 Eriocalysin E
7276 Eriodictyl 7-O--D-(6'-ethyl ester)-glucuronopyranoside
C22H26O6 (386.45). mp 178~179.5C, []D23 = +92.7 (c = 0.27, MeOH).
C23H24O12 (492.44). Yellow needles (MeOH), mp 158~161C, []D20 = 58.1
(c = 0.56, MeOH). Source: NIU JIN TIAO Dichotomanthes tristaniaecarpa.

Ref: 2263.
O
H
H
O
OH
OO
OH
OH
7272 Eriocarpin
OH
OH
Desglucosyrioside C29H38O11 (562.62). Pharm: LD50 (male Swiss Webster
OH
mus, ip) = 6.5mg/kg. Source: MAO GUO MA LI JIN Asclepias eriocarpa.

Ref: 658.
7277 Eriodictyl 7-O--D-(6'-methyl ester)-glucuronopyranoside

O
OH
OH H
O
(c = 0.61, MeOH). Source: NIU JIN TIAO Dichotomanthes tristaniaecarpa.
O
OH
O OH
H
O
C22H22O12 (478.41). Yellow needles (MeOH), mp 121~123C, []D = 71.3

Ref: 2263.
OH
OO
OH
OH
7273 Eriocarpin B
3,15,23-Trihydroxy-olean-12-en-16-one C30H48O4 (472.71). Colorless
OH
OH
OH
crystals (MeOH), R[20, D] = +11.02 (c = 0.003, MeOH); colorless lamellar
crystals, mp 218~220C. Source: MAO GUO YU TENG Derris eriocarpa,

YUN NAN GE TENG Pueraria peduncularis. Ref: 665, 2262.
7278 Eriodictyol
[552-58-9] C15H12O6 (288.26). mp 267C. Pharm: Antibacterial
(Pseudomonas maltophilia, Enterobacter cloacae); diuretic (rbt); induces
gene expression of pea nodule bacteria and accrete host Pisum sativum;
larvacide (inhibits Heliothis zea larva growth); aldose reductase inhibitor (rat
H
H
HO
eye lens, 10-5mg/L, InRt = 90%); anti-inflammatory (modulator of cytokine
O
OH
network: inhibits LPS-stimulated TNF- release in RAW264.7 macrophages,
IC50 50mol/L)[4416]. Source: BA DAN XING REN Prunus amygdalus, DA
HO
CHI JI Onopordum acanthium, HUANG QIN Scutellaria baicalensis, JIN JI
7274 Eriocarpin C
ZE LAN Eupatorium subhastatum, LI MU Lyonia ovalifolia, OU BO HE
15-Hydroxy-16-oxo-olean-12(13)-en-3-O--glucuronopyranoside C36H56O9
Mentha longifolia, YOU GAN YE Phyllanthus emblica (branch and leaf). Ref:
(632.84). Colorless crystals (MeOH), R[20, D] = 20.67 (c = 0.0052, MeOH).
6, 658, 660, 4205, 4416.
Source: MAO GUO YU TENG Derris eriocarpa. Ref: 2262.

OH
O
HO
OH
H
OH
OO
OH
OH
OH
OH
7279 (S)-Eriodictyol-7-O-(6''-O-trans-p-coumaroyl)--D-glucopyranoside
OH
C30H28O13 (596.55). Yellow amorphous powder, []D28 = 92.8 (c = 0.36, MeOH).
7275 Eriocaside A
C26H44O10 (516.63). []D21 = +0.83 (c = 0.12, MeOH). Source: MAO E
Source: YOU GAN YE Phyllanthus emblica (branch and leaf). Ref: 4205.
XIANG CHA CAI Rabdosia eriocalyx. Ref: 4067.

H
H
OH
OH
OH
OH
O
OH
O
O
OO
OH
HO
OO
OH
OH
OH
H
OH
OH
OH
OH
OH
296
7280 (2R)-Eriodictyol-7,4'-di-O--D-glucopyranoside
7284 (2S)-Eriodictyol-7-O--D-glucopyranosiduronic acid
C27H32O16 (612.55). Pale yellow amorphous solid. Pharm: Antioxidant
C21H20O12 (464.39). Yellow powder, []D26 = 35.6 (c = 0.20, MeOH).
(hydroxyl radical, IC50 = 0.18mmol/L, control EGCG, IC50 = 0.58mmol/L;
Pharm: Aldose reductase inhibitor (rat lens, IC50 = 2.1mol/L, control
superoxide anion, IC50 = 0.25mmol/L, EGCG, IC50 = 0.53mmol/L). Source:
Epalrestat, IC50 = 0.072mol/L). Source: YE JU HUA Chrysanthemum
HU JI SHENG Viscum coloratum (branch and leaf: yield = 0.0008%dw).
indicum (flower: yield = 0.0027%). Ref: 4214.
Ref: 920.
OH
OH
OH
HO
OO
OO
HO
O
HO
OH
OH
OH
OH
OH
OH
OH
OH
OH
OH
OH
7285 Eriodictyol-7-glucoside
7281 Eriodictyol-7,3-diglucoside
[In DNP] C21H22O11 (450.40). mp 175~177C. Source: SHUI YANG ZHI
C27H32O17 (628.55). Source: SHAN ZHA Crataegus pinnatifida. Ref: 2.
YE Salix purpurea, YOU GAN YE Phyllanthus emblica (branch and leaf).

Ref: 6, 4205.
OH
OH
HO
OO
OH
OH
OH
OH
HO
OH
OH
OH
O
HO
OO
OH
OH
OH
OH
OH
7286 Erioflorin
OH
C19H24O6 (348.40). Source: Viguiera eriophora ssp. eriophora (aerial parts),
7282 (S)-Eriodictyol-7-O-(6''-O-galloyl)--D-glucopyranoside
C28H26 O15 (602.51). Yellow amorphous powder, []D28 = 79.4 (c = 0.41,
Viguiera puruana (aerial parts). Ref: 5090.
MeOH). Source: YOU GAN YE Phyllanthus emblica (branch and leaf).
Ref: 4205.
OH
OH
HO
OO
OH
OH
7287 Eriojaposide A
OH
OH
(6R,9R)-3-Oxo--ionyl-9-O--xylopyranosyl-(1''6')--glucopyranoside
OH
HO
OH
Source: PI PA YE Eriobotrya japonica (branch and leaf). Ref: 3061.
7283 (2R)-Eriodictyol-7-O--D-glucopyranosiduronic acid

C21H20O12 (464.39). Yellow powder, []D24 = 54.5 (c = 0.10, MeOH).
Pharm: Aldose reductase inhibitor (rat lens, IC50 = 1.5mol/L, control

Epalrestat, IC50 = 0.072mol/L)[4214]. Source: LU SHAN SHI WEI Pyrrosia
sheareri (dried leaf: content = 0.043%)
[5508]
, SHI WEI Pyrrosia lingua (dried
HO
HO
leaf: content scope of 3 origins = 0.026%~0.168%, mean content =

0.0763%)[5508], XI NAN SHI WEI Pyrrosia gralla (dried leaf: content =
0.037%)[5508], YE JU HUA Chrysanthemum indicum (flower-head: yield =
0.0023%)[4214], YOU BING SHI WEI Pyrrosia petiolosa (dried leaf: content
scope of 12 origins = 0.861%~2.743%, mean content = 1.613%)
[5508]
, ZHAN
MAO SHI WEI Pyrrosia drakeana (dried leaf: content = 0.051%)[5508]. Ref:
O
O O
HO
HO
OH
OH
7288 Eriojaposide B
(6R,9R)-3-Oxo--ionyl-9-O--rhamnopyranosyl-(1''6')--glucopyranoside
Source: PI PA YE Eriobotrya japonica (branch and leaf). Ref: 3061.
4214, 5508.
OH
OH
HO
OO
OH
OH
HO
OH
OH
HO
O
HO
HO
O
OH
OH
297
7289 Erosnine
7294 Ervahanine A
[In DNP] C18H8O6 (320.26). mp 350C (dec). Source: DI GUA ZI
C42H50N4O4 (674.89). Source: SAN FANG HUA XU HONG YUE GUI
Pachyrhizus erosus. Ref: 6.
Tabernaemontana corymbosa. Ref: 3403.
O
O
N
H H
O
N
7290 Erosone
[15236-21-2] C20H16O6 (352.35). mp 218C. Source: DI GUA ZI Pachyrhizus
N
H
erosus. Ref: 6.
H
H
7295 Erybraedin C
C25H28O4 (392.50). []D25 = 17 (c = 0.5, MeOH). Pharm: Cytotoxic (KB,

O
IC50 = (23.70.5)mol/L, control Helenalin, IC 50 = (0.640.08)mol/L,
Melphalan, IC50 = (6.00.5)mol/L; Mono-Mac-6, IC 50 =
(28.61.4)mol/L, Helenalin, IC 50 = (3.10.3)mol/L; Jurkat-T, IC 50 =
7291 Erucic acid
(21.40.5)mol/L, Helenalin, IC 50 = (1.140.08)mol/L, Melphalan, IC50
cis-13-Docosenoic acid [112-86-7] C22H42O2 (338.58). mp 33.5~34.0C, bp
= (9.10.8)mol/L). Source: Bituminaria morisiana (leaf). Ref: 5077.
241~243C/5mmHg. Source: BO NIANG HAO Descurainia sophia, GUI

ZHU XIANG Cheiranthus cheiri, HAN LIAN HUA Tropaeolum majus, LAI
FU ZI Raphanus sativus, YUN TAI ZI Brassica campestris [Syn. Brassica
HO
campestris var. oleifera]. Ref: 6, 658, 660.
O
H
OH
OH
7296 Erychroside
[630-65-9] C34H50O13 (666.77). mp 243~246C, []D = +18 (methanol).
Pharm: Cardiotonic; antihypertensive. Source: GUI ZHU TANG JIE
Erysimum cheiranthoides. Ref: 6, 661.
H
H
7292 Ervadivaricatine A
C43H56N4O5 (708.95). mp 217~220C. Source: DAN BAN GOU YA HUA
Ervatamia divaricata. Ref: 802.
H
H
OO
H
O
H
O
H
N
N
H
OH
OH
OO
OH
OH
OH
N
O
OH
7297 Erychrosol
7293 Ervadivaricatine B
C34H52O13 (668.79). Source: GUI ZHU TANG JIE Erysimum cheiranthoides. Ref: 6.
C43H56N4O5 (708.95). mp 190C. Source: DAN BAN GOU YA HUA

O
Ervatamia divaricata. Ref: 802.

O
HO
H
O
H
O
H
N
N
H
OO
OH
OO
OH
OH
N
O
OH
OH
OH
298
7298 Erycibe alkaloid II
7303 Erycordine
C10H17NO3 (199.25). White mucilage, []D20 = 5.56 (c = 0.90, CHCl3);
[13428-83-6] C35H54O14 (698.81). Pharm: Cardiotonic; increases coronary
benzoate: white tiny acicular crystals (benzene or acetone), mp 160~161C.
flow; antihypertensive. Source: GUI ZHU TANG JIE Erysimum
Pharm: Antihypertensive (rbt, iv, 0.5mL of 0.025% solution); causes miosis.
cheiranthoides, HUAN YANG SHEN YE TANG JIE Erysimum crepidifolium.
Source: DING GONG TENG Erycibe obtusifolia. Ref: 661.
Ref: 6, 658.
OH
O
O
HO
7299 Erycibelline
2,7-Dihydroxynortropane [107633-95-4] C7H13NO2 (143.19). Alkaline
OO
colorless oleaginous, []D10 = 12.5 (c = 0.57, ethanol). Source: AO MAI

DING GONG TENG Erycibe elliptilimba. Ref: 68.
OH
HO
OO
OH
OH
NH
OH
OH
OH
HO
OH
7304 Erycristagallin
7300 Erycibenin A
C25H26O4 (390.48). mp 179~180C. Pharm: Antimalarial (antiplasmodial in
C20H20O7 (372.38). Pharm: Hepatoprotective (mus primary cultured
vitro, Plasmodium falciparum, W2 strain, IC50 = (20.13.6)mol/L, control
hepatocytes, antihepatotoxin induced by D-galactosamine (GalN), IC50 =
Quinine, IC50 = (0.210.01)mol/L; D6 strain, IC50 = (19.00.9)mol/L,
79mol/L, control Silybin IC50 = 41mol/L). Source: GUANG BU DING
Quinine, IC50 = (0.0420.002)mol/L). Source: A BI XI NI YA CI TONG
GONG TENG Erycibe expansa. Ref: 4095.
Erythrina abyssinica (root cortex). Ref: 5420.
HO
O
O
HO
OH
OH
HO
OH
OH
7301 Erycibenin B
hepatocytes, antihepatotoxin induced by D-galactosamine (GalN), 100mol/L,
InRt = (31.90.3)%, weak, control Silybin, 100mol/L, InRt = (77.05.5)%).
Source: GUANG BU DING GONG TENG Erycibe expansa. Ref: 4095.
OH
7305 Erylatissin A
7,3'-Dihydroxy-4'-methoxy-5'-(,-dimethylallyl)isoflavone C21H20O5
(352.39). Brown paste. Pharm: Antibacterial (Escherichia coli, MIA = 5.00g,
control Chloramphenicol, MIA = 0.001g; Staphylococcus aureus, MIA =
HO
0.10g, Chloramphenicol, MIA = 0.0001g; Bacillus subtilis, MIA = 0.10g,

O
HO
Chloramphenicol, MIA = 0.0001g); antifungal (Candida mycoderma, MIA =

0.02g, control Miconazole, MIA = 0.0001g); antioxidant (DPPH scavenger,
OH
TLC, MIA = 0.5g, IC50 = 780g/mL; control Quercetin, MIA < 0.05g, IC50
OH
= 7g/mL, Gallic acid, MIA < 0.05g, IC50 = 4g/mL; Ascorbic acid, MIA <
7302 Erycibenin C
0.10g, IC50 = 18g/mL). Source: JI KUAN CI TONG Erythrina latissima
(stem wood). Ref: 5247.
hepatocytes, antihepatotoxin induced by D-galactosamine (GalN), 100mol/L,

InRt = (10.52.7)%, weak, control Silybin, 100mol/L, InRt = (77.05.5)%).
HO
O
OH
Source: GUANG BU DING GONG TENG Erycibe expansa. Ref: 4095.

O
O
O
O
H
299
7306 Erylatissin B
7310 Erypoegin D
7,3'-Dihydroxy-6'',6''-dimethyl-4'',5''-dehydropyrano [2'',3'':4',5']isoflavone
C22H24O6 (384.43). Colorless oil. Source: SHAN DI CI TONG Erythrina
C20H16O5 (336.35). Yellowish paste. Pharm: Antibacterial (Staphylococcus
poeppigiana. Ref: 1972.
aureus, MIA = 1.00g, Chloramphenicol, MIA = 0.0001g; Bacillus subtilis,

MIA = 1.00g, Chloramphenicol, MIA = 0.0001g); antifungal (Candida
mycoderma, MIA = 1.00g, control Miconazole, MIA = 0.0001g);

antioxidant (DPPH scavenger, TLC, MIA = 10g, IC50 > 1000g/mL; control
OH
Quercetin, MIA < 0.05g, IC50 = 7g/mL, Gallic acid, MIA < 0.05g, IC50 =
OH
4g/mL; Ascorbic acid, MIA < 0.10g, IC50 = 18g/mL). Source: JI KUAN
CI TONG Erythrina latissima (stem wood). Ref: 5247.
7311 Erypoegin E
C20H18O4 (322.36). Yellowish oil. Source: SHAN DI CI TONG Erythrina
HO

OH
O
O
HO
7307 Erylatissin C
()-7,3'-Dihydroxy-4'-methoxy-5'-(,-dimethylallyl)flavanone C21H22O5
O
(354.41). Yellow solid, mp 56~59C, []D = 78 (c = 0.025, MeOH). Pharm:

Antibacterial (Escherichia coli, MIA = 0.50g, control Chloramphenicol,
MIA = 0.001g; Staphylococcus aureus, MIA = 0.10g, Chloramphenicol,
MIA = 0.0001g; Bacillus subtilis, MIA = 0.01g, Chloramphenicol, MIA =
0.0001g); antifungal (Candida mycoderma, MIA = 0.01g, control
Miconazole, MIA = 0.0001g); antioxidant (DPPH scavenger, TLC, MIA =
0.5g, IC50 = 710g/mL; control Quercetin, MIA < 0.05g, IC50 = 7g/mL,
OH
7312 Erypoegin F
C21H20O5 (352.39). Amorphous powder. Pharm: Antibacterial (13 strains of
methicillin-resistant Staphylococcus aureus (MRSA), for 13/13 active).
Source: SHAN DI CI TONG Erythrina poeppigiana (root). Ref: 3400.
OH
HO
Gallic acid, MIA < 0.05g, IC50 = 4g/mL; Ascorbic acid, MIA < 0.10g,
IC50 = 18g/mL). Source: JI KUAN CI TONG Erythrina latissima (stem
O
wood). Ref: 5247.
OH
O
O
HO
7313 Erypoegin G
C22H22O6 (382.42). Amorphous powder, []D = 0. Pharm: Antibacterial
inactive (13 strains of methicillin-resistant Staphylococcus aureus (MRSA),
for 13/13 inactive). Source: SHAN DI CI TONG Erythrina poeppigiana (root).
7308 Eryphrinine
C18H19NO4 (313.36). Source: JI GUAN CI TONG Erythrina crysragalli (the
compound was isolated from the plant in 1973). Ref: 5505.
Ref: 3400.
O
OH
O
OH
7314 Erypoegin H
C20H18O4 (326.36). Amorphous powder. Pharm: Antibacterial (13 strains of

methicillin-resistant Staphylococcus aureus (MRSA), for 13/13 active).
Source: SHAN DI CI TONG Erythrina poeppigiana (root). Ref: 3400.
7309 Erypoegin C
C21H22O6 (370.41). Colorless oil. Source: SHAN DI CI TONG Erythrina
HO
HO
OH
OH
OH
300
7315 Erypoegin I
7319 Erysenegalensein O
C21H22O6 (370.41). Amorphous powder, []D = 71 (c = 0.1, MeOH). Pharm:
5,2',4'-Trihydroxy-6-(,-dimethylallyl)-3'''-hydroxy-2''',2'''-dimethyldihydropy
Antibacterial inactive (13 strains of methicillin-resistant Staphylococcus
rano[5''',6''';8,7]isoflavone C25H26O7 (438.48). Pale-yellow oil. Source: SAI
aureus (MRSA), for 13/13 inactive). Source: SHAN DI CI TONG Erythrina
NEI JIA ER CI TONG Erythrina senegalensis. Ref: 2344.
poeppigiana (root). Ref: 3400.

HO
OH
OH
O
OH
OH
OH
7320 Erysimoside
7316 Erypoegin J
C35H52O14 (696.80). mp 170~173C. Pharm: Cardiotonic. Source: CHANG
SHUO HUANG MA Corchorus olitorius, GUI ZHU TANG JIE Erysimum
Antibacterial inactive (13 strains of methicillin-resistant Staphylococcus
cheiranthoides, HUANG MA YE Corchorus capsularis, HUANG MA ZI
aureus (MRSA), for 13/13 inactive). Source: SHAN DI CI TONG Erythrina
Corchorus capsularis, KANG PI DU MAO XUAN HUA Strophanthus kombe,
poeppigiana (root). Ref: 3400.
LING LAN Convallaria keiskei [Syn. Convallaria majalis], MENG GU CE JIN
ZHAN HUA Adonis mongolica, TANG JIE Erysimum diffusum. Ref: 6, 658.
O
OH
H
H
H
OO
7317 Erysenegalensein E
C25H26O6 (422.48). Colorless amorphous, []D = +4.8 (c = 0.056, EtOH).
HO
Pharm: Antifungal (Trichophyton mentagrophytes, 500~1000g/mL)[2347];

cytotoxic (KB, EC50 = 6.25g/mL). Source: CI TONG Erythrina variegata
OH
OH
OO
OH
OH
[Syn. Erythrina indica] (stem cortex), PAN YUAN YU TENG Derris

scandens. Ref: 2347, 5220.
OH
OH
7321 Erysimosol
3-O-Digilanidobioside [11006-14-7] C35H54O14 (698.81). Source: GUI ZHU
TANG JIE Erysimum cheiranthoides. Ref: 6.
OH
O
HO
OH
HO
OH
H
OO
7318 Erysenegalensein N
5,7,2',4'-Tetrahydroxy-6-(2''-hydroxy-3''-methylbut-3''-enyl)-8-(,-dimet
hylallyl) isoflavone C25H26O7 (438.48). Pale-yellow oil, [] D20 = 3.3 (c
= 0.8, MeOH). Source: SAI NEI JIA ER CI TONG Erythrina
HO
OH
OH
OO
OH
OH
OH
senegalensis. Ref: 2344.
OH
7322 Erysodine
[7290-03-1] C18H21NO3 (299.37). mp 204~205C. Source: QIAO MU CI
TONG Erythrina arborescens. Ref: 6.
HO
OH
OH
HO
OH
O
OH
301
7323 Erysoline
7327 Erysotrine
[504-84-7] C6H11NO2S2 (193.29). mp 59~60C. Pharm: Antibacterial
[27740-43-8] C19H23NO3 (313.40). Free alkali: mp 95~97C (light petroleum
(gram-positive bacteria, gram-negative bacteria, acid-fast bacteria, EC =
ether); hydrochloride: mp 206~208C (etherethanol); bitter acid salt: mp
125-500g/mL); antiprotozoal (Trichomonas vaginalis and Trypanosoma
162~163, []D21 = +142 (c = 0.4, ethanol). Pharm: Antineoplastic;
equiperdum, in vitro, EC = 1.0g/mL, Castellanella gambiense, in vitro, EC =
neuromuscular blocker; uterine stimulant. Source: GOU QI XIAO BO
0.5-2.5g/mL); antiviral (in vitro); cytotoxic (EAC in vitro, 500g/mL, after
Berberis zycium, SHUAN ZHUANG CI TONG Erythrina suberosa. Ref: 661.
24h completely inhibition). Source: A FU HAN TANG JIE Erysimum
perofskianum, QUN XIN CAI Cardaria draba, MAO DU XING CAI
Lepidium draba. Ref: 661.
S
N
7328 Erysovine
[466-72-8] C18H21NO3 (299.37). mp 178~179C. Pharm: Ganglionic blocker
(curariform action). Source: CI TONG Erythrina variegata [Syn. Erythrina
S
O
indica], FU KE CI TONG Erythrina folkersii, QIAO MU CI TONG Erythrina

arborescens, SHU WEI CAO HUA CI TONG Erythrina salviiflora. Ref: 6,
658.
7324 Erysonine
[7290-05-3] C17H19NO3 (285.35). Pharm: Neuromuscular blocker. Source: JIA
LE BI CI TONG Erythrina caribea, HEI CI CI TONG Erythrina
melanacantha. Ref: 658.
O
N
HO
O
OH
7329 Erythrabssin II
C25H28O4 (392.50). Pharm: Antimalarial (antiplasmodial in vitro,
HO
Plasmodium falciparum, W2 strain, IC50 = (6.50.6)mol/L, control Quinine,

IC50 = (0.210.01)mol/L; D6 strain, IC50 = (8.11.4)mol/L, Quinine, IC50
= (0.0420.002)mol/L). Source: A BI XI NI YA CI TONG Erythrina

abyssinica (root cortex). Ref: 5420.
7325 Erysopine
HO
C17H19NO3 (285.35). mp 242~243C. Pharm: Ganglionic blocker (curariform

action). Source: A BI XI NI YA CI TONG Erythrina abyssinica, CI TONG
Erythrina variegata [Syn. Erythrina indica], FU KE CI TONG Erythrina
OH
folkersii, QIAO MU CI TONG Erythrina arborescens, SHU WEI CAO HUA

CI TONG Erythrina salviiflora, YING HE CI TONG Erythrina lithosperma.
Ref: 6, 658.
7330 Erythraline
[466-77-3] C18H19NO3 (297.36). mp 106~107C. Pharm: Ganglionic blocker
OH
HO
(curariform action). Source: HAI TONG PI Erythrina variegata var. orientalis.

O
Ref: 6, 658.
O
O
O
7326 Erysothiopine
[In DNP] C19H21NO7S (407.45). Hydrate crystals (solution of ethanol in
water), mp 168~169C, []D25 = +194 (ethanol). Pharm: Neuromuscular
blocker. Source: HUI CI TONG Erythrina glauca. Ref: 658.
7331 Erythratidine
[41431-22-5] C19H25NO4 (331.42). Pharm: Neuromuscular blocker. Source:
HEI CI CI TONG Erythrina melanacantha, JIA LE BI CI TONG Erythrina
caribea. Ref: 658.
O
HO
O
O
O
O
HO
N
O
OH
302
7332 Erythrinassinate B
7337 Erythroculine
C37H64O4 (572.92). Source: CI TONG Erythrina variegata [Syn. Erythrina
[22150-96-5] C20H25NO4 (343.43). Source: HENG ZHOU WU YAO
indica] (stem cortex). Ref: 5220.
Cocculus laurifolius. Ref: 6.

O
N
O
HO
O
7338 Erythrodiol
Olean-12-en-3,28-diol C30H50O2 (442.73). mp 215~217C. Source: BING
PIAN Dryobalanops aromatica, BING PIAN Dryobalanops aromatica,
FENG XIANG JI SHENG Viscum articulatum, MANG GUO SHU PI
7333 Erythrinin C
[63807-85-2] C20H18O6 (354.36). Source: Glycyrrhiza sp. Ref: 2431.
HO
Mangifera indica. Ref: 2, 6.
O
H
OH
OH
OH
HO
7334 Erythritol
Threitol [149-32-6] C4H10O4 (122.12). Amorphous powder, []D = 0, mp
7339 Erythrodiol 3-O-palmitate
D(+) 88.5~89.0C, L() 88C, dl 72 C; mp 121.5C, bp 329~331C. Pharm:
C46H80O3 (681.15). Source: HUANG LONG DAN Gentiana lutea (rhizome
Coronary vasodilator. Source: BAO CHUN HUA Primula malacoides, BEI
and root). Ref: 4307.
23
SHA SHEN Glehnia littoralis (fruit), SHI LUO ZI Anethum graveolens (fruit),
YING SU KE Papaver somniferum, ZHANG YE BAN XIA Pinellia
pedatisecta, ZHEN MO Armillariella mellea. Ref: 6, 586, 658, 3525, 4177.
HO
H
O
OH
OH
H
H
OH
OH
H
O
7340 -Erythroidine
[466-80-8] C16H19NO3 (273.33). Acicular crystals (pentane), mp 58~60C,
7335 Erythrocentauric acid
[]D27 = +136 (c = 0.5, water), instable in air. Pharm: Neuromuscular blocker.
5-Carboxyl-3,4-dihydrogen-1H-2-benzopyran-1-one C10H8O4 (192.17).
Source: MEI ZHOU CI TONG Erythrina americana. Ref: 658.
Tubbiness colorless transparent needles, mp 251~253C. Source: QIN JIAO

Gentiana macrophylla. Ref: 4594, 4824.
H
O
O
O
7341 -Erythroidine
OH
[466-81-9] C16H19NO3 (273.33). Crystals (absolute ethanol), mp
7336 Erythrocentaurin
99.5~100.0C, []D25 = +88.8. Pharm: Hypnotic; inhibits respiration;
C10H8O3 (176.17). Colorless needles, mp 145~147C (CHCl3). Source: QIN
antihypertensive; neuromuscular blocker; LD50 (mus, ip) = 29.5mg/kg. Source:
JIAO Gentiana macrophylla. Ref: 4594, 4824.
MEI ZHOU CI TONG Erythrina americana. Ref: 658.
O
O
303
7342 Erythrophlamine
7346 Erythroxyloside B
C25H39NO6 (449.59). Crystals (ethanolpetroleum ether), mp 149~157C,
[]D20 = 62.5 (c = 0.911, ethanol). Pharm: Cardiotonic. Source: FEI ZHOU
Source: JIAN PU ZHAI GU KE Erythroxylum cambodianum (aerial parts).
GE MU Erythrophleum africanum, JI NEI YA GE MU Erythrophleum
Ref: 4461.
guineense, KAO MING GE MU Erythrophleum couminga, XIANG YA HAI

AN GE MU Erythrophleum ivorense, YE XIANG GE MU Erythrophleum
OH
OH
suaveolens. Ref: 658.

O
OH
OH
OH OH
7347 Erythrozeylanine A
1R,3R,5S,6R-6-Acetoxy-3-(3',4',5'-trimethoxybenzoyloxy)tropane C20H27NO7
(393.44). Colorless semisolid, []D25 = 22.1 (c = 0.3, CHCl3). Source: XI
LAN GU KE Erythroxylum zeylanicum (root). Ref: 3919.
H
H
HO
OH
OO
OO
N
O
7343 Erythrophleguine
[4829-28-1] C25H39NO6 (449.59). mp 77~78C, []D = 38 (ethanol). Pharm:

Cardiotonic; enhances myocardial contractility; slows heart rate. Source: JI
O
O
NEI YA GE MU Erythrophleum guineense, KAO MING GE MU

Erythrophleum couminga, XIANG YA HAI AN GE MU Erythrophleum
O
O
ivorense, YE XIANG GE MU Erythrophleum suaveolens. Ref: 658.

O
cis-3-(Cinnamoyloxy)tropane C17H21NO2 (271.36). Source: XI LAN GU KE

Erythroxylum zeylanicum (root). Ref: 3919.
H
O
7348 Erythrozeylanine B
OH
H
O
7344 Erythrosuamine
C25H39NO6 (449.59). Source: JI NEI YA GE MU Erythrophleum guineense.
Ref: 1521.
7349 Erythrozeylanine C
cis-6-Acetoxy-3-(cinnamoyloxy)tropane C19H23NO4 (329.40). Source: XI
LAN GU KE Erythroxylum zeylanicum (twig, leaf). Ref: 3919.

N
H
H
O
OH
H
H
H
H
7345 Erythroxyloside A
7350 Eryvarin F
Source: JIAN PU ZHAI GU KE Erythroxylum cambodianum (aerial parts).
3-(2,4-Dihydroxyphenoxy)-7-hydroxy-6,8-di(3,3-dimethylallyl)chromen-4-on
Ref: 4461.
e C25H26O6 (422.48). Amorphous powder. Source: CI TONG Erythrina

variegata [Syn. Erythrina indica]. Ref: 2040.
HO
OH
OO
O
OH
HO
OH
OH OH
OH
OH
O
O
O
OH
304
7351 Eryvarin G
7355 Eryzerin B
3-(2,4-dihydroxyphenoxy)-8-(3,3-dimethylallyl)-2,2-dimethylpyrano[5,6:6,7]
(3R)-7,4'-Dihydroxy-2'-methoxy-6,8-di(,-dimethylallyl)isoflavanone C26H30O5
chromen-4-one C25H24O6 (420.47). Amorphous powder. Source: CI TONG
(422.53). Amorphous powder, []D = 41 (c = 0.1, MeOH). Pharm:
Erythrina variegata [Syn. Erythrina indica]. Ref: 2040.
Antibacterial (Methicillin-Resistent Staphylicoccus aureus (MRSA), MIC range

= 25~50g/mL, MIC50 > 50g/mL, MIC90 > 50g/mL, proportion of sensitive
strains at 12.5g/mL = 0/13). Source: Erythrina zeyheri (root). Ref: 3451.
OH
HO
O
O
OH
O
7352 Eryvarinol A
23
OH
7356 Eryzerin C
Source: CI TONG Erythrina variegata [Syn. Erythrina indica] (root: yield =
(3R)-7,2',4'-Trihydroxy-6,8-di(,-dimethylallyl)isoflavan C25H30O4 (394.52).
0.0015%). Ref: 4671.
Amorphous powder, []D = 9 (c = 0.1, MeOH). Pharm: Antibacterial

(Methicillin-Resistent Staphylicoccus aureus (MRSA), MIC range =
3.13~6.25g/mL, MIC50 = 6.25g/mL, MIC90 = 6.25g/mL, proportion of sensitive
OH

O
HO
OH
H O
HO
OH
H OH O
7353 Eryvarinol B
OH

CI TONG Erythrina variegata [Syn. Erythrina indica] (root: yield =
7357 Eryzerin D
0.0021%). Ref: 4671.
2',4'-Dihydroxy-8-,-dimethylallyl-2'',2''-dimethylpyrano-[5,6:6,7]isoflavan
C25H28O4 (392.50). Amorphous powder, []D = +3 (c = 0.1, MeOH). Pharm:
Antibacterial (Methicillin-Resistent Staphylicoccus aureus (MRSA), MIC
OH
range = 6.25~12.5g/mL, MIC50 = 12.5g/mL, MIC90 = 12.5g/mL,
O
HO
O
H O
proportion of sensitive strains at 12.5g/mL = 13/13). Source: Erythrina

OH
zeyheri (root). Ref: 3451.
H OH O
OH
7354 Eryzerin A
()-7,2',4'-Trihydroxy-8,3'-di(,-dimethylallyl)isoflavanone C25H28O5
(408.50). Amorphous powder, []D = 0. Pharm: Antibacterial
OH
(Methicillin-Resistent Staphylicoccus aureus (MRSA), MIC range =

12.5~25g/mL, MIC50 = 25g/mL, MIC90 = 25g/mL, proportion of sensitive
7358 Eryzerin E
(6aS,11aS)-3,6a-Dihydroxy-9-methoxy-4,10-di(,-dimethylallyl)pterocarpan
Antibacterial (Methicillin-Resistent Staphylicoccus aureus (MRSA), MIC range =
6.25~25g/mL, MIC50 = 6.25g/mL, MIC90 = 12.5g/mL, proportion of sensitive
HO
HO
O
HO
OH
OH
305
7359 (+)-Eschscholtzidine
7363 Escin IVg
C21H23NO3 (337.42). Source: HOU KE GUI Cryptocarya chinensis (wood).
22-Tigloylprotoaescigenin 3-O-[-D-glucopyranosyl (12)]
Ref: 3092.
[-D-glucopyranosyl (14)]--D-glucopyranosiduronic acid C53H84O23

(1089.25). White amorphous powder, []D25 = 25.0 (c = 1.00, MeOH).
Source: QI YE SHU Aesculus chinensis (seed). Ref: 3528.
OH
O
H
O
HO
7360 (+)-Eschscholtzidine-N-oxide
OO
C20H21NO5 (355.39). Colorless needles (MeOH), mp 193~194C, []D =

+145.3 (c = 0.1278, MeOH). Source: HOU KE GUI Cryptocarya chinensis
OH
HO
OH
OH
OH
OH
O N+
OH
OO
HO
OH
(wood). Ref: 3092.
OH
OH
OH
7364 Escin IVh

7361 Escin Ia
22-Angeloylprotoaescigenin 3-O-[-D-glucopyranosyl (12)]
21-O-Tigloyl-22-O-acetylprotoaescigenin-3-O-[-D-glucopyranosyl(12)][
-D-glucopyranosyl(14)]--D-glucopyranosiduronic acid C55H86O24
(1089.25). White amorphous powder, []D25 = 60 (c = 1.05, MeOH). Source:
(1131.28). Pharm: Anti-inflammatory (mus, assay of Dimethyl
QI YE SHU Aesculus chinensis (seed). Ref: 3528.
benzene-induced inflammation, dose 30mg/kg, InRt = 79.3%, control

Dexamethasone, dose 1mg/kg, InRt = 55.6%). Source: QI YE SHU Aesculus
OH
O
chinensis (seeds). Ref: 2578.

H
HO
OH
OH
OO
OH
HO
OO
OH
OH
OH
OH
OO
HO
OH
H
OH
OO
OH
OH
OH
OO
HO
OO
OH
HO
OH
OH
HO
O
H
OH
OH
OH
OH
OH
7365 Escin VIb
7362 Escin IIIa
16-Angeloyl-21-acetylprotoaescigenin 3-O-[-D-glucopyranosyl (12)]
MeOH). Source: QI YE SHU Aesculus chinensis (seed). Ref: 3528.
(1131.28). White amorphous powder, []D25 = 55 (c = 1.00, MeOH). Source:

QI YE SHU Aesculus chinensis (seed). Ref: 3528.
O
O
H
HO
OO
OH
OH
OH
OH
OH
HO
OH
OH
OO
OH
OH
OO
HO
HO
OH
OH
OO
HO
OH
OH
OH
HO
OH
OH
OH
OH
OH
O
O
306
7366 Esculentoic acid A
7370 Esculentoside C
C30H48O3 (456.72). Colorless powder, mp 248~251C, []D25 = 16.4 (c =
Phytolaccoside D [65931-92-2] C42H66O15 (810.99). mp 220~222C, []D =
0.64, CHCl3). Pharm: Cytotoxic (A2780 ovarian cancer cell line, IC50 =
+40 (c = 0.3, MeOH). Pharm: Anti-inflammatory. Source: MEI SHANG LU
6.4mg/mL, marginally active). Source: MU SHU DI SHANG BU FEN
Phytolacca americana [Syn. Phytolacca decandra], SHANG LU Phytolacca
Manihot esculenta. Ref: 5379.
esculenta [Syn. Phytolacca acinosa]. Ref: 1535, 3106, 3108.

O
O
HO
H
HO
OH
H
OO
OH
HO
7367 Esculentoic acid B

0.48, CHCl3:MeOH = 1:1). Pharm: Cytotoxic (A2780 ovarian cancer cell line,
OO
OH
OH
OH
OH
OH
IC50 = 4.8mg/mL, marginally active). Source: MU SHU DI SHANG BU FEN
7371 Esculentoside D
Manihot esculenta. Ref: 5379.
C37H58O12 (694.87). Source: SHANG LU Phytolacca esculenta [Syn.
O
HO
Phytolacca acinosa]. Ref: 1535.

O
O
H
H
O
HO
OH
H
HO
7368 Esculentoside A
OO
OH
Phytolaccoside E [65497-07-6] C42H66O16 (826.98). Powder, mp 257~258C,

[]D21 = +51.3 (c = 0.99, EtOH). Source: MEI SHANG LU Phytolacca
[5523]
americana [Syn. Phytolacca decandra] (dried root: content = 0.86%
),
OH
OH
OH
7372 Esculentoside E
SHANG LU Phytolacca esculenta [Syn. Phytolacca acinosa] (dried root:
[65949-36-7] C35H54O11 (650.81). Source: SHANG LU Phytolacca esculenta
mean content of 11 origins = 0.37%[5523]). Ref: 660, 1521, 1535, 5523.
[Syn. Phytolacca acinosa]. Ref: 1536.
O
O
HO
OO
HO
OH
OH
OH
O
OH
OH
OH
OH
HO
OO
OO
OH
O
OH
OH
OH
H
OH
OH
7373 Esculentoside F
7369 Esculentoside B
[95263-31-3] C41H64O16 (812.96). Source: SHANG LU Phytolacca esculenta
C35H54O11 (650.81). Source: SHANG LU Phytolacca esculenta [Syn.
[Syn. Phytolacca acinosa]. Ref: 1536.

O
Phytolacca acinosa]. Ref: 1535.

O
OH
O
HO
H
OO
OH
OH
H
OH
OO
OH
OH
HO
OH
OH
OH
H
H
OO
OH
OH
HO
OH
O
OH
307
7374 Esculentoside H
7377 Esculeoside C
Phytolaccasaponin B [66656-92-6] C48H76O21 (989.13). Needles +3H2O, mp
3-O--Lycotetraosyl(5S,25S)-22,26-epimino-16,23-epoxy-23-methoxy-
218~220C, []D29 = +38.3 (c = 0.93, EtOH). Source: MEI SHANG LU
22(N)-ene-3,20,27-trihydroxycholestane 27-O--D-glucopyranoside
Phytolacca americana [Syn. Phytolacca decandra], SHANG LU Phytolacca
C57H93NO29 (1256.37). Amorphous powder, []D24 = 56.7 (c = 0.9,
esculenta [Syn. Phytolacca acinosa]. Ref: 1521, 1537.
pyridine). Source: YING TAO FAN QIE Lycopersicon esculentum var.

cerasiforme (ripe fruit: yield = 0.00009%fw). Ref: 1453.
N
OH
HO
OO
HO
OH
OH
OH
OO
HO
OH
HO
OO
OH
O
OO
OH
OO
HO
HO
HO
H
OH
O
OH
OH
OH
OO
OH
HO
OO
OH
OH
OH
OH
OH
OH
OH
OH
OH
7375 Esculeogenin B
7378 Esculeoside D
(5,22S,23R,25S)-22,26-Epimino-16,23-epoxy-3,23,27-trihydroxycholestan
3-O--Lycotetraosyl 3,16-dihydroxy-5-pregn-20-one 16-O-[(4S)-2,5-
e C27H45NO4 (447.66). Amorphous powder, []D = 96.2 (c = 0.05, pyridine).
epimino-2-methoxy-4-(-D-glucopyranosyloxy) methyl-pentanoic acid]-ester
Source: FAN QIE Lycopersicon esculentum. Ref: 4484.
C57H93NO30 (1272.37). Amorphous powder, []D24 = 20.7 (c = 1.0,

pyridine). Source: YING TAO FAN QIE Lycopersicon esculentum var.
HN
H
H
cerasiforme (ripe fruit: yield = 0.00009%fw). Ref: 1453.
OH
OH
HO
HO
HO
H
OH
OH
7376 Esculeoside A
HO
OO
OH
OH
C58H95NO29 (1270.39). white powder, []D = 52.5 (MeOH). Pharm:
proliferation reagent, see M. Ishiyama, et al., Talanta, 1999, 44, 1299).

Source: FAN QIE Lycopersicon esculentum. Ref: 4317.
OH
OH
7379 Eseramine
[6091-57-2] C16H22N4O3 (318.38). Pharm: Cholinesterase inhibitor. Source:
DU BIAN DOU Physostigma venenosum. Ref: 658.
H
OH
OH
HO
OH
OH
O O OH
OH
OH OH
7380 Eseridine
Geneserine [25573-43-7] C15H21N3O3 (291.35). Pharm: Cholinesterase
inhibitor. Source: DU BIAN DOU Physostigma venenosum. Ref: 658.
N
OH
NH
OH
OH
OO
HO
O
OH
OO
OO
N
N
OH
HO
OH
OH
H
N
O
O
OO
HO
OH
Cytotoxic (MCF7 cells, IC50 = 24.5mol/L, control Tomatine, IC50 =

15mol/L, cytotoxicity of compounds was measured using the WST-8
OH
OH
H
N
OH
OO
OO
O
O
O
308
7381 Eserine
7385 Estragole
Physostigmine; Cogmine; Physostol [57-47-6] C15H21N3O2 (275.35).
4-Methoxyallylbenzene [140-67-0] C10H12O (148.21). bp 215~216C, bp
Trapezoidal half-prismatic crystals (ether or benzene), mp 105~106C, []D17
102C/16mmHg. Pharm: Antibacterial; antispasmodic; leukopoietic; promotes
= 76 (c = 1.3, chloroform), []D25 = 120 (benzene), soluble in ethanol,
liver regeneration; sedative; LD50 (mus, orl) = 4000mg/kg. Source: HUA
[5507]
benzene, chloroform, slightly soluble in water.
Pharm: BChE inhibitor
JIAO Zanthoxylum bungeanum, HUI XIANG Foeniculum vulgare, QIAN HU
(IC50 = (0.040.0001)mol/L[2563], IC50 = (0.8570.008)mol/L[4217], IC50 =
Angelica decursiva [Syn. Peucedanum decursivum], SHUI HUI XIANG
(0.8750.008)mol/L[5216]); BChE inhibitor (horse serum BChE, IC50 =
Limnophila rugosa, XI XIN Asarum sieboldii, LIAO XI XIN Asarum
(0.8570.008)mol/L)[4241]; AChE inhibitor (IC50 = (0.410.001)mol/L[4217],
heterotropoides var. mandshuricum, HUO XIANG Agastache rugosus, BA
IC50 = (0.0410.001)mol/L[5216]); AChE inhibitor (electric eel AChE, IC50 =
JIAO HUI XIANG Illicium verum, OU ZHOU CHI SONG Pinus sylvestris,
(0.0410.001)mol/L)[4241]; antidote (poisoning from anticholinergic); used in
RI BEN XIN YI Magnolia kobus. Ref: 2, 4, 6, 658, 660, 1521.
treatment of glaucoma (0.2%~0.5%) and myoparalysis[658]; LD50 (mus, ip) =

2.5mg/kg[658]. Source: DU BIAN DOU Physostigma venenosum (in 1864,
isolated from the plant for the first time[5507]; in 1969, isolated from the plant
O
by R.K.Hill, et al.[5505]). Ref: 658, 2563, 4217, 4241, 5216, 5505, 5507.
7386 Estriol
N
N
Estratriol [50-27-1] C18H24O3 (288.39). mp 282~283C. Pharm: Leukopoietic

(promotes growth of white blood cells); used in treatment of menopathy and
female climacteric syndrome. Source: ZI HE CHE Homo sapiens. Ref: 5, 6,
658.
O
NH
OH
OH
7382 Espeletone
C14H18O3 (234.30). Pharm: Antifungal (Trichophyton mentagrophytes
ATCC28185, MIC = 100g/mL, control Miconazole, MIC = 8g/mL;
Trichophyton rubrum ATCC28188, MIC = 100g/mL, Miconazole, MIC =
8g/mL). Source: Eupatorium aschenbornianum. Ref: 5472.
HO
7387 Estrone
3-Hydroxy-1,3,5(10)-estratrien-17-one [53-16-7] C18H22O2 (270.37). Crystals
(acetone), mp () 251~254C, mp (+) 254.5~256.0C, []D25 = +158~168
(dioxane). Pharm: Estrogenic activity. Source: LU RONG Cervus nippon;
Cervus elaphus, SUAN SHI LIU Punica granatum, WU LOU ZI Phoenix

dactylifera, ZI HE CHE Homo sapiens, YUE JI SHI LIU Punica granatum cv.
O
nana, YE ZI Cocos nucifera (fruit; the compound was isolated from the plant
by A.Butenandt et al. in 1938)[5505]. Ref: 6, 658, 5501, 5505.
7383 -Estradiol
[50-28-2] C18H24O2 (272.39). mp 223C. Pharm: Promotes normal growth of
female sexual organs and secondary sex characters. Source: LU RONG
Cervus nippon; Cervus elaphus, SHE XIANG Moschus moschiferus; Moschus

H
berezovskii; Moschus sifanicus, ZI HE CHE Homo sapiens. Ref: 2, 658, 5501.
HO
OH
7388 Ethane-1,2-diol 1-O--D-apiofuranosyl-(16)--D-glucopyranoside

C13H24O11 (356.33). Colorless syrup, []D21 = 47 (c = 0.7, MeOH). Source:
ZI RAN QIN Cuminum cyminum (fruit). Ref: 3395.
HO
O O
HO
OO
OH
7384 -Estradiol
17-Oestradiol [57-91-0] C18H24O2 (272.39). mp 178C. Pharm: Promotes
OH OH
normal growth of female sexual organs and secondary sex characters. Source:
OH
OH
OH
BAI FAN DOU Phaseolus vulgaris, LU RONG Cervus nippon; Cervus
7389 Ethane-1,2-diol 1-O--D-glucopyranoside
elaphus, SHE XIANG Moschus moschiferus; Moschus berezovskii; Moschus
C8H16O7 (224.21). Colorless syrup, []D21 = 17 (c = 0.6, MeOH). Source:
sifanicus, ZI HE CHE Homo sapiens. Ref: 2, 658, 5501.
HUI QIN Pimpinella anisum (fruit). Ref: 3402.
OH
H
H
HO
OO
HO
OH
H
OH
OH
OH
309
7390 Ethanolamine
7396 8-Ethoxy atractylenolide III
2-Aminoethanol [141-43-5] C2H7NO (61.08). bp 171C. Source: XI JIAO
C18H26O3 (290.41). Source: BAI ZHU Atractylodes macrocephala [Syn.
Rhinoceros unicornis; Rhinoceros sondaicus; Rhinoceros sumatrensis. Ref: 6.
Atractylis macrocephala]. Ref: 2.
OH
O
NH2
O
O
7391 2-(Ethenylbutadiynyl)-5-(propinyl)-thiophene
C13H8S (196.27). Source: MO LI HUA Jasminum sambac. Ref: 6.
7397 N-Ethoxycarbonyllaurotetanine
S
C22H25NO6 (399.45). Yellowish powder. Source: XIA YE SHAN HU JIAO

Lindera angustifolia (root). Ref: 4875.
O
7392 2-(5-Ethenyl-5-methyl-2-tetrahydrofuranyl)-6-methyl-5-hepten-3-one
C15H24O2 (236.36). Source: WU WEI ZI Schisandra chinensis. Ref: 2.

O
O
OH
7398 4-Ethoxycarbonyl-2-quinolinone
[5466-27-3] C12H11NO3 (217.23). Colorless acicular crystals, mp 208~209C.
7393 4-Ethenyl-2,2,4-trimethyl-3-(1-methylethenyl)-cyclohexane-methanol
Source: YA DAN ZI Brucea javanica [Syn. Brucea sumatrana; Rhus
C15H26O (222.37). Source: SHENG JIANG Zingiber officinale. Ref: 2.
javanica]. Ref: 2, 156.
OH
N
H
7394 9-Ethoxy-aristololactam
7399 Ethoxychelerythrine
C19H15NO5 (337.34). Source: MIAN MAO MA DOU LING Aristolochia
C23H23NO5 (393.44). White lamellar crystals (ammonia absolute ethanol), mp
mollissima. Ref: 127.
207~208C; Pharm: Cytotoxic (Ehrlich ascites carcinoma cells)[5369];

antineoplastic (cervical carcinoma, thyroid carcinoma); antibacterial;
anti-inflammatory (used in treatment of cervicitis). Source: BO LUO HUI
O
NH
Macleaya cordata. Ref: 658, 5369.
O
O
O
O
N
O
O
7395 9-Ethoxy-aristololactone
9-Ethoxy-aristololide C19H14O6 (338.32). Source: MIAN MAO MA DOU
LING Aristolochia mollissima. Ref: 127.
O
C24H30O7 (430.50). Pharm: CYP3A4 inhibitor and CYP2D6 inhibitor (in vitro,
CYP3A4, IC50 = 0.44mol/L; CYP2D6, IC50 = 87.9mol/L; control
O
O
O
O
O
7400 Ethoxyclusin
Ketoconazole, CYP3A4, IC50 = 0.72mol/L; control Quinidine, CYP2D6,

IC50 = 0.082mol/L). Source: BI CHENG QIE Piper cubeba (fruit: yield =
0.00005%dw). Ref: 4797.
O
O
O
O
O
O
310
7401 Ethoxydihydroisomoreollin
7406 2-(1-Ethoxy-2-hydroxy)propyl-4-methoxyphenol
C35H42O8 (590.72). mp 143C. Source: TENG HUANG Garcinia morella. Ref: 6.
C12H18O4 (226.27). Colorless liquid. Source: YANG HONG SHAN

Pimpinella thelungiana. Ref: 371.
OH
O
H
O
OH
O
O
OH
7407 2-(1-Ethoxy-2-hydroxy)propyl-4-methoxyphenol-2-methyl-butyrate
C17H26O5 (310.39). Colorless liquid. Source: YANG HONG SHAN
Pimpinella thelungiana. Ref: 371.
7402 3-Ethoxy-4,5-dihydroxy-benzoic acid
OH
C9H10O5 (198.18). White powder, mp > 300C. Source: AN MO LE
Phyllanthus emblica. Ref: 2434.
O
HO
OH
7408 3-Ethoxy-leptocarpin
HO
C22H30O6 (390.48). Source: Viguiera puruana (aerial parts). Ref: 5090.

OH
O
7403 5-(1-Ethoxy-ethyl)-2-hydroxy-7-methoxy-1,8-dimethyl-9,10-di-
hydrophenanthrene
O
O
O
O
O
7409 4-[1-Ethoxyl-1-(4'-hydroxy-3'-methoxy)benzyl]methyl-2-(4-hydroxy-3-methoxy)benzyl-3-hydroxymethyl-tetrahydro-furan
C22H28O7 (404.46). White powder, mp 114~116C. Source: CAO YE BAI
HO
JIANG Patrinia scabra. Ref: 2467.
7404 6-(1-Ethoxyethyl)plumbagin
C15H16O4 (260.29). Orange needles (hexane), mp 73C, []D30 = 0.06 (c =
O
O
OH
0.36, CHCl3). Pharm: Ichthyotoxin (MLC = 0.9mg/L, control Juglone, MLC =

0.2mg/L). Source: HAI SHI Diospyros maritima (fruit). Ref: 4185.
HO
OH
O
O
7410 7-Ethoxy-12-methoxy-8,11,13-abietatrien-11-ol
OH
C23H36O3 (360.54). Source: DU SONG SHI Juniperus rigida. Ref: 6.

O
7405 4-Ethoxy-6-hydroxymethyl--pyrone
C8H10O4 (170.17). White needles, mp 94.5~96.8C. Pharm: DPPH scavenger
HO
(SC50 > 100mol/L)[4247]; antioxidant (superoxide anion radical scavenger,

superoxide dismutase method, IC50 for Formazan formation activity >
100mol/L)[4247]. Source: XIAN REN ZHANG Opuntia dillenii (fresh stem:
yield = 0.00013%)[4247]. Ref: 2468, 4247.
7411 4-Ethoxy-3-methoxybenzoic acid

C10H12O4 (196.20). Source: FEN CHA DANG GUI Angelica furcijuga
OH
O

O
O
OH
O
311
7412 4-Ethoxymethylphenyl-4'-hydroxybenzylether
7417 16-Ethoxystrychnine
C16H18O3 (258.32). Source: TIAN MA Gastrodia elata. Ref: 2.
C23H26N2O3 (378.48). mp 224~225C. Source: LV SONG GUO Strychnos

ignatii. Ref: 6.
OH
O
H
N
7413 3-Ethoxymethyl-5,6,7,8-tetrahydro-8-indolizinone
H
O
O
H
C11H15NO2 (193.25). Pharm: Antifungal (Penicillium avellaneum UC-4376,

MIA = 250.0g/disk, control Amphotericin B, MIA = 0.08g/disk);
7418 Ethyl acetate
antibacterial (Staphylococcus aureus, MIA = 400.0g/disk, control
Ethyl ethanoate [141-78-6] C4H8O2 (88.11). bp 77.1C. Source: JIU Liquor,
Rifampicin, MIA = 1.0g/disk; Mycobacterium tuberculosis, MIA =
300.0g/disk, Rifampicin, MIA = 1.0g/disk; Streptococcus oneumonia,

MIA = 300.0g/disk, Rifampicin, MIA = 1.0g/disk). Source: DIAN
HUANG JING Polygonatum kingianum (dried rhizome). Ref: 5484.
7419 Ethyl aldehyde

O
Acetaldehyde [75-07-0] C2H4O (44.05). Source: HAI JIU CAI Triglochin
maritimum, NIU BANG GEN Arctium lappa. Ref: 6.

O
7414 8-Ethoxyprecriwelline
28
C20H25NO5 (359.43). Amorphous, []D = +116.6 (c = 0.06, CHCl3). Pharm:
AChE inhibitor (IC50 = (114587)mol/L, control Galanthamine, IC50 =

(1.90.2)mol/L)[4952]. Source: LIN JING ZHONG ZI WEN SHU LAN
Crinum bulbispermum. Ref: 2369, 4952.
O
7420 Ethylamine
Aminoethane [75-04-7] C2H7N (45.08). bp 16.6C. Source: LING MAO
XIANG Viverra zibetha. Ref: 6.
NH2
N
O
7421 Ethyl benzoate
Ethyl benzenecarboxylate [93-89-0] C9H10O2 (150.18). bp 212.9C. Source:
XUAN CAO GEN Hemerocallis fulva. Ref: 6.

O
7415 8-Ethoxysachaconitine
C23H41NO4 (419.61). Amorphous solid, []D25 = 17.6 (c = 0.08, CHCl3).

Source: BAN HUA WU TOU Aconitum variegatum (aerial parts). Ref: 5270.
7422 Ethyl-n-buthy-uralsaponin A esters
H
O
3-Hydroxy-11-oxo-olean-12-en-30-oic acid-3-O--D-(n-butyl-glucurono-
OH
pyranosyl ester)-(12)--D-(ethyl-glucuronopyranosyl ester C48H74O16

(907.12). Colorless powder, mp 178C. Source: GAN CAO Glycyrrhiza
uralensis. Ref: 2148.
7416 Ethoxysanguinarine
OH
C22H19NO5 (377.40). White lamellar crystals (ammonia absolute ethanol), mp
210~211C. Pharm: Antibacterial; antineoplastic (cervical carcinoma, thyroid
carcinoma); anti-inflammatory (used in treatment of cervicitis). Source: BO
LUO HUI Macleaya cordata. Ref: 658.
OO
OH
O
O
OH
O
O
OH
OH
OH
H
H
312
7423 Ethyl butyrate
7428 (24S)-Ethylcholesta-5,22,25-trien-3-ol
Ethyl butanoate [105-54-4] C6H12O2 (116.16). bp 119.9C. Source: JIU Liquor.
C29H46O (410.69). mp 152~153C. Source: CHOU MO LI Clerodendron
Ref: 6.
fragrans, SHUI HU MAN Clerodendron inerme. Ref: 6.
O
O
H
H
7424 Ethyl caffeate

C11H12O4 (208.22). Colorless acicular crystals, mp 138~140C (acetone).
Source: JIA BAI HE Notholirion hyacinthinum [Syn. Notholirion
bulbuliferum], NAN CHUAN GUAN CHUN HUA Microtoena prainiana
(stem: 0.00014%dw)[4752]. Ref: 663, 4752.
O
HO
7429 24-Ethylcholesta-5,9(11),22-trien-3-ol
C29H46O (410.69). Crystalline solid, mp 158~160C, []D = 47 (CHCl3).
Source: KU LANG SHU Clerodendrum inerme. Ref: 3382.
O
HO
OH
7425 Ethyl chlorogenate

C18H22O9 (382.37). Cream white acicular crystals (acetone), mp 106~110C.
HO
Source: JI ZI MU Sinoadina Racemosa [Syn. Adina racemosa] (leaf, flower
7430 Ethylcinnamate
and twig: yield = 0.00073%dw)[4723], XI NAN REN DONG Lonicera bournei.
trans-Ethyl cinnamate; Ethyl trans-3-phenylpropenoate [103-36-6] C11H12O2
Ref: 439, 4723.
(176.22). bp (cis) 125C/12mmHg. (trans) 271C. Source: ROU GUI

Cinnamomum cassia [Syn. Cinnamomum aromaticum] (bark: content =
OH
0.042%)[5508], SHAN NAI Kaempferia galanga. Ref: 6, 5508.
HO
HO
OH
O
HO
7431 Ethylcyclohexane
7426 24-Ethylcholesta-5,22-dien-3-ol palmitic acid ester
[1678-91-7] C8H16 (112.22). Source: SHAN ZHA Crataegus pinnatifida. Ref: 2.
Stigmasteryl palmitate C45H78O2 (651.12). Colorless columnar crystals

(CH3OH), mp 193~194C. Source: WU WEN ZI BEI TAI Plagiochasma
intermedium, CHE QIAN Plantago asiatica, HUI XIANG GEN Foeniculum
vulgare. Ref: 6, 857.
7432 Ethyl 3,4-dihydroxybenzoate

C9H10O4 (182.18). Pharm: DPPH scavenger (SC50 = 4.9mol/L)[4247];
H
H
O
antioxidant (superoxide anion radical scavenger, superoxide dismutase

method, IC50 for Formazan formation activity = 11mol/L). Source: XIAN
REN ZHANG Opuntia dillenii (fresh stem: yield = 0.00014%). Ref: 4247.
O
O
7427 24-Ethyl-5-cholestan-3-ol
OH
[83-45-4] C29H52O (416.74). Source: JIAO GU LAN Gynostemma

pentaphyllum. Ref: 2.
OH
7433 1-Ethyl-4,8-dimethoxy--carboline
C15H16N2O2 (256.31). Source: KU SHU PI Picrasma quassioides [Syn.
H

O
H
H
HO
H
N
H
313
7434 3-Ethyl-2,3-dimethyl-pentane
7439 1-Ethyl--D-galactoside
Eleutheroside C C8H16O6 (208.21). mp 142C. Source: CI WU JIA

Acanthopanax senticosus [Syn. Eleutherococcus senticosus], CI WU JIA PI
Acanthopanax senticosus [Syn. Eleutherococcus senticosus]. Ref: 2, 6.
HO
7435
Ethyl N-docosanoylanthranilate
HO
O
OH
7436
O
OH
[209523-04-6] C31H53NO3 (487.77). Source: XI ZANG QIN JIAO Gentiana

tibetica. Ref: 702.
7440 1-Ethyl--D-galactoside

NH
HO
OO
HO
OH
7436 5-O-Ethylembelin
C19H30O4 (322.45). Orange crystals, mp 59~60C. Pharm: Cytotoxic (in vitro,
OH
HL-60, IC50 = 2.5g/mL; Bel7402, IC50 = 2.7g/mL; HeLa, IC50 = 3.9g/mL;
7441 Ethyl gallate
U937, IC50 = 1.3g/mL; control Colchicine, HL-60, IC50 = 1.6g/mL;
Gallic acid ethyl ester [831-61-8] C9H10O5 (198.18). White rhombic crystals
Bel7402, IC50 = 0.4g/mL; HeLa, IC50 = 0.1g/mL; U937, IC50 =
(chloroformmethanol), mp 155~158C. Pharm: Antibacterial (Bacillus
0.1g/mL)[4746]. Source: LA ZHU GUO Aegiceras corniculatum (stem and

twig: yield = 0.00050%). Ref: 4746.
O
dysenteriae); antifibrotic; platelet aggregation inhibitor (in vitro); inhibits

OH-free radicals damaging AT-III (Antithrombase-III) (0.6 mmol/L, InRt =
48.5%); collagenase inhibitor (hmn in vitro, IC50 = 2g/mL); analgesic.
OH
Source: A LA BO JIN HE HUAN Acacia arabica, CHA TIAO QI Acer

ginnala, DA HUA HONG JING TIAN Rhodiola crenulata [Syn. Rhodiola
O
O
euryphylla], HE ZI Terminalia chebula, LI SHU PI Castanea mollissima, MU

MIAN HUA Bombax malabaricum [Syn. Gossampinus malabarica], SHE PU
7437 -1-C-Ethyl-fagomine
TAO Ampelopsis brevipedunculata, SHENG DI HONG JING TIAN Rhodiola
C8H17NO3 (175.23). []D = +45.7 (c = 0.71, H2O). Pharm: Enzymes inhibitor
sacra, WAN SHOU JU Tagetes erecta, XI XI LI QI SHU Rhus coriaria. Ref:
(-glucosidase: rice, IC50 = 490mol/L, control DMDP, IC50 = 300mol/L;
552, 660, 900.
yeast, IC50 > 1000mol/L, DMDP, IC50 = 3.6mol/L; rat intestinal maltase,
O
IC50 > 1000mol/L, DMDP, IC50 = 290mol/L; -glucosidase, almond, IC50 >
1000mol/L, DMDP, IC50 = 13mol/L; -galactosidase, bovine liver, IC50 =

29mol/L, DMDP, IC50 = 2.2mol/L; trehalase, porcine kidney, IC50 >
HO
OH
OH
1000mol/L, DMDP, IC50 = 200mol/L; amyloglucosidase, Aspergillus niger,

IC50 > 1000mol/L, DMDP, IC50 = 19mol/L). Source: RI BEN SAN YE
SHA SEN Adenophora triphylla var. japonica (fresh whole herbs). Ref: 3915.
7442 Ethyl geranate

[13058-12-3] C12H20O2 (196.29). bp 110~120C. Source: YUN XIANG CAO
Cymbopogon distans. Ref: 6.
H
N
HO
O
O
HO
OH
7438 Ethyl--D-fructoside
C8H16O6 (208.21). Source: DANG SHEN Codonopsis pilosula. Ref: 2.
7443 Ethyl -D-glucopyranoside

C8H16O6 (208.21). Colorless syrup, []D23 = 26. Source: BEI SHA SHEN Glehnia
littoralis (fruit), SHI LUO ZI Anethum graveolens (fruit). Ref: 3525, 4177.
OO
HO
OO
HO
HO
OH
OH
OH
OH
OH
314
7444 Ethyl heptadecanoate
7450 24-Ethylidene lophenol
Ethyl margarate [14010-23-2] C19H38O2 (298.51). Source: CHUAN XIONG
[474-40-8] C30H50O (426.73). mp 162~164C. Source: GAN ZHE Saccharum
sinensis. Ref: 6.
7445 5-O-Ethyl-hirsutanonol
C21H26O6 (374.44). Pharm: Antioxidant (superoxide radical scavenger, IC50 =
2.9mol/L; DPPH scavenger, IC50 = 4.3mol/L). Source: CHI YANG Alnus
japonica (leaf). Ref: 4535.
HO
7451 trans-3-Ethylidene-2-pyrrolidinone
Corydalactam [930-94-9] C6H9NO (111.14). mp 172~174C. Source: JU HUA
HUANG LIAN Corydalis pallida. Ref: 6.
HO
OH
HO
OH
H
O
N
H
7446 Ethyl (6-O-p-hydroxybenzoyl)--D-glucopyranoside
7452 Ethylisoheptadecanoate
C15H20O8 (328.32). Source: ZI YE Catalpa ovata (fallen leaf). Ref: 4290.

OO
O
OH
HO
OH
OH
O
7447 N-Ethyl-1-hydroxy-17-veratroyldictizine
25
C31H43NO7 (541.69). Amorphous solid, []D = +30.0 (c = 0.11, CHCl3).
7453 Ethylisooctadecanoate
Source: BAN HUA WU TOU Aconitum variegatum (aerial parts). Ref: 5270.

O
OH
O
OH
OH O
7454 Ethylisopropyl sulfide

7448 Ethylidene-3,3'-biplumbagin
2-Methyl-3-thiapentane [5145-99-3] C5H12S (104.22). Source: SHENG
C24H18O6 (402.41). Orange-red plates (hexaneC 6H 6), mp 200~201C. Pharm:
JIANG Zingiber officinale. Ref: 2.
Ichthyotoxin (MLC > 10mg/L, control Juglone, MLC = 0.2mg/L). Source:

HAI SHI Diospyros maritima (fruit). Ref: 4185.
O
Ethyl dodecanoate [106-33-2] C14H28O2 (228.38). Source: BAI ZHI Angelica

dahurica [Syn. Angelica porphyrocaulis]. Ref: 2.
OO
OH
S
7455 Ethyllaurate
HO
7449 Ethylidene-3,6'-biplumbagin
O
C24H18O6 (402.41). Orange-red plates (hexaneC6H6), mp 185~186C, []D28 =

1.50 (c = 1.28, CHCl3). Pharm: Ichthyotoxin (MLC > 10mg/L, control Juglone,
7456 Ethylleptol B
MLC = 0.2mg/L). Source: HAI SHI Diospyros maritima (fruit). Ref: 4185.
C17H24O4 (292.38). Yellowish oleaginous substances, []D10 = +3.26 (c = 0.307,

Me2CO). Source: SAN CHA KU Evodia lepta [Syn. Ilex lepta]. Ref: 393.
O
O
O HO
OH
315
7457 Ethyl lithospermate
7463 Ethyl-2-methylbut-2-enoate
C30H28O12 (580.55). Brown yellow gum, []D23 = +65.6 (c = 0.25, MeOH).
[5837-78-5] C7H12O2 (128.17). Pharm: Flavorant. Source: WEN PO Cydonia
Pharm: Antioxidant (DPPH scavenger, IC50 = 0.1028mmol/L, control Propyl
oblonga. Ref: 658.
gallate, IC50 = 0.03mol/L; superoxide radical inhibitor, inactive, control
Propyl gallate, IC50 = 0.106mmol/L; iron chelating assay, inactive, control
Propyl gallate, IC50 = 0.064mmol/L). Source: MING XIAN HUA ZHU

CHANG ZHU LIU LI CAO Lindelofia stylosa (aerial parts). Ref: 4533.
7464 5-Ethyl-2-methylheptane
OH
OH
O
OH
O
O
H
O
O
O
7465 (2E)-2-Ethyl-2-nonacosenal
OH
C31H60O (448.82). White crystals, mp 65~66C. Source: JI DAN SHEN
O
OH
Codonopsis convolvulacea. Ref: 779.
7458 Ethyl-m-digallate
OH
OH
O
OH
O
OH
O
H
H
OH
7466 Ethylnotopterol
5-{(2E,5E)-3,7-Dimethyl-7-[(1-ethoxy)ethoxy-2,5-octadienyloxy]} psoralen
C23H26O5 (328.26). Colorless ropy substance. Source: QIANG HUO
7459 1-Ethyl-4-methoxy--carboline
Notopterygium incisum. Ref: 325.
C14H14N2O (226.28). Source: KU SHU PI Picrasma quassioides [Syn.

O

O
N
H
7467 Ethyloctadecanoate
7460 Ethyl p-methoxy-cis-cinnamate
Ethyl stearate [111-61-5] C20H40O2 (312.54). Source: CHUAN XIONG
C12H14O3 (206.24). Pharm: Anti-cancer-promoted activity (IC50 = 5.5mol/L).
Source: SHAN NAI Kaempferia galanga. Ref: 2252.

O
7461 5-Ethyl-1-methoxy-2,3-methylenedioxybenzene
7468 Ethyl O--D-oleandropyranosyl-(14)-O-3-O-methyl-6-deoxy-
-D-allopyranoside
C16H30O8 (350.41). Source: ROU LEI NIU NAI CAI Marsdenia roylei. Ref: 1875.
O
O
7462 1-Ethyl-2-methylbenzene
OO
[611-14-3] C9 H12 (120.20). Source: SHAN ZHA Crataegus pinnatifida.

Ref: 2.
OO
O
OH
O OH
316
7469 Ethylpalmitate
7476 Ethyl pyroglutamate
Ethyl hexadecanoate [628-97-7] C18H36O2 (284.49). mp () 24C, () 19.3C.
C7H11NO3 (157.17). Source: SAN QI Panax pseudo-ginseng var. notoginseng
Source: CHUAN XIONG Ligusticum chuanxiong [Syn. Ligusticum wallichii],
DANG SHEN Codonopsis pilosula, JIN YIN HUA Lonicera japonica, SAN QI
Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]. Ref: 2, 6, 638.
N
H
7477 4-Ethylresorcinol

7470 Ethyl-p-digallate
OH

HO
OH
OH
OH
O
O
OH
O
OH
7478 Ethyl rosmarinate

C20H20O8 (388.38). Pharm: Antioxidant (DPPH scavenger, IC50 = 0.0412mmol/L,
control Propyl gallate, IC50 = 0.03mol/L; superoxide radical inhibitor, inactive,
control Propyl gallate, IC50 = 0.106mmol/L; iron chelating assay, inactive, control
Propyl gallate, IC50 = 0.064mmol/L). Source: MING XIAN HUA ZHU CHANG
ZHU LIU LI CAO Lindelofia stylosa (aerial parts). Ref: 4533.
7471 Ethylpentadecanoate
[41114-00-5] C17H34O2 (270.46). Source: CHUAN XIONG Ligusticum
chuanxiong [Syn. Ligusticum wallichii]. Ref: 2.
HO
O
O
OH
OH
HO
7479 5-Ethyl-1,2,3-trimethoxybenzene
7472 m-Ethylphenol
C8H10O (122.17). Source: DANG GUI Angelica sinensis, YIN CHEN HAO
Artemisia capillaris. Ref: 2, 660.
O
O
7480 Eucalyptin
HO
[3122-88-1] C19H18O5 (326.35). mp 198.5~200.0C. Source: AN YE
7473 p-Ethylphenol
Eucalyptus globulus, NING MENG AN YE Eucalyptus citriodora. Ref: 6.
C8H10O (122.17). Source: DANG GUI Angelica sinensis, YIN CHEN HAO
Artemisia capillaris. Ref: 2, 660.
O
O
OH
HO
7474 Ethyl-p-methoxycinnamate
p-Methoxycinnamic acid ethyl ether [24393-56-4] C12H14O3 (206.24). Pharm:
Cytotoxic (HeLa). Source: SHAN NAI Kaempferia galanga, TU LIANG
JIANG Hedychium spicatum. Ref: 6, 658.
7481 Eucalyptol
[470-82-6] C10H18O (154.25). Colorless liquid, camphor-like odor, mp 1.5C,
bp 176~177C. Pharm: Analgesic; antiasthmatic; antibacterial;
anti-inflammatory; anthelmintic; antipyretic. Source: AN YE Eucalyptus
globulus (95.13% in volatile oil), BAI QIAN CENG Melaleuca leucadendra,
BIN HAO Artemisia maritima, DA YE AN YE Eucalyptus robusta, GAO
LIANG JIANG Alpinia officinarum (dried rhizome: mean content of 6 origins

O
O
7475 Ethylpropionate
[105-37-3] C5H10O2 (102.13). Source: SHENG JIANG Zingiber officinale,
CHUAN XU DUAN Dipsacus asperoides. Ref: 2, 660.
= 0.35%)[5508], LUO LE Ocimum basilicum, MEI GUO XIA LA MEI

Calycanthus floridus, QING GUO Canarium album, SHU ZHI BAN RI HUA
Csitus ladaniferus, TU QIANG HUO Hedychium coronarium, ZHANG MU
Cinnamomum camphora (wood: content = 0.21%[5501]), ZI SUI HUAI
Amorpha fruticosa. Ref: 661, 5501, 5508.
O
O
O
317
7482 Eucalyptus wax
7487 Eucommin A
C33H64O2 (492.88). Pharm: Used in treatment of diseases in lung and
(+)-Medioresinol monoglucoside [99633-12-2] C27H34O12 (550.56). Pharm:
bronchus. Source: Eucalyptus sp., Acacia sp. Ref: 658.
Immunomodulator Source: DU ZHONG Eucommia ulmoides, HUANG

CHAN Allemanda neriifolia. Ref: 2.
O
OH
O
7483 Eucarvone
H
O
[503-93-5] C10H14O (150.22). bp 99~100C/22mmHg. Source: LIAO XI XIN

Asarum heterotropoides var. mandshuricum. Ref: 2, 660, 1521.
HO
OO
O
OH
OH
OH
7488 Eucommiol
Ref: 2.
7484 Euchrenone
OH
C25H26O4 (390.48). Source: GUANG GUO GAN CAO Glycyrrhiza glabra.
OH
Ref: 2431.
HO
O
HO
OH
7489 EucommiosideI
Ref: 2.
OH
O
O
HO
7485 (2S)-Euchrenone A7
HO
HO
Anticancer Flavonoid PMV70P691-90 C20H20O5 (340.38). Pharm: Aromatase

6.4mol/L)
. Source: GOU SHU Broussonetia papyrifera. Ref: 3090,
5038.
OH
OH
inhibitor (in vitro, IC50 = 3.4mol/L; control Aminoglutethimide, IC50 =

[3090, 5038]
OH
7490 Eucommioside-II
Ref: 2.
OH
HO
OH
HO
OH
OH
OH
OH
HO
OH
7491 (+)-Eudesma-5,7(11)-diene
C15H24 (204.36). Colorless oil. Source: Tritomaria polita (essential oil). Ref:
7486 (2S)-Euchrenone A16

5,7-Dihydroxy-8-(,-dimethylallyl)-[6''',6'''-dimethyl-4''',5'''-dihydropyrano-(2
3446.
''',3''':4',3')]-flavanone C25H28O5 (408.50). Yellow oil, []D24 = 213 (c = 0.05,

CHCl3). Source: TAI WAN SHAN DOU GEN Euchresta formosana. Ref:
1977.
7492 ()-Eudesma-3,11-dien-5-ol
C15H24O (220.36). Source: KAN MAI NIANG ZHUANG SHA CAO Cyperus
O
HO
OH
OH
318
7493 Eudesma-4(15),11(13)-dien-12,5-olide
7499 ()-Eudesma-2,4(15),11-triene
C15H20O2 (232.33). Source: LIU LENG JU Laggera alata (aerial parts: yield
= 0.00083%dw). Ref: 4709.
O
H
7494 Bis-[8-eudesma-4(15),7(11)-dien-12,8-olide]
C30H38O4 (462.63). Colorless prisms, mp 211~212C (CH2Cl2), 210~212 C,
7500 Eudesma-3,5,11-triene
[]D20 = +255.8 (c = 0.122, CHCl3). Source: Trattinickia rhoifolia (resin). Ref:
4213.

H
O
O
O
O
H
7495 (+)-Eudesma-4(15),7(11)-dien-8-one
7501 ()-Eudesm-3-ene-6-acetoxy-7-ol
Selina-4(15),7(11)-dien-8-one; Selina-4(14),7(11)-dien-8-one C15H22O
C17H28O3 (280.41). Colorless needle crystals, mp 141~142C. Source: LIE E
20
(218.34). Colorless oil, []D = +92.6 (c = 0.034, methanol). Pharm:
TAI Chiloscyphus polyanthus. Ref: 2188.
Anti-inflammatory (mus, reduces blood capillary permeability caused by

acetic acid, 300mg/kg, InRt = (31.611.9)%). Source: BAI ZHU Atractylodes
OH
macrocephala [Syn. Atractylis macrocephala], BEI CANG ZHU Atractylodes

chinensis, CANG ZHU Atractylodes lancea, GUAN CANG ZHU
Atractylodes japonica, SHUANG YE XI XIN Asarum caulescens. Ref: 660,
661.
O
7502 ent-4(15)-Eudesmene-1,6-diol
C15H26O2 (238.37). Amorphous, []D26 = 36.8 (c = 0.16, CHCl3), []D12 =
31.5 (c = 0.13, MeOH). Source: ZHAO WA JIA KE TAI Jackiella javanica.

7496 (+)-Eudesma-3,7(11)-dien-8-one
Ref: 5303.

Ref: 3446.
OH
O
H
OH
7497 (+)-Eudesma-3,11-dien-8-one
7503 7-Eudesmene-1,4-diol
Ref: 3446.
C15H26 O2 (238.37). Colorless plates, mp 107~109C. Pharm:

Antiplasmodial (Plasmodium falciparum strains, IC50 = 4.17g/mL,
O
control Chloroquine, IC 50 = 0.0028g/mL)[2383] . Source: Reneilmia

cincinnata (fruits). Ref: 2383.
H
OH
7498 Eudesma-2,4,11-triene
HO
319
7504 Eudesm-4(15)-ene-1,6-diol
7508 (+)-Eudesm-3-ene-7-ol
1,6-Dihydroxy-eudesman-4(15)-ene C15H26O2 (238.37). Colorless oil,
C15H26O (222.37). Greenish oil. Source: LIE E TAI Chiloscyphus polyanthus.
[]D = +4.5 (c = 0.2, CHCl3); []D17 = +7 (c = 0.50, CHCl3); White powder,
Ref: 2188.
[]D20 = 27.1 (c = 1.47, CHCl3); colorless needles (petroleum ether-EtOAc),

[]D20 = +45 (c = 0.1, CHCl3). Pharm: Cytotoxic (inhibits growth of Bel7402
OH
cell, 0.0001mol/L, InRt = 29.1%, control Etoposide, InRt = 96.0%)[5073];

anti-HIV-1 inactive (in vitro, HOG.R5)[4688]. Source: DIE DA LAO Litsea
verticillata (leaf and twig: 0.00049%dw), FEI CHENG FEI PENG Erigeron
7509 Eudesm-3-en-7-ol
philadelphicus (aerial parts), HUANG HUA HAO Artemisia annua (seed),
(+)-(2R,4aS,8aR)-1,2,3,4,4a,5,6,8a-Octahydro-4a,8-dimethyl-2-(1-methylethy
SU MEN BAI JIU CAO Erigeron sumatrensis (aerial parts), YI NIAN PENG
l)-2-naphthalenol C15H26O (222.37). Colorless oil. Source: YING ZHI YE
Erigeron annuus (aerial parts), ZHONG JIAN JIN JI ER Caragana
TAI Lepidozia vitrea (essential oil). Ref: 5209.
intermedia (aerial parts). Ref: 3435, 4338, 4688, 4786, 5073.

OH
OH
7510 Eudesm-4-en-7-ol
()-1,2,3,4,4a,5,6,7-Octahydro-4a,8-dimethyl-2-(1-methylethyl)-naphthalen-2
OH
-ol C15H26O (222.37). Colorless oil. Source: DONG YA ZHI YE TAI
7505 4(15)-Eudesmene-1,5-diol
1,5-Dihydroxyeudesman-4(15)-ene C15H26O2 (238.37). Colorless
monoclinic crystals (petroleum etherEtOAc), [] D20 = +122 (c = 0.7, CHCl3);
Lepidozia fauriana (essential oil), YING ZHI YE TAI Lepidozia vitrea

[]D17 = +30 (c = 0.10, CHCl3). Pharm: Antifungal (Pyricularia oryzae P-2b,
OH
MIC = 20g/mL)[4786]; glucose consumption activity (C2C12 muscle cell assay,

IC = 10.7g/mL; in animal tests, it showed the same effect on oral glucose
tolerance in db/db mouse as metformin, MIC = 100mg/mL)[4786]. Source: YI
NIAN PENG Erigeron annuus (aerial parts), ZHONG JIAN JIN JI ER
Caragana intermedia (aerial parts). Ref: 4338, 4786, 5073.
7511 Eudesm-4(15)-en-7-ol
()-(2R,4aS,8aR)-Decahydro-4a-methyl-8-methylene-2-(1-methylethyl)-2-na
phthalenol C15H26O (222.37). Colorless oil. Source: YING ZHI YE TAI
OH
Lepidozia vitrea (essential oil). Ref: 5209.

OH
OH
7512 Eudesmin
1,7-Dihydroxyeudesman-4(15)-ene C15H26O2 (238.37). Colorless oil,
C22H26O6 (386.45). mp 107~108C. Pharm: Tuberculostatic (in vitro); calcium
[]D17 = +30 (c = 0.13, CHCl3); colorless needles (petroleum ether-EtOAc),
antagonist (gpg, colon bands). Source: BAN PI AN Eucalyptus hemiphloia,
[]D20 = +35 (c = 0.1, CHCl3). Pharm: Antifungal (Pyricularia oryzae P-2b,
WANG CHUN YU LAN Magnolia biondii [Syn. Magnolia fargesii], XI
MIC = 12g/mL)[4786]. Source: YI NIAN PENG Erigeron annuus (aerial
BING MU JIANG ZI Litsea gracilipes, ZHAI YE NAN YANG SHAN
parts), ZHONG JIAN JIN JI ER Caragana intermedia (aerial parts). Ref:
Araucaria angustifolia, ZHOU YE MU LAN Magnolia praecocissima (seed),
4786, 5073.
Haplophyllum sp. Ref: 6, 658, 660, 4181.
OH
O
O
OH
O
H
H
O
20
C15H26O2 (238.37). Colorless needles (petroleum ether-EtOAc), []D = 12

(c = 0.1, CHCl3). Pharm: Antifungal (Pyricularia oryzae P-2b, MIC =
16g/mL)[4786]. Source: ZHONG JIAN JIN JI ER Caragana intermedia (aerial
parts). Ref: 4786.
OH
7513 -Eudesmol
[473-16-5] C15H26O (222.37). mp 75C, bp 156C/10mmHg. Source: CANG
ZHU Atractylodes lancea, HOU PO Magnolia officinalis, AO YE HOU PO
Magnolia biloba. Ref: 6, 660.
OH
H
H
OH
320
7514 -Eudesmol
7518 Eugeniin
[473-15-4] C15H26O (222.37). mp 76C. Pharm: NO production inhibitor (mus
Tellimagrandin II; Cornustannin 2 [58970-75-5] C41H30O26 (938.68). Pharm:
peritoneal macrophages, induced by LPS, 100mol/L, InRt = (98.51.8)%,
Antiviral (herpes simplex virus); inhibits lipolysis (rat fat cells, induced by
control L-NMMA, 100mol/L, InRt = (79.20.9)%, p<0.01)[4150]. Source: AO
adrenaline); antioxidant (SOD-like activity, EC50 = 94.8mol/L, control Gallic
YE HOU PO Magnolia biloba, BEI CANG ZHU Atractylodes chinensis
acid, EC50 = 31.7mol/L, L-Ascorbic acid, EC50 = 34.6mol/L)[3408];
[5531]
(dried rhizome: content = 2.20%
), CANG ZHU Atractylodes lancea
(dried rhizome: content scope of 5 origins = 0.44%~1.56%, mean content =

[5531]
0.84%
), FANG FENG Saposhnikovia divaricata [Syn. Ledebouriella
antioxidant (DPPH scavenger, EC50 = 0.44mol/L, control Gallic acid, EC50 =

5.88mol/L, L-Ascorbic acid, EC50 = 6.25mol/L)[3408]. Source: BAI SHAO
Paeonia albiflora [Syn. Paeonia lactiflora], BAI SHAO Paeonia albiflora
seseloides] (root: content = 1.549% in male, content = 1.727% in female)[5501],
[Syn. Paeonia lactiflora] (fresh fruit: yield = 0.063%fw)[4695], CHI SHAO
GAN SONG Nardostachys chinensis, GUAN CANG ZHU Atractylodes
Paeonia lactiflora wild, DING XIANG Syzygium aromaticum [Syn. Eugenia
japonica (dried rhizome: content = 0.02%)[5531], HOU PO Magnolia officinalis,
caryophyllata], HU TAO REN Juglans regia, RI BEN MA SANG Coriaria
LIU SHAN Cryptomeria fortunei, PING E SHU Curcuma zedoaria [Syn.
japonica, SHAN ZHU YU Cornus officinalis [Syn. Macrocarpium officinale],
Curcuma aeruginosa], SHENG JIANG Zingiber officinale. Ref: 2, 6, 660,
XIN SHAO NA CAO Tellima grandifolia, Rosa sp., Quercus sp., Fuchsia sp.
4150, 5501, 5531.
Ref: 2, 658, 3408, 4695.

OH
OH
HO
H
HO
OH
OH
O
HO
O
O
OO
O
HO
7515 -Eudesmol
O
OH
HO
2,2,15, IC50 = 0.01g/mL). Source: YI LAN Cananga odorata (fruit). Ref:
OH
O
OH
C15H26O (222.37). Pharm: Cytotoxic (in vitro, HepG2, IC50 = 1.5g/mL, Hep
OH
O
OH
OH
OH
3055.
7519 Eugenin
C11H10O4 (206.20). Pharm: Cytotoxic (hmn peripheral blood T cells, dose =

5.0g/mL, T cell survival rate = 98%)[3498]; immunosuppressant (inhibits IL-2
OH
secretion costimulated by CD28, dose = 5.0g/mL, InRt = 59%). Source:

HONG CHAI HU Bupleurum scorzonerifolium (root). Ref: 3498.
O
7516 -Eudesmol 11--L-rhamnoside
25
C21H36O5 (368.52). Gum, []D = 11.5 (c = 0.24, CHCl3). Pharm: Cytotoxic

(in vitro, HepG2, IC50 = 3.9g/mL, Hep2,2,15, IC50 = 10.6g/mL). Source:
OH
YI LAN Cananga odorata (fruit). Ref: 3055.
OH
7520 Eugenitin
[480-12-6] C12H12O4 (220.23). mp 162C. Source: DING XIANG Syzygium
OH OH
aromaticum [Syn. Eugenia caryophyllata]. Ref: 6.

OH
7517 Eudesobovatol A
[125196-77-2] C33H44O4 (504.72). Pharm: CNS depressant; used in treatment
of neurosis and gastrointestinal disease; neurotrophic. Source: RI BEN HOU
PO Magnolia obovata. Ref: 658.

7521 Eugenol
4-Allyl-2-methoxyphenol [97-53-0] C10H12O2 (164.21). mp 9C, bp
254~255C. Pharm: Antibacterial (Staphylococcus aureus, Klebsiella
OH
O
OH
pneumoniae, Escherichia coli, Shigella shigae, Bacillus proteus etc., IC =

1:2000~1:8000)[5501]; antifungal (pathogen fungi, EC = 1:8000~1:16000)[5501];
antioxidant[5501]; CNS activity (rbt, iv, anesthesia action, lowers blood
pressure, inhibits respiration and anticonvulsion)[5501]; platelet aggregation
inhibitor (rbt platelets induced by thrombin, 100g/mL, add thrombin
0.1u/mL, AggRt = (91.90.4)%, control AggRt = (92.60.4)%; add AA,
321
100mol/L, 100g/mL, AggRt = (0.00.0)%, 2g/mL, AggRt = (86.33.9)%,
7522 Eugenol--D-glucopyranoside
control AggRt = (87.80.3)%, Aspirin 50g/mL, AggRt = (11.710.1)%; add
3-Hydroxyestragole--D-glucopyranoside C16H22O7 (326.35). Amorphous
collagen 10g/mL, 100g/mL, AggRt = (17.15.6)%, 2g/mL, AggRt =
powder, []D23 = 34 (c = 0.4, MeOH). Pharm: Neurite outgrowth enhancer
(88.21.0)%, control AggRt = (89.30.5)%, Aspirin 100g/mL, AggRt =
inactive (PC12D cells, nerve growth factor-mediated, 10-100mol/L)[4745].
(81.30.5)%; add PAF 2ng/mL, 100g/mL, AggRt = (91.01.0)%, control
Source: HUI QIN Pimpinella anisum (fruit), SHE XIANG CAO Thymus
AggRt = (93.00.6)%)[4938]; antipyretic (rbt with IL-induced fever, stronger
vulgaris, YE GAN CAO Scoparia dulcis (aerial parts: yield = 0.0015%). Ref:
than acetyl aminophenol, antipyretic mechanism involves inhibition of PG
2592, 3402, 4745.
synthesis in brain)[5501]; anti-inflammatory (rat, swollen foot model caused

O
by carrageenan; mouse, edema on ears caused by oleum crotonis; gpg, edema

on ears caused by benzoic acid)
[5501]
; smooth muscle relaxant (smooth muscle
in blood vessel, intestine and isolated uterus, smooth muscle in gpg trachea
ED50 = (395)mol/L, smooth muscle in gpg ileum ED50 = (6.81.0)g/mL,
but causes constriction of rat isolated bladder)[5501]; anti-androgenic
(testosterone-5-reductase inhibitor)
[5501]
; LD50 (rat, orl) = 1.93g/kg, (rat, orl)
HO
OH
OH
OH
7523 Eugenol methyl ether
= 2.68g/kg; (mouse, orl) = 3g/kg[5501]. Source: BAI CHANG Acorus calamus,
Methyl eugenol [93-15-2] C11H14O2 (178.23). bp 248~249C. Pharm:
CHA SHU Sassafras tzumu, CHAI HU Bupleurum chinense, DA LIANG
Antispasmodic. ; CNS depressant; antipyretic; skeletal muscle relaxant.
JIANG Alpinia galanga, DING XIANG Syzygium aromaticum [Syn. Eugenia
Source: JU JIANG YE Piper betle, LIAO XI XIN Asarum heterotropoides var.
caryophyllata] (dried bud: content scope = 11.2%~15.3%[5501], mean content =
mandshuricum, LUO LE Ocimum basilicum, ROU DOU KOU Myristica
12.49%[5508]), DU HENG Asarum forbesii, DUO XIANG GUO Pimenta
fragrans (kernel: content = 1.052%)[5508], SHAN ZHU YU Cornus officinalis
dioica, FAN SHI LIU YE Psidium guajava, FEI LONG ZHANG XUE
[Syn. Macrocarpium officinale], SHENG JIANG Zingiber officinale, SHI
Toddalia asiatica [Syn. Toddalia aculeata; Paullinia asiatica], GAO LIANG
CHANG PU Acorus tatarinowii, SI JING JIE BA DOU Croton nepetaefolius,
JIANG Alpinia officinarum, GUANG HUO XIANG Pogostemon cablin [Syn.
XI XIN Asarum sieboldii, YIN CHEN HAO Artemisia capillaris, occurs in
Mentha cablin], GUI PI Cinnamomum japonicum, HUANG HAO Artemisia
many plants (in many essential oils). Ref: 2, 4, 658, 660, 5501, 5508.
scoparia [Syn. Artemisia capillaris var. scoparia], JIA JING JIE Nepeta
cataria, JIAN ZI SU YE Perilla frutescens var. acuta [Syn. Perilla frutescens
var. purpurascens], JIN YIN HUA Lonicera japonica, JIU LI XIANG
Murraya paniculata [Syn. Chalcas paniculata], JU JIANG YE Piper betle,
KE SHI HAO Artemisia klotzschiana, KONG SHI CHUN Ulva pertusa, LUO
LE Ocimum basilicum, MA HUA Cannabis sativa, MEI GUI HUA Rosa
rugosa, MO YAO Commiphora myrrha [Syn. Commiphora molmol], ROU
O
O
7524 Eugenone
[480-27-3] C13H16O5 (252.27). mp 97~98C. Source: DING XIANG Syzygium
aromaticum [Syn. Eugenia caryophyllata]. Ref: 6.
DOU KOU Myristica fragrans (kernel: content = 0.456%)[5508], SAN TIAO

O
JIN Cinnamomum tamala, SANG YE Morus alba, SHE XIANG SHI CAO
Achillea moschata, SHI CHANG PU Acorus tatarinowii, SHI ZHU Dianthus

chinensis, SHI XIANG RU Mosla chinensis [Syn. Orthodon chinensis], SHUI
XIAN HUA Narcissus tazetta var. chinensis, TAI WAN CHA MU Sassafras
randainense, TAI WAN HU JIAO Piper taiwanense (stem), TIAN NIU ZHI
Origanum majorana, XI XIN Asarum sieboldii, XIANG ZHANG
Cinnamomum parthenoxylum [Syn. Cinnamomum porrectum], XIAO CAO
WU Delphinium yunnanense, XIN YI Magnolia liliflora, YANG SHI CAO
Achillea millefolium, YE XIANG SHU Cestrum nocturnum, YIN CHEN
7525 Eugenylglucoside
3,4-Dihydroxy-allylbenzene-4-O--D-glucopyranoside C15H20O7 (312.32).
White powder. Source: BAI MEI HUA Prunus mume (flower: yield =
0.050%fw), JIAN YE LONG XUE SHU Dracaena cochinchinensis. Ref:
2114, 4641.
HAO Artemisia capillaris, YIN XING CAO Siphonostegia chinensis, YUE
HO
GUI ZI Laurus nobilis, ZHANG MU Cinnamomum camphora, Ocimum sp.,

occurs in many plants. Ref: 2, 4, 11, 638, 658, 660, 4938, 5501, 5508.
HO
OO
OH
OH
OH
7526 Eugenyl--rutinoside
C22H32O11 (472.49). Yellow-white powder. Source: BO SI YI MU CAO
Leonurus persicus. Ref: 2499.
O
OH
OH
OO
OO
OH
OH OH
OH
OH
322
7527 Euglobal Ia1
7531 Euglobal III
[77844-93-0] C23H30O5 (386.49). Pharm: Inhibits granulation. Source: AN YE
[76449-26-8] C28H38O5 (454.61). Colorless acicular crystals (ethanol), mp
Eucalyptus globulus. Ref: 658.
169~170C, []D20 = +229 (c = 1.0, chloroform). Pharm: Anti-inflammatory;

antineoplastic (EBV-EA induced by TPA, InRt = 100% with molecular ratio
of Euglobal-III/TPA 1000, while InRt over 70% with ratio 500). Source: AN
HO
YE Eucalyptus globulus. Ref: 981, 984, 1013.
H
O
OH
HO
O
H
7528 Euglobal Ib
OH
[77844-94-1] C23H30O5 (386.49). Colorless acicular crystals (chloroform), mp

118~120C, []D = +2.27 (c = 0.65, chloroform). Pharm: Anti-inflammatory;
antineoplastic (EBV-EA induced by TPA, InRt = (70~80)% with molecular
7532 Euglobal V
ratio of Euglobal-Ib/TPA 1000, while InRt = 50% with ratio 100). Source: AN
[77809-89-3] C28H38O5 (454.61). Colorless rhombic crystals, mp 184~185C,
YE Eucalyptus globulus. Ref: 977, 982.
[]D20 = 206 (c = 1, chloroform). Pharm: Anti-inflammatory; antineoplastic

(EBV-EA induced by TPA, InRt = 80% with molecular ratio of
Euglobal-V/TPA 1000, while InRt over 40% with ratio 500). Source: AN YE
HO
Eucalyptus globulus. Ref: 981, 984, 1042.
OH
HO
O
H
7529 Euglobal Ic
OH
[77794-60-6] C23H30O5 (386.49). Colorless rhombic crystals (ethanol), mp

108~110C, []D20 = 3.12 (c = 1.0, chloroform). Pharm: Anti-inflammatory;
7533 Eukovoside
antineoplastic (EBV-EA induced by TPA, InRt over 80% with molecular ratio
C30H38O15 (638.63). Amorphous powder. Source: DUAN XIAN XIAO MI
of Euglobal-Ic/TPA 1000, while InRt = (20~30)% with ratio 100). Source: AN
CAO Euphrasia regelii. Ref: 2432.
H
HO
OH
OH
OH
OH
OH OH
O
OH
OO
HO
OH
O
7534 Euonymine
7530 Euglobal Iia
C38H47NO18 (805.79). White powder. Source: LEI GONG TENG
[77844-92-9] C23H30O5 (386.49). Colorless rhombic crystals (chloroform), mp
Tripterygium wilfordii (root heart). Ref: 4559.
115~117C, []D = +26.7 (c = 0.7, chloroform). Pharm: Anti-inflammatory;

antineoplastic (EBV-EA induced by TPA, InRt over 80% with molecular ratio
of Euglobal-Iia/TPA 1000, while InRt (20~30)% with ratio 100). Source: AN

O
O
O
H
HO
O OH
O
H
OH
O
O
O
O
323
7535 Euonymoside A
7538 Euoverrine B
[155740-04-8] C35H54O14 (698.81). Colorless thin crystals (methanol), mp
C43H49NO18 (867.87). Amorphous white powder, mp. 148~149C, []D24 =
172~173C, []D25 = +33.9 (c = 2.42, chloroform:methanol = 4:1). Pharm:
+10.9 (c = 0.55, CHCl3). Source: YOU DIAN WEI MAO Euonymus
Cytotoxic (A549 in vitro, IC50 = 0.06g/mL, SK-OV-3, IC50 = 0.4g/mL).
verrucosides, FU FANG TENG Euonymus fortunei, SHUAN CHI WEI MAO
Source: XI BO SHI WEI MAO Euonymus sieboldianus Ref: 994, 1148, 1521.
Euonymus phellomana. Ref: 1928.
O
O
OH
H
H
OH
OO
O
H
OH
O
HO
O
O O
OH O
HO
O
OH
OH
7539 Eupachifolin D
OH
C22H27ClO8 (454.91). Source: CHENG GAN SHENG MA Eupatorium

lindleyanum (whole herb: yield = 0.00036%dw)[4762], HUA ZE LAN
7536 Euophelline
C47H51NO17 (901.93). Amorphous white powder, mp 168~169C, []D24 =
Eupatorium chinense (whole herb: yield = 0.0023%)[4739]. Ref: 4739, 4762.
+2.2 (c = 0.45, CHCl3). Source: YOU DIAN WEI MAO Euonymus

Cl
OH
O
O
O
O
OH
O
O
HO
O
O
O
O O
HO
O
7540 Eupachinilide A
8-Angelyloxy-3,4,14-trihydroxy-5H,6H,7H-guai-1(10),11(13)-diene-6
,12-olide C20H26O7 (378.43). White powder, []D20 = 65.8 (c = 0.58,
CH3OH). Pharm: Cytotoxic (in vitro, HL-60, IC50 = 10.8g/mL; Bel7402,
IC50 = 72.2g/mL; control Hydroxycamptothecin, HL-60, IC50 = 0.024g/mL;
Bel7402, IC50 = 0.62g/mL). Source: HUA ZE LAN Eupatorium chinense

(whole herb: yield = 0.0036%). Ref: 4739.
OH
7537 Euoverrine A
C48H51NO18 (929.94). Amorphous white powder, mp 145~146C, []D24 =
+5.5(c = 0.55, CHCl3). Source: YOU DIAN WEI MAO Euonymus
O
HO

O
O
O
O
7541 Eupachinilide B
8-(4'-Hydroxytiglyloxy)-3,4-epoxy-2-hydroxy-1H,5H,6H,7H-guai-
O
O
HO
O
O
O
O
HO
1(10),11(13)-diene-6,12-olide C20H24O7 (376.41). White powder, []D20 =

O
O
O O
67.1 (c = 0.50, CH3OH). Source: HUA ZE LAN Eupatorium chinense

HO
O
O
OH
O
O
324
7542 Eupachinilide C
7546 Eupachinilide G
C20H25ClO7 (412.87). Gum, []D20 = 66.9 (c = 0.50, CH3OH). Source:
8-(2',3'-Epoxy-2'-methylbutanoxy)-4-hydroxy-14-oxo-5H,6H,7H-guai-
CHENG GAN SHENG MA Eupatorium lindleyanum (whole herb: yield =
1(10),2,11(13)-triene-6,12-olide C20H22O7 (374.39). Gum, []D20 = 216.5 (c
0.0265%dw)[4762], HUA ZE LAN Eupatorium chinense (whole herb: yield =
= 0.65, CH3OH). Source: HUA ZE LAN Eupatorium chinense (whole herb:
[4739]
0.00032%)
. Ref: 4739, 4762.
Cl
OH
HO
yield = 0.00023%). Ref: 4739.

H
O
O
O
OH
HO
O
7543 Eupachinilide D
8-Angelyloxy-4-hydroxy-14-oxo-5H,6H,7H-guai-2,10(14),11(13)-trien
7547 Eupachinilide H
e-6,12-olide C20H22O6 (358.39). White powder, []D20 = 204.0 (c = 1.53,
8-(2',3'-Dihydroxy-2'-methybutanoxy)-2-hydroxy-6H,7H-germacra-1(10
CH3OH). Source: HUA ZE LAN Eupatorium chinense (whole herb: yield =
)-E,4E,11(13)-triene-6,12-olide C20H28O7 (380.44). White powder, []D20 =
0.0036%). Ref: 4739.
+34.7 (c = 0.54, CH3OH). Source: HUA ZE LAN Eupatorium chinense

O
O
HO
OH O
O
O
OH
OH
7544 Eupachinilide E
8-(4'-Hydroxytiglyloxy)-14-chrorine-3,4-epoxy-2,10-dihydroxy-1H,5
H,6H,7H-guai-11(13)-ene-6,12-olide C20H25ClO8 (428.87). White powder,
[]D20 = 59.4 (c = 0.60, CH3OH). Pharm: Cytotoxic (in vitro, HL-60, IC50 =
7548 Eupachinilide I
1.3g/mL; Bel7402, IC50 = 18g/mL; control Hydroxycamptothecin, HL-60,
8-(4'-Acetoxyangelyloxy)-2-hydroxy-6H,7H-germacra-1(10)-E,4E,11(13
IC50 = 0.024g/mL; Bel7402, IC50 = 0.62g/mL)[4739]. Source: CHENG GAN
)-triene-6,12-olide C22H28O7 (404.46). White powder, []D20 = +76.1 (c =
SHENG MA Eupatorium lindleyanum (whole herb: yield = 0.00059%dw)[4762],
0.65, CH3OH). Pharm: Cytotoxic (in vitro, HL-60, IC50 = 0.94g/mL;
HUA ZE LAN Eupatorium chinense (whole herb: yield = 0.0032%)
[4739]
. Ref:
4739, 4762.
0.024g/mL; Bel7402, IC50 = 0.62g/mL). Source: HUA ZE LAN
Cl
OH
HO
Bel7402, IC50 = 3.6g/mL; control Hydroxycamptothecin, HL-60, IC50 =

Eupatorium chinense (whole herb: yield = 0.0018%). Ref: 4739.
O
HO
O
O
OH
O
7545 Eupachinilide F
O
O
O
8-(4'-Hydroxytiglyloxy)-2-acetoxy-14-chlorine-3,4-epoxy-10-hydroxy1H,5H,6H,7H-guai-11(13)-ene-6,12-olide C22H27ClO9 (470.91). White

powder, []D20 = 52.3 (c = 0.84, CH3OH). Pharm: Cytotoxic (in vitro,
7549 Eupachinilide J
HL-60, IC50 = 0.87g/mL; Bel7402, IC50 = 3.7g/mL; control
8-(4'-Acetoxyangelyloxy)-2,3-dihydroxy-6H,7H-germacra-
Hydroxycamptothecin, HL-60, IC50 = 0.024g/mL; Bel7402, IC50 =
1(10)E,4E,11(13)-triene-6,12-olide C22H28O8 (420.46). White powder, []D20
0.62g/mL). Source: HUA ZE LAN Eupatorium chinense (whole herb: yield
= +40.8 (c = 0.55, CH3OH). Source: HUA ZE LAN Eupatorium chinense
= 0.0027%). Ref: 4739.
Cl
O
HO
OH
HO
O
O
O
O
OH
O
O
O
O
325
7550 Eupachlorin
7554 Eupacunolin
[20071-50-5] C20H25NO7 (412.87). Colorless lamellar crystals (methanol), mp
[79491-59-1] C22H28O8 (420.46). Colorless acicular crystals
219~221C (dec), []D27 = 110 (c = 0.35, ethanol). Pharm: Antineoplastic;
(methanolchloroform), mp 164~165C, [] D26 = +46 (c = 1.02, acetone).
cytotoxic (KB, ED50 = 0.21g/mL). Source: YUAN YE ZE LAN Eupatorium
Pharm: Antineoplastic; cytotoxic (KB, ED50 = 3.7g/mL). Source: XIE YE ZE
rotundifolium. Ref: 661.
LAN Eupatorium cuneifolium. Ref: 661.
OH
Cl
H
HO
OH O
O
O
O
HO
HO
7555 Eupacunoxin
[33853-88-2] C22H28O8 (420.46). Colorless acicular crystals (ether), mp

7551 Eupachlorin acetate
171~172C, []D26 = +27 (c = 1.0, acetone). Pharm: Antineoplastic; cytotoxic
[20501-52-4] C22H27ClO8 (454.91). Colorless acicular crystals (benzene), mp
(KB, ED50 = 2.1g/mL). Source: XIE YE ZE LAN Eupatorium cuneifolium.
161~164C (vacuum, dec), []D26 = 192 (c = 0.63, methanol). Pharm:
Ref: 661.
Antineoplastic (rat W256); cytotoxic (KB, ED50 = 0.18g/mL). Source: YUAN
HO
YE ZE LAN Eupatorium rotundifolium. Ref: 661.
O
O
Cl
OH
7556 Eupafolin
5,7,3',4'-Tetrahydroxy-6-methoxyflavone; 6-Methoxyluteolin [520-11-6]
HO
C16H12O7 (316.27). Yellow acicular crystals, mp 257~259C. Pharm:
Cytotoxic (KB, ED50 = 18g/mL). Source: JIN JI ZE LAN Eupatorium
subhastatum, LI ZHI CAO Salvia plebeia, MAO LIAN HAO Artemisia

vestita, MI DIE XIANG Rosmarinus officinalis, PENG LAI CAO Lippia
7552 Eupachloroxin
nodiflora, XIE YE ZE LAN Eupatorium cuneifolium, YIN DU JIA JING JIE
[20071-52-7] C20H25ClO8 (428.87). Amorphouspowder. Pharm:
Nepeta hindostana. Ref: 5, 474, 658.
Antineoplastic; cytotoxic (KB, ED50 = 0.21g/mL). Source: YUAN YE ZE
OH
OH
HO
HO
Cl
OH O
O
OH
7557 Eupafolin-7-glucoside
HO
Nepitrin; 6-Methoxyluteolin-7-glucoside C22H22O12 (478.41). mp 252~256C
(dec). Pharm: Antioxidant (DPPH free radical scavenger, DPPH radical
15mol/L: 10mol/L, ScRt = 38.1%; control BHA, 10mol/L, ScRt = 23.0%;

Vitamin E, 10mol/L, ScRt = 41.1%)[3846]. Source: DA MA YE ZE LAN
Eupatorium cannabinum, JIA HUI SE JIU LI XIANG PO PO NA Veronica
7553 Eupacunin
[33854-15-8] C22H28O7 (404.46). Colorless acicular crystals (methanolether),
25
thymoides ssp. pseudocinerea[3846], LI ZHI CAO Salvia plebeia, MAO DI
mp 166~167C, []D = +55 (c = 1.24, acetone). Pharm: Antineoplastic (rat,
HUANG Digitalis purpurea, MAO HUA MAO DI HUANG Digitalis lanata,
P388, W256, in vivo); cytotoxic (KB, ED50 = 2.1g/mL). Source: XIE YE ZE
PENG LAI CAO Lippia nodiflora, XIANG RI KUI YE Helianthus annuus,
LAN Eupatorium cuneifolium, ZHEN YE ZE LAN Eupatorium lancifolium.
XUAN FU HUA Inula britannica, YANG SHI CAO Achillea millefolium. Ref:
Ref: 661.
6, 660, 1388, 3846.

OH
OH
HO
O
O
O
HO
OO
OH
OH
O
OH
OH
326
7558 Eupaformonin
7563 Eupaglehnin D
[55520-20-2] C17H22O5 (306.36). Colorless prismatic crystals, mp 216~218C.
C21H28O6 (376.45). Oil, []D20 = +19.7 (c = 0.39, CHCl3). Source: KU YE DAO
Pharm: Cytotoxic (hmn throat epicytoma cells, in vitro). Source: TAI WAN
ZE LAN Eupatorium sachalinense [Syn. Eupatorium glehni]. Ref: 4226.
ZE LAN Eupatorium formosanum. Ref: 661.
O
O
OH
OH
O
H
7564 Eupaglehnin E
7559 Eupaformosanin
C17H23ClO6 (358.82). Oil, []D24 = +63.8 (c = 0.5, EtOH). Source: KU YE DAO
[64439-43-6] C20H26O7 (378.43). Pharm: Antineoplastic; cytotoxic. Source:
TAI WAN ZE LAN Eupatorium formosanum. Ref: 658.
OH
O
HO
O
H
HO
OH
OH
Cl
7565 Eupaglehnin F
C19H25ClO7 (400.86). Oil, []D20 = +40.0 (c = 0.3, CHCl3). Source: KU YE DAO
7560 Eupaglehnin A
C21H29O6 (376.45). Oil, []D24 = +55.3 (c = 0.86, EtOH). Source: KU YE

O
DAO ZE LAN Eupatorium sachalinense [Syn. Eupatorium glehni]. Ref:

O
4226.
O
OH
Cl
7566 Eupahyssopin
OH
Eupassopin [57718-77-1] C20H26O7 (378.43). Colorless prismatic crystals
(chloroform), mp 125C, []D25 = 138.9 (c = 1.45, chloroform). Pharm:
7561 Eupaglehnin B
C22H28O7 (404.46). Oil, []D20 = +52.5 (c = 0.5, CHCl3). Source: KU YE
Antiarthritic (animal model); antineoplastic (rat, W256); anti-inflammatory

(animal model); cytotoxic (mus EAC cells, inhibits biosynthesis of DNA,
RNA, protein and cholesterol). Source: SHEN XIANG CAO YE ZE LAN
4226.
Eupatorium hyssopifolium. Ref: 661.

O
O
OH
HO
O
OH
O
O
7567 Eupalinilide A
8-(4'-Hydroxytigloyloxy)-14-chloro-4,10-dihydroxy-1H,5H,6H,7H-g
7562 Eupaglehnin C
C20H26O5 (346.43). Oil, []D = +48.0 (c = 1.5, CHCl3). Source: KU YE
uai-2,11(13)-dien-6,12-olide C20H25ClO7 (412.87). Colorless gum, []D20 =
34.3 (c = 0.47, CHCl3). Source: CHENG GAN SHENG MA Eupatorium
4226.
20
OH
Cl
OH
OH
O
O
O
HO
O
O
O
327
7568 Eupalinilide B
7572 Eupalinilide F
8-(4'-Hydroxytigloyloxy)-4-hydroxy-1H,5H,6H,7H-guai-2,10-(14),11
8-(4'-Hydroxytigloyloxy)-2,10,14-trihydroxy-1H,5H,6H,7H-guai-3,1
(13)-trien-6,12-olide C20H24O6 (360.41). Colorless gum, []D20 = 84.9 (c =
1(13)-dien-6,12-olide C20H26O8 (394.43). Colorless gum, []D20 = 38.0 (c =
0.67, CHCl3). Pharm: Cytotoxic (in vitro, P388, IC50 = 0.21g/mL; A549, IC50
1.3, CH3OH). Pharm: Cytotoxic inactive (in vitro, P388, A549; control
= 0.75g/mL; control Pseudolaric acid B, P388, IC50 = 0.32g/mL; A549, IC50
Pseudolaric acid B, P388, IC50 = 0.32g/mL; A549, IC50 = 0.86g/mL). Source:
= 0.86g/mL). Source: CHENG GAN SHENG MA Eupatorium lindleyanum
CHENG GAN SHENG MA Eupatorium lindleyanum (whole herb: yield =
(whole herb: yield = 0.00045%dw). Ref: 4762.
0.0034%dw). Ref: 4762.
OH
O
OH
OH
HO
OH
OH
O
O
H
O
O
O
7569 Eupalinilide C
8-(4'-Hydroxytigloyloxy)-2,14-epoxy-10-hydroxy-1H,5H,6H,7H-gua
7573 Eupalinilide G
i-3,11(13)-dien-6,12-olide C20H24O7 (376.41). White powder, []D20 = 7.0 (c
8-(4'-Hydroxytigloyloxy)-3,4:10,14-diepoxy-2-hydroxy-1H,5H,6H,
= 1.0, CHCl3). Pharm: Cytotoxic (in vitro, P388, IC50 = 1.2g/mL; A549, IC50
7H-guai-11(13)-en-6,12-olide C20H24O8 (392.41). Colorless gum, []D20 =
= 11g/mL; control Pseudolaric acid B, P388, IC50 = 0.32g/mL; A549, IC50 =
44.3 (c = 0.47, CHCl3). Source: CHENG GAN SHENG MA Eupatorium
0.86g/mL). Source: CHENG GAN SHENG MA Eupatorium lindleyanum

OH
OH
OH
O
O
HO
O
O
7570 Eupalinilide D
7574 Eupalinilide H
14-Chloro-2,8,-10-trihydroxy-1H,5H,6H,7H-guai-3,11(13)-dien-6,12
8-Tigloyloxy-14-chloro-3,4-epoxy-2,10-dihydroxy-1H,5H,6H,7H-g
-olide C15H19ClO5 (314.77). Colorless gum, []D20 = 59.4 (c = 0.8, CHCl3).
uai-11(13)-en-6,12-olide C20H25ClO7 (412.87). Colorless gum, []D20 = 45.0
Source: CHENG GAN SHENG MA Eupatorium lindleyanum (whole herb:
(c = 1.5, CHCl3). Source: CHENG GAN SHENG MA Eupatorium
yield = 0.00055%dw). Ref: 4762.
Cl
HO
OH
HO
Cl
OH
OH
H
O
O
O
O
O
7571 Eupalinilide E
7575 Eupalinilide I
8-Tigloyloxy-14-chloro-2,10-dihydroxy-1H,5H,6H,7H-guai-3,
8-(4'-Hydroxytigloyloxy)-3,4-epoxy-2,10,14-trihydroxy-1H,5H,6H,
11(13)-dien-6,12-olide C20H25ClO6 (396.87). White powder, []D20 = 56.2
7H-guai-11(13)-en-6,12-olide C20H26O9 (410.42). Colorless gum, []D20 =
(c = 1.0, CHCl3). Pharm: Cytotoxic (in vitro, P388, inactive; A549, IC50 =
43.4 (c = 1.0, CH3OH). Pharm: Cytotoxic inactive (in vitro, P388, A549;
0.028g/mL; control Pseudolaric acid B, P388, IC50 = 0.32g/mL; A549, IC50
control Pseudolaric acid B, P388, IC50 = 0.32g/mL; A549, IC50 = 0.86g/mL).
= 0.86g/mL). Source: CHENG GAN SHENG MA Eupatorium lindleyanum
Source: CHENG GAN SHENG MA Eupatorium lindleyanum (whole herb:
yield = 0.00086%dw). Ref: 4762.
Cl
HO
OH
HO
OH
OH
O
H
O
O
O
OH
O
O
O
O
328
7576 Eupalinilide J
7581 Eupaserrin
8-(4'-Hydroxytigloyloxy)-3,4-epoxy-2-acetoxy-10,14-dihydroxy-1H,5
[38456-36-9] C22H28O7 (404.46). Crystals (ethermethanol), mp 153~154C,
H,6H,7H-guai-11(13)-en-6,12-olide C22H28O10 (452.46). Colorless gum,
[]D25 = +71.2 (c = 0.94, methanol). Pharm: Antineoplastic (mus, P388,
[]D20 = 46.7 (c = 0.68, CHCl3). Source: CHENG GAN SHENG MA
30mg/kg); cytotoxic (KB, ED50 = 0.23g/mL). Source: BAN JU CHI
Eupatorium lindleyanum (whole herb: yield = 0.00055%dw). Ref: 4762.
ZHUANG ZE LAN Eupatorium semiserratum, HUA ZE LAN Eupatorium

chinense (whole herb: yield = 0.0014%)[4739], KU YE DAO ZE LAN
OH
OH
Eupatorium sachalinense [Syn. Eupatorium glehni], ROU MAO XIANG RI

KUI Helianthus mollis. Ref: 661, 4226, 4739.
OH
O
O
HO
O
O
7577 Eupalitin
6,7-Dimethoxy-3,5,4'-trihydroxyflavone [In DNP] C17H14O7 (330.30). Source:

O
CU YING MAO DIAN ZI CAO Onosma hispida (whole herb), YIN CHEN
HAO Artemisia capillaris. Ref: 2, 4490.
7582 Eupatilin
5,7-Dihydroxy-3',4',6-trimethoxyflavone [22368-21-4] C18H16O7 (344.32).
OH
O
Crystals (ethyl acetate), mp 234~236C. Pharm: Cytotoxic (KB, ED50 = 38 or

45g/mL). Source: BAN JU CHI ZHUANG ZE LAN Eupatorium
semiserratum, HONG ZU HAO Artemisia rubripes, JU PI Citrus reticulata,

O
OH
OH
YE JU HUA Chrysanthemum indicum. Ref: 661, 4214.
7578 Euparin
[532-48-9] C13H12O3 (216.24). mp 121~122C. Source: CHENG GAN
SHENG MA Eupatorium lindleyanum, PEI LAN Eupatorium fortunei, ZHAI

HO
TOU TUO WU Ligularia stenocephala (root). Ref: 6, 4536.

O
O
OH
HO
7583 Eupatin
3,5,3'-Trihydroxy-6,7,4'-trimethoxy flavone [19587-65-6] C18H16O8 (360.32).
7579 Euparotin
[10191-01-2] C20H24O7 (376.41). Acicular crystals (ethyl acetatepetroleum
Golden bar crystals (methanol), mp 243~245C. Pharm: Cytotoxic (KB, ED50
ether), mp 199~200C (vacuum), []D = 124 (c = 1.25, ethanol). Pharm:
= 4.6g/mL). Source: BAN JU CHI ZHUANG ZE LAN Eupatorium
Antineoplastic; cytotoxic (KB, ED50 = 0.21g/mL). Source: YUAN YE ZE
semiserratum, HUANG HUA HAO Artemisia annua. Ref: 2, 660, 661.
32

HO
OH
O
O
HO
O
OH
OH
7584 Eupatocunin
7580 Euparotin acetate

30
[10215-89-1] C22H26O8 (418.45). mp 156~157C (vacuum), []D = 191 (c
[33853-87-1] C22H28O7 (404.46). Colorless prismatic crystals
= 0.54, ethanol). Pharm: Antineoplastic; cytotoxic (KB, ED50 = 0.21g/mL).
(methanolether), mp 163~164C, [] D26 = 129 (c = 1.36, acetone). Pharm:
Source: YUAN YE ZE LAN Eupatorium rotundifolium. Ref: 661.
Antineoplastic; cytotoxic (KB, ED50 = 0.11g/mL). Source: XIE YE ZE LAN

Eupatorium cuneifolium. Ref: 661.
O
O
O
OH
O
HO
O
H
O
O
O
O
H
329
7585 Eupatocunoxin
7590 Eupatoretin
[39204-36-9] C22H28O8 (420.46). Acicular crystals (acetone), mp 200~201C,
3,3'-Dihydroxy-4',5,6,7-tetramethoxyflavone [19587-69-0] C19H18O8
[]D26 = 209 (c = 1, acetone). Pharm: Antineoplastic; cytotoxic (KB, ED50 =
(374.35). Yellowish acicular crystals (benzene), mp 146~148C. Pharm:
1.7g/mL). Source: XIE YE ZE LAN Eupatorium cuneifolium. Ref: 661.
Cytotoxic (KB). Source: BAN JU CHI ZHUANG ZE LAN Eupatorium
OH
semiserratum. Ref: 661.
OH
O
O
O
7586 Eupatolide
OH
O
[6750-25-0] C15H20O3 (248.32). Crystals (chloroform), mp 188~190C. Pharm:
Antineoplastic; anti-inflammatory; cytotoxic (HEP2, ED 50 = 0.469g/mL,
7591 Eupatorin
W-18Va-2, ED50 = 0.034g/mL, KB, HeLa, normal Rk and EAC-E4 cells).
3',5-Dihydroxy-4',6,7-trimethoxyflavone [855-96-9] C18H16O7 (344.32).
Source: KU YE DAO ZE LAN Eupatorium sachalinense [Syn. Eupatorium
Crystals (dioxanewater), mp 196~198C. Pharm: Antioxidant (ferric
glehni], TAI WAN ZE LAN Eupatorium formosanum. Ref: 661, 4226.
thiocyanate method, 0.5mmol/L, peroxidation value = 11.7%, control BHA,

0.5mmol/L, peroxidation value = 4.5%, control Vitamin E, 0.5mmol/L,
peroxidation value = 14.7%)[4508]. Source: BAN JU CHI ZHUANG ZE LAN
H
H
Eupatorium semiserratum, GAO ZE LAN Eupatorium altissimum, TIAN
OH
SHE CAO Lippia dulcis (aerial parts), XIONG RUI ZHUANG ZHI GUAN
O
CAO Orthosiphon stamineus [Syn. Orthosiphon aristatus; Orthosiphon

grandiflorus; Orthosiphon spicatus] (aerial parts: yield = 0.00028%dw)[3053].
Ref: 661, 3053, 4508.
7587 Eupatolin
[29725-50-6] C23H24O12 (492.44). mp 200~201C. Source: PEI LAN
OH
Eupatorium fortunei. Ref: 6.
O
O
OH
HO
O
OH
OO
O
O
OH
OH
7592 Eupatoriochromene
6-Acetyl-7-hydroxy-2,2-dimethyl-2H-1-benzopyran [19013-03-7] C13H14O3
(218.25). Pharm: Phototoxic (yeast and bacteria). Source: HE AN ZE LAN
OH OH
Eupatorium riparium. Ref: 658.
7588 Eupatolitin
3,5,3',4'-Tetrahydroxy-6,7-dimethoxyflavone [29536-44-5] C17H14O8 (346.30).
Source: HUANG HUA HAO Artemisia annua, YIN CHEN HAO Artemisia
capillaris. Ref: 2, 660.
O
HO
OH
O
OH
OH
OH
7593 Eupatoriopicrin
[6856-01-5] C20H26O7 (378.43). mp 157~161C (dilute ethanol), [] D20 =
+95 (chloroform). Pharm: Antineoplastic; cytotoxic (KB, HeLa, normal Rk
cells and EAC-E4 cells). Source: PEI LAN Eupatorium fortunei, DA MA YE
ZE LAN Eupatorium cannabinum, KU YE DAO ZE LAN Eupatorium
7589 Eupatoranolide
sachalinense [Syn. Eupatorium glehni]. Ref: 6, 661, 4226.
C17H22O4 (290.36). Colorless crystals, mp 182~184C. Source: ZI JING ZE

LAN HUA Eupatorium adenophorum. Ref: 882.
OH
O
O
O
H
O
O
HO
OH
O
O
330
7594 Eupatoroxin
7598 Euphocharacin C
[20071-51-6] C20H24O8 (392.41). mp 197~200C, []D26 = 98 (c = 1.10,
methanol). Pharm: Antineoplastic; cytotoxic (KB, ED50 = 2.8g/mL). Source:
CHCl3). Pharm: Cancer cell P-Glycoprotein inhibitor (cellular
YUAN YE ZE LAN Eupatorium rotundifolium. Ref: 661.
P-glycoprotein-mediated daunomycin efflux, InRt = (1232)%, relative

standard Cyclosporin A(CsA) InRt = 100%). Source: DI ZHONG HAI DA JI
HO
Euphorbia characias (whole herb). Ref: 5003.
O
HO
OH
HO
H
O
7595 Eupatundin
O
O
O
[20071-53-8] C20H24O7 (376.41). mp 188~189C (vacuum), []D29 = 80 (c =

0.44, ethanol). Pharm: Antineoplastic; cytotoxic (KB, ED50 = 0.39g/mL).
7599 Euphocharacin D
Source: YUAN YE ZE LAN Eupatorium rotundifolium. Ref: 661.
C37H49NO12 (699.80). Colorless amorphous solid, []D25 = +8.0 (c = 0.1,

HO

H
HO
O
O
HO
O
O
7596 Euphocharacin A
O H
O
C39H45NO12 (719.79). Colorless amorphous solid, []D25 = 22.17 (c = 0.1,
O
O
7600 Euphocharacin E

O
HO

O
O
O H
O
O
O
N
OH
O
O
O
O
H
O
O
O
O
7597 Euphocharacin B
C37H43NO11 (677.76). Colorless amorphous solid, []D25 = +117.69 (c = 0.1,
7601 Euphocharacin F

N
HO
O
O H
O
O
O
O
O
O
N
O
O
O
OH
O H
O
O
O
O
331
7602 Euphocharacin G
C34H45NO10 (627.74). White amorphous solid, []D25 = 25.0 (c = 0.1,
N
O

O
O H
O
O
O
O
N
OH
7606 Euphocharacin K
O
O
O
O H
O

O
O
7603 Euphocharacin H
N
O

O
O H
HO
O
O
7607 Euphocharacin L
O
O
O
O H
O

O
O
7604 Euphocharacin I
25
C35H45NO11 (655.75). Colorless amorphous solid, []D = 22.0 (c = 0.1,
HO
N
O
O
O

O H
HO
O
O
N
O
7608 Euphoheliosnoid A
O
O
O
O H
O
C37H43NO9 (645.76). Colorless oil, []D20 = +19 (c = 1.36, CHCl3). Source:

ZE QI Euphorbia helioscopia (whole herb). Ref: 5076.
O
O
O
O
O
7605 Euphocharacin J

O
O
O
N
O
O
H
O
O
332
7609 Euphoheliosnoid B
7613 Euphopubescene
C37H43NO9 (645.76). Colorless oil, []D20 = +25 (c = 1.00, CHCl3). Source:
3,7,8,9,14,15-Hexaacetoxy-2H-jatropha-5E,11E-diene C32H46O12
ZE QI Euphorbia helioscopia (whole herb). Ref: 5076.
(622.72). White amorphous powder, []D25 = 139 (c = 0.14, CHCl3). Pharm:

Cytotoxic (in vitro MCF7 cell lines, GI50 = (72.05.8)mol/L, Doxorubicin,
Doxorubicin, GI50 = (93.07.0)mol/L). Source: DUAN ROU MAO DA JI

Euphorbia pubescens (whole herb). Ref: 4949.
O
O
Doxorubicin, GI50 = (94.08.7)mol/L; SF268 cell lines, GI50 > 100mol/L,
O
O
H
GI50 = (42.88.2)mol/L; NCI-H460 cell lines, GI50 = (40.90.8)mol/L,
O
O
O
O
O
O
7610 Euphoheliosnoid C
C33H42O10 (598.70). Colorless oil, []D20 = +33 (c = 0.58, CHCl3). Source: ZE
O
O
QI Euphorbia helioscopia (whole herb). Ref: 5076.
O
O
7614 Euphopubescenol
5,8,15-Triacetoxy-3-benzoyloxy-4-hydroxy-9,14-dioxo-13H-jatropha-
O
O
6(17),11E-diene C33H40O11 (612.68). White amorphous powder, []D25 = +29
O
O
H
OH
(c = 0.12, CHCl3). Pharm: Cytotoxic (in vitro MCF7, GI50 = (68.63.2)mol/L,

Doxorubicin, GI50 = (42.88.2)mol/L; NCI-H460, GI50 = 75mol/L,
Doxorubicin, GI50 = (94.08.7)mol/L; SF268, GI50 > 100mol/L,

O
Doxorubicin, GI50 = (93.07.0)mol/L). Source: DUAN ROU MAO DA JI

Euphorbia pubescens (whole herb). Ref: 4949.
O
O
7611 Euphol
Euphadienol; Eupha-8,24-dien-3-ol [514-47-6] C30H50O (426.73). mp 116C.
Pharm: Antihypertensive (anesthetic dog, iv, 0.31~10mg/kg, blood pressure is
lowered by 20~30mmHg to 50~93mmHg for 0.75-4.5 hours, ED50 (iv) =
HO
O
O
2.18mg/Kg); cytotoxic (P388, ED50 = 2.4g/mL); antineoplastic (EBV-EA
induced by TPA, mol ratio/TPA = 1000, relative percentage of EBV-EA = 0%

(positive control value 32pmol, 20ng TPA = 100%), viability of Raji cells =
7615 Euphorbetin
70%; reference compound -Carotene, relative percentage = 8.6%)[4606].
[35897-99-5] C18H10O8 (354.28). Source: QIAN JIN ZI Euphorbia lathyris.
Source: BA WANG BIAN Euphorbia royleana, GAN SUI Euphorbia kansui,
Ref: 6.
HUO YANG LE Euphorbia antiquorum (latex: yield = 0.38%fw)[4606], XI YE

DA JI Euphorbia esula var. cyparissoides. Ref: 6, 1812, 1813, 4606.
HO
HO
OH
OH
O
HO
7616 Euphorbia factor Ti2

7612 -Euphol
C32H42O7 (538.69). Pharm: Irritant. Source: LU YU SHU Euphorbia tirucalli.
C30H50O (426.73). Source: GAN SUI Euphorbia kansui (dried root). Ref:
Ref: 658.
4690.
O
O
OH
HO
H
OH
333
7617 Euphorbiasteroid
7622 Eupteleasaponin I
5,10-Diacetyl-6,20-epoxy-3-phenyl-acetyllathyrol C32H40O8 (552.67). mp
C52H82O21 (1043.22). Source: DUO XIONG RUI LING CHUN MU Euptelea
199.5C. Pharm: Laxative. Source: QIAN JIN ZI Euphorbia lathyris, XUE
polyandra (fresh leaf). Ref: 3537.
TONG Macaranga tanarius. Ref: 6, 661, 5501.

O
O
HO
7618 Euphorbol
127~128C,
1.0 (c = 0.20). Pharm: Antineoplastic (EBV-EA
induced by TPA, mol ratio/TPA = 1000, relative percentage of EBV-EA = 0%
OH
OH
OH
OH
OH
OH O O
OH
O
OH
-Euphorbol [566-14-3] C31H52O (440.76). Needles, mp 123~126C, mp

[]D25 =
HO
OO
(positive control value 32pmol, 20ng TPA =100%), viability of Raji cells =
70%; reference compound -Carotene, relative percentage = 8.6%). Source:
OH OH
BA WANG BIAN Euphorbia royleana, GAN SUI Euphorbia kansui, HUO

YANG LE Euphorbia antiquorum (latex). Ref: 6, 4606.
H
7623 Eupteleasaponin II
HO
H
O
7619 Euphoscopin B
C33H42O9 (598.706). Source: ZE QI Euphorbia helioscopia (whole herb). Ref: 5076.
O
O
H
O
HO
O
O
OH
OO
OH
O
OH
OH
OH
OH
OH
OH
OO
HO
OO
OO
OH OH
OH OH
7620 Euphoscopin C
C38H44O9 (644.77). Source: ZE QI Euphorbia helioscopia (whole herb). Ref: 5076.
H
O
O
H
7624 Eupteleasaponin III

O
O
7621 Euponin
OO
[70469-59-9] C20H24O6 (360.41). Pharm: Larvacide (insect larva growth

HO
inhibitor). Source: CHENG GAN CAO Eupatorium japonicum. Ref: 658.

HO
OH O O
O
O
O
H
OO
OH
O
OH
OH OH
OH
O
OH
OH
OH OH
O
O
OH
OH
OH
OO
HO
OH
334
7625 Eupteleasaponin IV
7628 Eupteleasaponin VI
Eupteleogenin 3-O--L-rhamnopyranosyl(12)-[-D-glucopyranosyl(13)]-
-D-glucopyranoside C47H72O18 (925.09). Colorless fine crystals (CHCl3MeOH),

mp 184~187C, []D25 = +46.8 (c = 0.1, MeOH). Source: DUO XIONG RUI
LING CHUN MU Euptelea polyandra (fresh leaf). Ref: 3537.
O
O
OH
OO
HO
OH
OH
OO
OO
OH
OH OH
HO
OH
OH
OH
HO
OH
OO
OH
OH
OO
O
OH
OH
OH
OO
OH OH
OH OH
7629 Eupteleasaponin VI acetate
7626 Eupteleasaponin V
Eupteleogenin 3-O-[-L-rhamnopyranosyl(12)][-D-glucopyranosyl
(13)]-6'-O-acetyl--D-glucopyranoside C49H74O19 (967.12). Colorless fine
crystals (CHCl3MeOH), mp 180~184C, []D26 = +31.9 (c = 0.1, MeOH).
Source: DUO XIONG RUI LING CHUN MU Euptelea polyandra (fresh leaf).
Ref: 3537.
O
OH
OH
OH
OH OO
OO
HO
HO
OH
O
OH
OH
OO
O
OH
OH
OO
OH
OH OH
OH OH
7630 Eupteleasaponin VII

7627 Eupteleasaponin V acetate
Eupteleogenin 3-O-[-L-rhamnopyranosyl(12)][-D-galactopyranosyl
(13)][-L-rhamnopyranosyl(14)]--D-glucopyranoside C53H82O22
(1071.23). Colorless fine crystals (CHCl3MeOH), mp 168~172C, []D26 =

+14.6 (c = 0.1, MeOH). Source: DUO XIONG RUI LING CHUN MU
Euptelea polyandra (fresh leaf). Ref: 3537.
O
OO
O
O
OH
OH
OH
OO
O
OH
HO
OH
OH
HO
OO
O O
OH
OO
OH
OH OH
OO
OH OH
OH OH
OH OH
335
7631 Eupteleasaponin VIII
7634 Eupteleasaponin XI
3,20,24-Trihydroxy-29-norolean-12-en-28-oic acid 24-O--D-glucopyra-
Oleanolic acid 3-O-{-L-rhamnopyranosyl(12)-[-L-rhamnopyranosyl
noside C35H56O10 (636.83). Colorless fine crystals (CHCl3MeOH), mp
(14)]--D-glucopyranosyl(13)}--D-xylopyranoside C53H86O20 (1043.26).
199~201C, []D26 = +73.9 (c = 0.1, MeOH). Source: DUO XIONG RUI
Colorless fine crystals (CHCl3MeOH), mp 241~245C, []D26 = +116 (c =
LING CHUN MU Euptelea polyandra (fresh leaf). Ref: 3537.
0.1, MeOH). Source: DUO XIONG RUI LING CHUN MU Euptelea

OH
OH
O
OO
HO
OH
OO
OH
O
OH
OO
OH
OH
OH
HO
HO
OH
OH
OO
OH
OH OH
7632 Eupteleasaponin IX
OH OH
3,20,24-Trihydroxy-29-norolean-12-en-28-oic acid
7635 Eupteleasaponin XII
24-O-[-L-rhamnopyranosyl(14)]-6'-O-acetyl--D-glucopyranoside
8-O--D-Glucopyranosylakebonoic acid 3-O--L-arabinopyranosyl(13)-
C43H68O15 (825.01). Colorless fine crystals (CHCl3MeOH), mp 221~225C,
[-L-rhamnopyranosyl(14)]--D-glucopyranoside C52H82O21 (1043.22).
[]D26 = +34.9 (c = 0.1, MeOH). Source: DUO XIONG RUI LING CHUN
MU Euptelea polyandra (fresh leaf). Ref: 3537.
OH
H
HO
OH
OH
OH
OH
OH
OO
0.1, MeOH). Source: DUO XIONG RUI LING CHUN MU Euptelea

OH
Colorless fine crystals (CHCl3MeOH), mp 175~177C, []D25 = +33.9 (c =
OH
OH
OH
OH
HO OHO O
OO
HO
OO
OH
OH OH
OH OH
7636 Europine
7633 Eupteleasaponin X
[570-19-4] C16H27NO6 (329.40). Pharm: Anticholinergic (rat); hepatotoxin.
Serratagenic acid 3-O--L-rhamnopyranosyl(14)--D-glucopyranoside
Source: OU ZHOU TIAN JIE CAI Heliotropium europaeum, YUAN YE
C42H66O14 (794.99). Colorless fine crystals (CHCl3MeOH), mp 237~239C,
TIAN JIE CAI Heliotropium rotundifolium. Ref: 658.
[]D26 = +12.1 (c = 0.1, MeOH). Source: DUO XIONG RUI LING CHUN
OH
HO
MU Euptelea polyandra (fresh leaf). Ref: 3537.

O
HO
H
O
OH
7637 Eurycarpin A
H
H
OO
HO
OH
OH
O
OH
7,2',4'-Trihydroxy-(3,3-dimethylally)isoflavone [166547-20-2] C20H18O5

(338.36). Powder (methanol), mp 85~87C. Source: HUANG GAN CAO
Glycyrrhiza kansuensis. Ref: 379.
H
HO
OO
OH
OH
OH OH
OH
336
7638 Eurycolactone
7644 Eurycolactone F

O
HO
OH
OH
HO
OH
HO
HO
O
O
OH
O
O
7645 Eurycolactone G
7639 Eurycolactone A
HO
OH
HO
O
HO
OH
OH
7646 Eurycomalactone
O
O
C19H24O6 (348.40). Pharm: Cytotoxic (A549 cancer cells, remarkable activity;

MCF7 cancer cells, IC 50 < 2.5g/mL); antileishmanial (IC50 = 0.21g/mL,
7640 Eurycolactone B
C18H19ClO5 (350.38). Source: Eurycoma sp. Ref: 4556.
control Thallioquin, IC50 = 0.21g/mL). Source: Eurycoma sp. Ref: 4556.

O
HO
OH
HO
O
Cl
O
O
7647 Eurycomalide A
7641 Eurycolactone C
HO
OH
HO
O
HO
H
O
7648 Eurycomalide B
7642 Eurycolactone D
HO
HO
HO
OH
H
7649 Eurycomalin A
7643 Eurycolactone E
OH
HO
OH
O
O
HO
O
HO
337
7650 Eurycomanol
7656 Euryopsin-3-one
C20H26O9 (410.42). Pharm: Cytotoxic (KB cells, IC50 = 3.6g/mL)[4556];
C15H18O2 (230.31). Colorless oil. Source: HUANG SE QIAN LI GUANG
antileishmanial (IC50 = 0.28g/mL, control Thallioquin, IC50 = 0.21g/mL).
Senecio flavus. Ref: 2409.
Source: Eurycoma sp. Ref: 4556.

O
OH
HO
OH
OH
OH
HO
O
7657 Euscaphic acid
2,3,19-Trihydroxyurs-12-en-28-oic acid [53155-25-2] C30H48O5 (488.71).

7651 Eurycomanol-2-O--glucopyranoside
C26H36O14 (572.57). Pharm: Antileishmanial (thallioquin-resistance
Leishmania sp., IC50 = 0.389~3.498mol/L, control Thallioquin, IC50 =
0.323~0.774mol/L). Source: Eurycoma sp. Ref: 4556.
OH
HO
OH
OH
OH
OH
involving T lymphocytes, B lymphocytes, and macrophages isolated from

peripheral blood, IC50 = 28.8mol/L; control Cyclosporine A, IC50 =
0.012mol/L)[3064]; cytotoxic inactive (HSC-2, IC50 > 200g/mL; HGF, IC50 >
laevigata, JUAN MAO QIANG WEI Rosa sericea, PI PA HE Eriobotrya
japonica, SAN YE SHU WEI CAO Salvia trijuga, TAI WAN PI PA
Eriobotrya deflexa (leaf)[3064], TUN XING GUO Pygeum topengii. Ref: 447,
OH
Pharm: Immunosuppressant (hmn mononuclear cells antiproliferation,
200g/mL)[5160]. Source: DI YU Sanguisorba officinalis, JIN YING ZI Rosa
OO
HO
Colorless powder crystals, mp 269~271C, []D18 = 22.4 (c = 0.05, pyridine).
570, 592, 643, 3064, 5160.
OH
7652 Eurycomaoside
C25H38O12 (530.57). []D25 = 10.9 (c = 0.5, MeOH). Source: CHANG YE
HO
KUAN MU Eurycoma longifolia (root). Ref: 4400.
HO
HO
OH
O
H
OH
HO
O
OH
7658 Euscaphic acid 2,3-monoacetonide
H
OH OH
C33H52O5 (528.78). White acicular crystals, mp 188~190C acetone-petroleum

ether). Source: JUAN MAO QIANG WEI Rosa sericea. Ref: 676.
7653 Eurylactone A
HO
OH
O
OH
7659 Euscapholide
7-Hydroxy-2-octen-5-olide C8H12O3 (156.18). Pharm: Anti-inflammatory
7654 Eurylactone B
(remarkably inhibits inflammation induced by k-carrageenan)[4546]. Source:

YE YA CHUN Euscaphis japonica (twig and leaf). Ref: 4546.
OH
O
HO
OH
OH
OH
H
O
11-Deacetyleurylene IC50 = 0.33g/mL). Source: Eurycoma sp. Ref: 4556.
238~242C (sublimation). Source: BIAN SE HE KE BAO Emericella

variecolor. Ref: 3386.
OH
OH
O
OO
O
1,2,3-Trihydroxy-6-methyl-8-methoxyanthraquinone C16H12O6 (300.27). mp
C34H58O8 (594.84). Pharm: Cytotoxic (KB cells, gtdrolysis product
7660 Evariquinone
7655 Eurylene
OH
H
O
H
O
OH
OH
OH
OH
HO
OH
HO
HO
O
338
7661 Evernic acid
level, and the effects of evodiamine were completely abolished by
[537-09-7] C17H16O7 (332.31). mp 169.6~170.1C. Source: XIAO LA BA
capsazepine (5.0mg/kg, sc), a competitive vanilloid receptor antagonist.
Cladonia verticillata. Ref: 6.
These results suggest that evodiamine exerts a protection against myocardial

ischemia-reperfusion injury in rats and that the protective effects of
O
O
O
OH
OH
O
OH
evodiamine are related to stimulation of CGRP release via activation of

vanilloid receptors)[4088]. Source: BO SHI WU ZHU YU Evodia rutaecarpa
var. bodinieri (dried and almost ripe fruit: content scope of 4 origins =
0.117%~1.229%, mean content = 0.544%)[5508], HUA NAN WU ZHU YU
7662 Everninic acid methyl ester 2-O--xylopyranosyl-(16)--
Evodia austrosinensis (dried and almost ripe fruit: content = 0.12%)

(3)
[5508]
, SHI
Evodia rutaecarpa var. officinalis (dried and almost ripe fruit: content
glucopyranoside
HU
scope of 14 origins = 0.093%~1.242%, mean content = 0.503%)[5508], WU
Source: NAO YANG HUA Rhododendron molle. Ref: 5396.
ZHU YU Evodia rutaecarpa (dried and almost ripe fruit: content scope of 14
origins = 0.203%~3.221%, mean content = 1.200%[5508]), YI HUA WU ZHU
O
O
OO
OO
OH
OH
0.114%~0.152%, mean content = 0.133%)[5508]. Ref: 2, 6, 347, 661, 1643,

4088, 5394, 5501, 5508.
OH
OH
OH
YU Evodia baberi (dried and almost ripe fruit: content scope of 2 origins =
OH
7663 Evocarpine
N
H H
[15266-38-3] C23H33NO (339.53). Note: evocarpine is a mixture, and the
N
N
following structure is its main component. Pharm: DGAT inhibitor (IC50 =

8.1g/mL)[4943]; leukotriene biosynthesis inhibitor (hmn polymorphonuclear
granulocytes, IC50 = 14.6mol/L, zileuton, IC50 = 10.4mol/L)[5031]. Source:
7666 Evodianinine
WU ZHU YU Evodia rutaecarpa (fruit). Ref: 2, 4943, 5031.
C19H13NO3 (299.33). Pale yellow crystals, mp 185~187C (CHCl3), []D23 =

0 (c = 0.5, CHCl3). Source: WU ZHU YU Evodia rutaecarpa (fruit). Ref:
4848.
7664 Evodiamide
C19H21N3O (307.40). Source: WU ZHU YU Evodia rutaecarpa. Ref: 2, 347,

877.
7667 Evodiaxinine
N
H
C20H15N3O (313.36). Yellow needles, mp 175~176C, []D23 = 0 (c = 0.5,
N
O
HN
CHCl3). Source: WU ZHU YU Evodia rutaecarpa (fruit). Ref: 4914.
7665 Evodiamine
8,13,13b,14-Tetrahydro-14-methylindolo[2',3':3,4]pyrido[2,1b]quinazolin-5(7
H)-one [518-17-2] C19H17N3O (303.37). Yellow lamellar crystals (ethanol),
mp 278C. []D15 = +352 (acetone), mp (+) 270~272C. Pharm: Analgesic

(has both stimulatory and desensitizing effects on sensory nerves, as
capsaicin does)[5394]; diuretic; raises body temperature; induces sweatiness;
7668 Evodinone
cytotoxic (induces apoptosis of HeLa cell); CGRP stimulator (Calcitonin
Rutaevin [33237-37-5] C26H30O9 (486.52). mp 295~297C (dec). Source: WU
gene-related peptide,CGRP, protects the myocardium against
ZHU YU Evodia rutaecarpa. Ref: 2, 6.
ischemia-reperfusion injury)[4088]; a detail study on protective effects of

evodiamine on myocardial ischemia-reperfusion injury in rats (Rats were
pretreated with evodiamine 10min before the experiment, and then the left
main coronary artery of rat hearts was subjected to 60min occlusion followed
O
O
by 180min reperfusion. Infarct size, the activity of serum creatine kinase,
serum concentrations of TNF- and plasma concentrations of CGRP were

measured. Pretreatment with evodiamine (30 or 60g/kg, iv) markedly
increased the content of CGRP in plasma concomitantly with a significant
reduction in infarct size, the activity of serum creatine kinase, and TNF-
O
OH
339
7669 Evodol
7674 Excisanin A
Limonindiosphenol [22318-10-1] C26H28O9 (484.51). mp 280~281C. Source:
1,7,12,14-Tetrahydroxy-ent-kaur-16-en-15-one C20H30O5 (350.46). mp
BAI XIAN PI Dictamnus dasycarpus, WU ZHU YU Evodia rutaecarpa. Ref:
262~264C, []D20 = 27.7 (c = 1.01, C5H5N). Pharm: Cytotoxic (in vitro,
2, 660, 1521.
P388, ED50 = 1.11g/mL)[3012]. Source: WEI YE XIANG CHA CAI Rabdosia

excisa (aerial parts: yield = 0.0069%dw). Ref: 3012, 4067.
O
O
OH
O
O
OH
OH
O
OH
O
H
OH
7670 Evofolin B
[168254-96-4] C17H18O6 (318.33). Yellow oil, []D26 = +16.7 (c = 0.30,
CH3OH). Pharm: Cytotoxic (quinone reductase induction assay in cultured
Hepa1c1c7 mouse hepatoma cells)[5038]. Source: HAI NAN JIAN MU
Dysoxylum hainanense, Couepia ulei. Ref: 2140, 5038.
HO
7675 Excisanin B
1,7,14-Trihydroxy-12-acetoxy-ent-kaur-16-en-15-one C22H32O6 (392.50).
mp 240~243C, []D20 = 13.9 (c = 1.00, C5H5N). Pharm: Cytotoxic (in vitro,
P388, ED50 = 0.63g/mL)[3012]. Source: WEI YE XIANG CHA CAI Rabdosia
excisa (aerial parts: yield = 0.0013%dw). Ref: 3012, 4067.
O
O
O
OH
OH
OH
O
H
OH
7671 Evonine
C36H43NO17 (761.74). mp 149~153C. Source: GUI JIAN YU Euonymus
alatus (the compound was isolated from the plant by H.Wada, et al. in 1971).
Ref: 5505.
7676 Excisanin C
C20H30O4 (334.46). []D21 = 112.7 (c = 0.15, MeOH). Source: WEI YE
O
O
XIANG CHA CAI Rabdosia excisa. Ref: 4067.
O
O
O
HO
OH O
OH
O
O
O
OH
O
OH
7677 Excisanin D
O
N
C22H32O6 (392.50). mp 140~142C, []D = 56 (c = 0.42, MeOH). Pharm:

Cytotoxic (in vitro, P388, IC50 = 0.72g/mL)[3012]. Source: WEI YE XIANG
7672 Exaltolide
Oxacyclohexadecan-2-one [106-02-5] C15H28O2 (240.39). Source: BAI ZHI
Angelica dahurica [Syn. Angelica porphyrocaulis]. Ref: 2.
CHA CAI Rabdosia excisa (aerial parts: yield = 0.0001%dw). Ref: 3012,
4067.
OH
O
H
O
O
7673 Excelsine
9-Hydroxy-monticamine [41645-62-9] C22H33NO6 (407.51). Colorless
quadratus crystals, mp 87~89C (acetone); 103~105C. Source: JI LIN WU
TOU Aconitum kirinense, ZI HUA GAO WU TOU Aconitum excelsum. Ref:
7678 Excisanin E
C22H32O7 (408.50). Yellow powder, []D = 46.1 (c = 0.64, MeOH). Source:
WEI YE XIANG CHA CAI Rabdosia excisa. Ref: 4067.
1521, 2515.
H
OH
N
O
OH
O
H
OH
O
OH
OH
OH
O
OH
H
O
OH
O
OH
340
7679 Excisanin F
7684 Excisanin K
C20H28O6 (364.44). []D20 = +27.3 (c = 0.55, MeOH). Source: WEI YE
1,7,14,18-Tetrahydroxy-ent-kaur-16-en-15-one C20H30O5 (350.46).
XIANG CHA CAI Rabdosia excisa. Ref: 4067.
Colorless powder (MeOH), mp 128~129C, []D = 109.2 (c = 0.23, MeOH).

Pharm: Cytotoxic (in vitro, P388, ED50 = 0.92g/mL). Source: WEI YE
XIANG CHA CAI Rabdosia excisa (aerial parts: yield = 0.00013%dw). Ref:
OH
OH
3012.
OH
H
O
OH
O
OH
OH
O
H
HO
7680 Excisanin G
Source: WEI YE XIANG CHA CAI Rabdosia excisa. Ref: 4067.
OH
C20H32O6 (368.47). mp 214~216C, []D20 = 100.8 (c = 0.51, MeOH).
7685 Excoecarin R1
C40H64O11 (720.95). Source: HAI QI Excoecaria agallocha (resinous resinous
OH
wood: yield = 0.0019%). Ref: 4674.
OH
OH
OH
H
H
HO
O
OH
H
O
HO
7681 Excisanin H
14,20-Epoxy-1,7,14-trihydroxy-ent-kaur-16-en-15-one C20H28O5
(348.44). Colorless powder (MeOH), mp 206~207C, []D = 87.9 (c = 0.07,
O
OH
HO
MeOH). Pharm: Cytotoxic (in vitro, P388, ED50 = 0.96g/mL). Source: WEI
YE XIANG CHA CAI Rabdosia excisa (aerial parts: yield = 0.00007%dw).
Ref: 3012.
7686 Excoecarin R2
C40H64O11 (720.95). Source: HAI QI Excoecaria agallocha (resinous wood:
yield = 0.0015%). Ref: 4674.
OH
O
OH
OH
OH
HO
H
O
7682 Excisanin I
O
O
HO
HO

7687 Excoecarin S
C20H32O6 (368.47). Colorless needles (MeOH), mp 254~256C, []D26 =
3012.
47.2 (c = 0.9, MeOH). Source: HAI QI Excoecaria agallocha (resinous

wood). Ref: 3461.
OH
OH
HO
HO
OH
O
OH
H
H
O
O
O
HO
H
H
7683 Excisanin J
7688 Excoecarin T1
C20H32O6 (368.47). As dimethyl ester: colorless needles (aqueous MeOH), mp
102~103C, []D30 = 8.1 (c = 1.0, CHCl3). Source: HAI QI Excoecaria
agallocha (resinous wood). Ref: 3461.
3012.
HO
HO
HO
O
OH
HO
O
O
OH
H
H
341
7689 Excoecarin T2
7693 Excoecarioside A
C20H32O6 (368.47). As dimethyl ester: colorless needles (aqueous MeOH), mp
C19H32O8 (388.46). Amorphous powder, []D25 = 10.3 (c = 1.36, MeOH). Source:
130~133C, []D30 = 14.7 (c = 0.5, CHCl3). Source: HAI QI Excoecaria
LU BEI GUI HUA Excoecaria cochinchinensis var. viridis. Ref: 4543.
agallocha (resinous wood). Ref: 3461.

OH
OO
HO
HO
OH
OH
O
OH
HO
7694 Excoecarioside B
C19H28O8 (384.43). Syrup, []D25 = +29.3 (c = 0.82, MeOH). Source: LU BEI
GUI HUA Excoecaria cochinchinensis var. viridis. Ref: 4543.
7690 Excoecarin V1
2,3,18-Trihydroxy-3,20-epoxybeyer-15-ene C20H30O4 (334.46). Colorless
prisms (MeOH), mp 177~179C, []D26 = 19.3 (c = 0.5, MeOH). Source:
HAI QI Excoecaria agallocha (fresh stem). Ref: 4386.
O
OO
HO
OH
HO
O
HO
OH
OH
HO
7695 Eximine
C19H20O8 (376.37). Source: YAO YONG HEI MIAN SHEN YE Breynia
7691 Excoecarin V2
officinalis (leaf). Ref: 2583.
ent-2,3-Secokaur-16-en-2,3-dioic acid C20H30O4 (334.46). Source: HAI QI

Excoecaria agallocha (fresh stem). Ref: 4386.
HO
O
O
O
OH
O
HO
OH
OH
OH
H
H
7696 Exoticin
3,5,6,7,8,3',4',5'-Octamethoxyflavone [13364-94-8] C23H26O10 (462.46). mp
7692 Excoecarin V3
124~125C. Source: JIU LI XIANG Murraya paniculata [Syn. Chalcas
ent-3,4-Seco-16-hydroxyatis-4(19)-en-3-oic acid C20H32O3 (320.48).
paniculata]. Ref: 6, 11.
Colorless plates (MeOH), mp 101~102C, []D28 = 53.7 (c = 1.0, MeOH).
Source: HAI QI Excoecaria agallocha (fresh stem). Ref: 4386.

O
O
O
H
O
HO
OH
H
H
O
O
7697 Exozoline
[70561-79-4] C22H25NO (319.45). Source: JIU LI XIANG Murraya
N
H
342
7698 Extensumside A
7700 Ezochasmanine
17-Uzarigenin-3-O--glucopyranosyl-(16)--glucopyranosyl-(14)--t
heveto-pyranosyl-(14)--cymaropyranoside C49H78O21 (1003.16). White
amorphous powder, mp 176~178C, []D25 = 12.5 (c = 0.4, MeOH). Pharm:

Cytotoxic (9 cancar cell lines, mean GI50 = 0.346g/mL: NCI-H460, GI50 =
(0.1070.016)g/mL; Colon205, GI50 = (0.1230.014)g/mL; MDA-MB-231,

GI50 = (0.5270.036)g/mL; MCF7, GI50 = (0.3850.019)g/mL;
MDA-MB-231, GI50 = (0.4700.018)g/mL; OVCAR-3, GI50 =
(0.4070.017)g/mL; A549, GI50 = (0.2960.008)g/mL; HT29, GI50 =
(0.4360.011)g/mL; ACHN, GI50 = (0.3610.022)g/mL; control Taxol, GI50
= (0.1020.009)g/mL, (0.0990.001)g/mL, (0.0280.006)g/mL,
(0.0300.001)g/mL, (0.0320.003)g/mL and (0.0880.004)g/mL),
respectively for last 6 cell lines). Source: CHI GUO TENG Myriopteron
extensum (whole herb). Ref: 4992.
O
H
H
OO
OO
O
OH
OO
OO
HO
OH
OH
OH
OH
OH
OH
OH
7699 Extensumside B
12-(3-Methylbut-2-enoyloxy)pregn-5-en-20-one 3-O-[-cymaropyranosyl(14)--cymaropyranosyl-(14)--thevetopyranosyl-(14)-(6-O-sulfo-glucopyranoside)] C53H84O22S (1105.31). White amorphous powder, mp
196~198C, []D25 = 12.0 (c = 0.4, MeOH). Pharm: Cytotoxic inactive
(NCI-H460, Colon205, MDA-MB-231, all GI50 > 100g/mL). Source: CHI
GUO TENG Myriopteron extensum (whole herb). Ref: 4992.
O
O
O
O
S
O
OO
OH
OO
O
OO
OH
OO
HO
O
OH
OH
H
HO
H
H
O
OH
OH
343
F
7701 cis-Fagaramide
C14H17NO3 (247.30). Pharm: Antioxidant (TLC-based assay, DPPH scavenger,
MIQ = 10g; control Quercetin, MIQ = 1g). Source: Fagara xanthoxyloides.
Ref: 5385.
7705 Fagomine
3,4-Dihydroxy-2-piperidinemethanol [53185-12-9] C6H13NO3 (147.18).
Pharm: Hypoglycemic (mus diabetes mellitus induced by SIZ, distinct
effect)[2170]; -Glucosidase inhibitor (IC50 = 15mmol/L)[4161]. Source: SANG
ZHI Morus alba. Ref: 2170, 4161.
OH
OH
OH
N
HN
O
O
7706 Falaconitine
[62926-57-2] C34 H 47 NO 10 (629.75). Pharm: Causes paralysis,
paroxysmal spasm, convulsion and death (gpg); similar action with

7702 trans-Fagaramide
aconitine (small animals). Source: FA KANG WU TOU Aconitum
N-Isobutyl-3,4-methylenedioxybenzethenylamide C14H17NO3 (247.30). Pharm:
falconeri. Ref: 658.
Antioxidant (TLC-based assay, DPPH scavenger, MIQ = 10g; control

Quercetin, MIQ = 1g)[5385]. Source: SHAN CI GU Asarum sagittarioides,
OH
Fagara xanthoxyloides. Ref: 660, 5385.
H
O
H
N
O
HO
N
H
O
O
O
H
O
7707 cis-Falcarindiol
1,9Z-Heptadecadiene-4,6-diyne-3R,8S-diol [55297-87-5] C17H24O2 (260.38).
Pharm: Analgesic; plant antitoxin; antibacterial (Staphylococcus aureus, MIC

7703 -Fagarine
= 2.2mg/mL; Streptomyces scabies, MIC = 1.5mg/mL; Bacillus subtilis, MIC
4,8-Dimethoxyfuro[2,3-b]quinoline [524-15-2] C13H11NO3 (229.24). mp
= 1.4mg/mL; Bacillus cereus, MIC = 1.6mg/mL; Pseudomonas aeruginosa,
142C. Pharm: Antiarrhythmic (in clinic); antibacterial; antifungal;
MIC = 1.4mg/mL)[5305]; antifungal (Aspergillus niger, MIC = 0.5mg/mL)[5305].
antispasmodic. Source: BAI XIAN PI Dictamnus dasycarpus, CHOU CAO
Source: BEI SHA SHEN Glehnia littoralis (root without cortex: content =
Ruta graveolens, CHOU SHAN YANG Orixa japonica (stem: yield =
0.146%)[5508], CHOU A WEI Ferula foetida (root: yield = 0.00026%)[4659],
0.00038%dw)[4774], GAO JIA SUO BAI XIAN Dictamnus caucasicus, HU
DIAN QIN Sinodielsia yunnanensis (root: yield = 2.90%), FANG FENG
JIAO HUA JIAO Zanthoxylum piperitum, MU(4) JU Aegle marmelos, QI
Saposhnikovia divaricata [Syn. Ledebouriella seseloides], HE SHI FENG
HAN NING HUA JIAO Zanthoxylum tsihanimposa, ZHU YE JIAO
Daucus carota (root), LI JIANG QIAN HU Peucedanum govanianum var.
Zanthoxylum planispinum, ZHU YE JIAO GEN Zanthoxylum planispinum.
bicolo, LONG YAN DU HUO Aralia fargesii, NAN HE SHI Daucus carota,
Ref: 6, 658, 4774.
SONG YE FANG FENG Seseli yunnanense, Niphogeton ternata. Ref: 2, 549,

557, 571, 658, 4156, 4305, 4659, 5305, 5508.
OH
O
N
O
7704 Fagaronine
OH
C21H20NO4 (350.40). Pharm: Cytotoxic (binds to calf thymus DNA by
7708 trans-Falcarindiol
intercalation and toxic to topoisomerases I and II) [5369]. Source: Fagara
1,9E-Heptadecadiene-4,6-diyne-3R,8S-diol; Farcarindiol C17H24O2 (260.38).
xanthoxyloides. Ref: 1521, 5369.
Brown oleaginous substance. Source: QIANG HUO Notopterygium incisum.

Ref: 452.
OH
O
HO
O
O
OH
344
7709 Falcarinol
7714 Fangchinoline
C17H24O (244.38). Source: Niphogeton ternata. Ref: 4156.
Demethyltetrandrine C37H40N2O6 (608.74). mp 237~238C (acetone); mp

177~179C (CH3OH). Pharm: Cytotoxic (HeLa in vitro, ED50 = 4.1g/mL);
antihypertensive; platelet aggregation inhibitor (due to collagen); analgesic;
anti-inflammatory (modulator of cytokine network: prevents
integrin-mediated neutrophil adhesion and fMLP- or leukotriene B4-induced
OH
transmigration, IC50 = 1~5g/mL)[4416]; IL-6 inhibitor (in vitro, IC50 >
7710 Fallacinol
6mol/L)[4416]; LD50 (mus, ip) 50mg/kg. Source: FANG JI Stephania
1,8-Dihydroxy-3-hydroxymethyl-6-methoxyanthraquinone [569-05-1]
tetrandra (dried root: mean content of 6 origins = 0.759%[5508]), RU LAN
Stephania hernandifolia. Ref: 2, 4, 5, 44, 658, 660, 4416, 5501, 5508.
OH
OH
OH O
N
OH
7711 Fallaxose C
C51H60O27 (1105.03). []D = 6.8. Source: JIA HUANG HUA YUAN ZHI
Polygala fallax [Syn. Polygala aureocauda]. Ref: 2184.
O
HO
O
7715 Faradiol
OH
OH
O
OO
O
HO
HO
O
O
HO
OH
Source: KUAN DONG HUA Tussilago farfara. Ref: 1521.
OH
OH
OH
20-Taraxastene-3,16-diol [20554-95-4] C30H50O2 (442.73). mp 236~237C.
H
O
OH
HO
HO
C52H62O28 (1135.06). []D = 6.5. Source: JIA HUANG HUA YUAN ZHI
O
HO
O
DONG HUA Tussilago farfara. Ref: 145.
OH
OH
HO
HO
HO
HO
O
O
O
OH
OH
7716 Farfaratin
C23H34O5 (390.52). White hyaloid crystals, mp 100~101C. Source: KUAN
O
O
OH
7712 Fallaxose D
OH
OH
O
O
7717 Farfugin A
HO
[36061-18-4] C15H18O (214.31). Source: LIAN PENG CAO Farfugium
7713 Fallaxose E
C59H74O34 (1327.23). []D = +16.1. Source: JIA HUANG HUA YUAN ZHI
japonicum. Ref: 6.
O
O
OH
O
HO
O
O
OH
OH
7718 Farfugin B
OH
OH
OH
OH
HO
O HO
O
O
OH
OH
O
OH
HO
OH
[36061-19-5] C15H18O (214.31). Source: LIAN PENG CAO Farfugium
japonicum. Ref: 6.
O
O
O
345
7719 Fargesin
7723 Fargoside A
[31008-19-2] C21H22O6 (370.41). Colorless rhombic crystals, mp
3,20-Dihydroxy-29-norolean-12-en-28-oic acid 3-O--D-xylopyranosyl-
130.0~130.5C (methanol), []D22 = 111.7 (c = 0.57, chloroform); mp
(12)--D-glucopyranoside C40H64O13 (752.95). Amorphous solid, []D25 =
139C. Pharm: Platelet aggregation inhibitor (strong, induced by PAF, IC50
+24.4 (c = 1.0, MeOH). Source: WU YE GUA TENG Holboellia fargesii
= 10mol/L, PAF receptor antagonist, ED50 = 1.3mol/L); phytogrowth
(root). Ref: 4109.
inhibitor (100g/mL, Amaranthus hypochondriacus, InRt = (92.11.8)%; E.
HO
crusgalli, InRt = (83.72.2)%)[5253]. Source: CI HUA JIAO Zanthoxylum

acanthopodium (stem cortex), WANG CHUN YU LAN Magnolia biondii
heptapata], Stauranthus perforatus (root). Ref: 6, 543, 660, 900, 1521,
4439, 5253.
OO
OH
OH
OH
H
HO
[Syn. Magnolia fargesii], YU LAN Magnolia denudata [Syn. Magnolia
OO
OH
O
H
OH
H
O
OH
7724 Fargoside B
3,20,24-Trihydroxy-29-norolean-12-en-28-oic acid 23-O--D-fucopyranos-
O
O
yl-(12)-[-L-arabinopyranosyl-(13)]--D-glucopyranoside C46H74O18
(915.09). Amorphous solid, []D22 = +39.6 (c = 1.0, MeOH). Source: WU YE
7720 ()-Fargesol
C22H28O7 (404.46). Source: ZHOU YE MU LAN Magnolia praecocissima
GUA TENG Holboellia fargesii (root). Ref: 4109.
(seed). Ref: 4181.
HO
O
O
OH
H
OH
OH
HO
O
O
O
7721 Fargesone A
HO
OO
OH
O
O
OH
OH
HO
OO
OH
OH
C21H24 O6 (372.42). Pharm: Calcium antagonist (gpg, colon bands).

Source: WANG CHUN YU LAN Magnolia biondii [Syn. Magnolia
OH
fargesii]. Ref: 658.

7725 Fargoside C
O
3,23-Dihydroxy-30-norolean-2,20(29)-dien-28-oic acid 3-O--L-arabino-
pyranosyl-(12)-[-D-glucopyranosyluronic acid-(13)]--L-arabinoO
pyranoside C45H68O18 (897.03). Amorphous solid, []D25 = +54.0 (c = 0.6,

MeOH). Source: WU YE GUA TENG Holboellia fargesii (root). Ref: 4109.
7722 Fargesone B
C21H24O6 (372.42). Source: YU LAN Magnolia denudata [Syn. Magnolia
heptapata]. Ref: 4439.
H
O OH
HO
O
O
O
O
H
H
OO
O
OH
OH
H
OH
OH
OO
OH OH
OH
O
OH
346
7726 Fargoside D
7730 -Farnesene
3,23-Dihydroxy-30-norolean-12,20(29)-dien-28-oic acid 3-O-methyl
C15H24 (204.36). bp 121~122C/9mmHg. Source: BO SHI QIE Solanum
-D-glucopyranosyluronate-(13)--L-arabinopyranoside C41H62O14
berthaultii, CHAN CHU DAN Bufo bufo gargarizans; Bufo melanostictus,
(778.94). Amorphous solid, []D23 = +65.6 (c = 0.5, MeOH). Source: WU YE
GUANG HUO XIANG Pogostemon cablin [Syn. Mentha cablin], HUA
GUA TENG Holboellia fargesii (root). Ref: 4109.
DONG LAN CI TOU Echinops grijsii, HUANG HUA HAO Artemisia annua,
HUO XIANG Agastache rugosus, PI PA YE Eriobotrya japonica, REN
SHEN Panax ginseng [Syn. Panax schinseng], SHENG JIANG Zingiber
officinale, TAN XIANG Santalum album, XI YANG SHEN Panax
O
H
O OH
H
OO
quinquefolium. Ref: 2, 660.
OH
OH
OH
OH
OH
OH
7731 Farnesiferol A
7727 Fargoside E
[511-33-1] C24H30O4 (382.50). mp () 155.0~155.5C, mp () 152~156C.
3,23-Dihydroxy-olean-12-en-28-oic acid 3-O-methyl -D-glucopyranos-
Source: A WEI Ferula assafoetida. Ref: 6.
yluronate-(13)--L-arabinopyranoside C42H66O14 (794.99). Amorphous

solid, []D28 = +18.3 (c = 0.8, MeOH). Source: WU YE GUA TENG
O
Holboellia fargesii (root). Ref: 4109.

HO
H
H
O OH
OO
O O
O
OH
7732 Farnesiferol B
[54990-68-0] C24H30O4 (382.50). mp 112.5~113.5C. Source: A WEI Ferula
assafoetida. Ref: 6.
OH
OH
OH
OH
HO
OH
7728 (E,E)--Farnesene
7733 Farnesiferol C
[21499-64-9] C15H24 (204.36). Source: GAN JIANG Zingiber officinale.
[512-17-4] C24H30O4 (382.50). mp 83.5~84.5C. Source: A WEI Ferula
Ref: 2.
assafoetida. Ref: 6.
7734 Farnesol
3,7,11-Trimethyl-2,6,10-dodecatrien-1-ol [4602-84-0] C15H26O (222.37). bp
7729 (Z,Z)--Farnesene
C 15 H 24 (204.36). bp 128~130C/12mmHg. Source: DU SONG SHI
Juniperus rigida, HONG CHAI HU Bupleurum scorzonerifolium, JU PI
Citrus reticulata, MU
(3)
JU Matricaria chamomilla [Syn. Matricaria
recutita], PI PA Eriobotrya japonica, PI PA YE Eriobotrya japonica,

SHENG JIANG Zingiber officinale, Malus sp., Pyrus sp. Ref: 2, 660.
160C/10mmHg. Pharm: Flavorant. Source: DAI DAI HUA Citrus aurantium

var. amara, HUANG KUI Abelmoschus moschatus [Syn. Hibiscus
abelmoschus], JIN YIN HUA Lonicera japonica, LA MEI HUA
Chimonanthus fragrans [Syn. Chimonanthus praecox], PI PA Eriobotrya
japonica, PI PA YE Eriobotrya japonica, PU TI SHU HUA Tilia miqueliana,
SHENG JIANG Zingiber officinale. Ref: 2, 6, 658, 660.
OH
347
7735 Farnesyl acetate
7740 Fastigilin C
C17H28O2 (264.41). bp 169~170C/10mmHg. Source: HUANG HUA HAO
[6995-12-6] C20H24O6 (360.41). mp 197~199C (acetone-isopropane ether),
Artemisia annua, MU HAO Artemisia japonica. Ref: 6, 660.
[]D23 = 85.8 (c = 1.11). Pharm: Antineoplastic (mus, P388 and Lewis lung
cancer, in vivo); cytotoxic (mus, P388 in vitro, ED50 = 0.004g/mL; mus, L1210
in vitro, ED50 < 0.01g/mL; KB, ED50 = 1.0g/mL). Source: BAI LAI SHI JU
Baileya multiradiata. Ref: 661.

OH
H
O
7736 Farrerol
[24211-30-1] C17H16O5 (300.31). mp () 223~224C. Pharm: Antibacterial
(Staphylococcus aureus, MIC = 25g/mL); antitussive (dispels phlegm, main

effective component in Rhododendron dauricum MAN SHAN HONG to treat
trachitis); inhibits tissue respiration in lung trachea (rat, in vitro); LD50 (mus,
7741 Fawcettiine
orl) = (150023)mg/kg. Source: MAN SHAN HONG Rhododendron
-Lofoline [6899-87-2] C18H29NO3 (307.44). mp 166~167C. Source: SHEN
dauricum (branchlet-leaf or flower: content = 0.1%[5501], content = 0.07%[5508];
JIN CAO Lycopodium japonicum [Syn. Lycopodium clavatum]. Ref: 6.
[5527]
leaf: mean content of 8 origins = 0.097%
), XIN XI LAN MA Phormium

OH
tenax. Ref: 4, 6, 658, 5501, 5508, 5527.

OH
HO
OH
7742 FB1
7737 Fascicularone A
C19H24O4 (316.40). Pharm: Anti-HIV. Source: SAN CHI LA RUI A Larrea
(1S,9S)-4,11,11-Trimethyl-2,5,6-trihydroxytricyclo[5,4,0,02,5]undec-3-en
tridentata. Ref: 2268.
-7-one C14H20O4 (252.31). Colorless needles, mp 75~77C, []D20 = +323.8 (c

= 0.56, CHCl3). Source: CU SHENG HUANG REN SAN Naematoloma
HO
fasciculare. Ref: 3775.

O
HO
H
OH
OH
OH
OH
7743 FB2
7738 Fascicularone B
(1S,8S)-4,7,10,10-Tetramethyl-3,6-dihydroxytricyclo[5,3,0,02,5]decan-2
,6-olide C15H22O4 (266.34). Colorless needles, mp 127~128C, []D20 = +63.5
(c = 0.88, CHCl3). Source: CU SHENG HUANG REN SAN Naematoloma
C19H24O4 (316.40). Pharm: Anti-HIV (strong). Source: SAN CHI LA RUI A

Larrea tridentata. Ref: 2268.
O
fasciculare. Ref: 3775.

O
O
HO
HO
H
OH
OH
OH
7744 FB3
7739 Fastigilin B
[6995-11-5] C20H26O6 (362.43). mp 259~261C (acetone-petroleum ether).
Pharm: Antineoplastic; cytotoxic. Source: BAI LAI SHI JU Baileya

multiradiata. Ref: 658.

OH
HO
O
O
O H
O
OH
348
7745 FB4
7750 -Fenchene
[33404-67-0] C10H16 (136.24). Source: HONG CHAI HU Bupleurum
scorzonerifolium, SHENG JIANG Zingiber officinale. Ref: 2.
HO
HO
7751 Fenchone
1,3,3-Trimethylbicyclo[2.2.1]heptan-2-one [1195-79-5] C10H16O (152.24). mp
OH
(+) 5.5C, () 6C, bp () 72~73C/12mmHg. Pharm: Local stimulant. Source:
7746 FB5
3'-Demethoxy-6-O-demethylisoguaicin C18H20O3 (284.36). Pharm: Anti-HIV;
antioxidant (Takamatsu DCFH method, myelomonocytic HL-60 cells, IC50 =
(1.60.4)g/mL; control NDGA, IC50 = (0.70.3)g/mL, Vitamin C, IC50 =
(1.90.7)g/mL, Trolox, IC50 = (1.40.5)g/mL)
[3850]
; cytotoxic (XTT assay,
HL-60 cells, IC50 = (13.62.6)g/mL; control NDGA, IC50 = (2.60.2)g/mL,

Vitamin C, IC50 > 10.0g/mL, Trolox, IC50 > 10.0g/mL)[3850]. Source: SAN
CHI LA RUI A Larrea tridentata. Ref: 1521, 2268, 3850.
BEI MEI YA BAI Thuja occidentalis, CE BAI YE Thuja orientalis [Syn.

Platycladus orientalis; Biota orientalis], FU SHE SONG Pinus radiata,
HUANG HUA HAO Artemisia annua, HUI XIANG Foeniculum vulgare,
LIU YE MU LAN Magnolia salicifolia, SHUI SHAN Metasequoia
glyptostroboides, XIA KU CAO Prunella vulgaris, XIANG LI Chenopodium
botrys, XIANG ZHI LENG SHAN Abies balsamea, XUAN YE XIANG
QING Anaphalis contorta, ZHANG MU Cinnamomum camphora. Ref: 6, 658,
660.
O
OH
HO
7752 Fenchyl alcohol
OH
1,3,3-Trimethyl-2-norbornanol C10H18O (154.25). bp 200C. Source: GANG

SONG Baeckea frutescens, SHENG JIANG Zingiber officinale. Ref: 2.
7747 Febrifugine
C16H19N3O3 (301.35). mp 139~140C. Source: CHANG SHAN Dichroa
febrifuga (in 1948, the compound was isolated from the plant by F.A.Kuehl, et
al.)
[5505]
HO
. Ref: 5505.
7753 Fenfangjine A
OH
[115556-32-6] C38H42N2O7 (638.77). Source: FANG JI Stephania tetrandra.
N
O
Ref: 2.
N
H
7748 Fenbaqia saponin
O O
C45H74O17 (887.08). Pharm: Hemolytic (chicken blood trial, distinct effect).

Source: HEI GUO BA QIA Smilax glauco-china. Ref: 2165.
O
H
OH
OO
OO
OH
OH
OH OH HO
N
O
O
H
OO
7754 Fenfangjine D
1,3,4-Tridehydrofangchinolium [115439-62-8] C37H37N2O6+ (605.72). Source:
FANG JI Stephania tetrandra. Ref: 2, 1521.
OH
OH
OH
OH O
7749 -Fenchene
[471-84-1] C10H16 (136.24). bp (+) 155~156C, () 153~154C/720mmHg, ()
154~156C. Source: XIE CAO Valeriana officinalis. Ref: 6.
N
O
+
O
O
349
7755 Feralolide
7760 Fern-9(11)-en-12-ol
[149418-38-2] C18H16O7 (344.32). mp 176~178C, []D25 = 44.9 (c = 0.025,
C30H50O (426.73). Source: ZHU ZONG CAO Adiantum capillus-veneris
MeOH). Source: HAO WANG JIAO LU HUI Aloe ferox. Ref: 730.
(fresh frond). Ref: 4230.

OH
O
HO
OH
O
OH
OH
7756 Fercomin
C20H24O5 (344.41). Pharm: Antibacterial (Staphylococcus aureus, MIC =
7761 Feroxidin
2.3mg/mL; Streptomyces scabies, MIC = 2.1mg/mL; Bacillus subtilis, MIC =
()-Feroxidin; (6R,8R)-5,6,7,8-Tetrahydro-8-methyl-1,3,6-naphthalenetriol
1.7mg/mL; Bacillus cereus, MIC = 1.4mg/mL; Pseudomonas aeruginosa,
[129622-85-1] C11H14O3 (194.23). White amorphous powder, mp 84C, []D20
MIC =1.00mg/mL); antifungal (Aspergillus niger, MIC = 1.0mg/mL). Source:
= 11.3 (c = 0.11, MeOH). Source: HAO WANG JIAO LU HUI Aloe ferox.
HE SHI FENG Daucus carota (root). Ref: 5305.
Ref: 731.
OH
O
O
HO
OH
7762 Feroxin A
OH
[142905-36-0] C17H24O8 (356.38). Source: HAO WANG JIAO LU HUI Aloe

ferox. Ref: 732.
7757 7-Fernene
C30H50 (410.73). mp 208.5~209.5C. Source: TIE SI QI Adiantum pedatum.
OH
Ref: 6.
HO
HO
OH
OH
OH
7763 Feroxin B
7758 9(11)-Fernene
[142905-37-1] C35H36O12 (648.67). Source: HAO WANG JIAO LU HUI Aloe
C30H50 (410.73). mp 170~171C. Source: GUAN ZHONG Dryopteris
ferox. Ref: 732.
crassirhizoma, SHUI LONG GU Polypodium niponicum, TIE SI QI Adiantum

OH
pedatum. Ref: 6, 660.

HO
OH
HO
OH
O
OH
7759 Fernenol
C30H50 O (426.73). mp 194C. Source: AI YE Artemisia argyi, LONG XU
7764 Ferruginol
CAO Poa sphondylodes, MAO CAO YE Imperata cylindrica var. major.
8,11,13-Abietatrien-12-ol [514-62-5] C20H30O (286.46). mp 57~59C, bp
Ref: 6.
175C/0.3mmHg, []D25 = +40.3 (c = 1.0, EtOH), []D25 = +43 (c = 1.0,

CHCl3), []D25 = +39.3 (c = 0.70, CHCl3); []D25 = +40.6. Pharm:
Antibacterial (Staphylococcus aureus, MIC = 31.2g/mL (MCC >
H
250g/mL), control Tetracycline, MIC = 1.56g/mL; Bacillus subtilis,

MIC = 7.8g/mL (MCC > 250g/mL), Tetracycline, MIC = 1.56g/mL;
HO
Enterococcus faecalis, MIC = 7.8g/mL (MCC > 250g/mL), Tetracycline,
350
MIC = 1.56g/mL; Listeria monocytogenes, MIC = 7.8g/mL (MCC =
7768 Ferulic acid
31.25g/mL), Tetracycline, MIC < 0.39g/mL; Salmonella enteriditis,
4-Hydroxy-3-methoxycinnamic acid [537-98-4] C10H10O4 (194.19). White
MIC > 250g/mL, Tetracycline, MIC = 1.56g/mL; Escherichia coli, MIC >
powder, mp 170~171C (Me2CO); mp 173~178C. Pharm: Antineoplastic;
250g/mL, Tetracycline, MIC = 1.56g/mL; Shigella sonnei, MIC >
antimitotic; cytotoxic (cyclooxygenase-1 inhibitor)[5038]; antibacterial;
250g/mL, Tetracycline, MIC = 6.25g/mL)
[5401]
; antifungal (Candida
antiestrogenic; antifungal; antihepatotoxin; platelet aggregation inhibitor;
albicans, MIC > 250g/mL, Miconazole, MIC = 8g/mL; Candida krusei,
antioxidant (DPPH scavenger, EC50 = 3.8g/mL = 19.6mol/L, control
MIC > 250g/mL, Miconazole, MIC = 2g/mL)[5401]; cytotoxic (Col2, IC50 =
Ascorbic acid, EC50 = 1.6g/mL = 9.1mol/L)[4154]; DPPH scavenger (SC50 =
9.7g/mL, control Ellpticine, IC50 = 0.3g/mL; LNCaP, IC50 = 17.1g/mL,
4.5mol/L)[4247]; antioxidant (superoxide anion radical scavenger, superoxide
Ellpticine, IC50 = 0.8g/mL; P388, IC50 = 16.3g/mL, Ellpticine, IC50 =
dismutase method, IC50 for Formazane formation activity > 100mol/L)[4247];
0.1g/mL; A2780, IC50 = 33.3g/mL, control Actinomycin D, IC50 =
antitubercular (Mycobacterium tuberculosis, MIC > 128g/mL, cytotoxic,
0.001g/mL; KB-VI, IC50 > 20g/mL; KB, IC50 > 20g/mL; Lu1, IC50 >
Vero cells, IC50 > 102g/mL, positive control Rifampin, MIC = 0.03g/mL,
20g/mL; BC-1, IC50 > 20g/mL)[5400]; cytotoxic (EBV-EA inhibitor
IC50 = 98.3g/mL, SI = 3277)[4986]; platelet aggregation inhibitor (100mol/L
TPA-induced, mol ratio/TPA = 1000, InRt = 100%)
[5352]
. Source: CHANG
AA-induced, 5g/mL, InRt = (100.00.0)%, p<0.001, control Aspirin,
GENG CU FEI Cephalotaxus harringtonia var. drupacea, DAN SHEN Salvia
50g/mL, InRt = (1000.0)%; 10g/mL collagen-induced, 100g/mL, InRt =
miltiorrhiza (dried root: content = 0.117%[5508]), DU SONG SHI Juniperus
(93.51.3)%, p<0.001, Aspirin, 50g/mL, InRt = (12.21.7)%; 2nmol/L
rigida, GAN XI SHU WEI CAO Salvia przewalskii, RI BEN XIANG BAI
PAF-induced, 100g/mL, InRt = (16.01.3)%, p<0.05, Aspirin, 50g/mL,
JING PI Thuja standishii, SAN YE SHU WEI CAO Salvia trijuga, XIONG
InRt = (9.61.2)%; 0.1g/mL thrombin-induced, 100g/mL, InRt =
RUI ZHUANG SHU WEI CAO Salvia staminea. Ref: 6, 116, 182, 4538,
(7.22.1)%); neuroprotectant (primary cultures of rat cortical cells injured by
5352, 5400, 5401, 5508.
glutamate, 0.1mol/L, cell viability = (54.81.1)%, p<0.01, control MK-801,

0.1mol/L, cell viability = (31.87.1)%, APV, 0.1mol/L, cell viability =
OH
(5.71.9)%, XNQX, 0.1mol/L, cell viability = (28.15.6)%)[3967]. Source: A

WEI Ferula assafoetida (balsam: content scope = 0.03%~0.09%[5501]), AI WA
JIN GU CAO Ajuga iva, BEI SHA SHEN Glehnia littoralis (underground
part), BEI XUAN SHEN Scrophularia buergeriana (root), CHA XIONG
Ligusticum sinense cv. chaxiong, CHOU A WEI Ferula foetida, CHUAN

XIONG Ligusticum chuanxiong [Syn. Ligusticum wallichii] (rhizome: mean
7765 Ferulagol A
7-[(E)-3'-Hydroxy-3',7'-dimethyl-4',6'-octadienyloxy]coumarin C19H22O4
(314.38). Source: Ferula ferulago (root). Ref: 5163.
content of 5 batch samples = 0.065%[5508]), DA CHE QIAN Plantago major,

DA SAN YE SHENG MA Cimicifuga heracleifolia (dried rhizome: content =
0.004%)[5508], DANG GUI Angelica sinensis (dried root: mean content =
0.058%[5508]), DANG SHEN Codonopsis pilosula (dried root: mean content =
OH
0.00221%)[5508], DI SHAO GUA Cynanchum thesioides, DUAN PIAN GAO

O
BEN Ligusticum brachylobum (root and rhizome: content = 0.02%)[5508], FEN

CHA DANG GUI Angelica furcijuga (flower), GAO BEN Ligusticum sinense
7766 Ferulagol B
(root and rhizome: mean content of 8 origins = 0.084%)[5508], GAO GUI
7-[(3'Z,5'E)-7'-Hydroxy-3',7'-dimethyl-3',5'-octadienyloxy]coumarin C19H22O4
CHUN HUANG JU Anthemis nobilis, GUAN MU TONG Aristolochia
(314.38). Source: Ferula ferulago (root). Ref: 5163.
manshuriensis (stem: yield = 0.00070%)[4706], HU HUANG LIAN Picrorhiza

kurrooa (dried rhizome: content scope = 0.82%~2.41%)[5508], HUANG LIAN
Coptis chinensis, HUI XIANG JING YE Foeniculum vulgare, JIA BAI HE
H
O
HO
Notholirion hyacinthinum [Syn. Notholirion bulbuliferum], JING MI Oryza

sativa, KE XI JIA SONG Pinus laricio, LAI FU Raphanus sativus, LAI FU ZI
Raphanus sativus, LAO SHU GUA Capparis spinosa, LI MENG YE Citrus
limonia, LIAO GAO BEN Ligusticum jeholense (root and rhizome: mean
7767 Ferulenol
content of 5 origins = 0.137%)[5508], LUAN BAN ZAO ZHUI Arenaria
C24H30O3 (366.50). Pharm: Antibacterial (Staphylococcus aureus, MIC=
kansuensis var. ovatipeatala (whole herb: mean content = 0.0406%)[5508],
2.4mg/mL; Streptomyces scabies, MIC = 2.2mg/mL; Bacillus subtilis, MIC =

2.0mg/mL; Bacillus cereus, MIC = 2.1mg/mL; Pseudomonas aeruginosa,
MIC =2.3mg/mL; Escherichia coli, MIC =4.8mg/mL)[5305]; antifungal
(Fusarium oxysporum, MIC = 4.6mg/mL; Aspergillus niger, MIC =
4.7mg/mL)[5305]. Source: HE SHI FENG Daucus carota (root). Ref: 5305.
MAO GENG XI XIAN Siegesbeckia orientalis var. glabrescens [Syn.

Siegesbeckia glabrescens], MI PI KANG Oryza sativa, MU ZEI Equisetum
hiemale, NING MENG GEN Citrus limon, NING MENG PI Citrus limon,
OU DANG GUI Levisticum officinale (dried root: mean content =
0.025%)[5508], QIANG HUO Notopterygium incisum, SHEN JIN CAO
Lycopodium japonicum [Syn. Lycopodium clavatum], SHENG MA
OH
Cimicifuga foetida (dried rhizome: content scope of 10 origins =

0.003%~0.063%, mean content = 0.018%)[5508], SHI DIAO BAI Asparagus
officinalis, SHU HUA JIE CAO Valeriana laxiflora (aerial parts and root),
351
SUAN ZAO REN Ziziphus jujuba var. spinosa, TAI WAN FENG DOU CAI
7771 2''-O-Feruloylaloesin
Petasites formosanus, TAI WAN FU RONG Hibiscus taiwanensis, TI MU
C29H32 O12 (572.57). Source: LU HUI Aloe vera [Syn. Aloe barbadensis].
CAO Phleum pratense, TIAN CAI Beta vulgaris, XI LA GANG LIU
Ref: 2.
Periploca graeca, XI ZANG HU HUANG LIAN Picrorhiza scrophulariiflora

(dried rhizome: content scope = 0.82%~2.41%[5508]), XIA TIAN WU
Corydalis decumbens [Syn. Corydalis amabilis], XIAN REN ZHANG
Opuntia dillenii (fresh stem: yield = 0.00053%), XIAO JIE JIN CAO
O
O
O
Huperzia selago [Syn. Lycopodium selago], XIN JIANG GAO BEN

Conioselinum vaginatum (root and rhizome: content = 0.30%)
[5508]
HO
, XING AN
SHENG MA Cimicifuga dahurica (dried rhizome: mean content of 3 origins =

0.010%
OH
OH
[5508]
), XUAN FU HUA Inula britannica, YANG CONG Allium cepa,
OH
O
OH
O
YAO YONG PU GONG YING Taraxacum officinale, YI YE TIE SHAN
Tsuga heterophylla, YI ZHU QIAN MA Urtica dioica, ZI BAI PI Catalpa

ovata, occurs in many plants (widely distributed in plants. firstly isolated from
Ferula foetida. found by Bate-Smith in 33% of investigated dicotyledonous
7772 3-O-trans-Feruloyleuscaphic acid
and 67% of monocotyledonous plants). Ref: 2, 4, 456, 476, 500, 507, 512, 601,
C40H56O8 (6648.9). Source: PI PA YE Eriobotrya japonica (stem and leaf).
602, 658, 660, 663, 2377, 2529, 3967, 4154, 4247, 4454, 4706, 4986, 5038,
Ref: 3061.
5501, 5508.
HO
OH
O
HO
OH
HO
O
HO
7769 6-O-E-Feruloylajugol
7773 6-O-Feruloyl--D-glucopyranoside
C16H20O9 (356.33). Pharm: Antioxidant inactive (hydroxyl radical scavenger,
IC50 > 400mol/L, control Ascorbic acid, IC50 = 51.8mol/L, superoxide

anion radical scavenger, IC50 > 400mol/L, control Ascorbic acid, IC50 =
86.2mol/L)[4289]. Source: XI ZANG HU HUANG LIAN Picrorhiza
scrophulariiflora (root). Ref: 4289.
HO
O
HO
HO
OH
HO
OH
O OH
OH
OH
7770 6-O-Z-Feruloylajugol
OH
OH

7774 1-O-Feruloyl--glucose
H
O
HO
racemosa] (leaf, flower and twig: yield = 0.0053%dw). Ref: 4723.
H
O
H
O
O
HO
O
O
HO
OH
OH
HO
HO
OO
OH
OH
OH
OH
352
7775 4'-O-[2'-O-E-Feruloyl-O--D-glucuronopyranosyl(12)-O--D-
7779 6'-O-E-Feruloylmonotropein
glucuronopyranoside]apigenin
C26H30O14 (566.52). Crystals, mp 143~144C (MeOH) []D20 = 30.2 (c =
C37H34 O20 (798.67). Amorphous yellow powder, mp 197~198C, []D20 =
0.24, MeOH). Source: JI SHI TENG Paederia scandens. Ref: 2561.
74.2 (c = 0.1, MeOH). Source: MU XU Medicago sativa (aerial parts).
Ref: 5167.
H
O
HO
HO
HO
OH
OH
OH
O
HO
O
O OH H
HO
O
O
O
OH
OH
OH
OH
HO
7780 10-O-E-Feruloylmonotropein
OH
C26H30O14 (566.52). Crystals, mp 147~148C (MeOH), []D20 = 26.0 (c =
0.23, MeOH). Source: JI SHI TENG Paederia scandens. Ref: 2561.
7776 8-O-Feruloylharpagide
C25H32O13 (540.53). Amorphous powder; mp 150152C, []D = 24.20 (c =

0.231, MeOH). Source: NAN FEI GOU MA Harpagophytum procumbens,
O
OH
OH
HO
OH
OH
OH
OH
O
OH
HO
HO
O
O
OH
O
O
HO
XUAN SHEN Scrophularia ningpoensis. Ref: 1855, 5458.

HO
OH
7781 N-cis-Feruloyloctopamine
C18H19NO5 (329.36). Colorless oil. Source: MA LING SHU Solanum
OH
tuberosum (tuber). Ref: 5321.
7777 N-trans-Feruloylmethoxytyramine
OH
N-trans-Feruloyl-3-methyldopamine C19H21NO5 (343.38). Yellowish

prismatic crystals (Me2CO), mp 105~106C. Pharm: Germination/growth
HO
N
H
inhibitor/stimulator (dicotyledon Lactuca sativa lettuce, Lycopersicon
OH
esculentum tomato, monocotyledon Allium cepa onion,
7782 N-trans-Feruloyloctopamine
0.0001~0.1mmol/L)[3499]; anti-HIV inactive (in vitro, acutely infected H9
C18H19NO5 (329.36). Colorless oil. Source: MA LING SHU Solanum
lymphocyte cells)[4706]; cytotoxic inactive (in vitro, MCF7 and A549)[4706].
tuberosum (tuber). Ref: 5321.
Source: BO CAI Spinacia oleracea, GUAN MU TONG Aristolochia
N
H
parts), ZHU MAO CAI Salsola collina (aerial parts). Ref: 3499, 4706, 4846.
HO
HO
OH
OH
manshuriensis (stem: yield = 0.00055%), LI Chenopodium album (aerial
HN
7783 2''-O-Feruloylorientin
OH

0.048, MeOH). Source: DUAN BAN JIN LIAN HUA Trollius ledebourii
7778 N-trans-Feruloyl-4'-O-methyldopamine
OH
C19H21NO5 (343.38). Pharm: Germination/growth inhibitor/stimulator

(dicotyledon Lactuca sativa lettuce, Lycopersicon esculentum tomato,
monocotyledon Allium cepa onion, 0.0001~0.1mmol/L). Source: LI
Chenopodium album (root, aerial parts). Ref: 3499.
O
O
O
HO
N
H
OH
HO
HO
OH
OH
OH
OH
OH
O
O
353
7784 3-trans-Feruloyloxy-16-hydroxylup-20(29)-ene
6.7g/mL, PD, InRt = 26.4%, A549, ED50 = 13.35g/mL, MCF7, ED50 =
C40H58O5 (618.91). White amorphous powder (CHCl3MeOH), mp 168C
4.76g/mL, HT29, ED50 = 23.58g/mL); cytotoxic (quinone reductase
(dec) []D20 = +18.7 (c = 0.15, MeOH). Source: FEI LV BIN PIAO SHU
induction assay in cultured Hepa1c1c7 mouse hepatoma cells, CD =
Celtis philippinensis. Ref: 2060.
8.5g/mL)[5038]; cytotoxic (mouse mammary organ culture assay, 75% at

10g/mL)[5038]; cytotoxic (P388, ED50 = 2.20g/mL, control Mithramycin,
ED50 = 0.58g/mL; A549, ED50 = 22.42g/mL, Mithramycin, ED50 =
0.073g/mL; HT29, ED50 = 6.22g/mL, Mithramycin, ED50 =

0.076g/mL)[5421]; cytotoxic inactive (in vitro, LNCaP, IC50 >
H
O
OH
H
O
100mol/L)[4607]; antioxidant (lipid peroxidation inhibitor, brain tissue,

caused by insufficient oxygen and sugar); platelet aggregation inhibitor
(due to ADP); prostaglandin biosynthesis inhibitor (IC50 = 210mol/L);
HO
insect antifeedant (termites, 750mg/L, antifeedant index = 38.7); positive
inotropic effect in heart (in vitro, increases calcium flow in frog, ventricular
7785 3-trans-Feruloyloxy-2-hydroxyurs-12-en-28-oic acid
22
myocyte); immunoenhancer[2100]; germination/growth inhibitor/stimulator
C40H56O7 (648.89). White amorphous powder, []D = +7.2 (c = 0.12,
(dicotyledon Lactuca sativa lettuce, Lycopersicon esculentum tomato,
MeOH). Source: PI PA YE Eriobotrya japonica (stem and leaf). Ref: 3061.
monocotyledon Allium cepa onion, 0.0001~0.1mmol/L)[3499]; anti-HIV

inactive (in vitro, acutely infected H9 lymphocyte cells)[4706]; cytotoxic
inactive (in vitro, MCF7 and A549)[4706]. Source: BAI HUA YOU MA
TENG Mucuna birdwoodiana, CANG BAI CHENG GOU FENG
OH
O
HO
Diploclisia glaucescens, CI JI LI Tribulus terrestris, CI TIAN QIE Solanum

khasianum, FAN LI ZHI Annona squamosa, GUAN MU TONG
Aristolochia manshuriensis (stem: yield = 0.00076%), HE SHOU WU
Polygonum multiflorum, HONG HAI JIAO Capsicum annuum (stem and

root: yield = 0.0016%dw)[4779], HUAI TONG Aristolochia moupinensis,
HO
HUANG HUA REN Sida acuta, HUO MA REN Cannabis sativa, LANG
7786 3-O-Feruloylquinic acid
DANG ZI Hyoscyamus niger (seed: yield = 0.0006%dw)[4607], LI
C17H20O9 (368.34). mp 196~197C. Source: DI SHAO GUA Cynanchum
Chenopodium album (aerial parts), MA LING SHU Solanum tuberosum
thesioides, XIANG RI KUI YE Helianthus annuus. Ref: 6.
(tuber), MAI DONG Ophiopogon japonicus (tuber)[4663], TAI WAN FU

RONG Hibiscus taiwanensis, TIAN QIE ZI Solanum indicum (root)[3087],
O
O
OH O
MO ZHI JIAO GU CUI Casearia membranacea (stem), Hypecoum sp.,

occurs in many plants. Ref: 715, 900, 1316, 2100, 2529, 3087, 3499, 4607,
OH
HO
4663, 4706, 4779, 5038, 5321, 5421.
OH
OH
O
HO
7787 6'''-Feruloylspinosin
H
N
C38H40O18 (784.73). Source: DA ZAO Ziziphus jujuba, SUAN ZAO REN

Ziziphus jujuba var. spinosa. Ref: 2.
OH
O
HO
7789 N-cis-Feruloyltyramine
O
OH
OH
O
O
HO
OH
O
OH
OH
OH
C18H19NO4 (313.36). Pharm: Cytotoxic (P388, ED50 = 2.71g/mL, control

Mithramycin, ED50 = 0.58g/mL; A549, ED50 = 35.94g/mL, Mithramycin,
ED50 = 0.073g/mL; HT29, ED50 = 18.41g/mL, Mithramycin, ED50 =
0.076g/mL)[5421]. Source: HONG HAI JIAO Capsicum annuum (stem and
OH
7788 N-trans-Feruloyltyramine
Moupinamide; (2,3)trans-N-(p-Hydroxyphenethyl)ferulamide C18H19NO4
root: yield = 0.00048%dw), MA LING SHU Solanum tuberosum (tuber), TAI

WAN FU RONG Hibiscus taiwanensis, MO ZHI JIAO GU CUI Casearia
membranacea (stem). Ref: 2529, 4779, 5321, 5421.
(313.36). Colorless pillar crystals, mp 97~99C; colorless lamellar crystals,
OH
(chloroformacetone), mp 142~143C, colorless needles. Pharm: Anti-HIV

(H9 lymphocytic cells, inhibits replication, IC50 (concentration that inhibits
uninfected H9 cell growth by 50%) > 25g/mL)[2529]; cytotoxic (hmn, A549
EC50 > 20g/mL, MCF7 EC50 > 20g/mL)[2529]; cytotoxic (BST, IC50 =
HO
O
O
N
H
354
7790 trans-p-Ferulylalcohol-4-O-[6-(2-methyl-3-hydroxypropionyl)]glu-
7794 Fetisinine
copyranoside
(3R,20S)-3-Hydroxyl-20-(5'-hydroxy-3'-methylpyridin-6'-yl)-5-pregnan-6-on
C20H28O10 (428.44). Source: HONG HAI JIAO Capsicum annuum. Ref: 3419.
e) C27H39NO3 (425.62). Amorphous colorless powder, []D25 = 118 (c =

0.10, MeOH). Source: XI BEI MU Fritillaria imperialis. Ref: 3372.
HO
OO
HO
OH
OH
OH
OH
H
H
7791 Ferutidin
Jaeschkeanadiol p-methoxybenzoate C23H32O4 (372.51). Source: YI LANG A
WEI Ferula kuhistanica (stem). Ref: 3977.
HO
H
H
7795 Filicenal
[13843-88-4] C30H48O (424.72). mp 272C. Source: TIE SI QI Adiantum
pedatum. Ref: 6.
HO
O
O
7792 Ferutinin
Jaeschkeanadiol p-hydroxybenzoate C22H30O4 (358.48). Pharm: Antibacterial
(MSSA, MIC = 8g/mL, control Ampicillin, MIC = 1g/mL; MRSA, MIC =
16g/mL, Ampicillin, MIC = 2g/mL; Staphylococcus epidermidis IFO 3762,
MIC = 16g/mL, Ampicillin, MIC < 0.125g/mL; Enterococcus faecalis
ATCC 21212, MIC = 31g/mL, Ampicillin, MIC = 1g/mL; Bacillus subtilis
IFO 3134, MIC = 16g/mL, Ampicillin, MIC < 0.125g/mL; Salmonella
7796 Filicene
[2472-29-9] C30H50 (410.73). mp 228.5~229.5C. Source: GUAN ZHONG
Dryopteris crassirhizoma, TIE SI QI Adiantum pedatum. Ref: 6.
typhimurium IFO 13245, MIC > 250g/mL, Ampicillin, MIC = 1g/mL;

Proteus mirabilis IFO 3849, MIC > 250g/mL, Ampicillin, MIC = 2g/mL;
Escherichia coli NIHJ JC-2, MIC > 250g/mL, Ampicillin, MIC =
4g/mL)[5207]. Source: YI LANG A WEI Ferula kuhistanica (root), YI LANG
A WEI Ferula kuhistanica (fruit). Ref: 3977, 5207.
7797 Filicinic acid

HO
[2065-00-1] C8H10O3 (154.17). mp 215C (dec). Source: GUAN ZHONG
Dryopteris crassirhizoma. Ref: 6.
HO
OH
OH
7793 Fetidine
O
[7072-86-8] C40H46N2O8 (682.82). mp (+) 132~135C. Pharm:

Anti-inflammatory; inhibits neuroaction; antihypertensive. Source: XIANG
TANG SONG CAO Thalictrum foetidum. Ref: 6, 658, 660.
7798 Filixic acid BBB

[4482-83-1] C36H44O12 (668.74). Pharm: Anthelmintic. Source: MIAN MA
Dryopteris filix-mas. Ref: 658.
O
O
HO
N
OH
HO
O
OH
HO
HO
OH
O
O
O
OH
355
7799 Fimbriatone
7803 Fissistigmoside
C16H10O5 (282.26). Yellowish powder, mp 272~273C. Source: LIU SU JIN
C17H24O10 (388.37). White crystals, mp 188~190C. Source: HEI FENG
SHI HU Dendrobium fimbriatum. Ref: 2469.
TENG Fissistigma polyanthum. Ref: 669.
HO
OH
O
OH
O
OH
OH
OH
O
OH
7800 Finaconitine
[81161-27-5] C32H44N2O10 (616.71). Crystals (ethanol), mp 220~221C, []D22
7804 Fistacacidin
= +44.7 (c = 1, methanol). Pharm: Analgesic. Source: GAN WAN WU TOU
[25375-34-2] C15H14O5 (274.28). mp 245~247C. Source: PO LUO MEN
Aconitum finetianum. Ref: 658.
ZAO JIA Cassia fistula. Ref: 6.
H
O
O
OH
OH
OH
OH
O
OH
N
NH
OH
OH
O
O
OH
7805 Flabelliformine
C16H25NO2 (263.38). []D25 = 78 (MeOH). Source: DONG BEI SHI SHAN
7801 Finitin
Huperzia miyoshiana. Ref: 5412.
[54192-33-5] C15H20O3 (248.32). mp 153~155C. Source: DONG BEI HUI

HAO Seriphidium finitum [Syn. Artemisia finita]. Ref: 6.
O
OH
7806 Flaccidin B
C41H66O12 (750.98). Pharm: Reverse transcriptase inhibitor of RNA tumor

virus. Source: E ZHANG CAO Anemone flaccida. Ref: 4060.
7802 Fisetin
3,7,3',4'-Tetrahydroxyflavone [528-48-3] C15H10O6 (286.24). Yellow acicular
crystals (dilute ethanol), mp 330C (dec), mp 348C, mp 350C; yellow thin
acicular, mp > 300C. Pharm: Antibacterial; antispasmodic (mus small
intestine, caused by acetylcholine, smooth muscle relaxant); inhibits
metabolism and release of arachidonic acid; antihistamine (inhibits histamine
OO
release, basophilic granulocyte); prostaglandin biosynthesis inhibitor;

5-lipoxygenase inhibitor; NADH oxidase inhibitor; iodine-induced thyronine
deiodinase inhibitor; aldose reductase inhibitor (rat eye lens, ID50 = 1mol/L);
protein kinase C inhibitor; succinic oxidase inhibitor; regulates allergic
reaction. Source: HAI ER CHA Acacia catechu, HUANG LIAN YA Pistacia
chinensis, LIAO SHANG RONG MAO HUA Anthyllis vulneraria, LIN BEI
OH
H
O
HO
HO
OH
OO
OH
OH
OH
ZI Toxicodendron succedaneum [Syn. Rhus succedanea], MANG GUO
7807 Flavanol
Mangifera indica, YE QI SHU YE Rhus sylvestris. Ref: 6, 661.
Flavan-4-ol C15H14O2 (226.28). mp 119C. Source: LUO TUO CI Alhagi

pseudalhagi, CHA SHU GEN Camellia sinensis [Syn. Thea sinensis]. Ref: 6.
O
OH
HO
OH
OH
OH
356
7808 Flavanone 4',5-dihydroxy-7-prenyloxyflavanone
7813 Flavidusin B
C20H20O5 (340.38). Fine needles, mp 69~70C. Source: GAO GUI YOU MU
C20H32O2 (304.48). mp 79~80C, []D22 = +109.0 (c = 0.65, CHCl3). Source:
YUN XIANG Teclea nobilis (aerial parts). Ref: 3503.
DAN HUANG XIANG CHA CAI Isodon flavidus. Ref: 4067.
OH
OH
OH
7809 Flavaspidic acid BB
7814 Flavinadenine dinucleotide
[114-42-1] C24H30O8 (446.50). mp () 92C; 150C, () 156C. Pharm:
[146-14-5] C27H35N9O15P2 (787.58). Source: QING WA Rana nigromaculata;
Antibacterial; antifungal; anthelmintic. Source: GAO JIA SUO LIN MAO
Rana plancyi, YUAN CAN ZI Bombyx mori. Ref: 6.
JUE Dryopteris caucasica, GUAN ZHONG Dryopteris crassirhizoma,

O
HUANG MAO LIN MAO JUE Dryopteris chrysocoma, MIAN MA

Dryopteris filix-mas. Ref: 6, 658.
OH
OH HO
HO
HN
OH
OH
OH
OH
OH OH
O
O
O
P
P
O
NH2
7810 Flavaspidinin
N
O
N
N
OH OH
[1763-14-0] C23H28O8 (432.47). mp 211~212C. Source: GUAN ZHONG

Dryopteris crassirhizoma. Ref: 6.
7815 (+)-Flavinantine
C19H21NO4 (327.38). Pharm: Cytotoxic (in vitro, HepG2, IC50 = 9.3g/mL;
OH
OH
Hep2,2,15, IC50 = 9.7g/mL)[3083]. Source: YOU GOU YING ZHAO

Artabotrys uncinatus (root and stem). Ref: 3083.
O HO
HO
OH
O
HO
7811 Flavidin
[83924-98-5] C15H12O3 (240.26). Pharm: Antispasmodic. Source: BEI MU
LAN Coelogyne ovalis, JIE JING SHI XIAN TAO Pholidota articulata. Ref:
658.
O
OH
7816 Flavin mononucleotide

[146-17-8] C17H21N4O9P (456.35). Source: YUAN CAN ZI Bombyx mori,
ZHANG LANG Blatta orientalis. Ref: 6.
HO
OH
7812 Flavidusin A
DAN HUANG XIANG CHA CAI Isodon flavidus. Ref: 4067.
OH
OH
H
H
N
O
N
H
OH
OH
H
OH
OH
O P O
OH
357
7817 Flavocommelin
7822 Flavumone A
[16049-42-6] C28H32O15 (608.56). mp 216~217C. Source: YA ZHI CAO
1-[3-(2,4-Dihydroxy-benzoyl)-4,5,6-trihydroxy-2-(4-hydroxy-phenyl)-benzof
Commelina communis. Ref: 6.
uran-7-yl] -3-(4-hydroxy-phenyl)-propenone C 30H20O10 (540.49). Yellow

crystals, mp 240~241C (Me2CO). Source: HUANG SAI JIN LIAN MU
O
HO
Ouratea flava (stem cortex). Ref: 3384.
O
HO
OH
O
OH
OH
OH
OH
OH
OH
OH
OH
HO
7818 Flavokawain A
2'-Hydroxy-4,4',6'-trimethoxychalcone C18H18O5 (314.34). Yellow plates
O
O
HO
(n-hexane-EtOAc), mp 112C, mp 114~115C. Source: CHANG YE GE NA
OH
OH
XIANG Goniothalamus gardneri (aerial parts). Ref: 5096.

OH
7823 Flavumone B
3-(2,4-Dihydroxy-benzoyl)-4-hydroxy-2,7-bis-(4-hydroxy-phenyl)-7,8-dihydr
o-furo[2,3-f]chromen-9-on C30H20O9 (524.49). Amorphous yellow solid.
OH
[]D25 = +29 (c = 0.5, MeOH). Source: HUANG SAI JIN LIAN MU Ouratea
flava (stem cortex). Ref: 3384.
7819 Flavone
HO
2-Phenylchromone [525-82-6] C15H10O2 (222.25). mp 97C. Pharm: Platelet
aggregation inhibitor (hmn); inhibits release of histamine from basophiles;
5-lipoxygenase inhibitor; cyclooxygenase inhibitor. Source: YIN FEN BAO
OH
CHUN Primula pulverulenta, WU LOU ZI Phoenix dactylifera. Ref: 6, 658.
OH
OH
O
OH
O
7824 Flazin
7820 Flavonol
C17H12N2O4 (308.30). Pharm: Cytotoxic (mouse mammary organ culture
[577-85-5] C15H10O3 (238.25). mp 169~170C. Source: BAI GUO YE Ginkgo
assay, 75% at 4g/mL)[5038]. Source: YA DAN ZI Brucea javanica [Syn.
biloba, BAI QU CAI Chelidonium majus, CHA SHU GEN Camellia sinensis
Brucea sumatrana; Rhus javanica]. Ref: 5038.
[Syn. Thea sinensis]. Ref: 6.
O
OH
N
H
HO
7821 Flavoxanthin
OH
5,8-Epoxy-5,8-dihydro-,eplsilon-carotene-3,3'-diol [512-29-8] C40H56O3

(584.89). mp 184C. Pharm: Yellow pigment. Source: CAO DI MAO GEN
7825 Flemichapparin B
Ranunculus acris, DA BAI DING CAO Senecio oryzetorum, JIN ZHAN JU
C17H12O5 (296.28). Pharm: Antioxidant (DPPH scavenger, ScRt = 5.26%,
Calendula officinalis, OU ZHOU QIAN LI GUANG Senecio vulgaris, QIAN
control BHT, ScRt = 71.5%)[3810]; antibacterial (Staphylococcus aureus ATCC
LI GUANG Senecio scandens [Syn. Senecio chinensis], WAN SHOU JU
25923, MIC > 512g/mL, control Vancomycin, MIC = 0.5g/mL; MRSA
Tagetes erecta, XI YANG JIE GU MU Sambucus nigra, XING REN Prunus
SK1, MIC > 512g/mL, Vancomycin, MIC = 1.0g/mL)[3810]; increases blood
armeniaca, YANG LI Prunus domestica, YAO YONG PU GONG YING
pressure (anesthetized rats, increases in mean arterial blood pressure,
Taraxacum officinale, YE MU XU Medicago falcata (whole herb: content
0.4mg/kg, 8.9mmHg)[3810]. Source: PAN YUAN YU TENG Derris scandens
scope = 7%~8%), YIN BAI JIN HE HUAN Acacia dealbata, Berberis sp.,
(stem). Ref: 3810.
Chrysanthemum sp., Narcissus sp., Rosa sp., Tulipa sp. Ref: 6, 658, 660.
H
H
HO
OH
O
O
358
7826 Flemichapparin C
7831 Floranol
C17H10O6 (310.27). Pharm: Antioxidant (DPPH scavenger, ScRt = 21.05%,
C21H22O7 (386.41). Source: DA HUA DI AO DOU Dioclea grandiflora (root).
control BHT, ScRt = 71.5%). Source: PAN YUAN YU TENG Derris
Ref: 4978.
scandens (stem). Ref: 3810.
HO
O
O
OH
OH
OH
7827 Flemiphilippinin C
7832 Floratheasaponin A
[133830-92-9] C26H26O6 (434.49). Yellowish acicular crystals
C59H92O26 (1217.38). Pharm: Antihyperlipidemic[4537]. Source: PU ER CHA
(methanolwater), mp 143~145C. Source: MAN XING QIAN JIN BA
Camellia sinensis var. assamica (flower). Ref: 4537.
Flemingia philippinensis [Syn. Moghania philippinensis]. Ref: 179.

O
O
OH
OH
OH
HO
O
O HO
OH
OH
OH
O
OH
OH
HO
O
H
OH
OO
OH
C22H32O6 (392.50). mp 224~226.5C, []D21 = 99.43 (c = 0.52, MeOH).
HO
7828 Flexicaulin A
Source: ROU JING XIANG CHA CAI Isodon flexicaulis. Ref: 4067.
O
OH
OO
OH
OH
OH
7833 Floridic acid methyl ester

C30H46O5 (486.70). Pharm: Anti-inflammatory[5341]; antiviral. Source: MIAN
MAO GOU TENG Uncaria lanosa. Ref: 5341.
7829 Flindersiamine
C15H15NO5 (289.29). Pharm: Antibacterial (Staphyloccocus aureus and
Streptococcus faecalis, moderate). Source: Esenbeckia yaaxhokob (leaf). Ref:
HO
4929.
O
H
O
HO
OH
7834 Floridinine
7830 Flindersine
[200067-94-3] C15H27NO5 (301.39). Oil, []D = 8.3 (c = 0.096, ethanol).
C14H13NO2 (227.27). Pharm: Photo-activated antibacterial (Staphylococcus
Pharm: Antifungal (Fusarium moniliforme). Source: Heliotropium floridum
aureus)[4989]; photo-activated antifungal (Candida albicans weak)[4989];

photo-activated DNA binding inactive (16 restriction enzymes)[4989] . Source:
var. latifolium. Ref: 1554.
JIAN YE YUN XIANG CAO Haplophyllum acutifolium, Sarcomelicope
OH
glauca. Ref: 4989, 5175.

HO
O
H
O
N
H
OH
359
7835 Floridiolide A
7839 Fluorocarpamine
Limbatolide C C20H28O4 (332.44). Gummy solid, []D23 = 98.231 (c = 0.063,
CHCl3). Pharm: AChE inhibitor (in vitro, IC50 = (103.70.5)mol/L, positive
control Galanthamine, IC50 = (0.50.01)mol/L)[4453]; BChE inhibitor (in vitro,

IC50 = (14.20.3)mol/L, positive control Galanthamine, IC 50 =
(8.50.1)mol/L)[4453]. Source: GE LUN BI YA BA DOU Croton

N
schiedeanus (aerial parts), YOU YAN AO TUO SI TE CAO Otostegia limbata
(root). Ref: 4447, 4453.

O
O
O
7840 Fluorocarpamine-N-oxide

O
OH
7836 Florilenalin
2,4-Dihydroxy-10(14),11(13)-guaiadien-12,8-olide [54964-49-7] C15H20O4
N O
(264.32). Oil. Pharm: Cytotoxic (hmn H.Ep.-2 cutis cancer in throat, 1g/mL).
O
Source: DUI XIN JU Helenium autumnale. Ref: 661.
O
H
HO
7841 Fluorocurine
O
O
HO
C21H27N2O2 (339.46). Source: Strychnos guianensis (stem cortex). Ref: 3943.
7837 Floripavine
N
(+)-Salutaridine [1936-18-1] C19H21NO4 (327.38). mp 197~198C. Pharm:

YING SU Papaver bracteatum, JIN DONG YING SU Papaver orientale,
HO
XIANG BA DOU Croton balsamifera, YI KANG BA DOU Croton salutaris,

YING SU Papaver somniferum. Ref: 6, 658.
Antineoplastic (W256). Source: YA PIAN Papaver somniferum, DA HONG
7842 Flustrabromine
C17H21BrN2O (349.27). Pharm: Affinity to nAChR (42 subtype, K i >
50000nmol/L, control ()-Nicotine, Ki = (0.8380.132)nmol/L; 7 subtype,

Ki > 50000nmol/L, ()-Nicotine, Ki = (1275)nmol/L)[5029]. Source: BEI HAI
HO
XIAN TAI CHONG Flustra foliacea Ref: 5029.

N
N
O
7838 Flourensadiol
C15H26O2 (238.37). Pharm: Phytotoxin (inhibits radicle growth, Amaranthus
NH
hypochondriacus, IC50 = 412mol/L, control 2,4-D, IC50 = 180mol/L;
Br
Echinochloa crusgalli, IC50 = 4200mol/L, control 2,4-D, IC50 =
7843 Flustramine A
230mol/L); CaM interactor (cAMP phosphodiesterase inhibitor, IC50 =
C21H29BrN2 (389.38). Pharm: Affinity to nAChR (42 subtype, Ki >
5.2mol/L, control Chlorpromazine, IC50 = 10.2mol/L, interacted with
50000nmol/L, control ()-Nicotine, Ki = (0.8380.132)nmol/L; 7 subtype,
bovine-brain calmodulin and inhibited the activation of the
Ki > 50000nmol/L, ()-Nicotine, Ki = (1275)nmol/L)[5029]. Source: BEI HAI
calmodulin-dependent enzyme cAMP phosphodiesterase). Source: FU
XIAN TAI CHONG Flustra foliacea. Ref: 5029.
CHUI FE LAO JU Flourensia cernua. Ref: 3433.

OH
H
N
Br
H
OH
360
7844 Flustramine B
7851 Foliamenthin
[71239-65-1] C21H29BrN2 (389.38). Source: BEI HAI XIAN TAI CHONG
[21848-66-8] C26H36O12 (540.57). mp 194~196C. Source: SHUI CAI
Flustra foliacea. Ref: 1521.
Menyanthes trifoliata (the compound was isolated from the plant by Battersby
et al. in 1968)[5505], SHUI CAI GEN Menyanthes trifoliata. Ref: 6, 5505.
HO
Br
OH
OH
OH
7845 Foetisulfide A
E-3-Methylsulfinyl-2-propenyl sec-butyl disulfide C8H16OS3 (224.41). Pale
HO
H
O
yellow oil, []D25 = 36.7 (c = 1.1, MeOH). Source: CHOU A WEI Ferula
foetida (root: yield = 0.0029%). Ref: 4659.

S S
7852 Folic acid
Pteroylglutamic acid; Cytofol; Folipac [59-30-3] C19H19N7O6 (441.41). mp
250C (dec), []D25 = +23 (c = 0.5, 0.1mol NaOH).[5507] Pharm:

7846 Foetisulfide B
Hematopoietic vitamin (used in treatment of megaloblastic anemia due to lack
Z-3-Methylsulfinyloxy-2-propenyl sec-butyl disulfide C8H16O2S3 (240.41).
of folic acid). Source: BEI HAI DANG GUI Angelica acutiloba var.
Pale yellow oil, []D = +8.8 (c = 0.9, MeOH). Source: CHOU A WEI
sugiyamae, BO CAI Spinacia oleracea, CHUAN XIONG Ligusticum
Ferula foetida (root: yield = 0.00051%). Ref: 4659.
chuanxiong [Syn. Ligusticum wallichii], CU LIU GUO Hippophae
25
rhamnoides, DONG DANG GUI Angelica acutiloba [Syn. Ligusticum
O
S
acutilobum], HONG CHE ZHOU CAO Trifolium pratense, HUANG QI
Astragalus membranaceus, LI ZHI Litchi chinensis, LIN QIN Malus asiatica,
MANG GUO Mangifera indica, REN SHEN Panax ginseng [Syn. Panax
7847 Foetisulfide C
schinseng], SANG YE Morus alba, YANG SHI GUO Syzygium cumini. Ref: 2,
E-3-Methylsulfinyloxy-2-propenyl sec-butyl disulfide C8H16O2S3 (240.41).
658, 660, 5507.
Pale yellow oil, []D25 = +27.5 (c = 1.2, MeOH). Source: CHOU A WEI
Ferula foetida (root: yield = 0.00077%). Ref: 4659.
H2N
O
S
N
N
H
N
OH
H
N
OH
7848 Foetisulfide D
O
Bis(3-methylthio-2E-propenyl) disulfide C8H14S4 (238.46). Colorless oil.
OH
Source: CHOU A WEI Ferula foetida (root: yield = 0.00026%). Ref: 4659.
S
S S
7849 Foetithiophene A
3,4,5-Trimethyl-2-thiophenecarboxylic acid C8H10O2S (170.23). Colorless
needles, mp 166.0~166.5C. Source: CHOU A WEI Ferula foetida (root: yield
= 0.00051%). Ref: 4659.
7853 Folinic acid

[58-05-9] C21H25N7O7 (487.48). mp 248~250C. Source: BA JIAO HUI
XIANG Illicium verum, BO CAI Spinacia oleracea, CAN DOU YE Vicia
faba, CU LIU GUO Hippophae rhamnoides, DANG GUI Angelica sinensis,
FENG MI Apis cerana, FENG RU Apis cerana, HEI DA DOU Glycine max,
HEI DA DOU YE Glycine max, HEI ZHI MA Sesamum indicum (black seed)
[Syn. Sesamum orientale (black seed)], HONG CHE ZHOU CAO Trifolium
OH
pratense, HONG CHE ZHOU CAO Trifolium pratense, HUANG QI

Astragalus membranaceus, LI ZHI Litchi chinensis, MANG GUO Mangifera
indica, MO GU Agaricus campestris, NIU RU Bos taurus domesticus;
7850 Foetithiophene B
3,4,5-Trimethyl-2-(methylsulfinyloxymethyl) thiophene C9H14O2S2 (218.34). Pale
Bubalus bubalis, SANG YE Morus alba, YAO YONG PU GONG YING

Taraxacum officinale. Ref: 6, 660.
yellow oil. Source: CHOU A WEI Ferula foetida (root: yield = 0.00051%). Ref: 4659.
S
S
O
N
HN
O
H2N
N
H
N
H
OH
H
N
O
O
OH
361
7854 Foliosidine
7859 Fomefficinic acid E
[2520-38-9] C16H21NO5 (307.35). mp 141~142C, []D = +42 (ethanol).
15-Acetoxy-3-oxo-24-methylenelanosta-7,9(11)-dien-21-oic acid C33H48O5
Pharm: Antiarrhythmic (cat, caused by CaCl2 or adrenine, 20~30mg/kg iv, the
(524.75). White amorphous powder, mp 207~209C, []D20 = +46.7 (c = 0.03,
action maintains 20~60min); LD50 (mus, iv) = 209mg/kg. Source: DA YE
CHCl3:MeOH = 1:1). Source: A LI HONG Fomes officinalis. Ref: 2566.
YUN XIANG CAO Haplophyllum perforatum. Ref: 658.

O
HO
OH
HO
7855 Fomannoxin acid

2-Isopropenyl-2,3-dihydrobenzofuran-5-carboxylic acid [84015-64-5] C12H12O3
(204.23). Source: BAI HUA LONG DAN Gentiana algida. Ref: 704.
7860 Fomitopinic acid A

24S,25-Dihydroxy-3-oxolanost-8-en-21-oic acid C30H48O5 (488.71).
Colorless needles (CHCl3), mp 182~184C, []D25 = +33.8 (c = 1.1, MeOH).

Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor, 10g/mL, InRt = 18.1%,
HO
COX-2 inhibitor, IC50 = 1.15mol/L; control Indomethacin, COX-1 inhibitor,
IC50 = 0.10mol/L; COX-2 inhibitor, IC50 = 0.60mol/L). Source: HONG

7856 Fomefficinic acid A
YUAN CENG KONG JUN Fomitopsis pinicola [Syn. Fomes pinicola;
24-Methylene-3-oxo-lanost-8-en-21-oic acid C31H48O3 (468.73). White
Polyporus pinicola] (sporocarp: yield = 0.0036%fw). Ref: 4798.
needles, mp 201~203C, []D20 = +4.6 (c = 0.06, CHCl3:MeOH = 1:1).

HO
O
HO
OH
Source: A LI HONG Fomes officinalis. Ref: 2566.
OH
7861 Fomitopinic acid B

24,25-Dihydroxy-3-acetoxylanost-8-en-21-oic acid C32H52O6 (532.77).
7857 Fomefficinic acid B

3,15-Dihydroxy-24-methylene-lanosta-7,9(11)-dien-21-oic acid C31H48O4
20
Amorphous powder, []D25 = +16.7 (c = 0.3, MeOH). Source: HONG YUAN
(484.73). White amorphous powder, mp 194~196C, []D = +25.8 (c = 0.05,
CENG KONG JUN Fomitopsis pinicola [Syn. Fomes pinicola; Polyporus
pinicola] (sporocarp: yield = 0.00058%fw). Ref: 4798.
O
HO
OH
O
H
HO
OH
HO
OH
H
O
7858 Fomefficinic acid D

15-Hydroxy-3-oxo-24-methylenelanost-8-en-21-oic acid C31H48O4 (484.73).
7862 Fomitopsic acid B
White amorphous powder, mp 205~207C, []D20 = +37.5 (c = 0.04,
C33H48O5 (524.75). Source: HONG YUAN CENG KONG JUN Fomitopsis
pinicola [Syn. Fomes pinicola; Polyporus pinicola] (sporocarp: yield =

0.017%fw). Ref: 1521, 4798.
O
HO
HO
OH
O
362
7863 Fomitopsin A
7867 Fomitoside B
3-Carboxyacetyloxy-24-exomethylene-12-hydroxy-23-oxo-lanost-8-en-26-oi
C 35 H 54 O 8 (602.82). Amorphous powder, []D 25 = 18.3 (c = 0.2,
c acid C34H50O8 (586.77). []D20 = +5.5 (c = 0.4, CHCl3). Source: CENG
MeOH). Source: HONG YUAN CENG KONG JUN Fomitopsis
KONG JUN Fomitopsis spraguei. Ref: 5302.
pinicola [Syn. Fomes pinicola; Polyporus pinicola] (sporocarp: yield =

0.00091%fw). Ref: 4798.
O
OH
HO
HO
OH
OH
OH
O
O
HO
7864 Fomitopsin B
C34H48O7 (568.76). Source: CENG KONG JUN Fomitopsis spraguei. Ref:
7868 Fomitoside C
5302.
3-Oxolanosta-8,24-dien-21-oic acid 21-O--D-xylopyranoside

C 35 H 54 O 7 (586.82). Amorphous powder, []D 25 = +31.4 (c = 2.4,
MeOH). Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor, IC 50 =
1.91mmol/L, COX-2 inhibitor, IC 50 = 5.11mmol/L; control

O
Indomethacin, COX-1 inhibitor, IC 50 = 0.10mol/L; COX-2 inhibitor,
IC 50 = 0.60mol/L). Source: HONG YUAN CENG KONG JUN
Fomitopsis pinicola [Syn. Fomes pinicola; Polyporus pinicola]

(sporocarp: yield = 0.0044%fw). Ref: 4798.
HO
O
O
HO
HO
OH
7865 Fomitopsin C
C34H50O7 (570.77). Source: CENG KONG JUN Fomitopsis spraguei. Ref:
5302.
7869 Fomitoside D
3-Oxolanosta-8,24(31)-dien-21-oic acid 21-O--D-xylopyranoside
O
H
C 36 H 56 O 7 (600.84). Amorphous powder, []D 25 = +36.6 (c = 0.6,

MeOH). Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor, IC 50 =
HO
3.33mmol/L, COX-2 inhibitor, IC 50 = 2.39mmol/L; control

Indomethacin, COX-1 inhibitor, IC 50 = 0.10mol/L; COX-2 inhibitor,
IC 50 = 0.60mol/L). Source: HONG YUAN CENG KONG JUN

Fomitopsis pinicola [Syn. Fomes pinicola; Polyporus pinicola]
7866 Fomitoside A
25
C35H54O8 (602.82). Amorphous powder, []D = +1.1 (c = 0.2, MeOH).

O
Source: HONG YUAN CENG KONG JUN Fomitopsis pinicola [Syn. Fomes
pinicola; Polyporus pinicola] (sporocarp: yield = 0.00055%fw). Ref: 4798.
HO
HO
OH
O
HO
HO
O
OH
OH
363
7870 Fomitoside E
7873 Fomitoside H
25-Hydroxy-3-acetoxylanost-8-en-21-oic acid 21-O--D-xylopyranoside
Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor, IC50 = 73.9mol/L,
Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor, 10g/mL, InRt = 57.2%,
COX-2 inhibitor, 10g/mL, InRt = 70.1%; control Indomethacin, COX-1
inhibitor, IC50 = 0.10mol/L; COX-2 inhibitor, IC50 = 0.60mol/L). Source:
HONG YUAN CENG KONG JUN Fomitopsis pinicola [Syn. Fomes pinicola;
O
HO
HO
O
HO
HO
OH
OH O
O
O
OH
H
OH
7874 Fomitoside I
Trametenolic acid 21-O--D-glucopyranoside C36H58O8 (618.86). Amorphous

powder, []D25 = +1.77 (c = 0.1, MeOH). Source: HONG YUAN CENG
KONG JUN Fomitopsis pinicola [Syn. Fomes pinicola; Polyporus pinicola]
7871 Fomitoside F
25
C37H58O8 (630.87). Colorless needles (MeOH), mp 185~186.6C, []D =
3.4 (c = 2.6, MeOH). Pharm: Anti-inflammatory (in vitro, COX-1 inhibitor,

10g/mL, InRt = 27.5%, COX-2 inhibitor, IC50 = 1.13mol/L; control
Indomethacin, COX-1 inhibitor, IC50 = 0.10mol/L; COX-2 inhibitor, IC50 =
HO
HO
HO
O
O
OH
0.60mol/L). Source: HONG YUAN CENG KONG JUN Fomitopsis pinicola

[Syn. Fomes pinicola; Polyporus pinicola] (sporocarp: yield = 0.010%fw).
Ref: 4798.
HO
O
HO
HO
7875 Fomitoside J
OH
Eburicoic acid 21-O--D-glucopyranoside C37H60O8 (632.89). Amorphous

powder, []D25 = +22.1 (c = 0.3, MeOH). Source: HONG YUAN CENG
KONG JUN Fomitopsis pinicola [Syn. Fomes pinicola; Polyporus pinicola]
O
O

H
HO
HO
HO
O
O
OH
7872 Fomitoside G
3-Acetoxylanosta-8,24(31)-dien-21-oic acid 21-O--D-xylopyranoside
C38H60O8 (644.9). Amorphous powder, []D25 = +5.0 (c = 0.7, MeOH). Pharm:
Anti-inflammatory (in vitro, COX-1 inhibitor, 10g/mL, InRt = 21.7%,
HO

7876 Fomlactone A
C33H50O5 (526.76). White needles (MeOH), mp 184~186C, []D 15 = +30 (c
= 0.02, CHCl3). Source: FEN ROU CENG KONG JUN Fomes cajanderi
(sporocarp: yield = 0.0018%dw). Ref: 4726.
O
O
HO
HO
O
OH
H
O
O
O
O
O
364
7877 Fomlactone B
7882 Formic acid
C31H48O4 (484.73). White needles (MeOH), mp 278~280C, []D 15 = +37 (c
Methanoic acid [64-18-6] CH2O2 (46.03). mp 8.4C, bp 100.5C. Pharm:
Astringent; corrosion. Source: BAI GUO Ginkgo biloba, BAI BU Stemona
tuberosa, QIAN MA Urtica cannabina, KUAN YE XIANG PU Typha

latifolia. Ref: 2, 658, 660.
O
O
OH
7883 Formononetin
Pratol; 7-Hydroxy-4'-methoxyisoflavone; Formonetin [485-72-3]
HO
C16H12 O4 (268.27). mp 265~266C; 257~258C; 256~257C. Pharm:

Diuretic (in clinic); estrogenic activity ; antihypercholesterolemic (male
7878 Fomlactone C
C31H46O4 (482.71). White crystals (MeOH), mp 246~250C, []D 15 = +40 (c
O
rat, hyperlipemia, due to Triton WR1339); hepatoprotective (mus primary

cultured hepatocytes, antihepatotoxin induced by D-galactosamine
(GalN), 100mol/L, InRt = (6.31.0)%, inactive, control Silybin,
100mol/L, InRt = (77.05.5)%)[4095] ; antimalarial (Plasmodium
falciparum PoW, IC50 > 50g/mL, control Chloroquine diphosphate, IC50 =
(0.0060.002)g/mL; Dd2, IC50 < 50g/mL, Chloroquine diphosphate, IC50
= (0.0630.01)g/mL)[5208]; antibacterial (Escherichia coli, MIA =
50.0g, control Chloramphenicol, MIA = 0.001g; Bacillus subtilis, MIA

= 50.0g, Chloramphenicol, MIA = 0.001g; Staphylococcus aureus,
MIA = 10.0g, Chloramphenicol, MIA = 0.001g)[3785] ; antifungal
(Candida mycoderma, MIA = 10.0g, Miconazole = MIA =
0.0001g) [3785]; antioxidant (DPPH scavenger, TLC detection limit =

7879 Fordimine
0.5g, IC50 = 960g/mL; control Quercetin, TLC detection limit < 0.05g,
[103548-82-9] C16H20N2O (256.35). Acicular crystals, mp 149~150C (dec).
IC50 = 7g/mL; Gallic acid, TLC detection limit < 0.05g, IC50 = 4g/mL;
Source: HUA NAN MA WEI SHAN Phlegmariurus fordii. Ref: 95.
Ascorbic acid, TLC detection limit < 0.10g, IC50 = 18g/mL)[3785].

Source: AO DA LI YA YAN DIAN Baptisia australis, BO TE LAN DA JI
Euphorbia portlandica (whole herb), CI GUO GAN CAO Glycyrrhiza
pallidiflora, CI MANG BING HUA Ononis spinosa, DI XIA CHE ZHOU
CAO Trifolium subterraneum, DUO MAI NAN MEI ROU DOU KOU
H
N
H
NH
Virola multinervia, GAN CAO Glycyrrhiza uralensis, GE GEN Pueraria

lobata [Syn. Pueraria thunbergiana; Pueraria pseudohirsuta], GUANG
GUO GAN CAO Glycyrrhiza glabra, HONG CHE ZHOU CAO Trifolium
7880 Foresticine
[91794-15-9] C24H39NO6 (437.58). Source: LI JIANG WU TOU Aconitum
forrestii [Syn. Aconitum likiangense]. Ref: 1521.
pratense, HUANG QI Astragalus membranaceus (dried root: mean

content of 5 origins = 0.0068%)[5519] , HUI HUI DOU Cicer arietinum,
KU SHEN Sophora flavescens [Syn. Sophora angustfolia], LUO HUA
NAN MEI ROU DOU KOU Virola caducifolia, MENG GU HUANG QI
H
O
H
H
N
H
O
O
OH
OH
OH
Astragalus mongholicus (dried root: mean content of 4 origins =

0.0032%[5508] ), MU XU Medicago sativa, SI TE WEN HUANG TAN
Dalbergia stevensonii, WU CI KE YA SHU Andira inermis (leaf), XI A
LA HUANG TAN Dalbergia cearensis, YI KA TUO YE HUANG TAN
Dalbergia ecastophyllum, ZI SUI HUAI Amorpha fruticosa, ZI TAN
Pterocarpus indicus, Baptisia spp., family Fabaceae spp., Bolusanthus
7881 Formaldehyde
speciosus (root wood), occurs in many plants. Ref: 6, 2, 6, 243, 372, 379,
Methanal [50-00-0] CH2O (30.03). mp 92C, bp 21C. Source: CU
658, 660, 1521, 3785, 4095, 5019, 5208, 5508, 5519.
vinegar, NIU BANG GEN Arctium lappa, YANG SHI CAO Achillea
millefolium. Ref: 6.
O
H
HO
365
7884 Formononetin-7-O--D-apiofuranosyl-(16)--D-glucopyranoside
7888 Formosadimer C
C27H30O13 (562.53). White powder, []D25 = +78.2 (c = 0.25, MeOH:H2O =
12-Acetoxy-7-butoxyethoxyabieta-6-yl 6,7-dehydroabieta-8,11,13-trien-
1:0.5). Source: FENG CHENG JI XUE TENG Millettia nitida var.
12-yl ether C48H70O5 (727.09). Gum, []D25 = +37.0 (c = 0.2, MeOH). Source:
hirsutissima (stem). Ref: 4455.
TAI WAN CUI BAI Calocedrus macrolepis var. formosana (bark). Ref:
4531.
HO
OO
OH
OH
OH OH
OH
7885 Formononetin-7-glucoside
Ononin; Ononoside [486-62-4] C22H22O9 (430.42). Source: GAN CAO
Glycyrrhiza uralensis (root and rhizome: mean content of 4 origins =
0.037%[5508]), GE GEN Pueraria lobata [Syn. Pueraria thunbergiana;
O
H
Pueraria pseudohirsuta], GUANG GUO GAN CAO Glycyrrhiza glabra (root
and rhizome: content = 0.032%)[5508], HUANG GAN CAO Glycyrrhiza

kansuensis (root and rhizome: content = 0.0279%[5508]), ZHANG GUO GAN
CAO Glycyrrhiza inflata (root and rhizome: content = 0.011%[5508]). Ref: 2,
660, 5508.
HO
{5,7,5'-Trihydroxy-6-(3-hydroxy-3-methylbutyl)-8-(,-dimethylallyl)-[6'''',6''''
OO
OH
-dimethylpyrano-(2'''',3'''':4',3')]}-coumaronochromone C30H32O8 (520.58).

Colorless needles, mp 221~223C. Source: TAI WAN SHAN DOU GEN
OH
OH
7889 Formosanatin A
Euchresta formosana. Ref: 1977.

O
7886 Formosadimer A
6,7-Dehydroabieta-8,11,13-trien-12-yl
HO
7-hydroxy-12-methoxyabieta-8,11,13-trien-6-yl ether C41H58O3 (598.92).
23
Gum, []D = +45.9 (c = 0.4, MeOH). Source: TAI WAN CUI BAI
Calocedrus macrolepis var. formosana (bark). Ref: 4531.
OH
HO
OH
7890 Formosanatin B
{5,7,5',4'''',5''''-Pentahydroxy-6,8-bis-(,-dimethylallyl)-[6'''',6''''-dimethyl-4'''',
OH
O
5''''-dihydropyrano-(2'''',3'''':4',3')]}-coumaronochromone C30H32O9 (536.58).
Yellow needles, mp 243~245C, []D24 = 40 (c = 0.05, CHCl3). Source: TAI
H
H
WAN SHAN DOU GEN Euchresta formosana. Ref: 1977.
OH
7887 Formosadimer B
HO
7-Butoxyethoxy-12-hydroxyabieta-6-yl
6,7-dehydroabieta-8,11,13-trien-12-yl ether C46H68O4 (685.05). Gum, []D25 =
HO
+85.8 (c = 0.3, MeOH). Source: TAI WAN CUI BAI Calocedrus macrolepis
OH
var. formosana (bark). Ref: 4531.
OH
7891 Formosanatin C
{5,5'-Dihydroxy-8-(,-dimethylallyl)-[6'',6''-dimethyl-4'',5''-dihydropyrano-(2
'',3'':7,6)]-[6'''',6''''-dimethylpyrano-(2'''',3'''':4',3')]}-coumaronochromone
O
C30H30O7 (502.57). Pale yellow Needles, mp 248~250C. Source: TAI WAN

SHAN DOU GEN Euchresta formosana. Ref: 1977.
O
HO
O
H
H
O
OH
OH
366
7892 Formosanatin D
7896 20-Formylbenzo[6,7]indolizino[1,2-b]quinolin-11 (13H)-one
{5,5'-Dihydroxy-8-[6'',6''-dimethyl-4'',5''-dihydropyrano-(2'',3'':7,8)]-[6'''',6''''-
C20H12N2O2 (312.33). Source: XI SHU Camptotheca acuminata. Ref: 4097.
dimethylpyrano-(2'''',3'''':4',3')]}-coumaronochromone C25H22O7 (434.45).

Yellow needles (CHCl3), mp 246~248C. Source: TAI WAN SHAN DOU
GEN Euchresta formosana. Ref: 1977.
O
O
7897 3-Formylcarbazole
C13H9NO (195.22). Pharm: Antitubercular (MIC > 128g/mL, control
OH
OH
Rifampin, MIC = (0.0400.017)g/mL)[5072]; cytotoxic (Vero, IC 50 >
102g/mL, Rifampin, IC50 = 100g/mL)[5072]; antibacterial (Mycobacterium

tuberculosis, MIC = 100g/mL, control Isoniazide, MIC = 0.040~0.090g/mL,
7893 Formosaninol
20
C40H56O4 (600.89). Colorless solid, []D = +36.3 (c = 0.48, CHCl3). Source:

RI BEN LIU SHAN Cryptomeria japonica (black heartwood). Ref: 4268.
Kanamycin sulfate, MIC = 2.0~5.0g/mL)[5367]; antifungal (Candida albicans,

IC50 = 13.6g/mL, control Amphotericin, IC50 = 0.01g/mL)[5367]. Source:
SHAN HUANG PI Clausena excavata, YING MAO XIAO YUN MU
Micromelum hirsutum (stem cortex). Ref: 5072, 5367.
O
OH
HO
O
N
H
7894 N-Formylanonaine
7898 1-Formyl--carboline
C18H15NO3 (293.33). Pharm: Platelet aggregation inhibitor (rat blood:
[20127-63-3] C12H8N2O (196.21). Orange crystals, mp 200~202C. Source:
2~5mol/L ADP-induced, IC50 = 930mol/L, control Acetylsalicylic acid,
KU SHU PI Picrasma quassioides [Syn. Picrasma ailanthoides]. Ref: 12.
IC50 > 1000mol/L; 2~5g/mL collagen-induced, IC50 = 6.9mol/L,

Acetylsalicylic acid, IC50 = 420mol/L; 1~4mol/L epinephrine-induced with
threshold concentration of collagen (0.8~1.0g/mL), IC50 = 0.24mol/L,
N
H
Acetylsalicylic acid, IC50 = 53mol/L; 10~40mol/L AA-induced with

Acetylsalicylic acid, IC50 = 66mol/L; 1~5mol/L U46619-induced with
7899 N-Formylcorydamine
Acetylsalicylic acid, IC50 = 340mol/L; 1~2mol/L hmn U46619 in 1mmol/L
[In DNP] C21H18N2O5 (378.39). mp 159.5~160.5C. Source: ZI HUA YU
acetylsalicylic acid induced, IC50 > 100mol/L, control Pentolamine, IC50 >
DENG CAO Corydalis incisa. Ref: 6.
[5381]
100mol/L, control Yohimbine, IC50 > 100mol/L)
. Source: RI BEN
O
HOU PO Magnolia obovata (leaf). Ref: 5381.
O
N
H
O
N
O
O
7900 N-Formylcytisine
7895 p-Formyl benzoic acid
[53007-06-0] C12H14N2O2 (218.26). Colorless acicular crystals, mp
C8H6O3 (150.14). Source: TAI WAN FU RONG Hibiscus taiwanensis. Ref:
174~176C, []D = 233 (c = 0.16, EtOH). Source: MU MA DOU
2529.
Thermopsis lanceolata. Ref: 699.

O
O
OH
H
N
O
O
367
7901 N-Formyl-N-deacetylcolchicine
7906 1-Formyl-3-hydroxyneogrifolin
C21H23NO6 (385.42). mp 264~266C. Source: CAO BEI MU Iphigenia indica.
C23H32O4 (372.51). Yellow needles, mp 83~84C. Source: RE BEN MO GU
Ref: 6.
Albatrellus ovinus. Ref: 2005.
N
H
O
HO
OH
OH
O
O
7902 14-Formyldihydrorutaecarpine
[68353-23-1] C19H15N3O2 (317.35). Source: WU ZHU YU Evodia rutaecarpa
(dried and almost ripe fruit: content scope of 7 origins = trace~0.21%, mean
content = 0.04%[5508]). Ref: 1521, 5508.
N
H H
7907 3-Formyl-6-methoxycarbazole
C14H11NO2 (225.25). Pharm: Antitubercular (MIC = (42.30.5)g/mL,
control Rifampin, MIC = (0.0400.017)g/mL); cytotoxic vero, IC50 =
101g/mL, Rifampin, IC50 = 100g/mL)[5072]. Source: YING MAO XIAO
YUN MU Micromelum hirsutum (stem cortex). Ref: 5072.
N
H
7903 3'-Formyl-4',6'-dihydroxy-2'-methoxy-5'-methylchalcone
7908 1-Formyl-4-methoxy--carboline
C18H16O5 (312.33). Orange yellow needles (MeOH), mp 123~124C. Source:
Kumujancine [92631-69-1] C13H10N2O2 (226.24). Yellowish needle crystals,
SHUI RONG Cleistocalyx operculatus (bud). Ref: 3768.
mp 209~210C. Source: KU MU Picrasma quassioides [Syn. Picrasma

ailanthoides]. Ref: 12.
O
O
HO
OH
N
H
7904 8-Formyl-7-hydroxycoumarin

7909 8-Formyl-7-methoxycoumarin
(viability = 60%), -Carotene, EBV-EA-positive cells = (34.31.1)%
Source: YOU PU TAO YPU ZA JIAO ZHONG Citrus grandis cv. x Citrus
paradisi. Ref: 5048.
Source: CHENG ZI Citrus junos, Citrus rugulosa, Citrus sulcata. Ref: 5048.
HO
O
O
7905 (2S)-8-Formyl-5-hydroxy-7-methoxy-6-methylflavanone
C18H16O5 (312.33). Yellow needles (MeOH), mp 154~155C, []D25 = 2.4 (c
7910 1-Formylneogrifolin
= 0.01, MeOH). Source: SHUI RONG Cleistocalyx operculatus (bud). Ref:
C23H32O3 (356.51). White plates, mp 98~102C. Source: RE BEN MO GU
3768.
Albatrellus ovinus. Ref: 2005.
O
O
O
OH
HO
OH
368
7911 17-Formyloxy-3-acetyloxy-28-nor-urs-12-ene
7915 Forrestin A
C32H50O4 (498.75). Colorless needles (MeOH), mp 203~204C, [] D20 = +59
(c = 0.05, CHCl3). Pharm: Cytotoxic (HL-60 cells, IC50 = (8324)mol/L).
ZI E XIANG CHA CAI Isodon forrestii. Ref: 4067.
Source: ZHI ZHUANG E AN Eucalyptus cladocalyx (leaf). Ref: 5259.

O
O
O
O
O
H
HO
O
O
O
O
7912 3-Formyloxyresibufogenin
7916 Forrestin B
C25H32O5 (412.53). Colorless solid, []D21 = +12.0 (c = 0.1, CH3OH). Pharm:
C24H36O8 (452.55). mp 228~229C. Source: ZI E XIANG CHA CAI Isodon
Cytotoxic (in vitro, KB, IC50 = 3.4g/mL; HL-60, IC50 = 1g/mL; MH-60,
forrestii. Ref: 4067.
IC50 = 8.1g/mL; BXPC3, IC50 = 1.6g/mL; MCF7, IC50 = 0.6g/mL; SF268,

HO
OH
IC50 = 0.38g/mL; NCI-H460, IC50 = 0.53g/mL; KM20L2, IC50 =

0.54g/mL; DU145, IC50 = 0.42g/mL). Source: CHAN SU Bufo bufo
gargarizans; Bufo melanostictus. Ref: 3082.
H
O
OH
OH
O
7917 Forrestin C
C26H38O9 (494.59). mp 291~292C, []D = 29.44 (c = 0.523, MeOH).
H
O
H
Source: XIAN HUA XIANG CHA CAI Rabdosia adenantha (leaf: yield =
O
0.00073%dw), ZI E XIANG CHA CAI Isodon forrestii. Ref: 4067, 4640.
7913 6-Formylumbelliferone

H
HO
OH
OH
O
7918 Forrestin D
C28H40O10 (536.63). mp 136~138C, []D = 46.01 (c = 0.489, MeOH).
Source: Citrus medica var. etrog. Ref: 5048.
Source: ZI E XIANG CHA CAI Isodon forrestii. Ref: 4067.
O
O
OH
HO
O
O
HO
7914 Forrestiin A
[163597-22-6] C20H26O4 (330.43). Acicular crystals, []D19 = +105.6 (c =
0.71, chloroform). Pharm: Cytotoxic (KB in vitro, IC50 = 18.96g/mL).
Source: YUAN BAN JIANG HUA Hedychium forrestii. Ref: 322.
O
O
7919 Forrestin E
C26H38O9 (494.59). mp 251~254C. Source: ZI E XIANG CHA CAI Isodon
forrestii. Ref: 4067.
O
O
O
OH
OH
O
HO
O
OH
O
369
7920 Forrestin F
7925 Forsythoside B
C34H44O19 (756.72). Colorless amorphous powder, []D20 = 66 (c = 0.1,
ZI E XIANG CHA CAI Isodon forrestii. Ref: 4067.
MeOH). Pharm: Antioxidant (in vitro inhibits LDL peroxidation,

Cu2+-induced and AAPH-induced)[5370]; inhibits minimally oxidized
LDL-induced cellular toxicity (cultured bovine aortic endothelial cells,
BAEC)[5370]; antioxidant (DPPH free radical scavenger, IC50 = 113mol/L,

O
H
O
O
O
control Ascorbic acid IC50 = 129mol/L)[5449]; antitrypanosomal
(Trypanosoma b. rhodesiense, IC50 = 5.8g/mL, control Melarsoprol, IC50 =

0.00098g/mL; Trypanosoma cruzi, IC50 > 90g/mL, control Benznidazole,
IC50 = 1.06g/mL)[5009]; antileishmanial (Leishmania donovani, IC50 =
11.4g/mL, control Miltefosine, IC50 = 0.102g/mL)[5009]; antimalarial
7921 Forrestin G
C26H34O7 (458.56). mp 204~206C, []D = 69.88 (c = 0.508, MeOH).
Source: ZI E XIANG CHA CAI Isodon forrestii. Ref: 4067.
O
0.0022g/mL)[5009]; cytotoxic (L6, IC50 = 70.1g/mL, control

Podophyllotoxin, IC50 = 0.008g/mL)[5009]. Source: LIAN QIAO Forsythia
suspensa, OU XIA ZHI CAO Marrubium vulgare (aerial parts), ZI HUA
GUAN MAO RUI HUA Verbascum wiedemannianum, ZONG KUI CAO

SU Phlomis brunneogaleata. Ref: 2, 5009, 5370, 5449.
H
O
(Plasmodium falciparum, IC50 > 50g/mL, control Artemisinin, IC50 =
HO
7922 Forsythenside A
OH OH
C22H26O10 (450.45). Source: LIAN QIAO Forsythia suspensa. Ref: 8.

OH
HO
OH
OH
OH OHO
OO
OH
OO
OH
HO
OH
OH
O
OH
OH
7923 Forsythenside B
7926 Forsythoside C
C14H16O5 (264.28). Source: LIAN QIAO Forsythia suspensa. Ref: 8.
Suspensaside C29H36O16 (640.60). Powder, mp 177~181C, []D18 = 18.7

(c = 1.7, MeOH). Pharm: Antibacterial; free radical scavenger; inhibits
metabolism of arachidonic acid (in leucocytes); 5-lipoxygenase inhibitor
O
H
(rat, peritoneum cells); cAMP phosphodiesterase inhibitor; used in
treatment of asthma and allergic disease. Source: LIAN QIAO Forsythia
suspensa. Ref: 47, 658.
7924 Forsythoside A
OH
Forsythiaside [79916-77-1] C29H36O15 (624.60). Pale-yellowish powder + 2H2O, mp

144~150C, []D20 = 18.6 (EtOH). Pharm: Immunomodulator (selectively inhibits
OH
OH O O
OO
HO
OH
OH OH
formation of 5-HETE and leukotriene LTB4, which are products of 5-lipoxygenase,

IC50 =1.92mol/L and 1.01mol/L respectively); 5-HETE production inhibitor (IC50 =
O
OH
2.50mol/L); antiallergic; antiasthmatic; cAMP phosphodiesterase inhibitor (in vitro,
OH
OH
IC50 = 110mol/L); leucine aminopeptidase inhibitor (competitive, Ki = 8.0mol/L);

antibacterial (strong action for 11 pathogenic bacteria, including plant pathogenic
7927 Forsythoside D
bacteria); free radical scavenger; 5-lipoxygenase inhibitor (rat peritoneum cells and
Decaffeoyl forsythoside C [84233-74-9] C20H30O13 (478.45). []D = 30.5
hmn leucocyte in vitro). Source: CHAO XIAN LIAN QIAO Forsythia koreana, GAN
(methanol). Pharm: Antibacterial (Staphylococcus aureus, MIC 2mmol/L).
DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa f. huechingensis],
Source: LIAN QIAO Forsythia suspensa. Ref: 1037.
LIAN QIAO Forsythia suspensa (green fruit: mean content = 1.31%, ripe fruit: mean
content = 0.64%[5508]). Ref: 2, 47, 658, 1639, 1640, 1641, 1642, 5508.
OH
OH
OH O O
OO
HO
OH
OH OH
O
O
OH
OH
OH
OH O O
H
OO
OH
OH OH
OH
OH
OH
OH
370
7928 Forticine
7932 Foveolin B
(20S,22S,25S)-5-Cevanine-3,6-diol C27H45NO2 (415.67). Colorless needle,
[220358-68-9] C31H54O5 (506.77). Source: DA YE SHU LAN Aglaia
mp 221~223C (dec), []D23 = 52 (c = 0.5, CHCl3). Pharm: AChE inhibitor
elliptifolia (leaf: yield = 0.00020%dw), FENG CHAO MI ZI LAN Aglaia
(IC50 > 500mol/L, control Eserine, IC50 = (0.410.01)mol/L); BChE
foveolata. Ref: 1521, 3031.
inhibitor (IC50 = (100.50.5)mol/L, control Eserine, IC 50 =

(0.860.01)mol/L). Source: XI BEI MU Fritillaria imperialis (bulb). Ref:
4217.
OH
O
HO
H
N
H
[114926-96-4] C21H24O5 (356.42). Source: ROU DOU KOU Myristica

fragrans. Ref: 909, 1521.
H
H
7933 Fragransol C
HO
HO
OH
HO
7929 Fortuneine
[87340-25-9] C20H25NO3 (327.43). Source: SAN JIAN SHAN Cephalotaxus

fortunei. Ref: 2.
7934 Frameroside
C27H38O15 (602.59). Colorless amorphous powder, [] D27 = 134 (c = 1.09,
MeOH). Source: MEI GUO BAI CEN Fraxinus americana (leaf). Ref: 5091.
N
OH
OO
O
OH
7930 Fortunellin
[20633-93-6] C28H32O14 (592.56). mp 214~216C. Source: JIN JU Fortunella
HO
margarita, JIN DAN Fortunella crassifolia. Ref: 6, 660.
OO
OH
OH
OH
O
HO
OO
OH
OH
OH O O
7935 Franchetine

OH
H
OH OH
OH
O
O
7931 Fouquierone
Dammar-25-ene-20,24-diol-3-one C30H50O3 (458.73). White powder, []D25 =
+58 (c = 0.16, CHCl3). Source: YA DAN ZI Brucea javanica [Syn. Brucea
sumatrana; Rhus javanica] (stem cortex). Ref: 4111.
H
O
7936 Franchitine
[88661-42-1] C31H41NO6 (523.68). White amorphous powder. Source: GONG
OH
H
OH
BU WU TOU Aconitum kongboense. Ref: 2211, 1521.

H
O
O
371
7937 Frangufoline
7942 Fraxetin
Sanjoinine A [19526-09-1] C31H42N4O4 (534.70). mp 244C. Source: MIAN
[574-84-5] C10H8O5 (208.17). mp 228C. Pharm: Antibacterial (Bacillus
ZAO Ziziphus mauritiana. Ref: 6.
dysenteriae, used in treatment of infant bacillary dysentery). Source: MAO

GUO QI Acer nikoense (stem cortex), XIAO YE CEN Fraxinus bungeana,
HUA BAI LA SHU Fraxinus ornus, XI MA BAI LA SHU Fraxinus

O
HN
O
floribunda, RI BEN QI YE SHU Aesculus turbinata, OU ZHOU QI YE SHU
O
N
H
N
H
Aesculus hippocastanum, BAI LA SHU Fraxinus chinensis. Ref: 2, 658, 660,

4304.
7938 Frangulanine
HO
OH
[25350-22-5] C28H44N4O4 (500.69). mp 275~277C. Pharm: Laxative. Source:

OU SHU LI Rhamnus frangula [Syn. Frangula alnus], ZHI JU GEN Hovenia
7943 Fraxidin
dulcis. Ref: 6, 658, 660.
O
O
HN
O
O
N
H
N
H
OH
7944 Fraxin
N
Fraxoside; Paviin; Fraxetin-8-glucoside [524-30-1] C16H18O10 (370.32). mp

205C, , easily soluble in hot water, hot EtOH, slightly soluble in cold water,
7939 Frangulin A
[521-62-0] C21H20O9 (416.39). Pharm: Laxative. Source: YAO SHU LI
Rhamnus cathartica, OU SHU LI Rhamnus frangula [Syn. Frangula alnus].
Ref: 658.
cold ether, insoluble in ether[5507]. Pharm: Antibacterial; antitussive (dispels

phlegm); diuretic; -hexosaminidase inhibiter inactive (RBL-2H3 cells,
inhibits release of -hexosaminidase, 100mol/L, InRt = (7.74.4)%)[4304].
Source: HUA BAI LA SHU Fraxinus ornus, JIAN YE CEN Fraxinus
OH
OH
szaboana [Syn. Fraxinus chinensis var. acuminata], LA MEI HUA

Chimonanthus fragrans [Syn. Chimonanthus praecox], LIU YE CEN
OH
Fraxinus stylosa, MAO GUO QI Acer nikoense (stem cortex), OU ZHOU
OO
BAI LA SHU Fraxinus excelsior[5507], OU ZHOU QI YE SHU Aesculus
hippocastanum, QIN LING BAI LA SHU Fraxinus paxiana[5507], TU ER QI
OH OH
SI TAN BAI LA SHU Fraxinus potamophila, XIAO YE CEN Fraxinus
7940 Frangulin B
bungeana, Symphoricarpos sp., Campanula sp. Ref: 2, 658, 660, 4304, 5507.
[14101-04-3] C20H18O9 (402.36). Pharm: Laxative. Source: YAO SHU LI

Rhamnus cathartica, OU SHU LI Rhamnus frangula [Syn. Frangula alnus].
Ref: 658.
OH
OH
HO
HO
OO
OH
HO
OH
O
O
OH
7945 Fraxinellone
OH OH
[28808-62-0] C14H16O3 (232.28). mp 108~110C; 120C. Pharm: Anti-fertility
7941 Fraxamoside
agent (rat, orl, 75mg/(kgd), pregnant rate = 6/10); platelet aggregation
C25H30O13 (538.51). Colorless amorphous powder, [] D22 = 137 (c = 0.12,
inhibitor; antihypertensive (relaxes aortal contraction induced by K+ and Ca2+,
MeOH). Source: MEI GUO BAI CEN Fraxinus americana (leaf). Ref: 5091.
ID50 25mol/L); coronary vasodilator (calcium selective antagonist). Source:
O
HO
O
O
BAI XIAN PI Dictamnus dasycarpus, KU LIAN PI Melia azedarach. Ref: 6,

1644, 1645, 1646.
H
H
HO
O
OO
OH
OH
O
OH
372
7946 Friedelan-1,3-dion-24-al
7950 Friedelan-3-ol
C30H46O3 (454.70). Source: SUO LA MU Salacia prinoides [Syn. Salacia
[5085-72-3] C30H52O (428.75). mp 302~304C. Pharm: Antifungal;
chinensis]. Ref: 6.
anti-inflammatory. Source: TIAO JING CAO Euonymus japonicus, DONG

FENG CAI Doellingeria scaber [Syn. Aster scaber], HE AN ZE LAN
Eupatorium riparium, HUO YANG LE Euphorbia antiquorum, LIANG YE
RONG Ficus nitida, MEI LI YIN BEI TENG Argyreia speciosa, QIU FENG
MU Bischofia javanica [Syn. Bischofia trifoliata], TIAN LAN ZE LAN
Eupatorium azureum, XUE TONG Macaranga tanarius, YANG YE YIN BEI
TENG Argyreia populifolia. Ref: 6, 658.

O
O
7947 Friedelan-1,3-dion-7-ol
C30H48O3 (456.72). Source: SUO LA MU Salacia prinoides [Syn. Salacia

HO
chinensis]. Ref: 6.
7951 Friedelan-3-one
Friedelin [559-74-0] C30H50O (426.73). Colorless thin acicular crystals, mp
O
257~264C, []D28 = 14.1 (c = 0.07, CHCl3). Pharm: Anti-inflammatory;
NFAT transcription factor inhibitor inactive (IC50 > 50mol/L, positive

control Cyclosporin A, IC50 = (0.310.01)mol/L)[4511]; cytotoxic (P388, ED50 =
OH
14.61g/mL, control Mithramycin, ED50 = 0.58g/mL; A549, ED50 =

30.72g/mL, Mithramycin, ED50 = 0.073g/mL; HT29, ED50 = 17.30g/mL,
Mithramycin, ED50 = 0.076g/mL)[5421] . Source: BIAN TAO Mangifera
persiciformis, CHAO XIAN LUO WAN Gymnaster koraiensis (leaf),
7948 Friedelane-3,7-dione
C30H48O2 (440.72). White powder, mp 286C. Source: Drypetes molunduana
(stem). Ref: 3989.
CHUAN DANG SHEN Codonopsis tangshen, CHUAN LI GUO Pyrus

pashia, DA FEI YANG CAO Euphorbia hirta, DANG SHEN Codonopsis
pilosula (dried root: mean content = 0.0095%[5508]), HAI TANG GUO
Calophyllum inophyllum (root cortex and nut), HEI XIAN TIAO TENG
HUANG Garcinia nigrolineata (leaf)[4735], HUANG HUA HAO Artemisia
annua, HUI BAO HAO Artemisia roxbugiana, HUO XIANG Agastache
rugosus, KUAI JING MA LI JIN Asclepias tuberosa, KUO JIA HE HUAN
Albizzia lebbeck, LONG XU CAO Poa sphondylodes, LU BIAN QING
Clerodendron cyrtophyllum, MANG GUO Mangifera indica, MAO LIAN
HAO Artemisia vestita, MENG GU LI Quercus mongolica, MO ZHI JIAO
GU CUI Casearia membranacea (stem), NAN ZHU ZI Vaccinium bracteatum,

QIU HUA DANG SHEN Codonopsis subglobosa, QUE MEI TENG
Sageretia theezans [Syn. Sageretia thea], QUN DAI CAI Undaria pinnatifida,
7949 Friedelane-3-one-29-ol
RI BEN HUANG BAI Phellodendron japonicum (leaf), SHI LIU PI Punica
C30H50O2 (442.73). Pharm: DPPH scavenger inactive (for 40mol/L DPPH
granatum, SU HUA DANG SHEN Codonopsis pilosula var. modesta [Syn.
radical, SC50 > 40mol/L)[4378]. Source: SUO LA MU Salacia prinoides [Syn.
Codonopsis modesta] (dried root: mean content = 0.0162%)[5508], TAI BAI
Salacia chinensis] (stem). Ref: 4378.
HUA Cladonia stellaris [Syn. Cladonia alpestris], TUN XING GUO Pygeum
topengii, XIAO SHE ZI WAN Aster albescens, YA ZHI CAO Commelina
OH
communis, ZI WAN Aster tataricus, occurs in many plants. Ref: 2, 447, 474,
503, 505, 515, 550, 572, 600, 611, 658, 660, 3866, 4502, 4511, 4735, 5421,
5501, 5508.
O
H
373
7952 Friedelan-3-yl acetate
7957 Fritillarizine
C32H54O2 (470.79). mp 317~319C. Source: QIU FENG MU Bischofia
[76733-86-3] C27H43NO2 (413.65). mp 141.5~143.0C, []D = 18.6 (c = 1.0,
javanica [Syn. Bischofia trifoliata]. Ref: 6.
CHCl3). Source: ZHE BEI MU Fritillaria verticillata var. thunbergii [Syn.

Fritillaria thunbergii]. Ref: 2201.
H
H
O
H
OH
H
H
H
HO
7953 1-Friedelen-3-one
C30H48O (424.72). mp 262~263C. Source: SUO LA MU Salacia prinoides
[Syn. Salacia chinensis]. Ref: 6.
7958 Fritillaziebinol
ent-Kauran-16-hydroxy-17-chloride C20H23ClO (324.94). Colorless square
crystals, mp 153~154C. Source: ZI HUA E BEI BEI MU Fritillaria ebeiensis
var. purpurea. Ref: 833.
Cl
OH
O
H
7954 D:C-Friedomadeir-7-en-3-yl acetate
C32H52O2 (468.77). White granular crystals, mp 213~214C, []D = 61.5 (c

= 0.75, CHCl3). Source: YOU AN DI JIN Euphorbia stygiana. Ref: 3383.
7959 Fritillebeinol
ent-3-Acetoxy-kauran-16,17-diol C22H36O4 (364.53). Colorless acicular
crystals, mp 163~164C. Source: E BEI BEI MU Fritillaria ebeiensis. Ref:
H
O
827.
H
O
OH
OH
H
O
7955 D-Friedomadeir-14-en-3-yl acetate
C32H52O2 (468.77). White powder, mp 220~221C, []D = +23.4 (c = 0.6,

CHCl3). Source: YOU AN DI JIN Euphorbia stygiana. Ref: 3383.
7960 Fritillebic acid

HU BEI BEI MU Fritillaria hupehensis. Ref: 2182.
H
O
H
O
OH
7956 D:C-Friedo-urs-7-en-3-one
H
O
C30H48O (424.72). Colorless needles, mp 212~214C, []D25 = 4.1 (c = 0.4,
CHCl3). Pharm: Antimutagenic (E. coli PQ37, antigenotoxicity test, for
7961 Fritillebin A
mutagen MNNG shows 20% reduction of induction factor, for mutagen NQO,
shows 25% reduction of induction factor)[4459]. Source: ZAO JIA CI Gleditsia
E BEI BEI MU Fritillaria ebeiensis. Ref: 578, 2182.
sinensis [Syn. Gleditsia horrida] (thorn). Ref: 4459.

O
O
H
O
H
OH
H
O
H
374
7962 Fritillebin B
7967 Fritillebinide C
C42H66O4 (634.99). Source: E BEI BEI MU Fritillaria ebeiensis. Ref: 906.

O
O
O
H
O
H
O
OH
H
O
7963 Fritillebin C
7968 Fritillebinide D
C44H68O6 (693.03). Colorless needles (EtOAc), mp 247~249C. Source: ZI
HUA E BEI BEI MU Fritillaria ebeiensis var. purpurea. Ref: 4806.
O
O
O H
OH
H
7969 Fritillebinide E
7964 Fritillebin D
C40H64O3 (592.95). mp 231~233C, []D = 86.4 (c = 0.16, CHCl3). Source:
C44H68O6 (693.03). Colorless needles (EtOAc), mp 247~248C. Source: ZI
HUA E BEI BEI MU Fritillaria ebeiensis var. purpurea. Ref: 4806.
25
O
O
H
O
OH
H
7970 6'-O--D-Fructofuranosylswertiamarin
7965 Fritillebinide A
ent-Kauran-16,17-acetal ent-16-kauran-17(S)-aldehyde C40H64O2 (576.95).
Source: RI BEN ZHANG YA CAI Swertia japonica. Ref: 2573.
Source: ZI HUA E BEI BEI MU Fritillaria ebeiensis var. purpurea. Ref: 682,
906.
OH
HO
H
H
O
HO
OH
H
O
OH
O
OH
OH
OH
7971 Fructose
C6H12O6 (180.16). mp L (+) 101~103C, D() 102~104C (dec). Pharm:
7966 Fritillebinide B
C42H66O4 (634.99). Source: ZI HUA E BEI BEI MU Fritillaria ebeiensis var.
purpurea. Ref: 906.
Provides energy and restores body fluid (for patients with diabetes and
hepatitis). Source: REN SHEN Panax ginseng [Syn. Panax schinseng],
DANG SHEN Codonopsis pilosula, YAO YONG PU GONG YING
Taraxacum officinale, XI SHU Camptotheca acuminata. Ref: 2, 660, 4097.
H
O
O OH
HO
H
H
H
HO
OH
OH
375
7972 Fruticolone
7976 (24S,25R)-1-[(-D-Fucopyranosyl)oxy]-6-hydroxy-3,5-cyclo-
C22H30 O6 (390.48). Pharm: Insect antifeedant (fifth instar larvae of
spirostan-24-yl -D-glucopyranoside
Spodoptera littoralis, dual-choice feeding assays, dose = 10g/cm2, FR50
= 0.690.11). Source: GUAN CONG XIANG KE KE Teucrium fruticans.
Source: DUO ZHI LONG XUE SHU Dracaena surculosa (whole herb). Ref:
Ref: 3761.
4216.
O
HO
O O
OH
OH
H
O
HO
OH
O
OH
OH
OH
OH
O
O
7977 (25S)-1-[(-D-Fucopyranosyl)oxy]-6-hydroxy-22-methoxy3,5-cyclofurostan-26-yl -D-glucopyranoside

7973 Frutinone A
Source: DUO ZHI LONG XUE SHU Dracaena surculosa (whole herb). Ref:
[38210-27-4] C16H8O4 (264.24). Pharm: Antifungal (Cladosporium
4216.
cucumerinum). Source: GUAN MU YUAN ZHI Polygala fruticosa. Ref:

OO
HO
658.
OH
OH
HO
OH
O O
OH
O
H
OH
OH
7974 Fucaxanthone A
C29H32O6 (476.57). Pharm: Antioxidant (DPPH scavenger, IC50 > 200mol/L,
7978 Fucosterol
control BHT, IC50 = 5.10g/mL; crude latex of Garcinia cowa, IC 50 =
Stigmasta-5,24(28)E-dien-3-ol [17605-67-3] C29H48O (412.71). mp 124C.
13.20g/mL). Source: YUN NAN SHAN ZHU ZI Garcinia cowa (latex). Ref:
Pharm: Antihypercholesterolemic (reduces the level of cholesterol in serum);
5281.
antithrombotic; ACE inhibitor (endothelial cells, inhibits synthesis of

glucocorticoid receptor). Source: QUN DAI CAI Undaria pinnatifida, SHUI
LONG GU Polypodium niponicum, YE ZI YOU Cocos nucifera. Ref: 6, 660,
1601, 1602, 1603.
H
OH
HO
7975 L-Fucitol
C6H14O5 (166.18). Amorphous powder, []D21 = 5 (c = 0.1, H2O). Source:
GE LU ZI Carum carvi. Ref: 1926.
HO
7979 Fucoxanthin
[3351-86-8] C41H56O6 (644.90). Pharm: Antineoplastic (mus, inhibits
occurrence of cutaneum carcinoma and duodenum carcinoma). Source: FAN
QIE Lycopersicon esculentum. Ref: 1521, 1582.
H
HO
HO
H
OH
H
H
H
OH
OH
H
O
OH
OH
O
376
7980 Fugapavine
7984 Fukanefuromarin G
Mecambrine [1093-07-8] C18H17NO3 (295.34). Pharm: Eclamptogenic (high
2,3-Dihydro-7-methoxy-2R*,3R*-dimethyl-2-[4-methyl-5-(4-methyl-2-furyl)-
dose); increases blood pressure (animal model); slows heart rate (animal
3(E)-pentenyl]-furo[3,2-c]coumarin C25H28O5 (408.50). Colorless oil, []D23 =
model); respiratory stimulant (animal model); LD50 (mus) = 4.1mg/kg. Source:
8.9 (c = 0.18, MeOH). Pharm: NO production inhibitor (macrophage-like
CHANG GUO YING SU Papaver dubium, WEI ER SHI LV RONG HAO
cell line RAW264.7 activated by LPS/IFN-, IC50 = (27.32.3)mol/L);
Meconopsis cambrica, YI XIAN YING SU Papaver fugax. Ref: 658.
cytotoxic inactive (MTT assay, 3~100mol/L, did not demonstrate any

significant cytotoxicity upon LPS/IFN- treatment for 24h.). Source: FU
KANG A WEI GEN Ferula fukanensis. Ref: 2574.

N
7981 Fugaxin
12,14-Dihydroxy-2,3-(tetrahydro-3',5'-dihydroxy-4'-methoxy-6'-methyl-
7985 Fukanemarin B
2H-pyran-2',4'-diylbisoxy)-card-4,20-dienolide C30H42O10 (562.66). Whitish
4-Hydroxy-7-methoxy-3-[1,2,6-trimethyl-7-(4-methyl-2-furyl)-hepta-2(E),5(E
amorphous. Source: YI XIAN HAI CONG Urginea fugax (bulb). Ref: 3871.
)-dienyl]-coumarin C25H28O5 (408.50). Yellow oil, []D23 = 0 (c = 0.23,

MeOH). Pharm: NO production inhibitor (macrophage-like cell line
RAW264.7 activated by LPS/IFN-, IC50 = (30.21.7)mol/L); inhibits the

inducible nitric oxide synthase (iNOS) gene expression (LPS/IFN- treatment
OH
increased the level of iNOS mRNA expression, and the compound inhibits
HO
O
H
OH
O
this increase, dose-dependent manner); cytotoxic inactive (MTT assay,
3~100mol/L, did not demonstrate any significant cytotoxicity upon
OH
LPS/IFN- treatment for 24h.). Source: FU KANG A WEI GEN Ferula
fukanensis. Ref: 2574.
7982 Fukanefuromarin E
OH
2,3-Dihydro-7-methoxy-2S*,3R*-dimethyl-3-[4-methyl-5-(4-methyl-2-furyl)-

2.0 (c = 0.36, MeOH). Pharm: NO production inhibitor (macrophage-like
inhibits the inducible nitric oxide synthase (iNOS) gene expression
(LPS/IFN- treatment increased the level of iNOS mRNA expression, and the
compound inhibits this increase, dose-dependent manner); cytotoxic inactive
7986 Fukinanolide
[19906-72-0] C15H22O2 (234.34). mp 80.5~80.6C. Source: FENG DOU CAI
H
(MTT assay, 3~100mol/L, did not demonstrate any significant cytotoxicity

upon LPS/IFN- treatment for 24h.). Source: FU KANG A WEI GEN Ferula
fukanensis. Ref: 2574.
7987 Fukinolic acid

[50982-40-6] C20H18O11 (434.36). Source: FENG DOU CAI Petasites
japonicus. Ref: 6.
OH
HO
7983 Fukanefuromarin F
O
2,3-Dihydro-7-methoxy-2R*,3R*-dimethyl-3-[4-methyl-5-(4-methyl-2-furyl)-

cytotoxic inactive (MTT assay, 3~100mol/L, did not demonstrate any
significant cytotoxicity upon LPS/IFN- treatment for 24h.). Source: FU

S
O
O
OH
OH
[18456-03-6] C21H28O6S (408.52). mp 207C. Source: FENG DOU CAI
O
HO
7988 S-Fukinolide
KANG A WEI GEN Ferula fukanensis. Ref: 2574.

O
OH
HO

+41.7 (c = 0.14, MeOH). Pharm: NO production inhibitor (macrophage-like
377
7989 Fukinolide
7994 Fulvine
[18455-98-6] C22H30O6 (390.48). mp 101~102C. Source: FENG DOU CAI
[6029-87-4] C16H23NO5 (309.37). Prismatic crystals (acetone), mp 212~213C,
[]D20 = 50.8 (c = 1, chloroform); hydrochloride: colorless prismatic crystals,

mp 285C (dec); bitter acid salt: yellow acicular crystals, mp 185C (dec).
O
O
Pharm: Antineoplastic (rat, Walker carcinoma); toxic (hepatic and pulmonary
toxicity); mutagen (drosophila); similar action with narceine (rat and gpg,
ileum). Source: AN HUANG ZHU SHI DOU Crotalaria fulva, MA DU LA

ZHU SHI DOU Crotalaria madurensis, YUAN ZHUI ZHU SHI DOU
O
Crotalaria paniculata, ZOU BO ZHUANG ZHU SHI DOU Crotalaria
crispata. Ref: 658.
7990 Fukinone
HO
[19593-06-7] C15H24O (220.36). bp 97C/0.8mmHg. Source: FENG DOU

CAI Petasites japonicus. Ref: 6.
H
O
O
7995 Fulvotomentoside A
C58H94O26 (1207.38). White thin acicular crystals, mp 215~217C, []D27.5 =
14.9 (c = 0.98, MeOH). Source: HUANG HE MAO REN DONG Lonicera
fulvotomentosa. Ref: 126.
7991 Fukugiside
[29082-55-1] C36H30O16 (718.63). mp 242~243C (dec). Pharm: Antioxidant
(DPPH radical scavenger, 10mol/L, ScRt = 56%, IC50 = 11.40mol/L;
control BHT, 10mol/L, ScRt = 43%, IC50 = 19.00mol/L)[4422]. Source:
HO
(flower). Ref: 6, 4422.

OH
SHAN ZHU ZI Garcinia multiflora, TIAN SHAN ZHU ZI Garcinia dulcis
OH
H
OH
OH
OH
OH
OH
O
O
OH
OH
OO
HO
OH
OH
O
OH
OH
O
OH
HO
OH
OH
OH
O
OH
OH
OH
OH
7996 Fumaric acid

(E)-2-Butenedioic acid [110-17-8] C4H4O4 (116.07). mp 250~260C. Pharm:
Analgesic; antibacterial; antineoplastic; anti-electroshock; antitussive. Source:
OH
DA CHE QIAN Plantago major, GAN ZHE Saccharum sinensis, HUANG
7992 Fukujusone
HAI YING SU Glaucium flavum, HUO YANG LE Euphorbia antiquorum, JI
3,8,14-Trihydroxypregn-5-en-20-one [25276-16-8] C21H32O4 (348.49). mp
CAI Capsella bursa-pastoris, JIN SHUA BA Cladonia fallax, JIU JIE CHA
224~227C. Source: FU SHOU CAO Adonis amurensis. Ref: 6.
Sarcandra glabra [Syn. Chloranthus glaber] (dried whole herb: content scope
of 6 origins = 0.052%~0.183%, mean content = 0.122%[5508]), LU SHAN SHI
FENG ZI Daphniphyllum calycinum, PING GUO HAI TANG Malus
OH
H
WEI Pyrrosia sheareri, MAI JIA GONG Lithospermum arvense, NIU ER

domestica, SHI RUI Cladonia rangiferina, WAN DOU Pisum sativum, WU
OH
HUA GUO Ficus carica, XIANG RI KUI ZI Helianthus annuus, YAN HU
HO
SUO Corydalis yanhusuo [Syn. Corydalis turtschaninovii f. yanhusuo], YAO
7993 Fukujusonorone
YONG QIU GUO ZI JIN Fumaria officinalis, YI ZHU QIAN MA Urtica
[26708-71-4] C20H26O3 (314.43). mp 88~90C. Source: FU SHOU CAO
dioica, YUN NAN FEI SHU Torreya yunnanensis (leaf and twig), ZI ZHI
Adonis amurensis. Ref: 6.
Ganoderma japonicum [Syn. Ganoderma sinense], occurs in many plants. Ref:
6, 658, 660, 4707, 5501, 5508.

H
OH
HO
H
HO
378
7997 Fumaricine
8002 -Funebrene
[24181-77-9] C21H23NO5 (369.42). Pharm: Used in treatment of skin disease,
[50894-66-1] C15 H 24 (204.36). Source: BAI SHU YE Cupressus
hepatitis, and inflammation (using the source plant YAO YONG QIU GUO ZI
funebris, DU HUO Angelica pubescens f. biserrata [Syn. Angelica
JIN Fumaria officinalis). Source: YAO YONG QIU GUO ZI JIN Fumaria
pubescens]. Ref: 2.

O
O
H
HO
8003 Fungisterol
Ergost-7-en-3-ol [53260-54-1] C28H48O (400.69). mp 152C. Source: XIANG
XUN Lentinus edodes. Ref: 6.
7998 Fumarprotocetraric acid

[489-50-9] C22H16O12 (472.37). mp 250~260C. Pharm: Cytotoxic (L1210, IC50
= (82.312.3)g/mL, control Etoposide, IC50 = (0.30.15)g/mL; 3LL, IC50 =
(75.99.7)g/mL, Etoposide, IC50 = (2.60.8)g/mL; DU145, IC50 >

100g/mL, Etoposide, IC50 = (0.90.2)g/mL; MCF7, IC50 > 100g/mL,
Etoposide, IC50 = (12.20.5)g/mL; K562, IC50 > 100g/mL, Etoposide, IC50 =
(2.11.3)g/mL; U251, IC50 > 100g/mL, Etoposide, IC50 =
(0.280.06)g/mL)[5027]. Source: JIN SHUA BA Cladonia fallax, SHI RUI
H
HO
Cladonia rangiferina, ZONG JUAN SHI RUI Cladonia convoluta. Ref: 6,

8004 Funiferine
5027.
HO
C38H42 N 2O6 (622.77). Pharm: Antitrypanosomal (inhibits trypomastigote form
O
O
OH
OH
OH
O
O
of Trypanosoma cruzi, strain Y, IC50 = 29.7g/mL, IC90 = 88.2g/mL);

antimalarial (Plasmodium falciparum D6, LC50 = 114.0ng/mL, SI = 92;
Plasmodium falciparum W2, LC50 = 183.3ng/mL, SI = 57); cytotoxic (KB,
LC50 = 10500ng/mL). Source: Guatteria boliviana (stem cortex). Ref:
3976.
7999 Fumotoshidin A
[89354-44-9] C20H32O4 (336.48). Source: BIAN YUAN LIN GAI JUE
Microlepia marginata. Ref: 1538.

N
OH
O
N
O
O
HO
H
O
OH
OH O
8000 Fumotoshidin B
8005 Funingenoside A
(8R)-3,4-Dihydrox-yl-14-oxo-5-15(148)-abeo-card-20(22)-enolide
OH
O
H
HO
OH
C44H66O19 (899.01). Colorless needles (MeOH), mp 261~265C, []D26 ~53.7

(c = 0.87, MeOH). Source: FU NING TENG Parepigynum funingense (root:
yield = 0.0026%dw). Ref: 4701.
8001 Fumotoshidin C

OH
HO
H
O
OH
HO
HO
HO
O
O
HO
HO
OH
OO
H
O
OH
379
8006 Funingenoside B
8010 Funtumine
(8R)-4-Acetoxy-3-[(O--D-glucopyranosyl-(16)-O--D-glucopyranosyl-(
[474-45-3] C21H35NO (317.52). Prismatic crystals (ethyl acetate), mp 126C,
14)--L-cymaropyranosyl)-oxy]-14-oxo-5-15(148)-abeo-card-20(22)-di
[]D = +95 (c = 1.7, chloroform). Pharm: Antipyretic; local anesthetic;
hydroenolide C44H68O19 (901.02). White powder, mp 271~275C, []D26 =
antihypertensive; promotes respiration; vasodilator. Source: GANG GUO HE
73.9 (c = 0.43, MeOH). Source: FU NING TENG Parepigynum funingense
ZHI XIE MU Holarrhena congolensis, SI JIAO SHU Funtumia elastica, TUI
(root: yield = 0.0073%dw). Ref: 4701.
RE ZHI XIE MU Holarrhena febrifuga. Ref: 658.

O
HO
O O
HO
HO
O
O
OH
OO
HO
HO
H2N
OH
8011 2-Furaldehyde
8007 Funingenoside C
Furan-2-carboxaldehyde [98-01-1] C5H4O2 (96.09). bp 162C. Source: CANG
(8R)-4-Acetoxy-3-[(O--D-glucopyranosyl-(14)--L-cymaropyranosyl)o
ZHU Atractylodes lancea, HONG CHE ZHOU CAO Trifolium pratense,
xy]-14-oxo-5-15-(148)-abeo-card-20(22)-dihydroenolide C38H58O14
HUANG HAO Artemisia scoparia [Syn. Artemisia capillaris var. scoparia],
(738.88). White powder, mp 256~259C, []D = 75.9 (c = 0.22, MeOH).
KONG SHI CHUN Ulva pertusa, LUO LE Ocimum basilicum, SHAN ZHU
Source: FU NING TENG Parepigynum funingense (root: yield = 0.0014%dw).
YU Cornus officinalis [Syn. Macrocarpium officinale], SHUI SONG Codium
Ref: 4701.
fragile, YIN CHEN HAO Artemisia capillaris, ZE XIE Alisma orientale [Syn.
13
Alisma plantago-aquatica var. orientale], ZI CAI Porphyra tenera. Ref: 2, 6,
660.
O
O
O
HO
HO
HO
OO
8012 2-Furancarboxylic acid
OH
Pyromucic acid [88-14-2] C5H4O3 (112.09). Leaflets (H2O), mp 133~134C,
8008 Funingenoside D
bp 230~232C, bp 141~144C/20mmHg. Source: BAI FAN DOU Phaseolus
(8R)-4-Acetoxy-3-[(O--D-glucopyranosyl-(16)-O--D-glucopyranosyl-
vulgaris, DANG SHEN Codonopsis pilosula, JIAN WEI YU Alocasia
(16)-O--D-glucopyranosyl-(14)--L-cymaopyranosyl)oxy]-14-oxo-5-
cucullata [Syn. Arum cucullatum], QIAN LI GUANG Senecio scandens [Syn.
15(148)-abeo-card-20(22)-dihydroenolide C50H78O24 (1063.16). White
Senecio chinensis], SHI YE Diospyros kaki, fungus Epicoccum sp. Ref: 2, 660,
powder, mp 248~253C, []D13 = 66.0 (c = 0.67, MeOH). Source: FU NING
1521, 2721, 2980, 5445.

O
TENG Parepigynum funingense (root: yield = 0.00035%dw). Ref: 4701.

O
HO
O
HO
HO
OH
HO
HO
O
O
OH
HO
HO
O O
OH
8013 Furandiol
C15H22O3 (250.34). Source: MEI WEI HONG GU Russula delica (sporocarp).
Ref: 4374.
O
O
OH
OH
8009 Funtumafrine C
(20S)-20-(N,N-dimethylamino)-5-pregna-3-one C23H39NO (345.57). White
O
OH
crystalline solid (CHCl3), mp 169~170C, []D25 = +50 (c = 0.06, CHCl3).
8014 Furanodiene
Pharm: BChE inhibitor (horse serum BChE, IC50 = (6.560.12)mol/L,
Isofuranodiene [19912-61-9] C15H20O (216.38). mp 44~45C. Pharm: NO
control Eserine, IC50 = (0.860.01)mol/L); AChE inhibitor (electric eel
production inhibitor (mus peritoneal macrophages, induced by LPS,
AChE, IC50 = (45.751.12)mol/L, control Eserine, IC50 =
(0.0410.001)mol/L). Source: YUN NAN YE SHAN HUA Sarcococca
(79.20.9)%, p<0.01)[4150]. Source: JI JI Chloranthus serratus, JIN SU LAN
coriacea [Syn. Sarcococca wallichii] (leaf). Ref: 4241.
Chloranthus spicatus, PING E SHU Curcuma zedoaria [Syn. Curcuma

aeruginosa], YIN XIAN CAO Chloranthus japonicus. Ref: 6, 660, 4150.
H
O
H
H
H
N
H
380
8015 Furanodienone
8021 S-Furanopetasitin
Isofuranodienone [24268-42-6] C15H18O2 (230.31). mp 89.5~90.5C; 70~71C.
[34335-97-2] C24H32O5S (432.58). mp 107~108C. Source: FENG DOU CAI
Pharm: NO production inhibitor (mus peritoneal macrophages, induced by
LPS, 100mol/L, InRt = (64.62.6)%, control L-NMMA, 100mol/L, InRt =

H
(79.20.9)%, p<0.01)[4150]. Source: PING E SHU Curcuma zedoaria [Syn.
Curcuma aeruginosa]. Ref: 6, 660, 4150.

H
O
H
O
O
8022 Furanopinguisanol
C15H22O2 (234.34). Source: YE TAI Trocholejeunea sandvicensis. Ref: 3909.
8016 Furanoeremophilane
[6750-13-6] C15H22O (218.34). bp 148C/16mmHg. Source: FENG DOU CAI
O
H
O
OH
8023 1-Furanoyl-2,3,7,8,11-pentaacetoxy-4,5-dihydroxy-dihydroagarofuran
8017 Furanoeremophilane-6,10-diol
[35101-40-7] C15H22O3 (250.34). mp 122C. Source: LIAN PENG CAO
Pharm: Immunosuppressant (inhibits lymphocyte transformation, 80g/mL,
Farfugium japonicum. Ref: 6.
InRt = 17%, control Dexamethasone, 50g/mL, InRt = 61%). Source: LEI

GONG TENG Tripterygium wilfordii (xylem). Ref: 4466.
OH
O
O
O
OH
8018 Furanofukinol
[In DNP] C15H22O3 (250.34). mp 178~180C (dec). Source: FENG DOU CAI
O
O
O
OH
O
OH
H
O
8024 1-Furanoyl-2,3,7,8,11-pentaacetoxy-5-hydroxy-dihydroHO
agarofuran
OH
8019 Furanojaponin
Pharm: Immunosuppressant (inhibits lymphocyte transformation, 80g/mL,
[34335-98-3] C20H28O3 (316.44). bp 110~130C/0.00005mmHg. Source:
InRt = 44%, control Dexamethasone, 50g/mL, InRt = 61%). Source: LEI
FENG DOU CAI Petasites japonicus. Ref: 6.
GONG TENG Tripterygium wilfordii (xylem). Ref: 4466.
O
O
O
O
8020 10-H-Furanoligularenone
O
OH
Furanoligularenone [16148-24-6] C15H18O2 (230.31). mp 95C. Pharm:

Anti-inflammatory (NO production inhibitor)
[4415]
; anti-inflammatory
(RAW264.7 stimulated by LPS, inhibits PGE2 production, IC50 =
8025 Furfuryl alcohol
1.93mol/L; inhibits expression of COX-2)[4415]. Source: HU LU QI
2-Hydroxymethylfuran [98-00-0] C5H6O2 (98.10). bp 170~171C. Source:
Ligularia fischeri, HU LU QI BIAN ZHONG Ligularia fischeri var.
CHA YE Camellia sinensis [Syn. Thea sinensis], SHUI SONG Codium
spiciformis. Ref: 6, 4415.
fragile. Ref: 6.
H
O
O
OH
381
8026 Furohyperforin
8030 Furosin
[219793-20-1] C35H52O5 (552.80). Oil, []D20 = +62.4 (c = 0.9, CHCl3).
C27H22O19 (650.46). Source: AN MO LE Phyllanthus emblica (branch and
Source: GUAN YE LIAN QIAO Hypericum perforatum (aerial parts: yield =
leaf). Ref: 3094.
0.00016%dw). Ref: 1521, 3032.
OH
OH
OH
O
OH
O
O O
OH
O
H
OH
O
HO
OH
HO OH O
OH
8031 cis-1-(2-Furyl)-4-(2-thienyl)-1-buten-3-yne
[20288-15-7] C12H8OS (200.26). bp 100~110C/0.3mmHg. Source: YANG
8027 Furomegistine I
SHI CAO Achillea millefolium. Ref: 6.
C15H15NO7 (321.29). Pharm: Cytotoxic (A549, IC50 = 90mol/L; HT29, IC50

= 100mol/L). Source: Sarcomelicope megistophylla (bark). Ref: 5155.
S
O
8032 Fuscaxanthone C
O
O
C26H30O6 (438.53). Pharm: Cytotoxic inactive (hmn small cell lung cancer
NCI-H187 cell line, control Ellipticine, IC50 = (0.350.15)g/mL). Source:
QIAO MU ZHUANG HUANG NIU MU Cratoxylum arborescens (stem

cortex). Ref: 5061.
8028 Furomegistine II
C14H13NO7 (307.26). []D = 0 (c = 0.1, CH2Cl2). Pharm: Cytotoxic (A549,
IC50 = 90mol/L; HT29, IC50 = 100mol/L). Source: Sarcomelicope
megistophylla (bark). Ref: 5155.
OH
O
O
8033 Fuscoporine
O
N
C20H14O9 (398.33). Dull-brown powder, mp > 300C. Source: HUA HE

KONG JUN Fuscoporia obliqua. Ref: 792.
OH
OH
8029 Furonewguinone B
O
O
OH
HO
O
OH
OH
8034 Fusicoserpenol A
4,12-Dihydroxy-8(17)-fusicoccene C20H34O2 (306.49). Colorless crystals
O
O
HO
(hexane), mp 87~90C, []D = +19.4 (c = 0.5, CHCl3). Pharm: Antifungal.

Source: PU FU QIANG DAO YAO Hypoestes serpens. Ref: 2063.
HO
O
OH
OH
H
OH
H
H
HO
382
8035 Futoamide
8040 Futoquinol
C18H23NO3 (301.39). mp 128~130C. Source: HAI FENG TENG Piper
Hancinone D [28178-92-9] C21H22O5 (354.41). White crystals (hexane), mp
kadsura [Syn. Piper futokadsura], SHAN JU Piper hancei. Ref: 6, 75.
96~97C, mp 97~98C, []D14 = 0 (c = 0.3, CHCl3). Pharm: PAF antagonist

(IC50 = 23mol/L). Source: HAI FENG TENG Piper kadsura [Syn. Piper
futokadsura], SHAN JU Piper hancei, ZHANG YE HU JIAO Piper
polysyphorum. Ref: 6, 130, 191, 1578.
N
H
O
O
8036 Futoenone
[19913-01-1] C20H20O5 (340.38). mp 197C. Source: HAI FENG TENG Piper
O
kadsura [Syn. Piper futokadsura]. Ref: 6.

O
8041 Futoxide
H
Crotepoxide [20421-13-0] C18H18O8 (362.34). mp 150~151C. Source: HAI
FENG TENG Piper kadsura [Syn. Piper futokadsura]. Ref: 6, 5501.
O
O
8037 Futokadsurin A
(7S,8S,7'S,8'R)-3,4,3'-Trimethoxy-4'-hydroxy-7,7'-epoxylignan C21H26O5 (358.44).
Colorless oil, []D25 = +12.3 (c = 1.09, CHCl3). Pharm: NO production inhibitor (mus,
macrophage-like cell line RAW264.7 activated by LPS/IFN, IC50 = 47.2mol/L,
control quercetin, IC50 = 26.8mol/L)[2537]. Source: HAI FENG TENG Piper kadsura
O
O
[Syn. Piper futokadsura]. Ref: 2537.

8042 Fuzinoside
O
Glycerol-2-O--D-galactofuranosyl (13)-galactofuranoside C15H28O13

(416.38). Yellowish powder. Source: FU ZI Aconitum carmichaeli. Ref: 4588.
OH
OH
8038 Futokadsurin B
(7R,8R,7'R,8'S)-3,4-Dimethoxy-3',4'-methylenedioxy-7,7'-epoxylignan
23
C21H24O5 (356.42). Colorless needles, mp 102C, []D = +33.7 (c = 1.18,

CHCl3). Pharm: NO production inhibitor (mus, macrophage-like cell line
HO
OH
O
OH
HO
OH
OH O
RAW264.7 activated by LPS/IFN, IC50 = 55.0mol/L, control quercetin, IC50
O
HO
= 26.8mol/L)[2537]. Source: HAI FENG TENG Piper kadsura [Syn. Piper

futokadsura]. Ref: 2537.
OH
C20H25NO4 (343.43). Brown solid, mp 210~212C(dec.), []D25 = +212 (c =

O
8043 Fuzitine
0.1, MeOH). Source: XIAN MAO HEI ZHONG CAO Nigella glandulifera
(seed). Ref: 4277.
8039 Futokadsurin C
(7R,8R,7'S,8'S)-3,4-Methylenedioxy-3',4'-dimethoxy-7,7'-epoxylignan C21H24O5
(356.42). Colorless oil, []D23 = 11.7 (c = 3.26, CHCl3). Pharm: NO production

inhibitor (mus, macrophage-like cell line RAW264.7 activated by LPS/IFN, IC50 =
79.2mol/L, control quercetin, IC50 = 26.8mol/L)[2537]. Source: HAI FENG TENG
Piper kadsura [Syn. Piper futokadsura]. Ref: 2537.
O
O
O
O
O
HO
HO
N
H
383
8049 Gajutsulactone B
C15H22O2 (234.34). Colorless oil, []D27 = 35.0 (c = 0.10, CHCl3), []D26 =

53.4 (c = 0.1, MeOH). Pharm: NO production inhibitor (mus peritoneal
8044 Gadesine
[70420-60-9] C23H35NO6 (421.54). mp 174~177C, []D = +76 (c = 0.27,
EtOH). Source: WU ZHU FEI YAN CAO Delphinium pentagynum. Ref:
1521.
H

O
H
OH
H
OH
H
OH
8050 L-Galactoheptulose
[29325-35-7] C7H14O7 (210.19). mp 110~115C (dec). Source: MU XU
8045 Gadoleic acid
Medicago sativa. Ref: 6, 1521.
[29204-02-2] C20H38O2 (310.52). mp (cis)23.0~23.5C, bp 170C/0.1mmHg.

OH
OH
OH
Source: LUO HUA SHENG YOU Arachis hypogaea. Ref: 6.
O
OH
HO
OH
OH
8051 3T-O--D-Galactopyranosylcinnamtannin B1
H
C51H46O23 (1026.92). Light-brown amorphous powder, []D = +17.1 (c = 1,
MeOH). Pharm: Antioxidant (inhibits NADPH-dependent lipid peroxidation
8046 Gagaminine
in microsomes and autoxidation of linoleic acid); antioxidant (DPPH
[41060-37-1] C36H43NO8 (617.75). mp 166~169C. Source: LUO MO
scavenger (effective). Source: KE KE Theobroma cacao. Ref: 2023.
Metaplexis japonica. Ref: 6.
OH
OH
OH
O
HO
OH
O
OH
HO
OH
OH
HO
HO
OH
OH
8047 Gaillardin
OH
[14682-46-3] C17H22O5 (306.36). Crystals, mp 199~200C (vacuum), []D30 =
OH
0.80~1.60g/mL or 2.30g/mL); antiprotozoal (amebic and Trichomonas
OH
OH
HO
15 (c = 1.08, chloroform). Pharm: Antineoplastic (KB, ED50 =
OH
HO
OH
vaginalis, 0.24~7.8g/mL). Source: TIAN REN JU Gaillardia pulchella,
8052 2-O--D-Galactopyranosyl-1-deoxynojirimycin
ZHONG GUO XUAN FU HUA Inula britannica var. chinensis. Ref: 661.
C12H23NO9 (325.32). Pharm: Hypoglycemic (mus diabetes mellitus induced
by SIZ, distinct effect). Source: SANG ZHI Morus alba. Ref: 2170.
O
H
H
N
HO
HO
OH
HO
HO
O
OH
OH
8048 Gajutsulactone A
O
OH
C15H22O2 (234.34). Colorless oil, []D28 = 128.4 (c = 0.10, CHCl3). Pharm:

NO production inhibitor (mus peritoneal macrophages, induced by LPS,
8053 6-O--D-Galactopyranosyl-1-deoxynojirimycin
C12H23NO9 (325.32). Source: Morus sp. Ref: 2513.
(79.20.9)%, p<0.01). Source: PING E SHU Curcuma zedoaria [Syn.

Curcuma aeruginosa]. Ref: 4150.
OH
HO
O
OH
O
OH OH
OH
H
N
OH
384
8054 3-O--D-Galactopyranosyl-(14)--D-galactopyranosyloleanolic acid
8057 3-O--D-Galactopyranosyl-(12)--D-glucuronopyranosyl-gypso-
C42H68O13 (781.00). Pharm: Cytotoxic (A2780, IC50 = (9.60.3)g/mL;
genin
control Actinomycin D, IC50 = 2~5ng/mL). Source: DA YE NAN YANG
C42H64O15 (808.97). White amorphous powder. Source: JIN TIE SUO
SHEN Polyscias amplifolia (infructescence), GUANG YE JUE MING Cassia
Psammosilene tunicoides. Ref: 2261.
laevigata [Syn. Cassia floribunda]. Ref: 5397.
H
OH
OH
H
HO
HO
OO
OO
HO
H
O
HO OH
O
HO
O
OH
OH
OH
OO
OH
OH
OH
OH
OH
8055 3-O--D-Galactopyranosyl-(12)--D-glucuronopyranosyl-21,
22-di-O-angeloylbarringtogenol C
21
C52H80O18 (993.21). []D = +2.3 (c = 0.13, MeOH). Source: NAN SU GE

LAN JIA SHAN LUO Harpullia austro-caledonica (stem cortex). Ref: 5269.
8058 3-O--D-Galactopyranosyl-(12)--D-glucuronopyranosylgypso-genin-28-O--D-xylopyranosyl(14)-[-D-6-O-acetylglucopyranosyl (13)]--L-rhamnopyranosyl(12)--D-fucopyranoside

C67H104O33 (1437.56). White powder. Source: JIN TIE SUO Psammosilene
tunicoides. Ref: 2261.
H
O
O
O
H
O
HO
OH
H
OH
OH
HO OH
HO OH
HO
OO
OO
OO
HO
O
OH
OH
OH
OH
HO
O
OH
OH
O-[-D-glucopyranosyl-(12)--L-rhamnopyranosyl-(12)--D-4-Otrans-p-methoxycinnamoyl-fucopyranosyl] quillaic acid

C72H106 O31 (1467.63). Source: HAN MAI PING CAO Silene jenisseensis.
Ref: 709.
OH
OH
8056 3-O-[-D-Galactopyranosyl-(12)--D-glucuronopyranosyl]-28-
OH
O
O
OO
HO
OO
O O OH
OH
OH
OH
8059 3-O-[-D-Galactopyranosyl-(12)--D-glucuronopyranosyl]
quillaic acid-28-O-[-L-arabinopyranosyl-(12)--L-arabinopyranosyl-(13)--D-xylopyranosyl-(14)--L-rhamnopyranosyl-(12)]-[6O-acetyl--D-glucopyranosyl-(13)]-4-O-acetyl--D-fucopyranoside
C79H122O43 (1757.83). White amorphous powder, []D20 = +13 (c = 0.10,
MeOH). Pharm: Proliferation stimulator (Jurkat-Tumor cell lines, at low
concentration). Source: YING ZI CAO Silene fortunei (root: yield =
0.0028%dw). Ref: 4658.
H
O
HO
OO
OH
OH
HO
H
O
O
OH
O
HO OH
OO
OH
OH
O HO
OH
OO
OH
OH
OH
O
HO
HO
HO
HO
OH
OO
OHO
O
OH
OH
HO
O
HO
HO
HO
O O
HO
OO
HO
OO
OH
OH
OO
HO
OO
OH
O O
O
O
OH
OH
OH
385
8063 3-O-[-D-Galactopyranosyl-(12)--D-glucuronopyranosyl]-
quillaic acid-28-O--L-rhamnopyranosyl-(12)-3-O-acetyl-4-O-cis-p-
sophoradiol methyl ester
methoxycinnamoyl -D-fucopyranoside
C43H70O13 (795.03). Source: HUAI Sophora japonica (bud). Ref: 4823.
C66H94O27 (1319.47). White amorphous powder. Pharm: Proliferation

stimulator or inhibitor (Jurkat-Tumor cell lines, stimulator at low
concentration, inhibitor at high concentration). Source: YING ZI CAO Silene
OH
fortunei (root). Ref: 4658.

O
OO
OH
OH
HO
O
OO
HO
OH
OH
O
OH
OO
O
HO HO
HO
OH
OH O
O
HO
HO
8064 6-O--D-Galactopyranosylharpagoside
C30H40O16 (656.64). Amorphous powder, mp 169~173C, []D = ~7.43 (c =
OH
0.336, MeOH). Source: XUAN SHEN Scrophularia ningpoensis. Ref: 1855.
OH
OH
HO
HO
O
OH
quillaic acid-28-O--L-rhamnopyranosyl-(12)-3-O-acetyl-4-O-trans-p-
methoxycinnamoyl -D-fucopyranoside
C66H94O27 (1319.47). White amorphous powder. Pharm: Proliferation
O
OH
OH
HO
stimulator or inhibitor (Jurkat-Tumor cell lines, stimulator at low

concentration, inhibitor at high concentration). Source: YING ZI CAO Silene
O
O
OH
OH
fortunei (root). Ref: 4658.
OH
8065 3-O--D-Galactopyranosyloleanolic acid

C36H58O8 (618.86). Pharm: Cytotoxic (A2780, IC50 = (10.80.5)g/mL;
control Actinomycin D, IC50 = 2~5ng/mL). Source: DA YE NAN YANG
O
HO H O
OH
OH
O O
HO
O O
OH
OH
OO
O
O
OH
HO
O
OH
SHEN Polyscias amplifolia (infructescence), DUAN HUA HU LU Lagenaria

breviflora, Brenania brieyi. Ref: 5397.
O
O
O
O
OH
OH
HO
H
OO
HO
OH
8062 3-O-[-D-Galactopyranosyl-(12)--D-glucuronopyranosyl]sophoradiol ethyl ester
OH
C44H72O13 (809.06). White amorphous powder. Source: HUAI Sophora
8066 2''-O--L-Galactopyranosylorientin
japonica (bud). Ref: 4823.
C27H30O16 (610.53). Yellow powder, mp 218~220C, []D20 = +28.9 (c =

OH
OH
O
HO
OO
OH
HO OH
OO
HO
OH
OH
HO
HO
O
O
OH
OH
OH
HO
HO
OH
HO
386
8067 3-O--D-Galactopyranosyl-(13)--L-rhamnopyranosyl-(12)-
8070 6'-O--D-Galactopyranosylswertiamarin
-L-arabinopyranosyl-23-hydroxyolean-12-en-28-oic acid
[245050-38-8] C47H76O17 (913.12). []D25 = +36.2 (c = 0.1, MeOH). Source:
DUO BAN LV TI CAO Caltha polypetala. Ref: 2338.

O
OH
HO
OH
OO
OH
OH
OH
OH
OH
H
O
OH
OH
H
OH
OH
OH
8071 6'-O--D-Galactopyranosylsyringopicroside
OO
Source: BAO MA ZI Syringa amurensis [Syn. Syringa reticulata var.

HO
HO
amurensis] (leaf). Ref: 4363, 4723.
O O OH
OH
OH
8068 3-O--D-Galactopyranosyl-(13)--L-rhamnopyranosyl-(12)-
HO
OH
O
O
OH
HO
-L-arabinopyranosyl-23-hydroxyolean-12-en-28-oic acid 28-O--Lrhamnopyranosyl-(14)--D-glucopyranosyl-(16)--D-glucopyranosyl
O
H
OO
OH
OH
ester
OH
[245050-37-7] C65H106O31 (1383.55). []D25 = 18.60 (c = 0.1, MeOH).

Source: DUO BAN LV TI CAO Caltha polypetala. Ref: 2338.
OH
8072 2''-O--L-Galactopyranosylvitexin
OH
H
OH
OO
OH
OH
HO
HO
H
HO
HO
OH
O O OH
OO
OH
OH
OH
OH
OH OH
OH
HO
OH
OH
OO
HO
O
O
OO
HO
HO
OH
HO
HO
OH
8073 3-O--D-Galactopyranosyl(12)-[-D-xylopyranosyl(13)]--D-
OH
6-O-ethylglucoronopyranosyl-quillaic acid
8069 3'-O--D-Galactopyranosylswertiamarin
C49H76O20 (985.14). White amorphous powder, mp 232~235C []D20 = 106.98 (c

= 0.43, MeOH). Source: JIN TIE SUO Psammosilene tunicoides. Ref: 2486.
O
O
HO
HO
HO
OH
OH
OH
OH
OH
OH
OO
O
H
O
OH
OH
OH
HO
HO
OH
OH
OH
O
OH
387
8074 3-O--D-Galactopyranosyl-(12)-[-D-xylopyranosyl(13)]--D-
8078 D-Galacturonic acid
glucuronopyranosyl-gypsogenin
[6294-16-2] C6H10O7 (194.14). mp () 156~159C (dec), mp () 160C (dec).
C47H72O19 (941.09). White amorphous powder. Source: JIN TIE SUO
Source: CHUN Brasenia schreberi, FEN TUAN HUA Hydrangea paniculata,
Psammosilene tunicoides. Ref: 2261.
HAI DAI Zostera marina, KU GUA Momordica charantia, LUO LE ZI

Ocimum basilicum, MU MIAN HUA Bombax malabaricum [Syn.
Gossampinus malabarica], YE YU Colocasia antiquorum, YI ZHU QIAN
OH
O
OH
OH
OH
OO
MA Urtica dioica, YU SHU SHU Zea mays. Ref: 6, 660.
OH
HO
O
OH
OH
OH
HO
HO
OO
OH
OH
OH
8079 Galanal A
[104086-74-0] C20H30O3 (318.46). Colorless rhombic Crystals, mp
167~169C, []D = 44 (c = 0.1, chloroform). Pharm: Antifungal (Candida
OH
8075 3-O--D-Galactopyranosyl(12)-[-D-xylopyranosyl(13)]--D6-O-methylglucoronopyranosyl-quillaic acid
guilliermondii, MIC = 12.5g/mL); cytotoxic (KB, ED50 = 3.25g/mL).

Source: DA LIANG JIANG Alpinia galanga. Ref: 1140.
H
25
C48H74O20 (971.11). White amorphous powder, mp 225~228C []D =
+12.31 (c = 0.325, MeOH). Source: JIN TIE SUO Psammosilene tunicoides.

Ref: 2486.
OH
H
O
OH
H
O
OO
O
O
OH
OH
8080 Galanal B
[104113-52-2] C20H30O3 (318.46). Colorless rhombic Crystals, mp
134.0~134.5C, []D = 48 (c = 0.1, chloroform). Pharm: Antifungal
(Candida guilliermondii, MIC = 12.5g/mL, Candida tropicalis, MIC =
OH
HO
OH
O
O
HO
OH OH
50g/mL); cytotoxic (KB, ED50 = 15.0g/mL). Source: DA LIANG JIANG

Alpinia galanga. Ref: 1140.
H
O
OH
8076 Galactosamine
[7535-00-4] C6H13NO5 (179.17). mp D() 185C. Source: LU RONG Cervus
OH
nippon; Cervus elaphus, YE YU Colocasia antiquorum. Ref: 2.
8081 Galangin
HO
HO
4H-1-Benzopyran-4-one,3,5,7-trihydroxy-2-phenyl [548-83-4] C15H10O5
O
OH
(270.24). Yellow acicular Crystals (MeOH), mp 214~216C. Pharm:

OH
Antimicrobial (bacteria on skin surface, such as Pseudomonas maltophilia,
NH2
Enterobacter cloacae, and Staphylococcus epidermidis); cyclo-oxygenase
8077 1-O--D-Galactosyl (61)--D-galactosyl-2,3-O-dihexadecanoyl-
inhibitor (ox spermia); mutagen (Salmonella aertrycke TA98 and TA100);
glycerol
antiemetic (young male chicks, copper sulfate induced emesis assay, 20mg/kg,
C47H88O15 (893.22). Yellowish gum. Source: XIAO YE GUAN ZHONG
InRt = 25.4%, p<0.01)[4649]. Source: BING TOU CAO Scutellaria
Matteuccia struthiopteris (rhizome). Ref: 4862.
galericulata, CHUI QI MU Alnus pendula, DA CHE QIAN Plantago major,

DA LIANG JIANG Alpinia galanga, FENG JIAO Apis mellifera ligustica,
OH
HO
GAO LIANG JIANG Alpinia officinarum (dried rhizome: content scope of 12
OH
O
OH
HO
origins = 0.35%~1.30%, mean content = 0.756%[5508]; yield = 0.063%dw[4649]),

Escallonia sp. Ref: 6, 463, 658, 4649, 5501, 5508.
OH
OO
OH
O
OH
OH
HO
388
8082 Galanolactone
[115753-79-2] C20H30O3 (318.46). Source: DA LIANG JIANG Alpinia
8086 ()-Galbacin
galanga, SHENG JIANG Zingiber officinale. Ref: 1140, 1542.
C20H20O5 (340.38). Pharm: NO production inhibitor (mus, macrophage-like

cell line RAW264.7 activated by LPS/IFN, IC50 = 47.7mol/L, control
quercetin, IC50 = 26.8mol/L)[2537]. Source: HAI FENG TENG Piper kadsura
[Syn. Piper futokadsura], YU LAN Magnolia denudata [Syn. Magnolia

heptapata]. Ref: 2537, 4439.
O
H
O
O
8083 Galanthamine
Jikon; Lycoremine; Galantamine [357-70-7] C17H21NO3 (287.36). Crystals

(benzene), mp 126~127C (benzene), []D20 = 118.8 (c = 1.378, ethanol),
8087 Galbanic acid
soluble in hot water, easily soluble in ethanol, acetone, chloroform, slightly
C24H30O5 (398.50). Source: A WEI Ferula assafoetida (root). Ref: 5243.
[5507]
soluble in benzene, ether.
Pharm: Analgesic; pesticide (kills Eurema
hecabe mandarina); cholinesterase inhibitor (reversibly inhibits cholinesterase

and easy passes BBB: AChE, IC50 = (0.500.01)mol/L, BChE, IC 50 =
(8.20.01)mol/L); AChE inhibitor (IC50 = (1.90.2)mol/L) [4952]. Source:
HO
BAI SHUI XIAN Narcissus papyraceus, DA YI ZHI JIAN Lycoris aurea, LU

CONG Lycoris squamigera, SHI SUAN Lycoris radiata [Syn. Amaryllis
radiata], SHUI XIAN GEN Narcissus tazetta var. chinensis, XIA XUE PIAN
8088 ()-Galbelgin
LIAN Leucojum aestivum, XUE HUA LIAN Galanthus nivalis, XUE PIAN
LIAN Leucojum vernum. Ref: 4, 6, 658, 2563, 4952, 5507.
cell line RAW264.7 activated by LPS/IFN, IC50 > 100mol/L, control

quercetin, IC50 = 26.8mol/L). Source: HAI FENG TENG Piper kadsura [Syn.
Piper futokadsura]. Ref: 2537.
OH
O
O
O
N
O
O
8084 Galanthindole
8089 (+)-Galbelgin
C17H15NO3 (281.31). Colorless amorphous solid. Source: TU ER QI XUE
C22H28O5 (372.47). Pharm: Neuroprotective (glutamate-induced neurotoxicity
HUA LIAN Galanthus plicatus ssp. byzantinus. Ref: 5443.
in primary cultures of cortical cells, 0.1mol/L, protection rate =

(20.93.2)%, p<0.05, MK-801: 1.0mol/L, protection rate = (83.62.0)%,
p<0.001, CNQX: 1.0mol/L, protection rate = (70.51.5)%, p<0.001).
Source: HONG NAN PI Machilus thunbergii. Ref: 4927.
N
O
OH
8090 Galdosol
8085 (+)-Galbacin
[528-64-3] C20H20O5 (340.38). Crystals (EtOAc), mp 115.5~116C, []D =
+117 (CHCl3). Pharm: Antibacterial (Mycobacterium tuberculosis H37Rv).
Source: RI BEN NAN Machilus japonica, SAN JIAO MA DOU LING
Aristolochia triangularis. Ref: 658, 1521.
rosmanol [52591-18-1] C20H24O5 (344.41). Pharm: Binding activity to

benzodiazepine receptor (IC50 = (0.80.1)mol/L, control Diazepam, IC50 =
(0.050.01)mol/L)[5366]. Source: YAO YONG DAN SHEN YE Salvia
OH
HO
O
O
O
O
O
389
8091 Galegine
8095 Gallic acid
[543-83-9] C6H13N3 (127.19). Moisture absorption bitter Crystals, mp
3,4,5-Trihydroxybenzoic acid [149-91-7] C7H6O5 (170.12). mp 235~240C
60~65C. Pharm: Hypoglycemic; toxin. Source: SHAN YANG DOU Galega
(dec). Pharm: Antiallergic; antibacterial (in vitro: Staphylococcus aureus,
Sarcina sp., -Streptococcus, Neisseria sp., Bacillus pyocyaneus, Bacillus

dysenteriae, Bacillus typhorus and Bacillus paratyphosus A, EC = 5mg/mL);
HN
antineoplastic (mus, pulmonary adenoma induced by morpholine and sodium

NH2
nitrite); cytotoxic (antioxidant assay)[5038]; antifungal (17 kinds of fungi in
HN
vitro, EC = 3%); anti-inflammatory; antimutagenic; antiviral (influenza virus);

astringent (intestinal tract of livestock animals); antiasthmatic; choleretic;
inhibits degradation of insulin, IL-10-like activity (proliferation assay,
dose-dependent, maximal at 30g/mL)[4445]; antioxidant (DPPH scavenger,
TLC, MIA < 0.05g, IC50 = 4g/mL)[5247]; DPPH scavenger (IC50 =
(12.40.2)mol/L, control Trolox, IC50 = (25.40.8)mol/L)[4244]; cell growth
8092 Galeopsin
[76475-16-6] C22H32O5 (376.50). Source: YI MU CAO Leonurus
heterophyllus [Syn. Leonurus artemisia]. Ref: 1543, 4493, 4534.
inhibitor (tsFT210 cell, 12.5g/L, inhibits G2/M stage); ACE inhibitor (IC50
> 500mol/L, control Lisinopril, IC50 = 1nmol/L); NEP inhibitor (IC50 =
480mol/L, control Phosphoramidon, IC50 = 9nmol/L); APN inhibitor inactive;
antibacterial (Erwinia carotovora, IZD = 13mm/100g, control Quercetin
sulfate, IZD = 21mm/10g; Staphylococcus aureus, IZD = 7mm/100g,

Quercetin sulfate, IZD = 14mm/10g; Corynebacterium accolens, IZD =
7mm/100g, Quercetin sulfate, IZD = 28mm/10g)[5250]; antifungal (Candida
OH
albicans, IZD = 7mm/100g, control Nystatin, IZD = 11mm/20g)[5250];

xanthine oxidase inhibitor (IC50 = 7.1g/mL, IC50 = 41.7mol/L; control
O
O
Quercetin, IC50 = 3.4g/mL, IC50 = 10mol/L)[5250]. Source: A LA BO JIN HE
HUAN Acacia arabica, BAI HUA QIAN HU Peucedanum praeruptorum,

BAI LIAN Ampelopsis japonica [Syn. Paullinia japonica], BAI SHAO
Paeonia albiflora [Syn. Paeonia lactiflora] (fresh fruit: yield = 1.13%fw)[4695],
8093 ()-Galgravin
cell line RAW264.7 activated by LPS/IFN, IC50 = 33.4mol/L, control
quercetin, IC50 = 26.8mol/L)[2537]. Source: HAI FENG TENG Piper kadsura
[Syn. Piper futokadsura], YU LAN Magnolia denudata [Syn. Magnolia
heptapata]. Ref: 2537, 4439.
BIAN XU Polygonum aviculare, CAO YUAN LAO GUAN CAO Geranium

pratense, CHANG YE SHUI MA Debregeasia longifolia, CHENG LIU
Tamarix chinensis, CU LIU GUO Hippophae rhamnoides, DA HUANG
Rheum officinale (stem and rhizome: mean content = 0.282%[5508]), DA YE
AN YE Eucalyptus robusta, DA YE KU NUO NI Cunonia macrophylla (leaf),
DI JIN CAO Euphorbia humifusa, DI YU Sanguisorba officinalis (dried root:
mean content of 6 origins = 0.25%)[5508], DIAN NAN HONG HOU KE
Calophyllum polyanthum (seed: yield = 0.0047%dw)[4767], DUO HUA SHAO
O
O
YAO Paeonia emodi (fruit), ER CHA GOU TENG Uncaria gambir, FAN
SHI LIU GAN Psidium guajava, HE TAO DA HUANG Rheum hotaoense
(stem and rhizome: content = 0.38%)[5508], HE ZI Terminalia chebula (fruit:
content scope = 1.04%~2.78%[5501, 5508], content = 1.04%[5508]), HONG KUAI
ZI Chamaenerion angustifolium [Syn. Epilobium angustifolium], HU LU BA
8094 Galiridoside
Trigonella foenum-graecum, HU TAO YE Juglans regia, HU ZHANG
Polygonum cuspidatum, HUA XIANG SHU YE Platycarya strobilacea,
persicus, TAI WAN JIN GU CAO Ajuga taiwanensis (whole herb). Ref: 2499,
HUANG LIAN YA Pistacia chinensis, HUANG LU Cotinus coggygria,
4483.
HUANG LU ZHI YE Cotinus coggygria var. cinerea, JI MU Loropetalum

chinense, KUAN DONG HUA Tussilago farfara, LU JIAO QI SHU Rhus
typhina, LU XIAN CAO Pyrola calliantha [Syn. Pyrola rotundifolia ssp.
OH
chinensis], LV BEI GUI HUA Excoecaria cochinchinensis var. viridis, MA

O
H
HO
OO
OH
OH
SANG Coriaria sinica [Syn. Coriaria nepalensis], MA SANG YE Coriaria

sinica [Syn. Coriaria nepalensis], MANG GUO Mangifera indica, MAO
YAN CAO Euphorbia lunulata (whole herb), MEI GUI HUA Rosa rugosa,
MO SHI ZI Quercus infectoria (parasitic bee: Cynips gallae-tinctoriae), MU
OH
DAN PI Paeonia moutan [Syn. Paeonia suffruticosa], NAN SUAN ZAO

Choerospondias axillaris (dried ripe fruit: mean content of 5 origins =
(2)
0.063%)[5508], NI LUO HE CHENG LIU Tamarix nilotica, PU
TAO Vitis
390
vinifera, QIAN NIU ZI Pharbitis nil, QIAN QU CAI Lythrum salicaria,
8098 (+)-Gallocatechin
QING GUO Canarium album (dried ripe fruit: content = 0.216%)[5508],
[970-73-0] C15H14O7 (306.27). Yellow powder, mp 188~190C, []D20 = 80
QUAN SHEN Polygonum bistorta, SAN WEI ZHI FAN YING TAO
(c = 0.5, CHCl3), mp (+) 185~188C, () 218C (dec). Pharm: Inhibitory
Eugenia sandwicensis, SHAN ZHU YU Cornus officinalis [Syn.
activity against NFAT transcription (IC50 = (24.50.9)mol/L, positive
Macrocarpium officinale] (dried ripe fruit: mean content of 8 origins =
control Cyclosporin A, IC50 = (0.290.01)mol/L) [2536]; inhibits cancer cell
[5508]
0.147%
), SHENG DI HONG JING TIAN Rhodiola sacra, SHI DI
Diospyros kaki (calyx: mean content = 0.029%)
[5508]
, SHI LIU PI Punica
invasion (MM1 cells, in vitro, 10g/mL, InRt = 24.2%)[4329]. Source: AN MO

LE Phyllanthus emblica (branch and leaf)[3094], BAI GUO YE Ginkgo biloba,
granatum, SHU ZHANG LAO GUAN CAO Geranium sibiricum, SHUI JIE
CHA YE Camellia sinensis [Syn. Thea sinensis], HUA CHA BIAO Ribes
GU DAN Epilobium hirsutum, SU MU Caesalpinia sappan, TANG GU TE
fasciculatum var. chinense. Ref: 6, 2536, 3094, 4329.
DA HUANG Rheum tanguticum (stem and rhizome: content = 0.93%[5508]),

WEI LING CAI Potentilla chinensis, WU JIU MU GEN PI Sapium sebiferum,
OH
WU JIU YE Sapium sebiferum, WU YA GUO Dillenia indica, XI FAN LIAN

Passiflora caerulea, XI XI LI QI SHU Rhus coriaria, XIAN HE CAO
OH
HO
OH
Agrimonia pilosa var. japonica, XIANG SI ZI Abrus precatorius, XIN XING

PU TAO Syzygium cordatum, YAN FU ZI Rhus chinensis [Syn. Rhus
OH
OH
semialata], YANG MEI SHU PI Myrica rubra (bark: content = 0.026%), YE

XIA ZHU Phyllanthus urinaria (whole herb: mean content = 0.115%[5508]),
YOU GAN MU PI Phyllanthus emblica, YOU GAN YE Phyllanthus emblica,
YOU SE ZI JIN NIU Ardisia colorata (fruit), YUE JI HUA Rosa chinensis,
ZANG BIAN DA HUANG Rheum emodi [Syn. Rheum australe] (stem and
8099 ()-Gallocatechin
C15H14O7 (306.27). Red amorphous powder, []D = 5.4 (c = 0.5, MeOH).
Source: XIAO GUO YE JIAO Musa acuminata (fruit). Ref: 3913.
rhizome: content = 0.042%)[5508], ZHANG YE DA HUANG Rheum palmatum
OH
(stem and rhizome: content = 0.30%[5508]), ZHU HONG SHI Diospyros
OH
cinnabarina, ZI WEI HUA Lagerstroemia indica., ZONG LV PI

Trachycarpus fortunei (petiole and fibre of sheath, roasted petiole: mean
HO
OH
[5508]
content of 5 origins = 0.029%
), occurs in many plants. Ref: 2, 4, 5, 6, 283,
OH
297, 658, 660, 3802, 4163, 4186, 4244, 4445, 4543, 4695, 4767, 4893, 5034,
OH
5038, 5247, 5250, 5375, 5501, 5508.

8100 Gallocatechin-(48)epicatechin
OH
[79199-56-7] C30H26O 13 (594.53). mp 223~227C. Source: KUN MING SHAN
HO
HAI TANG Tripterygium hypoglaucum. Ref: 612.

OH
HO
OH
OH
8096 Gallic acid-3-O-(6'-O-galloyl)glucoside

[87087-61-4] C20H20O14 (484.37). Source: AN MO LE Phyllanthus emblica
HO
OH
(branch and leaf)[3094], DA HUANG Rheum officinale, TANG GU TE DA
Ref: 2, 660, 3094.
OH
OH
HUANG Rheum tanguticum, ZHANG YE DA HUANG Rheum palmatum.

HO
OH
OH
OH
OH
OH
HO
HO
O
HO
8101 Gallocatechin-(48)-epigallocatechin
OO
OH
OH
OH
C30H26 O14 (610.53). Source: SAN XIAO CAO Trifolium repens (flower).
OH
Ref: 3970.
OH
OH
8097 Gallic acid-4-O-(6'-O-galloyl)-glucoside

[87087-62-5] C20H20O14 (484.37). Source: DA HUANG Rheum officinale,
ZHANG YE DA HUANG Rheum palmatum, TANG GU TE DA HUANG
OH
O
HO
Rheum tanguticum. Ref: 2, 660.

OH
OH
HO
OH
HO
O
OH
OH
OH
OH
OH
OH
HO
OO
OH
OH
OH
HO
OH
OH
391
8102 (+)-Gallocatechin-hexacetate
8106 8--C-(2'-Galloylglucopyranosyl)-5,7-dihydroxy-2-isopropylchromone
C27H26O13 (558.50). Source: BAI GUO Ginkgo biloba. Ref: 2.
C25H26O13 (534.48). Colorless amorphous powder. []D21 = 136.9 (c = 2.53,

MeOH). Source: GANG SONG Baeckea frutescens. Ref: 1895.
O
OH
O
O
O
HO
O
O
O
HO
OH
OH
O
OH
OH
HO
8107 1-Galloyl--D-glucopyranosyl-(14)--D-galactopyranoside
C19H26O15 (494.41). Oil, []D25 = +7.2 (c = 0.10, MeOH). Pharm: Antifungal
8103 ()-2-Galloyl-4-(E)-caffeoyl-L-threonic acid

20
C20H18O12 (450.36). Dark brown amorphous powder, mp 128~130C, []D =
(Candida albicans ATCC2091, MIC > 200g/mL, control Amphotericin B,
27 (c = 0.09, MeOH). Source: DENG TAI SHU Cornus controversa [Syn.
MIC = 1g/mL; Candida albicans 32, MIC > 200g/mL, Amphotericin B,
Bothrocaryum controversum] (leaf). Ref: 3918.
MIC = 4g/mL; Candida albicans 19, MIC = 100g/mL, Amphotericin B,

MIC = 2g/mL); cytotoxic inactive (MIC > 200g/mL); antibacterial inactive.
Source: Baseonema acuminatum (leaf). Ref: 5021.
OH
HO
O
O
HO
OH
OH
OH
OO
HO
OH
OO
HO
OH
OH
OH
OH
OH
OH
8108 1-O-Galloyl-glucose
OH
Glucogallin C13H16O10 (332.27). mp 212C (dec); mp () 179~181C, () 207.
OH
Source: AN MO LE Phyllanthus emblica (fruit juice, branch and leaf)[3094],

BAI SHAO Paeonia albiflora [Syn. Paeonia lactiflora] (fresh fruit: yield =
8104 4-O-(6'-O-Galloyl--D-glucopyranosyl)-cis-p-coumaric acid
0.0056%fw)[4695], DA HUANG Rheum officinale, HE ZI Terminalia chebula,
C22H22O12 (478.41). White amorphous powder, []D = 14.3 (c = 1.1, MeOH).
YOU GAN MU PI Phyllanthus emblica, YOU GAN YE Phyllanthus emblica,
Source: Monochaetum multiflorum (leaf). Ref: 5185.
TANG GU TE DA HUANG Rheum tanguticum, ZHANG YE DA HUANG

Rheum palmatum. Ref: 6, 660, 3094, 4695.
OO
OH
OH
OH
OH
H
OH
OH OH
HO
HO
OH
OO
OH
OH
O
OH
OH
8105 6--C-(2'-Galloylglucopyranosyl)-5,7-dihydroxy-2-isopropylchromone
C25H26O13 (534.48). Colorless amorphous powder, []D21 = 93.1(c = 2.50,
MeOH). Source: GANG SONG Baeckea frutescens. Ref: 1895.
8109 6-O-Galloyl-glucose
C13H16O10 (332.27). mp 166C (dec). Source: AN MO LE Phyllanthus
emblica (root)[3065], CAO YUAN LAO GUAN CAO Geranium pratense, DA
HUANG Rheum officinale, ZHANG YE DA HUANG Rheum palmatum,
TANG GU TE DA HUANG Rheum tanguticum, QUAN SHEN Polygonum
HO
HO
OH
bistorta. Ref: 2, 660, 3065.
HO
O
OH
HO
OH
HO
O
OH
OOH
OH
HO
OH
OH
OH
392
8110 1-O-Galloyl-glycerol
8115 5-O-Galloylpunicacortein D
C10H12O7 (244.20). Source: DA HUANG Rheum officinale. Ref: 2.
C59H42O34 (1294.97). Pale yellow amorphous powder. Source: SHI LIU XIN
OH
HO
OH
O
HO
HO
OH
HO
OH
HO
HO
8111 2''-O-Galloylisoorientin
C28H24O15 (600.49). Yellow amorphous powder, []D20 = 174 (c = 0.13,
HO
HO
HO
OH
HO
OH
HO
O
OH
O
OH
OH
8116 3-O-Galloyl quinic acid
HO
8112 2''-O-Galloylisovitexin
HO
OH
methanol). Source: SHEN YE TIAN ZHU KUI Pelargonium reniforme. Ref:
1994.
OH
HO
OH
O
OH
OH
HO
OH
HO
O
OH
OH
HO
OH
HO
HO
O
OH
OH
OH
OH
OH
1994.
H
O
HO
O
OH
HO
OH
HO
OH
OH
OH
8117 4-O-Galloyl quinic acid

HO
O
8113 2''-O-Galloylorientin
HO
OH

1994.
O
HO
OH
OH
O
O
HO
HO OH
OH
HO
O
OH
OH
OH
OH
HO
OH
HO
8118 1-O-Galloyl--L-rhamnose
O
C13H16O9 (316.27). Source: HONG HUA QI Acer rubrum. Ref: 2419.
8114 6'-O-Galloylprunasin
C21H21NO10 (447.40). White amorphous powder, []D = 17.0 (c = 1.9,
MeOH). Source: Monochaetum multiflorum (leaf). Ref: 5185.
HO
OH
HO
O
HO
O
HO
OH
OO
O
HO
OH
OH
H CN
OH
O
O
OH OH
393
8119 2''-O-Galloylvitexin
8123 Gamabufotalin-3-suberate
C32H46O8 (558.72). Source: CHAN SU Bufo bufo gargarizans; Bufo
melanostictus. Ref: 6.
O
1994.
O
OH
HO
OH
O
HO
HO
OH
OH
OH
H
O
HO
OH
OH
O
OH
8124 Gamatin
[479-85-6] C19H12O6 (336.30). mp 233~234C. Source: SHUI LIU DOU
Pongamia pinnata. Ref: 6.
8120 Galuteolin
[20344-46-1] C21H20O11 (448.39). mp 260~263C. Source: LIAN ZI XIN
Nelumbo nucifera, WEN JING Equisetum arvense. Ref: 6.
OH
OH
HO
O
O
8125 Gambireine
HO
C22H26N2O4 (382.46). Source: CHANG HUA GOU TENG Uncaria longiflora,
HOU YE GOU TENG Uncaria callophylla. Ref: 5341.
OH
OH
OH
OH
8121 Gamabufogenin
Gamabufotalin [465-11-2] C24H34O5 (402.54). mp 261~263C (dec). Pharm:
N
H H
Cytotoxic (in vitro, KB, IC50 = 0.75g/mL; HL-60, IC50 = 0.014g/mL;

MH-60, IC50 > 25g/mL)[3082]. Source: CHAN SU Bufo bufo gargarizans
(dried secretion: content = 0.22%[5508]); Bufo melanostictus (dried secretion:

content = 0.01%
[5508]
). Ref: 2, 6, 3082, 5508.
8126 Gambiriin C
O
O
[76236-89-0] C30H26O11 (562.54). Pharm: Tanning agent. Source: ER CHA

GOU TENG Uncaria gambir. Ref: 658.
OH
HO
HO
H
H
HO
OH
OH
OH
OH
HO
OH
OH
OH
8122 Gamabufotalininol
8127 Gambirine
C24H32O5 (400.52). mp 263~265C. Source: CHAN PI Bufo bufo gargarizans;
[29472-77-3] C22H28N2O4 (384.48). mp 163~165C, []D = +29 (chloroform).
Bufo melanostictus. Ref: 6.
Pharm: Uterine stimulant. Source: ER CHA GOU TENG Uncaria gambir,
HOU YE GOU TENG Uncaria callophylla. Ref: 6, 660, 661, 1521.

OH
H
H
O
N
H H
HO
OH
O
O
394
8128 Gambogic acid
8132 Ganbajunin C
-Guttiferin [2752-65-0] C38H44O8 (628.73). Yellow amorphous resin;
C34H26O8 (562.58). Source: JIN HUANG GE JUN Thelephora aurantiotincta.
pyridine salt Crystals, mp 147~149C. Pharm: Antineoplastic (mus, EAC, EC
Ref: 3423.
= 5mg/kg, S180, InRt = 61%~79%); antiprotozoal (non-pathogenicity, in vitro);

cytotoxic (cultural hmn liver cancer cells and HeLa, 4g/mL); laxative (mus).
Source: TENG HUANG Garcinia morella (dried balsam: content scope of 9
batch samples = 19.70%51.05%, mean content = 33.84%)[5508], TENG
[661]
HUANG SHU Garcinia hanburyi
HO
O
O
. Ref: 661, 5508.
O
HO
OH
OH
8133 Ganbajunin E
HO
OH
C34H26O8 (562.58). Source: JIN HUANG GE JUN Thelephora aurantiotincta.

Ref: 3423.
HO
8129 Gamboukokoensein A
O
OH
HO
O
1,2,3,19,23-Pentahydroxyurs-12-en-28-oic acid C30H48O7 (520.71).

White powder, mp > 300C. Source: Gambeya boukokoensis. Ref: 3463.
OH
HO
OH
8134 Gancaonin A
OH
HO
C21H20O5 (352.39). Source: GAN CAO Glycyrrhiza uralensis. Ref: 660.
HO
HO
OH
8130 Gamboukokoenside A
OH
2,3,6,28-Tetrahydroxyolean-12-en-23-oic acid 23-O--L-arabinopyranosyl

ester C35H56O10 (636.83). White powder, mp > 300C. Source: Gambeya
8135 Gancaonin B
boukokoensis. Ref: 3463.
[124596-86-7] C21H20O6 (368.39). Source: GAN CAO Glycyrrhiza uralensis.

Ref: 660.
HO
OH
OH
HO
OH
HO
OH
OO
8136 Gancaonin C
OH
[124596-87-8] C20H18O6 (354.36). Pharm: Antibacterial (Escherichia coli,
OH
MIA = 0.10g, control Chloramphenicol, MIA = 0.001g; Bacillus subtilis,

MIA = 0.05g, Chloramphenicol, MIA = 0.001g; Staphylococcus aureus,
OH
MIA = 0.05g, Chloramphenicol, MIA = 0.001g)[3785]; antifungal (Candida
8131 Gamboukokoenside B
6,28-Dihydroxy-3-oxoolean-12-en-23-oic acid 23-O--L-arabinopyranosyl
ester C35H54O9 (618.82). White powder, mp > 300C. Source: Gambeya
boukokoensis. Ref: 3463.
mycoderma, MIA = 0.05g, Miconazole = MIA = 0.0001g)[3785]; antioxidant

(DPPH scavenger, TLC detection limit = 0.5g, IC50 = 610g/mL; control
Quercetin, TLC detection limit < 0.05g, IC50 = 7g/mL; Gallic acid, TLC
detection limit < 0.05g, IC50 = 4g/mL; Ascorbic acid, TLC detection limit <
0.10g, IC50 = 18g/mL)[3785]. Source: GAN CAO Glycyrrhiza uralensis,
Bolusanthus speciosus (root wood)[3785]. Ref: 660, 2431, 3785.
OH
OH
O
OH
HO
OO
OH
O
OH
OH
OH
OH
395
8137 Gancaonin D
8141 Gancaonin P
C20H18O7 (370.36). Pharm: Aromatase inhibitor inactive (in vitro, IC50 >
Ref: 660.
40mol/L; control Aminoglutethimide, IC50 = 6.4mol/L)[3090]. Source: GOU

SHU Broussonetia papyrifera. Ref: 3090.
OH
OH
O
OH
HO
HO
OH
O
OH
OH
HO
8138 Gancaonin E
8142 Gancaonin P-3'-methylether
3,5,7,4'-Tetrahydroxy-3'-methoxy-6-isoprenyl flavone C21H20O7 (384.39).
Ref: 660.
Yellow lamellar Crystals. mp 160~162C. Source: GAN CAO Glycyrrhiza

O
OH
O
HO
OH
OH
HO
HO
O
OH
OH
8139 Gancaonin F
8143 Gancaonin X
C21H22O4 (338.41). Source: GAN CAO Glycyrrhiza Uralensis. Ref: 2431.

O
Ref: 660.
O
OH
O
O
8144 Gancaonin Y
OH
HO
8140 Gancaonin I
C21H22O5 (354.41). Pharm: Antibacterial (Enterococcus faecalis JCM7783

(VSE) (= ATCC19434), MIC = 3.13g/mL, control Linezolid, MIC =
1.56g/mL; Enterococcus faecalis JU1856(VRE, VanA), MIC = 3.13g/mL,

Linezolid, MIC = 0.78g/mL; Enterococcus faecalis JU1782(VRE, VanB),
MIC = 3.13g/mL, Linezolid, MIC = 0.78g/mL; Enterococcus faecium
8145 Gancaonin Z
JCM5804 (VSE) (= ATCC 29212), MIC = 6.25g/mL, Linezolid, MIC =
1.56g/mL; Enterococcus faecium JU1858 (VRE, VanA), MIC = 3.13g/mL,

Linezolid MIC = 0.78g/mL; Enterococcus faecium JU1777 (VRE, VanB),
HO
OH
MIC = 3.13g/mL, Linezolid, MIC = 1.56g/mL; Enterococcus gallinarum

JU2786 (VRE,VanC), MIC = 3.13g/mL, Linezolid, MIC = 0.78g/mL;
O
Staphylococcus aureus JCM2874 (MSSA) (=ATCC29213), MIC = 3.13g/mL,

Linezolid, MIC =1.56g/mL; Staphylococcus aureus (MRSA, 10 strains),
MIC = 3.13g/mL, Linezolid, MIC = 0.78g/mL; Staphylococcus aureus
8146 Ganervosin A
(MRSA, 8 strains), mean MIC80 = 3.13g/mL, Linezolid, mean MIC80 =
C24H32O8 (448.52). mp 224~226C. Source: XIAN MAI XIANG CHA CAI
0.78g/mL)
[5007]
. Source: GAN CAO Glycyrrhiza uralensis. Ref: 5007.
Rabdosia nervosa. Ref: 4067.

O
O
OH
O
HO
O
HO
O
OH
396
8147 Ganervosin B
8151 Ganode-8-en-ric acid B
C22H30O6 (390.48). mp 278~281C, []D20 = 80 (c = 0.23, C5H5N). Source:
Ganoderic acid B [81907-61-1] C30H44O7 (516.68). Amorphous powder.
XIAN MAI XIANG CHA CAI Rabdosia nervosa. Ref: 4067.
Pharm: HIV-1 protease inhibitor (IC50 = 0.17mmol/L); analgesic (best dose =

3~5mg/kg sc, InRt of twister reaction = (30~60)%, p<0.05). Source: LING
ZHI Ganoderma lucidum (dried sporocarp: mean content of 2 origins =
0.15%[5508]; yield = 0.0015%[4603]). Ref: 2235, 4603, 5508.
H
O
H
OH
OH
8148 Ganode-7,9-dien-ric acid X

Ganoderic acid X [86377-53-9] C32H48O5 (512.74). Pharm: Cytotoxic (mus
HO
OH
hepatosarcoma cell HTC, distinctly inhibits cell proliferation). Source: LING

ZHI Ganoderma lucidum. Ref: 2235.
8152 Ganode-8-en-ric acid C1
O
OH
H
O
Ganoderic acid C1 [95311-97-0] C30H42O7 (514.67). Crystals, mp 150~151C,

[]D15 = +175.4 (c = 0.057, CHCl3). Pharm: HIV-1 protease inhibitor (IC50 =
0.18~0.32mmol/L). Source: LING ZHI Ganoderma lucidum. Ref: 2235.
O
HO
OH
O
8149 Ganode-7,9-dien-ric acid Y

O
Ganoderic acid Y [86377-52-8] C30H46O3 (454.70). Pharm: Cytotoxic (mus

OH
8153 Ganode-8-en-ric acid D

H
Ganoderic acid D [97653-94-6] C30H42O8 (530.66). Crystals (EtOAc), mp
O
OH
201~203C, []D22 = +185 (c = 0.1, EtOH). Pharm: Antihistamine (inhibits

histamine release, mus must cells in vitro, induced by ConA, 0.4g/mL InRt =
15%). Source: LING ZHI Ganoderma lucidum (dried sporocarp: content
scope of 6 origins = 0.024%~0.686%, mean content = 0.334%[5508]). Ref:
2235, 5508.
HO
8150 Ganode-8-en-ric acid A
OH
O
Ganoderic acid A [81907-62-2] C30H44O7 (516.68). Amorphous powder,
OH
27
[]D = +153.8 (c = 0.156, CHCl3). Pharm: Analgesic (best dose = 3~5mg/kg
sc, InRt of twister reaction = (30~60)%, p<0.05); protein opopanax ester

transferase (FPT) selective inhibitor; cytotoxic inactive (mus lung carcinoma
OH
LLC cell, ED50 > 20g/mL; hmn carcinoma T-47D, ED50 > 20g/mL; S180,
ED50 > 20g/mL; mus sarcoma Meth-A, ED50 > 20g/mL; control adriamycin,
ED50 = 0.06g/mL, 0.02g/mL, 0.11g/mL, 0.13g/mL, respectively)[4204].
8154 Ganode-8-en-ric acid DM
Source: LING ZHI Ganoderma lucidum (dried sporocarp: content scope of 6
Ganoderic acid DM C30H44O4 (468.68). Yellowish acicular crystals
origins = 0.036%~1.560%, mean content = 0.340%[5508]; yield = 0.002%[4603]).
(chloroformmethanol), mp 203~205C. Source: LING ZHI Ganoderma
Ref: 188, 387, 2235, 4204, 4603, 5508.
lucidum (sporocarp: yield = 0.0017%)[4603]. Ref: 387, 4603.
H
O
OH
OH
O
OH
OH
397
8155 Ganode-8-en-ric acid F
8159 Ganode-8-en-ric acid U
Ganoderic acid F [98665-15-7] C32H42O9 (570.69). Pharm: ACEI (IC50 =
Ganoderic acid U C30H48O4 (472.71). Crystals, mp 196~199C, []D = +35.
4.7mol/L); EBV-EA activation inhibitor (Raji cells in vitro, TPA-induced,
Pharm: Cytotoxic (mus hepatosarcoma cell HTC, distinctly inhibits cell
IC50 = 293mol ratio/32pmol TPA, control -Carotene, IC50 = 400mol
proliferation). Source: LING ZHI Ganoderma lucidum. Ref: 2235.
ratio/32pmol TPA)
[4737]
. Source: LING ZHI Ganoderma lucidum (sporocarp:

H
yield = 0.0097%dw). Ref: 2235, 4737.
O
OH
H
O
O
O
OH
O
HO
8160 Ganode-8-en-ric acid V
O
O
Ganoderic acid V [86377-50-6] C32H48O6 (528.74). Pharm: Cytotoxic (mus
OH

8156 Ganode-8-en-ric acid H
Ganoderic acid H C32H44O9 (572.70). Pharm: HIV-1 protease inhibitor (IC50 =

0.18~0.32mmol/L); analgesic (best dose = 3~5mg/kg sc, InRt of twister
OH
reaction = (30~60)%, p<0.05). Source: LING ZHI Ganoderma lucidum
(sporocarp: yield = 0.0025%)[4603]. Ref: 2235, 4603.
O
O
8161 Ganode-8-en-ric acid W
OH
Ganoderic acid W C34H52O7 (572.79). Amorphous, mp 114~117C. Pharm:
Cytotoxic (mus hepatosarcoma cell HTC, distinctly inhibits cell proliferation).

Source: LING ZHI Ganoderma lucidum. Ref: 2235.
O
HO
OH
OH
H
O
O
8157 Ganode-8-en-ric acid LM2

Ganoderic acid LM2 C30H42O7 (514.67). mp 227~229C, []D = +132 Source:
LING ZHI Ganoderma lucidum. Ref: 2235.
(E)-7-Hydroxy-3,11,15,23-tetraoxolanosta-8,20(22)-dien-26-oic acid
C30H40O7 (512.65). Source: Ganoderma lipsiense. Ref: 3972.
OH
OH
O
OH
8162 Ganoderenic acid D
O
H
OH
OH
O
O
8158 Ganode-8-en-ric acid Ma

Ganoderic acid Ma C34H52O7 (572.79). Source: LING ZHI Ganoderma
lucidum. Ref: 1521.
OH
8163 Ganoderenic acid H

[120462-48-8] C30H40O7 (512.65). Source: SHU SHE Ganoderma
applanatum. Ref: 1521.
OH
OH
OH
O
O
HO
398
8164 Ganoderenic acid I
8168 Ganoderic acid C1
[120462-49-9] C30H42O7 (514.67). Source: SHU SHE Ganoderma
C30H42O7 (514.67). Pharm: Cytotoxic inactive (mus lung carcinoma LLC cell,
applanatum. Ref: 1521.
ED50 > 20g/mL; hmn carcinoma T47D, ED50 > 20g/mL; mus sarcoma S180,
ED50 > 20g/mL; mus sarcoma Meth-A, ED50 > 20g/mL; control
O
O
OH
Adriamycin, ED50 = 0.06g/mL, 0.02g/mL, 0.11g/mL, 0.13g/mL,

respectively). Source: LING ZHI Ganoderma lucidum. Ref: 4204.
OH
OH
HO
O
O
8165 Ganoderic acid AM1

C30H42O7 (514.67). Source: LING ZHI Ganoderma lucidum (sporocarp: yield
OH
= 0.0004%). Ref: 4603.

8169 Ganoderic acid E
O
H
C30H40O7 (512.65). Pharm: EBV-EA activation inhibitor (Raji cells in vitro,

OH
TPA-induced, IC50 = 281mol ratio/32pmol TPA, control -Carotene, IC50 =

400mol ratio/32pmol TPA)[4737]. Source: LING ZHI Ganoderma lucidum
(dried sporocarp: content scope of 6 origins = 0.342%~1.129%, mean content
= 0.784%[5508]; yield = 0.0066%dw[4737]). Ref: 4737, 5508.
O
HO
8166 Ganoderic acid B8

C30H44O7 (516.68). Pharm: Cytotoxic inactive (mus lung carcinoma LLC cell,
ED50 > 20g/mL; hmn carcinoma T-47D, ED50 > 20g/mL; mus sarcoma S180,
ED50 > 20g/mL; mus sarcoma Meth-A, ED50 > 20g/mL; control
OH
Ganoderic acid G [98665-22-6] C30H44O8 (532.68). Plates (EtOAcMeOH),

mp 218~220C, []D22 = +105.7 (c = 0.48, CHCl3). Pharm: Analgesic (best
dose = 3~5mg/kg sc, InRt of twister reaction = (30~60)%, p<0.05). Source:
OH
O
8170 Ganode-8-en-ric acid G
OH
O
LING ZHI Ganoderma lucidum (sporocarp: yield = 0.005%)[4603]. Ref: 2235,
OH
4603.
O
8167 Ganoderic acid C

OH
[98296-48-1] C30H46O7 (518.70). Pharm: Antihistamine (inhibits histamine
release, rat mastocyte in vitro, inhibits ConA-reduced histamine release,

0.4g/mL, InRt = 15%); cytotoxic (in vitro, HepG2, IC50 = 0.144nmol/L;
Hep2,2,15, IC50 = 0.105nmol/L; CCM2, IC50 = 31.3mol/L; P388, IC50 =
5mol/L) [3081]. Source: LING ZHI Ganoderma lucidum (dried sporocarp:
OH
O
O
HO
OH
content scope of 6 origins = 0.106%~0.901%, mean content = 0.472%[5508]).

8171 Ganoderic acid I
Ref: 387, 1521, 3081, 5508.
C30H44O8 (532.68). Source: LING ZHI Ganoderma lucidum (sporocarp: yield

= 0.0013%). Ref: 4603.
O
H
OH
HO
OH
OH
OH
O
HO
OH
OH
O
399
8172 Ganoderic acid N
8177 Ganoderic acid
7,20-Dihydroxy-3,11,15,23-tetraoxolanost-8-en-26-oic acid C30H42O8
(7,15,23S,24E)-7,15,23-Trihydroxy-3,11-dioxolanosta-8,24-dien-26-oic
(530.66). Source: Ganoderma lipsiense. Ref: 3972.
acid [294674-00-3] C30H44O7 (516.68). mp 243~245C, []D = +155.3.

Source: LING ZHI Ganoderma lucidum. Ref: 2235.
OH
O
O
OH
OH
OH
OH
OH
8173 Ganoderic acid T-Q
C32H46O5 (510.72). Pharm: EBV-EA activation inhibitor (Raji cells in vitro,
OH
TPA-induced, IC50 = 281mol ratio/32pmol TPA, control -Carotene, IC50 =
8178 Ganoderic acid
400mol ratio/32pmol TPA). Source: LING ZHI Ganoderma lucidum
[294674-02-5] C30H44O7 (516.68). []D = +160. Source: LING ZHI
Ganoderma lucidum. Ref: 2235.

O
O
OH
OH
OH
O
OH
O
O
OH
8179 Ganoderic acid

8174 Ganoderic acid Z
3,7,23-Trihydroxy-11,15-dioxolanosta-8,24-dien-26-oic acid [294674-05-8]
[86420-19-1] C30H48O3 (456.72). Pharm: Cytotoxic (mus hepatosarcoma cell
C30H44O7 (516.68). mp 249~251C, []D = +153.3. Source: LING ZHI
HTC, distinctly inhibits cell proliferation). Source: LING ZHI Ganoderma
lucidum. Ref: 2235.

H
O
OH
OH
OH
O
HO
HO
H
OH
8175 Ganoderic acid
8180 Ganoderic acid
C32H46O9 (574.72). []D = +55. Pharm: HIV-1 protease inhibitor(IC50 =
3,23-Dihydroxy-7,11,15-trioxolanosta-8,24-dien-26-oic acid. [294674-09-2]
0.18~0.32mmol/L). Source: LING ZHI Ganoderma lucidum. Ref: 2235.
OH
O
OH
HO
OH
OH
O
O
HO
8176 Ganoderic acid
8181 Ganoderic acid
C30H44O6 (500.68). mp 187~189C, []D = +60. Pharm: HIV-1 protease inhibitor (in
vitro, IC50 = 20mol/L). Source: LING ZHI Ganoderma lucidum. Ref: 341, 2235.
Ganoderma lucidum. Ref: 255, 2235.
O
OH
OH
OH
OH
OH
O
O
HO
HO
400
8182 Ganoderiol A
8186 Ganodermadiol
C30H50O4 (474.73). Needles (CHCl3), mp 232~234C, []D23 = +20 (c = 0.1,
C30H48O2 (440.72). Pharm: Cytotoxic (mus lung carcinoma LLC cell, ED50 >
EtOH). Pharm: HIV-1 protease inhibitor (IC50 = 0.18~0.32mmol/L). Source:
20g/mL; hmn carcinoma T-47D, ED50 > 20g/mL; mus sarcoma S180, ED50
> 20g/mL; mus sarcoma Meth-A, ED50 = 10.3g/mL; control Adriamycin,

ED50 = 0.06g/mL, 0.02g/mL, 0.11g/mL, 0.13g/mL, respectively). Source:
OH

OH
OH
OH
HO
HO
8187 Ganodermanondiol
8183 Ganoderiol B
C30H48O3 (456.72). Pharm: Cytotoxic (mus lung carcinoma LLC cell, ED50 =
[106518-62-1] C30H46O4 (470.70). Amorphous powder. Pharm: HIV-1
14.0g/mL; hmn breast carcinoma T47D, ED50 = 4.7g/mL; mus sarcoma S180,
protease inhibitor (IC50 = 0.17mmol/L). Source: LING ZHI Ganoderma
ED50 = 11.0g/mL; mus sarcoma Meth-A, ED50 = 9.2g/mL; control
lucidum (sporocarp: yield = 0.00025%)
[4603]
. Ref: 2235, 4603.

OH
OH
OH
OH
OH
O
8184 Ganoderiol D
8188 Ganodermanonol
[114567-45-2] C30H48O5 (488.71). Source: LING ZHI Ganoderma lucidum.
C30H46O2 (438.70). Pharm: Cytotoxic (mus lung carcinoma LLC cell, ED50 >
Ref: 387.
20g/mL; hmn breast carcinoma T47D, ED50 = 4.8g/mL; mus sarcoma S180,
ED50 = 10.0g/mL; mus sarcoma Meth-A, ED50 = 2.8g/mL; control
OH
OH

OH
OH
8189 Ganodermanontriol
[106518-63-2] C30H48O4 (472.71). Crystals, mp 168~170C, []D24 = +41 (c =
8185 Ganoderiol F
[114567-47-4] C30H46O3 (454.70). Yellowish plates (CHCl3MeOH), mp
116~120C, []D21 = +42 (c = 0.1, MeOH). Pharm: Anti-HIV-1 (MT-4 cell,
inhibits cytotoxic effect induced by HIV-1, IC100 = 7.8g/mL and this
concentration is 50% of that of cytotoxic concentration only); HIV-1 protease
inhibitor (IC50 = 0.18~0.32mmol/L). Source: LING ZHI Ganoderma lucidum.
Ref: 2235.
0.2, MeOH). Pharm: Anti-HIV-1 (MT-4 cell, inhibits cytotoxic effect induced
by HIV-1, IC100 = 7.8g/mL and this concentration is 50% of that of cytotoxic
concentration only); cytotoxic inactive (mus lung carcinoma LLC cell, ED50 >
20g/mL; hmn carcinoma T47D, ED50 > 20g/mL; mus sarcoma S180, ED50 >
20g/mL; mus sarcoma Meth-A, ED50 > 20g/mL; control adriamycin, ED50
= 0.06g/mL, 0.02g/mL, 0.11g/mL, 0.13g/mL, respectively)[4204]. Source:
LING ZHI Ganoderma lucidum. Ref: 2235, 4204.
OH
OH
HO
OH
OH
401
8190 Ganodermic acid R
8195 Ganolactone
[108026-93-3] C34H50O6 (554.77). Pharm: inhibits biosynthesis of cholesterol
Lucidenolactone C27H36O6 (456.58). White acicular Crystals, mp 294~296C,
(inhibits absorption of cholesterol in foods). Source: LING ZHI Ganoderma
[]D20 = +6 (c = 0.1148, chloroform). Source: LING ZHI Ganoderma lucidum.
lucidum. Ref: 2235.
Ref: 350, 3081.

O
H
O
H
O
O
OH
O
O
O
O
OH
8196 Ganolucidic acid A

8191 Ganodermic acid S
[98665-21-5] C30H44O6 (500.68). Pharm: HIV-1 protease inhibitor (distinct
[112430-63-4] C34H50O6 (554.77). Pharm: platelet aggregation inhibitor
effect). Source: LING ZHI Ganoderma lucidum. Ref: 2235.
(2mol/L, InRt = 50%, 7.5~10mol/L, InRt = 100%, IC50 = 2mol/L); inhibits
biosynthesis of cholesterol (inhibits absorption of cholesterol in foods. Source:
OH
OH
O
H
O
O
OH
8197 Ganolucidic acid B
[98683-75-1] C30H46O6 (502.70). Source: LING ZHI Ganoderma lucidum.
Ref: 2235.
O
OH
8192 Ganoderpurine
O
[133086-82-5] C11H15N5O (233.28). Oleaginous substance, mp 151~152C.
Source: BAO GAI LING ZHI Ganoderma capense. Ref: 164.
OH
HO
NH2
N
N
8198 Ganosporelactone A
C30H40O7 (512.65). White acicular Crystals, mp 238~240C, []D13 = +74.5 (c

= 0.057, chloroform). Source: LING ZHI Ganoderma lucidum. Ref: 192.
8193 Ganodine
[133086-81-4] C14H15NO2 (229.28). Source: BAO GAI LING ZHI
OH
Ganoderma capense. Ref: 164.
H
H
HO
8194 Ganoine
[133086-80-3] C11H17NO2 (195.26). Oleaginous liquid. Source: BAO GAI
LING ZHI Ganoderma capense. Ref: 164.
OH
8199 Ganosporelactone B
C30H42O7 (514.67). White acicular Crystals, mp 235~237C, []D12 = +68.8 (c
= 0.083, chloroform). Source: LING ZHI Ganoderma lucidum. Ref: 192.
OH
HO
H
H
O
O
HO
OH
402
8200 Ganosporeric acid A
8205 Garcibiphenyl B
[135357-25-4] C30H38O8 (526.63). Yellow acicular Crystals, mp 115~118C,
C18H20O3 (284.36). Colorless oil. Pharm: Cytotoxic (P388 ED50 = 6.63g/mL,
[]D28 = +48 (c = 0.1, chloroform). Source: LING ZHI Ganoderma lucidum
control Mithramycin ED50 = 0.06g/mL, HT29 ED50 = 12.7g/mL, control
(dried sporocarp: mean content of 2 origins = 0.14%[5508]) Ref: 188, 5508.
Mithramycin ED50 = 0.08g/mL). Source: TAI WAN LV DAO TENG
OH
O
HO
O
8201 Garajonone
C22H32O9 (440.49). Pharm: Antifeedant (Spodoptera littoralis, EC50 >
23nmol/cm2, Leptinotarsa decemlineata, EC50 > 23nmol/cm2). Source: YIN
DU E LI Persea indica (aerial parts). Ref: 5128.
HO
O
HO
OH
O
O
HUANG Garcinia linii. Ref: 4094.
OH
8206 Garcimangosone A
C28H28O6 (460.53). Yellow powder, mp 143~145C. Source: DAO NIAN ZI
Garcinia mangostana (fruit hull). Ref: 3066.
OH
OH
O
O
OH
OH
8202 Garbanzol
Aromadendrin-4',7-dimethyl ether [1226-22-8] C15H12O5 (272.26). mp
189~190C. Source: HUI HUI DOU Cicer arietinum, NING MENG AN YE
Eucalyptus citriodora. Ref: 6, 1521.
8207 Garcimangosone B
OH
HO
OH
OH
O
8203 Garcibenzopyran
C18H20O3 (284.36). Colorless amorphous powder, mp 82~83C. Pharm:
Cytotoxic (P388 ED50 = 3.98g/mL, control Mithramycin ED50 = 0.06g/mL,
HT29 ED50 = 6.90g/mL, control Mithramycin ED50 = 0.08g/mL). Source:
TAI WAN LV DAO TENG HUANG Garcinia linii. Ref: 4094.
8208 Garcimangosone C
OH
HO
OH
OH
O
OH
8204 Garcibiphenyl A
C13H12O3 (216.24). Colorless oil. Pharm: Cytotoxic (P388 ED50 = 10.2g/mL,
control Mithramycin ED50 = 0.06g/mL, HT29 ED50 = 13.5g/mL, control
Mithramycin ED50 = 0.08g/mL). Source: TAI WAN LV DAO TENG
HUANG Garcinia linii. Ref: 4094.
8209 Garcimangosone D
C19H20O9 (392.37). Yellow powder, mp 136~138C, []D25 = 64 (c = 0.5,
MeOH). Source: DAO NIAN ZI Garcinia mangostana (fruit hull). Ref: 3066.
OH
HO
OH
HO
HO
O
HO
HO
OO
OH
403
8210 Garcinianone A
8214 Garcinielliptone L
C28H32O6 (464.56). Yellow oil, []D25 = 0 (c = 0.48, CHCl3). Pharm:
9,9-Dimethyl-6,8-di(,-dimethylallyl)-3,4-[2-(2'-hydroxyisopropyl)-2,3-
Cytotoxic (BST, LD50 = 7.7mol/L; control Berberine, LD50 = 67mol/L);
dihydrofuran]-2-(1-oxo-2-methylpropyl)-8-H-cis-bicyclo[3.3.1]nona-1,5-
antioxidant (DPPH radical scavenger, IC50 = 107.4mol/L; control Catechin,
dione C30H44O5 (484.68). Colorless oil, []D = 41 (c = 0.29, CHCl3). Pharm:
IC50 = 2.53mol/L). Source: SHAN ZHU ZI Garcinia multiflora (stem: yield
Anti-inflammatory (rat mast cells stimulated with 10g/mL compound 48/80,
= 0.000042%dw). Ref: 4708.
in vitro: inhibits release of -glucuronidase, IC50 = 22.9mol/L; inhibits

release of histamine, IC50 > 30mol/L; control Mepacrine, inhibits release of
-glucuronidase, IC50 = 13.7mol/L; inhibits release of histamine, IC50
=23.3mol/L); anti-inflammatory (inhibits accumulation of NO2, culture
OH
media of RAW264.7 macrophage-like cells in response to 1g/mL LPS, IC50
O
HO
= 22.7mol/L; N9 microglial cells in response to lipopolysaccharide

(10ng/mL)/IFN- (10U/mL), IC50 = 12.8mol/L; control N-(3-Aminomethyl)
OH
benzylacetamidine, RAW264.7 cells, IC50 = 2.9mol/L; N9 cells, IC50 =

6.3mol/L). Source: FU MU Garcinia subelliptica (seed: yield =
8211 Garcinianone B
25
C28H32O6 (464.56). Yellow oil, []D = 0 (c = 0.21, CHCl3). Pharm:
0.00011%fw). Ref: 4773.
Cytotoxic (BST, LD50 = 25.8mol/L; control Berberine, LD50 = 67mol/L);

antioxidant (DPPH radical scavenger, IC50 = 144.8mol/L; control Catechin,
HO
IC50 = 2.53mol/L). Source: SHAN ZHU ZI Garcinia multiflora (stem: yield
H
O
= 0.000036%dw). Ref: 4708.
O
OH
O
O
HO
OH
8212 Garciniaxanthone E
8215 Garcinielliptone M
C28H32O6 (464.56). Pharm: Neurite outgrowth enhancer (PC12D cells,
9,9-Dimethyl-6,8-di(,-dimethylallyl)-3,4-[2-(2'-hydroxyisopropyl)-2,3-d
10mol/L, NGF-mediated neurite outgrowth, to enhance the ability of NGF,
ihydrofuran]-2-(1-oxo-2-methylpropyl)-8-H-cis-bicyclo[3.3.1]nona-1,5-dio
may be useful in the treatment of neurological disorders). Source: DA YE
ne C30H44O5 (484.68). Colorless oil, []D = +73 (c = 0.16, CHCl3). Pharm:
TENG HUANG Garcinia xanthochymus (wood). Ref: 4404.
Anti-inflammatory (rat mast cells stimulated with 10g/mL compound 48/80,

in vitro: inhibits release of -glucuronidase, IC50 = 13.6mol/L; inhibits
release of histamine, IC50 = 19.0mol/L; control Mepacrine, inhibits release of
-glucuronidase, IC50 = 13.7mol/L; inhibits release of histamine, IC50
=23.3mol/L); anti-inflammatory (inhibits accumulation of NO2, culture
OH
media of RAW264.7 macrophage-like cells in response to 1g/mL LPS, IC50

O
HO
OH
OH
8213 Garcinielliptone K
2-Benzoyl-9,9-dimethyl-6,8-di-(,-dimethylallyl)-3,4-[2-(2'-hydroxyiso
= 15.3mol/L; N9 microglial cells in response to lipopolysaccharide

(10ng/mL)/IFN- (10U/mL), IC50 > 30mol/L; control N-(3-Aminomethyl)
benzylacetamidine, RAW264.7 cells, IC50 = 2.9mol/L; N9 cells, IC50 =
6.3mol/L). Source: FU MU Garcinia subelliptica (seed, yield =
0.00008%fw). Ref: 4773.
propyl)-2,3-dihydrofuran]-8-H-cis-bicyclo[3.3.1]nona-3-ene-1,5-dione
C33H42O5 (518.7). Colorless oil, []D = +27 (c = 0.27, CHCl3). Source: FU
MU Garcinia subelliptica (seed: yield = 0.000027%fw). Ref: 4773.
HO
HO
H
O
O
O
404
8216 Garcinielliptone N
Staphylococcus aureus MRSA SK1, MIC = 16g/mL, Vancomycin, MIC =
3,3-Dimethyl-4,6-di(,-dimethylallyl)-2-(2-methyl-1-oxopropyl)cyclohex
2g/mL)[5319]. Source: TENG HUANG SHAN ZHU ZI Garcinia cambogia,
anone C22H36O2 (332.53). Colorless oil, []D = 42 (c = 0.38, CHCl3). Pharm:
TIAN SHAN ZHU ZI Garcinia dulcis (fruit), TIAN SHAN ZHU ZI Garcinia
Anti-inflammatory inactive (rat mast cells stimulated with 10g/mL
dulcis (flower), YIN DU TENG HUANG Garcinia indica, Garcinia bancana
compound 48/80, in vitro: inhibits release of -glucuronidase, IC50 >
(twig and leaf). Ref: 658, 4422, 4452, 5319.
30mol/L; inhibits release of histamine, IC50 > 30mol/L; control Mepacrine,
OH
inhibits release of -glucuronidase, IC50 = 13.7mol/L; inhibits release of

O
histamine, IC50 =23.3mol/L); anti-inflammatory inactive (inhibits
OH
OH
accumulation of NO2 , culture media of RAW264.7 macrophage-like cells in
response to 1g/mL LPS, IC50 > 30mol/L; N9 microglial cells in response to

lipopolysaccharide(10ng/mL)/IFN- (10U/mL), IC50 > 30mol/L; control
N-(3-Aminomethyl)benzylacetamidine, RAW264.7 cells, IC50 = 2.9mol/L;

N9 cells, IC50 = 6.3mol/L). Source: FU MU Garcinia subelliptica (seed,
yield = 0.000053%fw). Ref: 4773.
O
8219 Garcinone B
C23H22O6 (394.43). Pharm: Antitubercular (Mycobacterium tuberculosis, MIC

= 6.25g/mL)[4358]; antioxidant (DPPH scavenger, 10mol/L, ScRt = 15%,
control BHT, 10mol/L, ScRt = 43%)[5319]; antibacterial (Staphylococcus
aureus ATCC 25923, MIC = 8g/mL, control Vancomycin, MIC = 2g/mL;
Staphylococcus aureus MRSA SK1, MIC > 128g/mL, Vancomycin, MIC =
2g/mL)[5319]; cytotoxic inactive (KB cancer cell lines, BC-1, NCI-H187)[1619];
antioxidant inactive (DPPH scavenger, 50mol/L, ScRt = 6.9%; control BHT,
8217 Garcinielliptone O
6-Methoxylcarbonyl-3,3-dimethyl-4,6-di(,-dimethylallyl)-2-(2-methyl-1
-oxo-propyl)cyclohexanone C24H38O4 (390.57). Colorless oil, []D = 277 (c
= 016, CHCl3). Pharm: Anti-inflammatory inactive (rat mast cells stimulated
with 10g/mL compound 48/80, in vitro: inhibits release of -glucuronidase,
IC50 > 30mol/L; inhibits release of histamine, IC50 > 30mol/L; control
Mepacrine, inhibits release of -glucuronidase, IC50 = 13.7mol/L; inhibits
50mol/L, ScRt = 51.7%, IC50 = 28.9mol/L)[4423]. Source: DAO NIAN ZI

Garcinia mangostana (young fruit: yield = 0.0017%dw)[1619], DAO NIAN ZI
Garcinia mangostana (fruit hull), HUANG NIU MU Cratoxylum
cochinchinense (root), TIAN SHAN ZHU ZI Garcinia dulcis (fruit), TIAN
SHAN ZHU ZI Garcinia dulcis (flower). Ref: 1521, 1619, 3066, 4358, 4422,
4423, 5319.
release of histamine, IC50 =23.3mol/L); anti-inflammatory inactive (inhibits

accumulation of NO2, culture media of RAW264.7 macrophage-like cells in
response to 1g/mL LPS, IC50 > 30mol/L; N9 microglial cells in response to
HO
lipopolysaccharide(10ng/mL)/IFN- (10U/mL), IC50 > 30mol/L; control
N-(3-Aminomethyl)benzylacetamidine, RAW264.7 cells, IC50 = 2.9mol/L;
N9 cells, IC50 = 6.3mol/L). Source: FU MU Garcinia subelliptica (seed:

yield = 0.00028%fw). Ref: 4773.
OH
O
OH
8220 Garcinone C
C23H26O7 (414.46). Pharm: Cytotoxic (KB cancer cell lines, IC50 = 7.48g/mL,
control Ellipticine, IC50 = 1.33g/mL; BC-1, IC50 = 2.18g/mL, Ellipticine,
IC50 = 1.46g/mL; NCI-H187, IC50 = 3.66g/mL Ellipticine, IC50 =
0.39g/mL). Source: DAO NIAN ZI Garcinia mangostana (young fruit: yield
= 0.0068%dw). Ref: 1619.
8218 Garcinol
Camboginol; Guttiferone E [78824-30-3] C38H50O6 (602.82). Pharm:
Antibacterial (Staphylococcus aureus MRSA, MIC = 16g/mL)[4452];
OH
antifungal; antioxidant (DPPH scavenger, 10mol/L, ScRt = 74%, control

BHT, 10mol/L, ScRt = 43%)
[5319]
; antioxidant (DPPH radical scavenger,
10mol/L, ScRt = 59%, IC50 = 10.10mol/L; control BHT, 10mol/L, ScRt =

43%, IC50 = 19.00mol/L)[4422]; antibacterial (Staphylococcus aureus ATCC
25923, MIC = 16g/mL, control Vancomycin, MIC = 2g/mL;
OH
HO
HO
OH
405
8221 Garcinone D
8224 Garciosaterpene A
C24H28O7 (428.49). Pharm: Antitubercular (Mycobacterium tuberculosis, MIC
C32H50O4 (498.75). White needles, mp 120~121C, []D29 = +12 (c = 0.13,
= 25g/mL)[4358]; antioxidant (DPPH scavenger, 10mol/L, ScRt = 3%,
MeOH). Pharm: Anti-HIV-1 (HIV-1 reverse transcriptase assay, 200g/mL,
control BHT, 10mol/L, ScRt = 43%)[5319]; antioxidant inactive (DPPH
InRt = 96.2%, IC50 = 15.5g/mL). Source: MEI LI TENG HUANG Garcinia
scavenger, 50mol/L, ScRt = 6.9%; control BHT, 50mol/L, ScRt = 51.7%,
speciosa (trunk bark and stems). Ref: 5491.
IC50 = 28.9mol/L)[4423]; antibacterial (Staphylococcus aureus ATCC 25923,

MIC = 16g/mL, control Vancomycin, MIC = 2g/mL; Staphylococcus
aureus MRSA SK1, MIC = 32g/mL, Vancomycin, MIC = 2g/mL)[5319];
OH
cytotoxic (KB cancer cell lines, IC50 = 3.56g/mL, control Ellipticine, IC50 =
1.33g/mL; BC-1, IC50 = 2.81g/mL, Ellipticine, IC50 = 1.46g/mL;
NCI-H187, IC50 = 11.04g/mL Ellipticine, IC50 = 0.39g/mL)[1619]. Source:
DAO NIAN ZI Garcinia mangostana (fruit hull), DAO NIAN ZI Garcinia
H
O
mangostana (young fruit: yield = 0.030%dw)[1619], HUANG NIU MU
Cratoxylum cochinchinense (root), TIAN SHAN ZHU ZI Garcinia dulcis

(fruit). Ref: 1521, 1619, 3066, 4358, 4423, 5319.
OH
8225 Garciosaterpene B
C30H48O3 (456.72). White needles, mp 201~202C, []D29 = 121 (c = 0.008,
OH
O
HO
InRt = 38.1%). Source: MEI LI TENG HUANG Garcinia speciosa (trunk bark
and stems). Ref: 5491.
OH
8222 Garcinone E
C28H32O6 (464.56). Pharm: Cytotoxic (KB cancer cell lines, IC50 =
OH
2.67g/mL, control Ellipticine, IC50 = 1.33g/mL; BC-1, IC50 = 1.44g/mL,

Ellipticine, IC50 = 1.46g/mL; NCI-H187, IC50 = 3.74g/mL Ellipticine,
IC50 = 0.39g/mL)[1619]; cytotoxic (in vitro, HL-60, IC50 = 15.0mol/L)[4715].
Source: DAO NIAN ZI Garcinia mangostana (fruit hull, pericarp), DAO
H
HO
NIAN ZI Garcinia mangostana (young fruit: yield = 0.0078%dw)[1619]. Ref:

1619, 3066, 4715.
8226 Garciosaterpene C
C30H46O3 (454.70). White needles, mp 93~95C, []D29 = +125 (c = 0.008,
O
OH
InRt = 96.3%, IC50 = 12.2g/mL). Source: MEI LI TENG HUANG Garcinia
HO
speciosa (trunk bark and stems). Ref: 5491.
HO
OH
O
H
OH
8223 Garciosaphenone A
C33H42O6 (534.70). Yellow solid, mp 159~161C. Pharm: Anti-HIV-1 (HIV-1
reverse transcriptase assay, 200g/mL, InRt = 97.7%, IC50 = 23.9g/mL).
Source: MEI LI TENG HUANG Garcinia speciosa (trunk bark and stems).
H
O
Ref: 5491.
8227 Gardendiol
[160262-60-2] C10H14O4 (198.22). Source: ZHI ZI Gardenia jasminoides [Syn.
Gardenia florida]. Ref: 317, 1521.
OH
OH
HO
OH
OH
OH
O
O
O
H
HO
406
8228 Gardenin
8232 Gardnerilin A
5-Hydroxy-6,7,8,3',4',5'-hexamethoxy flavone [21187-73-5] C21H22O9 (418.40). mp
C35H66O8 (614.91). White amorphous powder, mp 94~95C, []D11 = +21.9 (c
163~164C. Source: ZHI ZI Gardenia jasminoides [Syn. Gardenia florida], YI ZHI
= 0.07, MeOH). Source: CHANG YE GE NA XIANG Goniothalamus
HAO Achillea alpina [Syn. Achillea sibirica]. Ref: 2, 33, 626.
gardneri. Ref: 774.

OH
OH
O
O
O
O
OH
O OH
OH
OH
O
OH
8233 Gardnerilin B
8229 Gardenolic acid A
C35H66O6 (582.91). White amorphous powder, mp 65~66C, []D11 = +12.78
C30H46O4 (470.70). Pharm: Anti-HIV-1 (syncytium assay: IC50 > 125g/mL,
(c = 0.11, MeOH). Source: CHANG YE GE NA XIANG Goniothalamus
EC50 = 110.0g/mL; HIV-1 RT assay: 200g/mL, InRt = 92.3%, IC50 <
gardneri. Ref: 774.
22.5g/mL, Fagaronine chloride IC50 = 10.9g/mL, Nevirapine IC50 =

1.8g/mL). Source: TAI GUO ZHI ZI Gardenia thailandica (leaf and twig).
Ref: 4963.
OH
[54835-76-6] C16H22O10 (374.35). Source: FEI LV BIN SHI ZI Gmelina

O
philippensis (aerial parts), ZHI ZI Gardenia jasminoides [Syn. Gardenia

OH
H
H
O
HO
8234 Gardoside
HO
OH
O OH
OH
O
8230 Gardenone
HO
OH
OH
OO
OH
OH
8235 Gartanin
H
C23H24O6 (396.44). Pharm: Cytotoxic (KB cancer cell lines, IC50 =
15.63g/mL, control Ellipticine, IC50 = 1.33g/mL; BC-1, IC50 = 15.54g/mL,
Ellipticine, IC50 = 1.46g/mL; NCI-H187, IC50 = 1.08g/mL Ellipticine, IC50

= 0.39g/mL)[1619], antioxidant (DPPH scavenger, 10mol/L, ScRt = 2%,
control BHT, 10mol/L, ScRt = 43%)[5319]. Source: DAO NIAN ZI Garcinia

8231 Gardenoside
mangostana (young fruit: yield = 0.0060%dw)[1619], TIAN SHAN ZHU ZI
[24512-62-7] C17H24O11 (404.37). mp 118~120C. Pharm: Laxative (mus, orl,
Garcinia dulcis (fruit). Ref: 1521, 1619, 3066, 5319.
ED50 = 1.2g/kg). Source: JING NI PING Genipa Americana (fruit), SHUI

ZHI Gardenia jasminoides var. grandiflora, ZHI ZI Gardenia jasminoides
OH
OH
[Syn. Gardenia florida] (dried ripe fruit: mean content = 3.75%[5508]). Ref: 2,
658, 4524, 5501, 5508.
O
OH
OH
O
O
H
8236 Gastrodamine
O
HO
OO
OH
OH
C14H15NO3 (245.28). Colorless acicular Crystals (CHCl3MeOH), mp

185~187C. Source: TIAN MA Gastrodia elata. Ref: 888.
OH
OH
N
OH
HO
OH
OH
407
8237 Gastrodin
8241 Gaultherin B
4-Hydroxybenzyl alcohol 4-O--D-glucopyranoside [62499-27-8] C13H18O7
(+)-Lyoniresinol-9,9'-diacetate C26H32O10 (504.54). White powder
(286.28). White solid, mp 96~98C, []D15 = 66.4 (water), soluble in water,
(acetone:water = 2:1), mp 120~121C, []D23 = +40 (c = 0.05, MeOH).
methanol, acetone, hot acetic ester, slightly soluble in ether.[5507] Source: LAN
Source: DIAN BAI ZHU SHU Gaultheria yunnanensis. Ref: 2295.
YU BAI JI Bletilla formosana (whole herb), SHAN HU LAN Galeola faberi,

SHI LUO ZI Anethum graveolens (fruit), TIAN MA Gastrodia elata (dried
O
O
tuber: content scope of 5 batch samples = 0.210%~0.943%, mean content =

0.467%[5513]). Ref: 4, 280, 4177, 4500, 5501, 5507, 5513.
HO
O
O
OO
HO
OH
OH
O
OH
OH
8242 Gaultheroside A
OH
(+)-Lyoniresinol-2-O--L-arabinopyranoside (D1) C27H36O12 (552.58). White

powder, mp 154~155C. Source: BAI ZHU SHU Gaultheria leucocarpa var.
8238 Gaudichaudic acid

C33H38O8 (562.67). Bright yellow amorphous powder, []D28 = 535, (c =
0.065, CHCl3). Pharm: Cytotoxic (hmn leukemia: doxorubicin-resistant K562,
IC50 = (0.610.05)g/mL, control Adriamycin, IC50 = (1.790.17)g/mL;
drug-sensitive K562, IC50 = (0.410.03)g/mL, Adriamycin, IC50 =
(0.110.01)g/mL). Source: TENG HUANG SHU Garcinia hanburyi (resin).
Ref: 1583.
cumingiana (root: content = 0.014%)[5508], DIAN BAI ZHU SHU Gaultheria

yunnanensis (root: content scope of 3 origins = 0.050%~0.128%, mean
content = 0.085%[5508]), FANG XIANG BAI ZHU Gaultheria fragrantissima
(root: content = 0.062%)[5508], SI LIE BAI ZHU Gaultheria tetramera (root:
content = 0.022%)[5508], WEI YE BAI ZHU Gaultheria griffithiana (root:
content = 0.045%)[5508]. Ref: 666, 5508.
OH
OH
O
HO
O
O
HO
OH
O
OH
OH
OH
OH
8243 GB1
8239 Gaudichaudione A
C33H38O7 (546.67). Yellow oil, []D = 571.7 (c = 0.1, CHCl3). Pharm:
Cytotoxic. Source: GAO DI CHA SHAN ZHU ZI Garcinia gaudichaudii.
[14736-58-4] C30H22O11 (558.50). Source: SHAN ZHU ZI Garcinia multiflora.

Ref: 6.
OH
Ref: 1521.
HO
O
O
O
HO
OH
OH
O
O
HO
OH
HO
OH
8240 Gaultherin A
8244 GB1a
5-Methoxy-(+)-isolariciresinol-9,9'-diacetate [243468-37-3] C25H30O9
(474.51). White powder (acetone:water = 2:1), mp 159~160C, []D23 = +30
Ref: 6.
(c = 0.08, MeOH). Source: DIAN BAI ZHU SHU Gaultheria yunnanensis.
OH
Ref: 2295.
O
O
HO
HO
O
O
O
OH
OH
O
OH
HO
OH
408
8245 GB2
8249 Gedunin
[2753-30-2] C28H34O7 (482.58). mp 157C, 218C. Source: KU LIAN PI
Ref: 6.
Melia azedarach. Ref: 6.

O
OH
O
HO
HO
OH
O
HO
O
OH
HO
O
OH
8250 Gein
8246 GB2a
Geoside [585-90-0] C21H30O11 (458.47). mp 146~147C, bp 183~184C.
Dihydromorelloflavone [18412-96-9] C30H22O11 (558.50). Buff powder, mp
Source: SHUI YANG MEI Geum japonicum, SHUI YANG MEI GEN Geum
214~216C (dec), []D = +28.2 (acetone). Pharm: Anti-HIV-1 RT (200g/mL,
japonicum. Ref: 6.
InRt = 96.0%, IC50 = 170mol/L); antiviral (EBV); antioxidant (DPPH radical

scavenger, 10mol/L, ScRt = 33%; control BHT, 10mol/L, ScRt = 43%, IC50
= 19.00mol/L)[4422]. Source: SHAN ZHU ZI Garcinia multiflora, TIAN
SHAN ZHU ZI Garcinia dulcis (flower). Ref: 6, 900, 1072, 4422.
OO
OO
OH
OH
OH
OH
OH
8251 Geissoschizine methyl ether
OH
O
OH
[60314-89-8] C22H26N2O3 (366.46). Pharm: Vasorelaxant (in vitro, isolated rat

aorta)[5341]; CNS activity (agonistic activity, against the central serotonergic
HO
HO
OH
receptor, binding to -adrenoceptor, 5-HT, dopamine and GABA receptors;
agonist of 5-HT1A receptor while blocking 5-HT2A receptor)[5341]. Source:

GOU TENG Uncaria rhynchophylla [Syn. Nauclea rhynchophylla]. Ref: 2,
OH
5341.
HO
OH
H
N
H
8247 GBB A
C43H44O6 (656.83). Source: CANG BAI QI SHE TAI Schistochila
N
H
glaucescens. Ref: 4549.
OH
8252 Gelsamydine
[120881-61-0] C29H36N2O6 (508.62). mp 194~196C, []D = 126.9C.
H
O
N
N
H OH
H
8248 GBB B
C43H44O6 (656.83). Source: CANG BAI QI SHE TAI Schistochila
O
H
glaucescens. Ref: 4549.

OH
8253 Gelsedine
[7096-96-0] C19H24N2O3 (328.41). mp 172.5~174.0C. Source: GOU WEN
O
O
N
H
409
8254 Gelselegine
8259 Gelsemiol 6'-trans-caffeoyl-1-glucoside
[131653-76-4] C20H26N2O4 (358.44). mp 167~168C, []D = 30. Source:
C25H32O12 (524.53). Colorless needle crystals (MeOH), mp 122~124C, []D27
GOU WEN Gelsemium elegans. Ref: 14.
= +3.4 (c = 0.23, MeOH). Pharm: Neurite outgrowth enhancer (PC12D cells,

NGF-mediated neurite outgrowth, to enhance the ability of NGF, may be
OH
H
O
useful in the treatment of neurological disorders, such as Parkinsons disease

(PD), Alzheimers disease (AD), Huntingtons disease (HD), amyotrophic
lateral sclerosis (ALS), and hmn immunodeficiency virus associated dementia
N
H
(HAD)). Source: HAI BIAN MA BIAN CAO Verbena littoralis (aerial parts).
Ref: 4383.
O
8255 Gelsemamide
O
[122297-34-1] C20H24N2O3 (340.43). mp 183~184C, []D = +228.3. Source:
H
OH

O
O
OO
O
OH
HO
O
NH
HO
OH
OH
8260 Gelsemoxonine
[135626-64-1] C19H22N2O5 (358.40). Powder, []D = 188.5. Source: GOU
8256 Gelsemicine
WEN Gelsemium elegans. Ref: 14.
[6887-28-1] C20H26N2O4 (358.44). mp 171C, []D24 = 140 (ethanol). Pharm:

Paralyses respiration (high dose); respiratory stimulant (low dose); uterine
stimulant; MLD (rbt, iv) = 0.08mg/kg. Source: CHANG LV GOU WEN
H
Gelsemium sempervirens. Ref: 661.

N
O H
NH2
H
O
N
H
8261 Gelseverine
[38990-03-3] C21H24N2O3 (352.44). Oil, []D = 4.5. Source: GOU WEN
8257 Gelsemine
O
Kiuminine [509-15-9] C20H22N2O2 (322.41). mp 178C. Pharm: Analgesic;
H
N
CNS stimulant; increases blood pressure (blocks decrease of blood pressure

due to injection of acetylcholine or electrostimulation of the vagus in heart);
toxin. Source: CHANG LV GOU WEN Gelsemium sempervirens, GOU WEN
Gelsemium elegans. Ref: 5, 6, 14, 658.
H
O
8262 Gemichalcone C
O
Isogemichalcone C; 3'-[-Hydroxymethyl (E)--methylallyl]-2,4,2',4'-tetra-
H
N
hydroxychalcone 11'-O-coumarate; Anticancer Flavonoid PMV70P691-020

C30H28O9 (532.55). Yellow powder (MeOH). Pharm: Cytotoxic (aromatase
H
O
N
H
inhibitor, a promising lead as potential cancer chemopreventive agents)[5038];
8258 Gelsemine N-oxide

[113900-76-8] C20H22N2O3 (338.41). Amorphous, []D = 16.9. Source:
H
N
N
H
aromatase inhibitor (in vitro, IC50 = 7.1mol/L; control Aminoglutethimide,

IC50 = 6.4mol/L) [3090]. Source: GOU SHU Broussonetia papyrifera, GOU
SHU Broussonetia papyrifera, SHUANG HUA JIN SI TAO Hypericum
geminiflorum. Ref: 3090, 3493, 5038.
O
OH
OH
OH
H
O
O
HO
OH
410
8263 Gemin A
8267 Genameside B
[82220-61-9] C82H56O52 (1873.33). Pharm: Antineoplastic (S180). Source:
C17H26O12 (422.39). Colorless syrup, []D26 = 63.8 (c = 1.9, MeOH). Source:
SHUI YANG MEI Geum japonicum. Ref: 658.
JING NI PING Genipa Americana (fruit). Ref: 4524.
OH
HO
O
O
HO
O
O
HO
HO
OH
HO
OH
O
O
OH
H
OO
OH
OH
HO
OH
OH
OH
OH
HO
OH
8268 Genameside C
OH
OH HO
HO
O
O
3.3, MeOH). Source: JING NI PING Genipa Americana (fruit). Ref: 4524.
OH
O
HO
Genipin -cellobioside C23H34O15 (550.52). White powder, []D26 = 0.4 (c =
OH
HO
HO
OH
O
OH
HO
OH
OH
HO
8264 Gemmacolide A
C30H39ClO14 (659.09). Source: DENG XIN LIU SHAN HU Junceella juncea
O
OO
OH
OH
OH
OH
H
HO
OO
OH
HO
(yield = 0.00018%). Ref: 4781.
HO
HO
HO
OH
8269 Genameside D
OH
10-O--D-Glucopyranosyl geniposide C23H34O15 (550.52). Colorless syrup,
Cl
[]D26 = +3.3 (c = 6.0, MeOH). Source: JING NI PING Genipa Americana
(fruit). Ref: 4524.
8265 Gemmacolide B
C33H45ClO14 (701.17). Source: DENG XIN LIU SHAN HU Junceella juncea

(yield = 0.00024%). Ref: 4781.
O
HO
OH
O
O
OH
OH
O
OO
O
O
H
OO
HO
OH
OH
Cl
O
O
OH
OH
8270 Geniculine
20-Ethyl-8-acetoxy-14-(p-hydroxybenzoyloxy)-1-,6,16,18-tetramethoxyac
onitane-3,13-diol C34H47NO11 (645.75). Amorphous powder, []D25.5 =
8266 Genameside A
+31.6 (c = 0.00372, CHCl3). Source: XI BAN WU TOU Aconitum
-Hydroxy-6,7-dihydrogardenoside C17H26O12 (422.39). Colorless syrup,
geniculatum. Ref: 2142.
[]D26 = 91.9 (c = 2.4, MeOH). Source: JING NI PING Genipa Americana

O
H
HO
HO
H
OO
OH
OH
OH
N
HO
H
O
O
O
O
H
O
HO
HO
OH
(fruit). Ref: 4524.
OH
411
8271 Genicunine A
8276 Geniposide
C22H35NO4 (377.53). White amorphous powder. Source: GONG GA SHAN
1--Glucogeniposide [24512-63-8] C17H24O10 (388.37). mp 163~164C.
WU TOU Aconitum liljestrandii. Ref: 2191.
Pharm: Analgesic (mus, ip, acetic acid-induced writhing model); laxative
(ED50 = 300mg/kg); cell growth inhibitor (transformed NIH3T3 cell line,
OH
25~100mol/L)[4979]. Source: AI LAI MU Cornus suecica, DU ZHONG
OH
Eucommia ulmoides (bark of 10 years old plant: content = 0.39%[5508]), GAN

DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa f.
N
OH
Huechingensis], JING NI PING Genipa Americana (fruit), SHUI ZHI

Gardenia jasminoides var. grandiflora, SHUI ZHI YE Gardenia jasminoides
var. grandiflora, WU SE MEI Lantana camara, ZHI ZI Gardenia jasminoides
8272 Genipic acid

27
[6902-76-7] C9H12O4 (184.19). []D = 105 (c = 1, ethanol). Pharm:

Antibacterial. Source: JING NI PING Genipa americana. Ref: 661.
[Syn. Gardenia florida] (dried ripe fruit: mean content = 3.25%[5508]), ZHI ZI
YE Gardenia jasminoides [Syn. Gardenia florida]. Ref: 2, 234, 658, 4524,
4979, 5501, 5508.
OH
HO
8273 Genipin
[6902-77-8] C11H14O5 (226.23). Pharm: Anticholinergic (mus ileum);
HO
HO
Source: ZHI ZI Gardenia jasminoides [Syn. Gardenia florida], JING NI

PING Genipa americana, DU ZHONG Eucommia ulmoides. Ref: 2, 658,
5501.
OH
antihistamine (gpg ileum); choleretic; inhibits gastric secretion

(pylorus-ligated rat); analgesic (mus, ip, acetic acid-induced writhing model).
OH
OH
8277 Geniposidic acid

[27741-01-1] C16H22O10 (374.35). Pharm: Laxative (ED50 > 800mg/kg).
Source: DU ZHONG Eucommia ulmoides (bark: mean content = 0.306%[5508]),
O
H
DU ZHONG YE Eucommia ulmoides (leaf: mean content = 0.085%)[5508], FEI
LV BIN SHI ZI Gmelina philippensis (aerial parts), JING NI PING Genipa

Americana (fruit), LONG CHUAN HUA Ixora chinensis, ROU CONG
RONG Cistanche deserticola, SHUI XIAN CAO Hedyotis corymbosa [Syn.
O
H
Oldenlandia corymbosa], ZHI ZI Gardenia jasminoides [Syn. Gardenia
OH
HO
florida] (dried ripe fruit: mean content = 0.29%[5508]). Ref: 2, 628, 658, 3954,
8274 Genipingentiobioside
4524, 5508.
OH
O
H
C23H34O15 (550.52). mp 193~195C (C2H5OH), 227~229C. Source: JING NI

PING Genipa Americana (fruit), SHUI ZHI Gardenia jasminoides var.
grandiflora, ZHI ZI Gardenia jasminoides [Syn. Gardenia florida] (dried ripe
fruit: mean content of 22 origins = 0.400%[5508]). Ref: 2, 4524, 5508.

O
HO
HO
O
H
OO
OH
OH
OH
OO
OH
OH
OH
OH
OH
OH
O
HO
OH
8278 Genistein
[446-72-0] C15H10O5 (270.24). mp 301~302C (dec). Pharm: Cytotoxic
cells)[5038]; cytotoxic (KB, ED50 = 7.4g/mL); cytotoxic (in vitro, Hs740T,
8275 Genipinic acid
ED50 = 4.38g/mL; Hs756T, ED50 = 5.82g/mL; Hs578T, ED50 = 3.5g/mL;
C11H14O6 (242.23). Very unstable moisture absorptive amorphous white
Hs742T, ED50 = 14.88g/mL; DU145, ED50 = 2.39g/mL; LNCaP-FGC, ED50
powder, []D26 = 126 (c = 1, ethanol). Pharm: Antibacterial. Source: JING
= 25.45g/mL)[4630]; antineoplastic (Inhibition of DMBA-induced
NI PING Genipa americana. Ref: 661.
preneoplastic lesions in vitro, MMOC assay, IC50 = 45.2mol/L; control

Sulforaphane, IC50 = 11mol/L)[4718]; catechol-O-methyltransferase inhibitor
O
HO
(competitive); histidine decarboxylase inhibitor (competitive); peroxidase

O
OH
O
inhibitor (competitive); lipase inhibitor (soy, competitive);

antihypercholesterolemic (rat, reduces the level of cholesterol and triglyceride
in serum, hyperlipemia caused by trinitrotoluene); CyP1A inhibitor (IC50 =
(4.90.5)mol/L)[5347]; QR inhibitor (cultured mouse Hepa1c1c7 cells, CD
412
= (17.18.5)mol/L, IC50 = (23.95.9)mol/L)[5347]; DPPH scavenger
8280 Genistein 7-O--D-glucopyranoside-4'-O-[(-D-glucopyranosyl)-
(SC50 > 250mol/L, 250mol/L scavenging rate = 2%)[5347];
(12)--D-glucopyranoside]
anti-Inflammatory (inhibit brain liposomal peroxidation, 62.5g/mL,
optical density of DMSO control = (52.80.3)%; positive control Propyl
(c = 0.001, DMSO). Source: HUAI Sophora japonica (pericarp). Ref: 3080.
gallate, 7.5mol/mL, optical density of DMSO control =

(20.60.2)%)[4984]; granular release inhibitor[4984]; hepatoprotective (mus
primary cultured hepatocytes, antihepatotoxin induced by
HO
O
HO
HO
D-galactosamine (GalN), IC50 = 29mol/L, control Silybin IC50 =
OH
41mol/L)[4095]; anti-inflammatory (modulator of cytokine network:
OH
HO
inhibits LPS-stimulated TNF- and IL-6 release in RAW264.7
HO
HO
HO
macrophages, IC50 = 5mol/L) [4416]; anti-inflammatory (NO production

inhibitor)[4415]; antioxidant (DPPH scavenger, TLC detection limit =
HO
HO
1.0g, IC50 = 1810g/mL; control Quercetin, TLC detection limit <
OH
0.05g, IC50 = 7g/mL; Gallic acid, TLC detection limit < 0.05g, IC50 =
4g/mL; Ascorbic acid, TLC detection limit < 0.10g, IC50 =
18g/mL)[3785]; antibacterial (Escherichia coli, MIA = 100.0g, control
Chloramphenicol, MIA = 0.001g; Staphylococcus aureus, MIA = 1.00g,
Chloramphenicol, MIA = 0.0001g; Bacillus subtilis, MIA = 5.00g,
Chloramphenicol, MIA = 0.0001g) [5247]; antifungal (Candida
mycoderma, MIA = 0.10g, control Miconazole, MIA = 0.0001g)[5247];
antioxidant (DPPH scavenger, TLC, MIA = 0.5g, IC50 = 354g/mL;
8281 Genistein 7-O--D-glucopyranoside-4'-O-[(-L-rhamnopyranosyl)(12)--D-glucopyranoside]

control Quercetin, MIA < 0.05g, IC50 = 7g/mL, Gallic acid, MIA <
0.05g, IC50 = 4g/mL; Ascorbic acid, MIA < 0.10g, IC50 =
18g/mL)
[5247]
. Source: DA DOU Glycine max (Soybean phytochemical
HO
O
HO
HO
OH
concentrate: yield = 0.013%dw)[4630] , DU HUI MAO DOU Tephrosia

[4718]
toxicaria (stem: yield = 0.000065%dw)
OH
, GE GEN Pueraria lobata
HO
[Syn. Pueraria thunbergiana; Pueraria pseudohirsuta], HONG CHE
HO
HO
ZHOU CAO Trifolium pratense, HUAI Sophora japonica, HUAI JIAO
Sophora japonica, HUANG HUA MU Piptanthus nepalensis, HUANG
HO
YU SHAN DOU Lupinus luteus, HEI DA DOU Glycine max, JI KUAN
O
OH
CI TONG Erythrina latissima (stem wood), PAN YUAN YU TENG
OH
Derris scandens (stem), RAN LIAO MU Genista tinctoria, SHAN DOU

GEN Sophora subprostrata [Syn. Sophora tonkinensis], Prunus sp., PAN
YUAN YU TENG Derris scandens (stem), GUANG BU DING GONG
TENG Erycibe expansa, Bolusanthus speciosus (root wood)[3785] . Ref: 2,
8282 Genistein 7-glucoside
4, 5, 658, 3785, 3810, 4095, 4416, 4415, 4630, 4718, 4984, 5038, 5247,
Genistin [529-59-9] C21H20O10 (432.39). mp 254~256C. Pharm: Estrogenic
5347.
activity ; inhibits growth of wheat coleoptile in vitro. Source: AI JING DOU
HO
Ulex nanus, DA DOU Glycine max (Soybean phytochemical concentrate:
yield = 0.011%dw)[4630], GE GEN Pueraria lobata [Syn. Pueraria

thunbergiana; Pueraria pseudohirsuta], HEI DA DOU Glycine max, HUAI
OH
Sophora japonica, HUAI Sophora japonica (pericarp)[3080], HUANG HUA
OH
MU Piptanthus nepalensis, HUANG YU SHAN DOU Lupinus luteus, RAN

LIAO MU Genista tinctoria. Ref: 6, 658, 660, 3080, 4630.
8279 Genistein 7-O--D-glucopyranoside-4'-O--D-glucopyranoside

C27H30O15 (594.53). Source: HUAI Sophora japonica (pericarp). Ref: 3080.
HO
HO
HO
OH
HO
OH
OH
O
HO
HO
HO
O
O
OH
OH
OH
OH
OH
413
8287 Genkwadaphnin
8283 Genistein 8-C-glucoside
[55073-32-0] C34H34O10 (602.64). Pharm: Daphne oleoides ssp. oleoides
[66026-80-0] C21H20O10 (432.39). Source: HUANG YU SHAN DOU Lupinus
luteus, GUANG LIANG HUANG TAN Dalbergia nitidula. Ref: 658.

O
HO
OH
O
OO
OH
HO
OH
OH
HO
OH
OH
OH
8288 Genkwadaphnin-20-palmitate
C50H64O11 (841.06). Amorphous powder, []D25 = +37.5 (c = 1.74, CHCl3).
8284 Genistein 7-O--L-rhamnopyranoside-4'-O-[(-D-glucopyranosyl)-
(12)--D-glucopyranoside]

O
HO
O
OO
O
O
OH
OH
OH
OH
HO
HO
HO
HO
HO
HO
8289 Genkwanin
4',5-Dihydroxy-7-methoxy flavone [437-64-9] C16H12O5 (284.27). mp 286C,
yl)-(12)--D-glucopyranoside]
293C. Pharm: Inhibits frog heart in vitro; inhibits intestinal and uterine
movement (animal in vitro); antihypertensive (dog, iv); uterine stimulant (dog,
iv); improves respiration (dog, iv). Source: CI CAO SU Phlomis pungens,
GUANG GUO GAN CAO Glycyrrhiza glabra, JI CHA KAI LA RUI A
Larrea divaricata, JIAO ZHI SHU WEI CAO Salvia glutinosa, MI DIE
XIANG Rosmarinus officinalis, SAN CHI LA RUI A Larrea tridentata, XI
YE YI MU CAO Leonurus sibiricus (aerial parts: yield = 0.00074%)[4744], YI
O
OH
OO
8285 Genistein 7-O--L-rhamnopyranoside-4'-O-[(-L-rhamnopyranos-
HO
HO
OH
MU CAO Leonurus heterophyllus [Syn. Leonurus artemisia] (aerial parts),

OH
OH
HO
HO
HO
YIN CHEN HAO Artemisia capillaris, YING TAO Prunus pseudocerasus,

YUAN HUA Daphne genkwa (dried bud: mean content of 19 origins =
0.390%[5535]). Ref: 2, 6, 658, 4493, 4744, 5501, 5508, 5535.
OH
HO
OH
OH
8286 Genkdaphin
OH
C20H16O7 (368.35). Colorless acicular Crystals, mp 118.0~119.5C, []D =

64.8 (c = 0.5, chloroform). Source: YUAN HUA Daphne genkwa. Ref: 175.
8290 Gentiacauleine
[15402-27-4] C15H12O6 (288.26). Pharm: Vasodilator (rat aortic preparations,
pre-contracted by 3mol/L arterenol, pIC50 = 5.000.03; pre-contracted by
O
O
20mol/L KCl, pIC50 = 4.900.15)
[5434]
. Source: XUE LONG DAN Gentiana
nivalis, KU HE LONG DAN Gentiana kochiana. Ref: 658, 5434.

O
H
O
O
H
O
HO
O
OH
414
8291 Gentialutine
8297 Gentianine
Venoterpine [17948-42-4] C9H11NO (149.19). mp 129~130C. Source: SHUI
[439-89-4] C10H9NO2 (175.19). mp 82~83C; mp 79~80C (ethanol)[5507].
CAI Menyanthes trifoliata, XI SHU Camptotheca acuminata, XI ZANG QIN
Pharm: Anti-inflammatory (arthritis induced by formaldehyde or egg white);
JIAO Gentiana tibetica. Ref: 6, 660, 1521.
antiulcerative; inhibits gastric secretion; bidirectional action to CNS system

(mus, central sedation at low dose, central stimulation at moderate dose and
HO
paralytic death at high dose); increases level of blood sugar (rat and mus, ip,
150~200mg/kg); inhibits frog heart in vitro; antihypertensive (gpg, anesthetic
dog and anesthetic rbt); reduces blood capillary permeability; antiallergic (rat,
protects against sensitive shock caused by egg white); Protects against

8292 Gentianadine
shock (gpg, induced by histamine); LD50 (mus, orl) = 460mg/kg, (mus, ip) =
[6790-32-5] C8H7NO2 (149.15). Pharm: Anti-inflammatory; antihypertensive;
350mg/kg, (mus, iv) = 250~300mg/kg, (mus, sc) 500mg/kg. Source: BAI
antipyretic; muscle relaxant; toxin. Source: AO LIE GE LONG DAN
HUA LONG DAN Gentiana algida, CU JING QIN JIAO Gentiana
Gentiana olgae, AO SHI LONG DAN Gentiana olivieri, TU ER QI SI TAN
crassicaulis (dried root: content = 0.41%[5508]), DA WU LI QIN JIAO
LONG DAN Gentiana turkestanorum. Ref: 658.
Gentiana dahurica (dried root: content = 0.89%[5508]), DIAN LONG DAN

Gentiana rigescens, GUAN HUA QIN JIAO Gentiana siphonantha (dried
root: content = 0.19%)[5508], HU LU BA Trigonella foenum-graecum, LONG

DAN Gentiana scabra, MA HUA JIAO Gentiana straminea (dried root:
content = 0.52%[5508]), QIN JIAO Gentiana macrophylla (dried root: content =

8293 Gentianaine
Gentiocrucine [58213-76-6] C6H7NO3 (141.13). mp 149~150C. Pharm:
Anti-inflammatory. Source: AO LIE GE LONG DAN Gentiana olgae, AO
1.43%[5508]), SHUI CAI Menyanthes trifoliata, TIAN SHAN QIN JIAO

Gentiana tianschanica, XI ZANG QIN JIAO Gentiana tibetica. Ref: 2, 4, 658,
660, 5501, 5507, 5508.
SHI LONG DAN Gentiana olivieri, GAO JIA SUO LONG DAN Gentiana
caucasa, TIAN SHAN QIN JIAO Gentiana tianschanica, TU ER QI SI TAN
LONG DAN Gentiana turkestanorum, ZHONG YA QIN JIAO Gentiana

kaufmanniana. Ref: 6, 658, 660.
O
8298 Gentianose
[25954-44-3] C18H32O16 (504.45). mp 209C. Source: LONG DAN Gentiana
NH2
O
scabra. Ref: 2.
8294 Gentianal
C10H11NO3 (193.20). Source: DIAN LONG DAN Gentiana rigescens. Ref: 2,
HO
660.
O
HO
O
OO
OH
OH
OH
O
OH
OH
OH
OH
OH
8295 Gentianamine
[22952-54-1] C11H11NO3 (205.22). Pharm: Anti-inflammatory. Source: AO
SHI LONG DAN Gentiana olivieri, TU ER QI SI TAN LONG DAN
8299 Gentiatibetine
[26005-36-7] C9H11NO2 (165.19). mp 161C. Source: SHUI CAI GEN
Menyanthes trifoliata. Ref: 6.
O
Gentiana turkestanorum. Ref: 658.

HO
OH
O
O
8300 Gentiobiose
8296 Gentianidine
[2202-12-2] C9H9NO2 (163.18). mp 131~132C. Source: DIAN LONG DAN
[5996-00-9] C12H22O11 (342.30). mp 190~195C. Source: ZANG HONG

HUA Crocus sativus. Ref: 6.
Gentiana rigescens, QIN JIAO Gentiana macrophylla, SHUI CAI

Menyanthes trifoliata. Ref: 2, 660.
O
HO
OO
OH
OH
OH
OH
O
O
HO
OH
OH
OH
415
8301 1-O-Gentiobiosyl-3,7-dimethoxy-8-hydroxyxanthone
20
content of 11 origins = 5.01%[15, 5508]), GUI ZHOU ZHANG YA CAI Swertia
C27H32O16 (612.55). Yellow Crystals, mp 184~186C, []D = 33.63 (c =
kouitchensis (whole herb: content = 3.61%)[5508], HONG HUA LONG DAN
0.33, DMSO). Source: XI DIAN ZHANG YA CAI Swertia punctata. Ref:
Gentiana rhodantha (root: mean content of 2 origins = 0.06%)[5508], HONG
2155.
ZHI ZHANG YA CAI Swertia erythrosticta (whole herb: content =

0.5081%)[5508], HUANG LONG DAN Gentiana lutea (the compound was
O
isolated from the plant by H.Inouye et al. in 1968)[5505], LONG DAN Gentiana
scabra (root: content scope = 1.28%~7.62%, mean content = 4.61%

O
HO
OO
OH
OO
OH
OH
[15, 5508]
),
MA HUA JIAO Gentiana straminea (dried root: mean content = 23.3%)[5508],

MAN ZHI LONG DAN Gentiana leptoclada (whole herb: content =
OH
0.01%)[5508], MAO ZHANG YA CAI Swertia pubescens (whole herb: content
OH
OH
OH
= 0.0158%)[5508], QIN JIAO Gentiana macrophylla (dried root: mean content

= 15.6%)[5508], SAN HUA LONG DAN Gentiana triflora (root: mean content
8302 Gentiodelphin
[84331-34-0] C51H53O28 (1113.97). Source: MU YE LONG DAN Gentiana
makinoi. Ref: 658.
= 3.68%[15, 5508]), TOU HUA LONG DAN Gentiana cephalantha (root:

content = 0.43%)[5508], XI NAN ZHANG YA CAI Swertia cincta (whole herb:
content = 0.06%)[5508], XIA YE ZHANG YA CAI Swertia angustifolia (whole
herb: content = 0.148%)[5508], XIAN MAI ZHANG YA CAI Swertia nervosa
OH
(whole herb: content = 0.13%)[5508], ZHANG YA CAI Swertia
HO
pseudochinensis (whole herb: content = 0.34%)[5508], ZHE JIANG ZHANG
O
OH
HO
YA CAI Swertia hickinii (whole herb: content = 1.84%)[5508], ZI HONG

O
OH
OH
+
HO
ZHANG YA CAI Swertia punicea (whole herb: mean content = 0.54%)[5508].
Ref: 2, 658, 660, 5501, 5505, 5508, 5534.

OH
OH
OH
O
OO
OH
OH
OO
HO
OH
OO
HO
OH
OH
OH
OH
8303 Gentioflavine
OH
OH
[18058-50-9] C10H11NO3 (193.20). mp 218~220C (dec). Source: LONG

DAN Gentiana scabra, TIAN SHAN QIN JIAO Gentiana tianschanica. Ref:
2, 660.
O
8305 Gentiopicroside tetraacetate

C24H28O13 (524.48). Source: LONG DAN Gentiana scabra. Ref: 2.
O
O
O
N
H
8304 Gentiopicroside
Gertiopicrin; Gentiopicrin [20831-76-9] C16H20O9 (356.33). mp 122C. Pharm:
Anti-inflammatory (swollen foot model caused by carrageenan); antiprotozoal

O
(plasmidium); gastric secretion promotor. Source: BAO JING ZHANG YA
O
O
CAI Swertia franchetiana (whole herb: content = 0.05%)[5508], BU SHI LONG

DAN Gentiana burseri, CHUAN DONG ZHANG YA CAI Swertia davidii
(whole herb: content = 0.13%)[5508], CU CAO LONG DAN Gentiana scabra
8306 Gentisein
var. buesgeri (root: mean content of 6 origins = 6.73%[5508]), CU HUA
1,3,7-Trihydroxyxanthone [529-49-7] C13H8O5 (244.21). Pharm: Antibacterial
ZHANG YA CAI Swertia fasciculata (whole herb: content = 0.054%) [5508],
(Mycobacterium tuberculosis). Source: CHAN YI TENG Securidaca
CU JING QIN JIAO Gentiana crassicaulis(root: mean content = 8.96%)[5534],
inappendiculata (stem), DI GEN JIN SI TAO Hypericum degenii, HUANG
CU ZHUANG LONG DAN Gentiana robusta (root: content = 3.63%)[5508],
LONG DAN Gentiana lutea. Ref: 658, 5238.
DA WU LI QIN JIAO Gentiana dahurica, DA ZI ZHANG YA CAI Swertia

macrosperma (whole herb: content = 0.02%)[5508], DAN HUANG ZHANG
HO
YA CAI Swertia punicea var. lutescens (whole herb: content = 0.0045%)[5508],

OH
DIAN LONG DAN Gentiana rigescens (root: mean content of 11 origins =

1.75%[15, 5508]), DONG BEI LONG DAN Gentiana manshurica (root: mean
OH
416
8307 Gentisic acid
Source: AN MO LE Phyllanthus emblica (branch and leaf)[3094], MAO GUO
[490-79-9] C7H6O4 (154.12). mp 204.5~205.0C. Pharm: Antibacterial;
QI Acer nikoense, GU KE Erythroxylum coca, RI BEN MA SANG Coriaria
antirheumatic and analgesic (sodium salt); antiviral. Source: DA CHE QIAN
japonica, YE WU TONG Mallotus japonicus, Geranium sp., Euphorbia sp.,
Plantago major, HUI XIANG JING YE Foeniculum vulgare, JU AN
Acer sp., Fuchsia sp. Ref: 658, 3094, 4416.
Eucalyptus grandis, JU YU Helianthus tuberosus, LAI FU Raphanus sativus,

LI MENG GEN Citrus limonia, LI MENG YE Citrus limonia, PU
(2)
TAO
OH
HO
cultivars, Gentiana sp. Ref: 6, 658, 660.

O
HO
HO
OH
OH
HO
OH
OO
O
HO
OH
OH
Vitis vinifera, SI ZI TAN Pterocarpus santalinus, ZAI PEI GAN JU Citrus
O
O
OH
O
O
H
O
HO
HO
OH
OH
OH
8308 Gephyromycin
8312 Geraniol
C19H18O8 (374.35). White crystalline solid (MeOH), mp 212C, []D20 = 51
Geranyl alcohol [106-24-1] C10H18O (154.25). mp 230C. Pharm: Antifungal
(c = 0.05, MeOH). Pharm: Glutaminergic agonist (neuronal cells)[5290].
(genus Trichophyton and Microsporum audouini, MIC = 0.39mg/mL); antiseptic;
Source: Streptomyces griseus. Ref: 5290.
anthelmintic (gpg, ascaricide); treatment of chronic bronchitis; antineoplastic

(leukemia); LD50 (rat, orl) = 4.8g/kg, (rbt, iv) = 50mg/kg. Source: BAN BIAN
SU Elsholtzia ciliata, CHAI HU Bupleurum chinense, DA MA SHI GE QIANG
WEI Rosa damascena, DA SUAN Allium sativum, FA GUO QIANG WEI Rosa
OH
OH
gallica, GAN JIANG Zingiber officinale, JIN YIN HUA Lonicera japonica, JIU
OH
LI XIANG Murraya paniculata [Syn. Chalcas paniculata], MANG NIU ER
OH
MIAO Erodium stephanianum, MEI GUI HUA Rosa rugosa, SHENG JIANG
Zingiber officinale, SHUI SONG Codium fragile, WU WEI ZI Schisandra
8309 Geraldone
chinensis, YUE GUI ZI Laurus nobilis, YUN XIANG CAO Cymbopogon
[21583-32-4] C16H12O5 (284.27). Pharm: Nodulation signal for metabiosis of
distans. Ref: 2, 4, 11, 638, 658, 660, 1582.
pea and Rhizobium leguminosarum. Source: DI XIA CHE ZHOU CAO

Trifolium subterraneum. Ref: 658.
OH
H
OH
HO
8313 Geranyl acetate

[105-87-3] C12H20O2 (196.29). bp 242~245C/764mmHg. Pharm: Insect
attractant. Source: TIAN MING JING Carpesium abrotanoides, HU LUO BO

Daucus carota var. sativa, HU LUO BO ZI Daucus carota var. sativa,
HUANG HAO Artemisia scoparia [Syn. Artemisia capillaris var. scoparia],

JU YUAN Citrus medica, MEI GUI HUA Rosa rugosa, NING MENG Citrus
8310 Gerambullol
limon, NING MENG PI Citrus limon, SHENG JIANG Zingiber officinale,
(E)-3-(Methylsulfonyl)-propenoic acid (2E,6E)-4-(8-hydroxy-3,7-dimethyl-
TIAN MING JING Carpesium abrotanoides, TU XIANG RU Origanum
2,6-octadienyloxy)-phenethyl amide C22H31NO5S (421.56). Colorless
vulgare, YE XIANG MAO Cymbopogon goeringii, YIN CHEN HAO
crystals (Et2O), mp 128~129C. Source: LV ZI SHAN XIAO JU Glycosmis
Artemisia capillaris. Ref: 6, 658, 660.
chlorosperma (leaf). Ref: 3956.

O
O
S
O
O
O
OH
N
O
8314 Geranyl N-Dimethylallylanthranilate

C22H31NO2 (341.50). Yellow oil. Pharm: Antibacterial (Staphyloccocus
aureus). Source: Esenbeckia yaaxhokob (leaf). Ref: 4929.
8311 Geraniin
[60976-49-0] C41H28O27 (952.66). Pharm: Inhibits adipose peroxidization (rat,

hepatic microsome); inhibits lipolysis (rat, adipose cells induced by adrenine);
promotes lipolysis (adipose cells induced by ACTH); TNF- release inhibitor
(BALB/3T3 cells, okadaic acid-stimulated, mean IC50 = 43mol/L)[4416] .
O
N
H
417
8315 2-Geranylemodin
8321 2-(1'-Geranyl-5'-hydroxy-2'-oxocyclohex-3'-enyl)acetic acid
C25H26O5 (406.48). Pharm: Cytotoxic (hmn small cell lung cancer
NCI-H187 cell line, IC50 = (3.080.73)g/mL, control Ellipticine, IC 50 =
Antiplasmodial (in vitro Plasmodium falciparum: D6, IC50 =
(0.350.15)g/mL). Source: QIAO MU ZHUANG HUANG NIU MU
1462.00ng/mL, control Mefloquine, IC50 = 11.67ng/mL; W2, IC50 =
Cratoxylum arborescens (stem cortex). Ref: 5061.
2552.94ng/mL, control Mefloquine, IC50 = 4.78ng/mL). Source:

Glossocalyx brevipes (leaf). Ref: 4973.
OH
OH
OH
HO
O
O
OH
8316 Geranylgeraniol
[24034-73-9] C20H34O (290.49). Source: YA MA Linum usitatissimum,
8322 4'-O-Geranylisoliquiritigenin
HONG CHUN Toona ciliata. Ref: 658.
C25H28O4 (392.50). Pharm: Antimalarial (antiplasmodial,

chloroquine-resistant W2 strain of Plasmodium falciparum, IC50 =
8.7mol/L, control Chloroquine, IC50 = 0.094mol/L, control Quinine, IC50
= 0.209mol/L; chloroquine-sensitive D6 strain of Plasmodium falciparum,
OH
8317 6-Geranylgeranyl 8'-methyl-6,8'-diapocaroten-6,8'-dioate
IC50 = 10.6mol/L, control Chloroquine, IC50 = 0.009mol/L, control
[247030-33-7] C43H60O4 (640.96). Source: HONG MU Bixa orellana (seed
Quinine, IC50 = 0.044mol/L). Source: Millettia usaramensis ssp.
coat). Ref: 2352.
usaramensis. Ref: 3454.
O
O
OH
OH
8318 6-Geranylgeranyl 6'-methyl-(9'E)-6,6'-diapocaroten-6,6'-dioate
C45H62O4 (666.99). Source: HONG MU Bixa orellana (seed coat). Ref: 2352.
8323 7-Geranyloxy-1,3-dihydroxyxanthone
O
H
O
C23H24O5 (380.44). Yellow needles (CH2Cl2hexane) mp 138~1408C.

O
Source: HUANG NIU MU Cratoxylum cochinchinense. Ref: 1907.
O
O
OH
8319 6-Geranylgeranyl 6'-methyl-(9'Z)-6,6'-diapocaroten-6,6'-dioate

C45H62O4 (666.99). Source: HONG MU Bixa orellana (seed coat). Ref: 2352.
OH
H
O
8324 5-Geranyloxy-7-hydroxycoumarin
O
C19H22O4 (314.38). Pharm: EBV-EA inhibitor (TPA-induced, IC50 = 331 Mol

O
8320 8-Geranyl-7-hydroxycoumarin
ratio/32 pmol TPA, control -Carotene, IC50 = 400 Mol ratio/32 pmol TPA).
Source: YUAN DONG JIU LI XIANG Murraya siamensis (leaf). Ref: 5255.
C19H22O3 (298.39). Source: DONG FENG JU GEN Atalantia buxifolia [Syn.

Severinia buxifolia] (root cortex). Ref: 3075.
OH
HO
O
418
8325 3-Geranyloxy-6-methyl-1,8-dihydroxyanthraquinone
8330 3'-Geranyl-2',3,4,4'-tetrahydroxychalcone
C25H26O5 (406.48). Yellow brown crystals, mp 120~121C. Pharm:
2',3,4,4'-Tetrahydroxy-3'-geranylchalcone C25H28O5 (408.50). Yellow powder,
Antitrypanosomal (Trypanosoma brucei, IC50 = (14.48.1)g/mL, control
mp 131~132C. Pharm: Antifungal (Cladosporium cladosporioides, TLC
Melarsoprol, IC50 = (0.00150.0009)g/mL; Trypanosoma cruzi, IC 50 >
bioautography method, 2g/spot, control Benlate)[3813]; antioxidant (DPPH
[5008]
90g/mL, control Benznidazole, IC50 = (0.390.15)g/mL)
scavenger, TLC bioautography method, 1g/spot, control Vitamin E,
antileishmanial (Leishmania donovani, IC50 = (12.01.0)g/mL, control
1g/spot)[3813]; 5-reductase inhibitor (IC50 = 104mol/L, control -Linolenic
Miltefosine, IC50 = (0.230.03)g/mL; Plasmodium falciparum, IC50 =
acid, IC50 =116mol/L)[3979]. Source: GAO GUI BO LUO MI Artocarpus
(25.61.4)g/mL, control Chloroquine, IC 50 = (0.0550.02)g/mL, control
nobilis (leaf), MIAN BAO GUO Artocarpus incisa [Syn. Artocarpus
Artemisinin, IC50 = (0.00110.0006)g/mL)[5008]; cytotoxic (L6, IC50 >
communis] (leaf). Ref: 3813, 3979.

OH
90g/mL, control Podophyllotoxin, IC50 = 0.0075g/mL; brine shrimp

lethality, IC50 = 21.3g/mL, control Cyclophosphamide, IC 50 =
HO
OH
16.33g/mL)[5008]; cytotoxic inactive (hmn small cell lung cancer NCI-H187

cell line, control Ellipticine, IC 50 = (0.350.15)g/mL)
[5061]
. Source: DONG
OH
FANG WEI SI MU Vismia orientalis (stem cortex), QIAO MU ZHUANG

HUANG NIU MU Cratoxylum arborescens (stem cortex). Ref: 5008, 5061.
OH
OH
8331 Gerardianin A
C24H32O7 (432.52). mp 135C. Source: XIA JI XIAN WEN XIANG CHA CAI
Isodon lophanthoides var. gerardiana. Ref: 4067.
OH
O
O
8326 8-Geranyloxy psoralen

C21H22O4 (338.41). mp 51~53C. Source: YUN NAN QIANG HUO
Pleurospermum rivulorum. Ref: 551.
8332 Gerardianin B
O
C24H32O7 (432.52). mp 158C. Source: XIA JI XIAN WEN XIANG CHA CAI
Isodon lophanthoides var. gerardiana. Ref: 4067.
O
O
8327 Geranyloxy sinapyl alcohol
C21H30O4 (346.47). Pharm: Cytotoxic (in vitro, A549, IC50 = 34mol/L;

HL-60, 6.7mol/L; KB, 3.0mol/L). Source: LIAN YE TUO WU Ligularia
nelumbifolia (root, yield = 0.0040%dw). Ref: 4632.

O
OH
8333 Gerberinol I
HO
[84153-78-6] C21H16O6 (364.36). Acicular crystals, mp 262~264C. Pharm:
8328 Geranyloxy sinapyl aldehyde
Antibacterial (Staphylococcus aureus, MIC 125g/mL). Source: DA DING
C21H28O4 (344.45). Pharm: Cytotoxic (in vitro, A549, IC50 = 22mol/L;
CAO Gerbera anandria [Syn. Leibnitzia anandria]. Ref: 77, 921, 1121.
OH
HL-60, 12mol/L; KB, 2.6mol/L). Source: LIAN YE TUO WU Ligularia
OH
nelumbifolia (root, yield = 0.0018%dw). Ref: 4632.

O
O
O
O O
8334 Gerberinside
O
[76474-54-9] C16H18O8 (338.32). Acicular crystals, mp 153~154C, [] D21 = 109
O
H
(c = 0.127, methanol). Pharm: Antibacterial (Bacillus pyocyaneus, infected mus, in

vivo, survival rate = (57.8~71.0)%, ED50 = 46.2mg/kg, in vitro no effects). Source:
8329 9-Geranyl-terpineol
C20H34O (290.49). Colorless oil, []D
31.2
= 51.3 (c = 0.046, MeOH). Source:
DA DING CAO Gerbera anandria [Syn. Leibnitzia anandria]. Ref: 900.
DI ER CAO Hypericum japonicum. Ref: 762.

OH
HO
OH
OH
O
O
OH
419
8335 5E,10(14)-Germacradien-1,4-diol
8341 Germacra-1(10),4,11(13)-trien-12-ol
C15H26O2 (238.37). Colorless prisms (n-hexaneEtOAc), mp 120~122C.
C15H24O (220.36). Colorless or slight-yellow oil. Source: MU XIANG
Pharm: Antiplasmodial (Plasmodium falciparum strains, IC50 = 1.63g/mL,
Saussurea lappa [Syn. Aucklandia lappa]. Ref: 5190.
control Chloroquine, IC 50 = 0.0028g/mL)[2383]. Source: YI NIAN PENG

Erigeron annuus (aerial parts), SU MEN BAI JIU CAO Erigeron sumatrensis
(aerial parts), Reneilmia cincinnata (fruits). Ref: 2383, 4338.
OH
OH
8342 (+)-Germacrene A1
C15H24 (204.36). Colorless oil. Source: MU XIANG Saussurea lappa [Syn.
OH
Aucklandia lappa]. Ref: 5190.
8336 1(10)E,5E-Germacradien-4-ol
C15H26O (222.37). Brown oil, []D26 = 118 (c = 0.80, CHCl3). Pharm:
Antiplasmodial (Plasmodium falciparum strains, IC50 = 1.54g/mL, control
Chloroquine, IC50 = 0.0028g/mL). Source: Reneilmia cincinnata (fruits). Ref:
2383.
8343 Germacrene B
[15423-57-1] C15H24 (204.36). Source: CHENG ZI PI Citrus junos. Ref: 6.
OH
8337 Germacranolide
C17H22O4 (290.36). Source: YUE GUI ZI Laurus nobilis. Ref: 6.
O
O
8344 Germacrene D
[23986-74-5] C15H24 (204.36). Source: CHENG ZI PI Citrus junos. Ref: 6.
O
O
8338 Germacra-1(10),4,11(13)-trien-12-al
C15H22O (218.34). Slight-yellow oil with strong mossy odor.
Source: MU XIANG Saussurea lappa [Syn. Aucklandia lappa]. Ref: 5190.
8345 1-cis,5-cis Germacrone

C15H22O (218.34). bp 100C/1mmHg. Source: MAN SHAN HONG
H
Rhododendron dauricum. Ref: 6.
8339 Germacra-1(10),4,11(13)-trien-12-oic acid

C15H22O2 (234.34). White crystals. Source: MU XIANG Saussurea lappa
H
O
[Syn. Aucklandia lappa]. Ref: 5190.
HO
8346 1-cis,5-trans Germacrone
8340 Germacra-1(10),4,7(11)-trien-9-ol
C15H22O (218.34). bp 100C/1mmHg. Source: MAN SHAN HONG
C15H24O (220.36). bp 62~63C/13mmHg. Source: XI XIN Asarum sieboldii.
Rhododendron dauricum. Ref: 6.
Ref: 6.
OH
H
O
H
420
8347 1-trans,5-trans Germacrone
8352 Germerine
1(10)E,4E-Germacrone C15H22O (218.34). Pharm: NO production inhibitor
[508-67-8] C37H59NO11 (693.88). mp 193~195C (dec). Source: LI LU
(mus peritoneal macrophages, induced by LPS, 100mol/L, InRt =
Veratrum nigrum. Ref: 6.
(32.71.3)%, control L-NMMA, 100mol/L, InRt = (79.20.9)%,

p<0.01)[4150]; antitussive (mus); LD50 = (mus, orl) = 970mg/kg. Source: MAN
SHAN HONG Rhododendron dauricum (leaf: content scope =
[5501]
0.045%~0.060%)
, PING E SHU Curcuma zedoaria [Syn. Curcuma
aeruginosa]. Ref: 4150, 5501.
OH
OH
OH
H
OH
OH
H
OH
O
8353 Germine
8348 (+)-Germacrone 4,5-epoxide
[508-65-6] C23H47NO8 (509.65). Pharm: Causes arrhythmia and bradycardia;
antihypertensive. Source: LV LI LU Veratrum viride. Ref: 658.

N
H
HO
8349 Germanaism A
OH
OH
OH
OH
H
OH
OH
Iriskashmirianin 4'-O--D-glucoside C24H24O12 (504.45). White amorphous

solid, mp 187 C, []D24 = +61.6 (c = 0.83, MeOH). Source: DE GUO YUAN
8354 Gerontoxanthone A
WEI Iris germanica (rhizome). Ref: 4223.
C23H22O6 (394.43). Pharm: Cytotoxic (HSC-2 cells, CC50 > 0.51mmol/L; HGF,
CC50 > 0.51mmol/L). Source: GOU JI Cudrania cochinchinensis (root: yield
= 0.00095%dw). Ref: 3025.
O
O
O
O
HO
OH
OH
OH
8350 Germanaism B
Nigricin 4'-O--D-glucoside C23H22O11 (474.43). Amorphous solid, []D24 =
+50.2 (c = 0.57, MeOH). Source: DE GUO YUAN WEI Iris germanica
OH
8355 Gerontoxanthone B
C23H22O6 (394.43). Pharm: Cytotoxic (HSC-2 cells, CC50 = 0.39mmol/L; HGF,
OH
OH
O
OH
8351 Germanicol
[465-02-1] C30H50O (426.73). mp 175~176C (MeOHCHCl 3), lit. (Yamada
et al., 1965) 176~177C, []D25 = +6.0. Source: SHAN WO JU Lactuca
indica, XIE WEI JU Koelpinia linearis (aerial parts). Ref: 6, 3912.
OH
OH
8356 Gerontoxanthone E
C24H26O6 (410.47). []D20 = +2.2 (c = 0.5, MeOH). Source: ZHE TENG
Cudrania fruticosa (root). Ref: 5074.
O
OH
HO
= 0.00017%dw). Ref: 3025.
HO
OH
HO
O
OH
421
8357 Gerontoxanthone G
8361 Gerronemin B
C23H24O6 (396.44). Pharm: Cytotoxic (HSC-2 cells, CC50 > 0.51mmol/L; HGF,
1,2-Dihydroxy-3-[12-(2,3-dihydroxyphenyl)-(Z)-dodec-4-enyl]benzene
C24H32O4 (384.52). Colorless oil. Pharm: Cytotoxic (HL-60 IC50 = 2.5g/mL,
= 0.0024%dw). Ref: 3025.
U937 IC50 = 3~4g/mL, L1210 IC50 = 2.5g/mL, COS-7 IC50 = 15g/mL,

HeLa-S3 IC50 > 40g/mL; inhibits cellular macromolecular biosyntheses);
anti-inflammatory (blocks inducible expression of proinflammatory enzymes
OH
hCOX-2 and iNOS promoter driven reporter gene, IC50 = 1~5mg/mL). Source:
Gerronema spp. Ref: 2022.
HO
OH
H
H
OH
8358 Gerontoxanthone H
OH

OH
CC50 = 0.20mmol/L). Source: GOU JI Cudrania cochinchinensis (root: yield

OH
= 0.00062%dw). Ref: 3025.
8362 Gerronemin C
1,2-Dihydroxy-3-[14-(2,3-dihydroxyphenyl)tetradecyl]benzene C26H38O4
O
(414.59). Colorless oil. Source: Gerronema spp. Ref: 2022.
OH
HO
OH
OH
OH
OH
OH
8359 Gerontoxanthone I
8363 Gerronemin D
1,2-Dihydroxy-3-[14-(2,3-dihydroxyphenyl)-(Z)-tetradec-6-enyl]benzene
C26H36O4 (412.57). Colorless oil. Pharm: Cytotoxic (HL-60 IC50 = 4g/mL,
= 0.00115%dw). Ref: 3025.
U937 IC50 = 1~2g/mL, L1210 IC50 = 2.5g/mL, COS-7 IC50 = 15g/mL,

HeLa-S3 IC50 > 40g/mL; inhibits cellular macromolecular biosyntheses);
anti-inflammatory (blocks inducible expression of proinflammatory enzymes
OH
hCOX-2 and iNOS promoter driven reporter gene, IC50 = 1~5mg/mL). Source:
Gerronema spp. Ref: 2022.
HO
OH
OH
H
H
OH
OH
8360 Gerronemin A
1,2-Dihydroxy-3-[12-(2,3-dihydroxyphenyl)dodecyl]benzene C24H34O4
(386.54). Colorless oil. Pharm: Cytotoxic (HL-60 IC50 = 2.5g/mL, U937 IC50
OH
OH
= 1~2g/mL, L1210 IC50 = 2.5g/mL, COS-7 IC50 = 15g/mL, HeLa-S3 IC50 >
8364 Gerronemin E
40g/mL; inhibits cellular macromolecular biosyntheses); anti-inflammatory
1,2-Dihydroxy-3-[14-(2,3-dihydroxyphenyl)-(Z,Z)-tetradeca-3,6-dienyl]benze
(blocks inducible expression of proinflammatory enzymes hCOX-2 and
ne C26H34O4 (410.56). Colorless oil. Pharm: Cytotoxic (HL-60 IC50 =
iNOS promoter driven reporter gene, IC50 = 1~5mg/mL). Source: Gerronema
2.5g/mL, U937 IC50 = 2g/mL, L1210 IC50 = 2.5g/mL, COS-7 IC50 =
spp. Ref: 2022.
15g/mL, HeLa-S3 IC50 > 40g/mL; inhibits cellular macromolecular

biosyntheses). Source: Gerronema spp. Ref: 2022.
OH
OH
OH
OH
OH
H
OH
OH
OH
422
8365 Gerronemin F
8370 Gesneroidin E
1,2-Dihydroxy-3-[16-(2,3-dihydroxyphenyl)-(Z,Z)-hexadeca-5,8-dienyl]benze
C30H42O11 (578.66). mp 149~151.5C, []D = 4.5 (c = 0.50, CHCl3). Source:
ne C28H38O4 (438.61). Colorless oil. Pharm: Cytotoxic (HL-60 IC50 =
JU TAI XIANG CHA CAI Isodon gesneroides. Ref: 4067.
4~5g/mL, U937 IC50 = 1.5g/mL, L1210 IC50 = 2.5g/mL, COS-7 IC50 =

15g/mL, HeLa-S3 IC50 > 40g/mL; inhibits cellular macromolecular
biosyntheses); anti-inflammatory (blocks inducible expression of
proinflammatory enzymes hCOX-2 and iNOS promoter driven reporter gene,

O
IC50 = 1~5mg/mL). Source: Gerronema spp. Ref: 2022.

OH
H
O
HO
H
H
OH
OH
O
8371 Gibberellin A1
[545-97-1] C19H24O6 (348.40). mp 255~258C (dec). Source: YU JIN XIANG
OH
Tulipa gesneriana, YU JIN XIANG GEN Tulipa gesneriana. Ref: 6.

8366 Gesneroidin A
C22H32O4 (360.50). mp 167C, []D = 130.9 (c = 0.84, CHCl3). Source: JU
O
HO
HO
H
H
TAI XIANG CHA CAI Isodon gesneroides. Ref: 4067.
OH
H
O
OH
8372 Gibberellin A3
Gibberellic acid [7700605] C19H22O6 (346.38). Crystals (ethyl acetate), mp

233~235C (blister), []D19 = +86 (c = 2.12). Pharm: Estrogenic activity
8367 Gesneroidin B
(female rat, ovariotomy model, 35mg/kgd for 7 days, effectively treats
C22H30O4 (358.48). mp 186C, []D = +17.9 (c = 1.12, CHCl3). Source: JU
uterine atrophy); phytohormone. Source: QIAN NIU ZI Pharbitis nil, YUAN
YE QIAN NIU ZI Pharbitis purpurea. Ref: 6, 658, 660.
O
H
H
HO
OH
H
O
OH
8373 Gibberellin A5
8368 Gesneroidin C
C28H38O10 (534.61). mp 202C, []D = 69.5 (c = 0.92, CHCl3). Source: JU
[561-56-8] C19H22O5 (330.38). mp 260~261 (dec). Source: QIAN NIU ZI
Pharbitis nil, YUAN YE QIAN NIU ZI Pharbitis purpurea, YU JIN XIANG
22
GEN Tulipa gesneriana. Ref: 6, 660.
O
O
OH
O
H
H
O
O
O
OH
OH
8374 Gibberellin A8
8369 Gesneroidin D
[7044-72-6] C19H24O7 (364.40). mp 210~215C (dec). Source: YU JIN
C28H38O9 (518.61). mp 129.5~130.5C, []D = +8.67 (c = 0.75, CHCl3).
XIANG GEN Tulipa gesneriana, YUAN YE QIAN NIU ZI Pharbitis
Source: JU TAI XIANG CHA CAI Isodon gesneroides. Ref: 4067.
purpurea. Ref: 6, 660.
O
O
O
HO
O
H
O
O
O
O
O
HO
H
OH
H
O
OH
423
8375 Gibberellin A9
8380 Gigantol
[427-77-0] C19H24O4 (316.40). mp 208~211C. Source: YU JIN XIANG GEN
C16H18O4 (274.32). Pharm: Platelet aggregation inhibitor (50mol/L, InRt =
Tulipa gesneriana. Ref: 6.
10%; 100mol/L, InRt = 31%). Source: MI HUA SHI HU Dendrobium

densiflorum (stem). Ref: 5171.
OH
O
H
O
OH
OH
8376 Gibberellin A13

Fujic acid [2922-24-9] C20H28O7 (380.44). mp 194~196C (dec). Source: YU
8381 Gigantriocin
JIN XIANG GEN Tulipa gesneriana. Ref: 6.
[134955-490] C35H64O6 (580.90). mp 69~71C, []D25 = +18 (CHCl3) Source:

JIN PING GE NA XIANG Goniothalamus leiocarpus, DA GE NA XIANG
HO
Goniothalamus giganteus. Ref: 420, 1521.
OH
HO
HO
H
O
OH
OH
OH
O
O
8377 Gibberellin A20

[19143-87-4] C19H24O5 (332.40). Source: QIAN NIU ZI Pharbitis nil, WAN
8382 [6]-Gingediacetate
DOU Pisum sativum, YUAN YE QIAN NIU ZI Pharbitis purpurea. Ref: 6,
C21H32O6 (380.49). Source: SHENG JIANG Zingiber officinale. Ref: 2.
660.
O
O
O
OH
H
O
HO
OH
8383 [6]-Gingediol
8378 Gigaconitine
[53318-09-5] C17H28O4 (296.41). Source: SHENG JIANG Zingiber officinale.
C24H39NO7 (453.58). Colorless needles, mp 164~166C (acetone). Source: JI
Ref: 2.
LIN WU TOU Aconitum kirinense. Ref: 2515.

OH
OH
OH
O
OH
N
O
HO
8384 [8]-Gingediol
OH
OH

Ref: 2.
8379 Gigantetronenin
C37H66O7 (622.93). Pharm: Cytotoxic (in vitro HepG2, EC50 = 0.086 g/mL,
OH
Hep3B, EC50 = 3.85g/mL; control Doxorubicin, HepG2, EC50 = 0.38g/mL,

Hep3B, EC50 = 0.36g/mL). Source: SHAN FAN LI ZHI Annona montana
(seed). Ref: 5035.
OH
O
OH
8385 [10]-Gingediol
H
O
O
HO
OH

Ref: 2.
H
OH
OH
HO
O
OH
OH
424
8386 [6]-Gingerdione (enol form)
8392 Gingerglycolipid B
[61871-71-4] C17H24O4 (292.38). Pharm: Prostaglandin biosynthesis inhibitor
C33H58O14 (678.82). White amorphous powder, []D = +50.9 (c = 7.5, MeOH).
(in vitro). Source: SHENG JIANG Zingiber officinale, GAN JIANG Zingiber
Pharm: PAF antagonist. Source: XI LAN ROU GUI Cinnamomum zeylanicum.
officinale. Ref: 2, 658.
Ref: 2199.
OH
OO
HO
OH
OH
OH
8387 [6]-Gingerdione (keto form)
OO
HO
OH
OH
C17H24O4 (292.38). Source: GAN JIANG Zingiber officinale. Ref: 2.
OH
OH
8393 Gingerglycolipid C
O
C33H60O14 (680.84). White amorphous powder, []D = +26.9 (c = 10.0,

MeOH). Pharm: PAF antagonist. Source: XI LAN ROU GUI Cinnamomum
zeylanicum. Ref: 2199.
OH
8388 [10]-Gingerdione
C21H32O4 (348.49). Pharm: Anti-inflammatory (prostaglandin biosynthesis
inhibitor, IC50 = 4.9mol/L); antihepatotoxin (rat liver cells, in vitro,
1.0mg/mL, liver toxicosis induced by CCl4 GPT = (722)%, P<0.01); inhibits
onset of senility (inhibits formation of active oxygen); prostaglandin
OO
HO
OH
OH
OO
HO
OH
synthetase inhibitor (IC50 = 2.0mol/L). Source: GAN JIANG Zingiber
OH
OH
H
O
OH
officinale. Ref: 2, 1815, 1816, 1817, 1818.
8394 [4]-Gingerol
O
OH

O
OH
OH
8389 Gingerenone A
Dehydroxytetrahydrocurcumin [128700-97-0] C21H24O5 (356.42). Pharm:
Antifungal (in vitro). Source: GAN JIANG Zingiber officinale, SHENG
HO
JIANG Zingiber officinale. Ref: 2, 658.

8395 [6]-Gingerol
C17H26O4 (294.39). bp 277~279C/6mmHg. Pharm: CYP3A4 inhibitor (IC50 =
O
O
36.4mol/L, control Ketoconazole, IC50 = 0.245mol/L)[4669]; CYP2D6

inhibitor inactive (IC50 > 100mol/L, control Quinidine, IC50 =
OH
HO
0.078mol/L)[4669]; antemetic; anti-seronine; cyclo-oxygenase inhibitor.
8390 Gingerenone B
Source: FANG XIANG JIANG Zingiber aromaticum (rhizome: yield =
[128700-98-1] C22H26O6 (386.45). Source: GAN JIANG Zingiber officinale,
0.0023%dw)[4669], GAN JIANG Zingiber officinale, SHENG JIANG Zingiber
officinale (rhizome: mean content of 4 origins = 0.700%[5508]). Ref: 2, 6, 658,

4669, 5508.
O
O
O
OH
HO
O
HO
8396 [8]-Gingerol
8391 Gingerenone C
[128701-01-9] C20H22O4 (326.40). Source: GAN JIANG Zingiber officinale,
Ketoconazole IC50 = 0.24mol/L)[4449]; CYP2D6 inhibitor (IC50 = 68.7mol/L,

control Quinidine IC50 = 0.068mol/L)[4449]. Source: FANG XIANG JIANG
Zingiber aromaticum (rhizome), GAN JIANG Zingiber officinale. Ref: 2, 4449.
O
O
HO
OH
OH
HO
OH
425
8397 [10]-Gingerol
harringtonia, SAN JIAN SHAN Cephalotaxus fortunei, YUAN ZHI JUAN
BAI Selaginella sanguinolenta (dried whole herb: content = 0.363%)[5508],
Ketoconazole IC50 = 0.24mol/L)[4449]; CYP2D6 inhibitor inactive (IC50 >
ZHI MU Anemarrhena asphodeloides, Dacrydium sp. Ref: 2, 442, 658, 4415,
100mol/L, control Quinidine IC50 = 0.068mol/L)[4449]. Source: FANG
5501, 5505, 5508.
XIANG JIANG Zingiber aromaticum (rhizome), GAN JIANG Zingiber
OH
officinale. Ref: 2, 4449.

OH
HO
OH
HO
OH
8398 [12]-Gingerol
C23H38O4 (378.56). Source: GAN JIANG Zingiber officinale. Ref: 2.
8402 Ginkgetin 7''-O--D-glucopyranoside

C38H32O15 (728.67). Yellow amorphous powder, []D20 = +5.5 (c = 0.004,
OH
MeOH). Source: BAI GUO YE Ginkgo biloba. Ref: 4512.
OH
HO
8399 4-Gingesulfonic acid

O
C15H22O6S (330.40). Pale brownish amorphous powder, mp 180~190C (dec),

[]D21 = +1.0 (c = 2.00, MeOH). Source: SHENG JIANG Zingiber officinale.
Ref: 3361.
OO
HO
OH
OH
OH
OH
OH
OH
8403 Ginkgolic acid
HO
Ginkgoic acid [22910-60-7] C22H34O3 (346.51). Yellowish oil, mp 41~43C. Pharm:

Antibacterial (in vitro, Mycobacterium tuberculosis); antineoplastic; antimicrobial;
8400 6-Gingesulfonic acid

C17H26O6S (358.46). White amorphous powder, mp 177~181C (dec),
[]D21 = +0.7 (c = 1.00, MeOH). Source: SHENG JIANG Zingiber
officinale. Ref: 3361.
O
O
prostaglandin biosynthetase inhibitor; molluscacide; prolyl endopeptidase inhibitor

(Ki = 0.87)mol/L, IC50 = (0.860.04)mol/L, control Oleic acid IC50 =
(31.32.4)mol/L, Salicylic acid IC50 = (165070)mol/L, Z-Pro-prolinal IC50 =
(0.002190.00022)mol/L)[4098]. Source: BAI GUO Ginkgo biloba (dried ripe seed:
OH
O
content = 0.0222%[5508]), BAI GUO YE Ginkgo biloba, DU XIAN ZI Anacardium

occidentale. Ref: 4, 658, 4098, 5501, 5508.
O
OH
HO
OH
H
H
8401 Ginkgetin
[481-46-9] C32H22O10 (566.53). Yellow powder, mp 330C (dec). Pharm:
Antihypercholesterolemic (reduces the level of cholesterol in serum and
normalizes the ratio between phospholipid to cholesterol); treatment of angina
pectoris; phospholipase A2 inhibitor[4415]; anti-inflammatory (reduces
arthritic inflammation in rat adjuvant-induced arthritis as well as abdominal
constriction caused by acetic acid, ID50 = 8.9mg/kg)[4415] ; anti-inflammatory
(inhibits croton oil-induced ear skin oedema by down-regulation of
COX-2)[4415]; anti-inflammatory (NO production inhibitor)[4415]. Source:
BAI GUO Ginkgo biloba, BAI GUO YE Ginkgo biloba (leaf: mean content =
0.653%[5508]; the compound was first isolated from the plant by Kichi
Nakazawa in 1941[5505]), CHAO XIAN YIN YANG HUO Epimedium
koreanum, HAN SHENG JUAN BAI Selaginella stauntoniana (dried whole
herb: content = 0.164%)[5508], MAO ZHI JUAN BAI Selaginella braunii
(dried whole herb: content = 0.121%)[5508], RI BEN CU FEI Cephalotaxus
8404 Ginkgolide A
[15291-75-5] C20H24O9 (408.41). Crystals (ethanol), mp 300C, []D24 = 53.4 (c =
1, ethanol).[5507] Pharm: Enhances effects of cytotoxic drugs against cancer
metastasis; platelet aggregation inhibitor (rbt, due to PAF, in vitro, IC50 = 94mol/L);
insect antifeedant; PAF receptor antagonist; nerve protectant (mus, 50mg/kg),
Antiasthmatic; insect antifeedant. Source: BAI GUO Ginkgo biloba, BAI GUO
GEN Ginkgo biloba, BAI GUO YE Ginkgo biloba (leaf: mean content of 12
samples = 2.56%[5508]). Ref: 6, 658, 900, 5507, 5508
OH
O
H
O
O
O
O
H
O
OH
426
8405 Ginkgolide B
8409 Ginsenol
[15291-77-7] C20H24O10 (424.41). Crystals (ethanol), mp 300C, []D24 =
C15H26O (204.36). Source: REN SHEN Panax ginseng [Syn. Panax
52.6 (c = 1, ethanol).[5507] Pharm: Antibacterial (Bacillus fusiformis);
schinseng]. Ref: 5330.
enhances effects of cytotoxic drugs against cancer metastasis; increases

fertility; platelet aggregation inhibitor (rbt, mus and pig, due to PAF, in vitro);
insect antifeedant; PAF receptor antagonist; nerve protectant; reduces
H
OH
nephrotoxicity of cyclosporine; anti-hypotension (PAF-induced, ID50 =

(38.52.7)mol/kg, control CV-3988, ID50 = (2.41.2)mol/kg)[5050];
anti-inflammatory (to determine release of lysosome enzyme from
8410 Ginsenoside F1
polymorphonuclear (PMN) leukocytes induced by PAF of rats, 10mol/L,
C36H62O9 (638.89). Source: REN SHEN Panax ginseng [Syn. Panax
InRt = 58.9%)[3891, 5013]. Source: BAI GUO Ginkgo biloba, BAI GUO GEN
Ginkgo biloba, BAI GUO YE Ginkgo biloba (leaf: mean content of 12

samples = 1.40%[5508]). Ref: 6, 900, 3891, 5013, 5050, 5507, 5508.
OH
O
OH
OH
OH
O
OH
OH
OH
O
O
OO
HO
HO
OH
8406 Ginkgolide C
[15291-76-6] C20H24O11 (440.41). Crystals (ethanol), mp 300C, []D24 =
14.7 (c = 1, ethanol). Pharm: Platelet aggregation inhibitor (rbt, in vitro, due
to PAF, IC50 = 17mol/L); PAF receptor antagonist. Source: BAI GUO GEN
Ginkgo biloba, BAI GUO YE Ginkgo biloba (leaf: mean content of 12
samples = 1.48%[5508]). Ref: 6, 900, 5508.
OH
O
2)-O--D-glucopyranoside C42H70O12 (767.02). mp 177~180C, []D20 =

+10.8 (c = 0.5, MeOH). Source: REN SHEN Panax ginseng [Syn. Panax
schinseng]. Ref: 8.
OH
H
O
O
OH
3,6,12-Trihydroxy-20(22),24-dammardiene-6-O--L-rhamnopyranosyl(1
8411 Ginsenoside F4
OH
H
HO
OH
HO
8407 Ginkgolide J
OH
[107438-79-9] C20H24O10 (424.41). Crystals, mp 322C, []589nm20 = 2.5 (c =
OH
OH
O
O
1, dioxocyclohexane). Pharm: Platelet aggregation inhibitor (due to PAF);

PAF receptor antagonist. Source: BAI GUO Ginkgo biloba. Ref: 943, 1036,
1078.
OH OH
OH
O
O

OH
8412 Ginsenoside I
schinseng]. Ref: 8.
OH
O
O
HO
OH
8408 Ginkgolide M
OH
H
OH
[15291-78-8] C20H24O10 (424.41). Crystals (ethanol), mp > 280C (dec), []D
OH
= 39 (c = 1, dioxocyclohexane). Pharm: PAF receptor antagonist. Source:

BAI GUO GEN Ginkgo biloba. Ref: 6, 1035, 1036, 1164.
H
H
O
O
HO
OH
O
O
O
OH
OH
O
O
HO
OH
OH
OH
OH
OH
OH
427
8413 Ginsenoside Ia
8416 Ginsenoside II
20(S)-Protopanaxatriol-3,20-di-O--D-glucopyranoside C42H72O14 (801.03).
3-O--D-Glucopyranosyl-(12)-O--D-glucopyranosyl-20-O--D-glucopyr
White powder, mp 190~191C. Source: REN SHEN Panax ginseng [Syn.
anosyl-3,12,20(S)-trihydroxy-24-hydrogenperoxide-dammar-25-ene

schinseng]. Ref: 8.
HO
O
O
HO
OH
OH
H
OH
OH
OH
H
OH
OH
OO
OH
OH
H
HO
OH
H
O
O
HO
OH
OH
OH
OH
OH
O
O
HO
OH
OH
OH
8414 Ginsenoside Ib
3,12,20(S),24-Tetrahydroxy-20-O--D-glucopyranosyl-3-O--D-glucopyra
noside C42H72O14 (801.23). White powder, mp 187~188C. Source: REN
8417 Ginsenoside III
SHEN Panax ginseng [Syn. Panax schinseng]. Ref: 8.

schinseng]. Ref: 8.
HO
OH
OH
OH
H
OH
OH
OH
OH
OH
H
O
O
HO
OH
OO
HO
OO
HO
OH
OH
OH
OH
O
O
HO
OH
OH
OH
H
H
OH
8415 Ginsenoside Ic
3,6,12-Trihydroxy-20(22),24-dammar-20(H),24-diene-6-O--L-rhamnopy
ranosyl(12)-O--D-glucopyranoside C42H70O12 (767.02). White powder.
Source: REN SHEN Panax ginseng [Syn. Panax schinseng]. Ref: 8.
8418 Ginsenoside La
[123617-34-5] C42H70O13 (783.02). White powder (methanol), mp 179~180C,
[]D20 = 18.4 (pyridine). Source: REN SHEN Panax ginseng [Syn. Panax
OH
H
schinseng]. Ref: 155, 1521.

H
O
H
HO
H
HO
OH
OH
OH
O
O
H
HO
OO
OH
OH
OH OH
OH
HO
O
OH
OH
OH
428
8419 Ginsenoside Ra0
20(S)-Protopanaxadiol 3-O--D-glucopyranosyl-(12)--D-glucopyranosyl-
(12)--D-glucopyranoside, 20-O--D-glucopyranosyl-(12)--D-glucopy-
Panax schinseng]. Ref: 2, 1521.
noside [112722-00-6] C60H102O28 (1271.47). White acicular crystals, mp

HO
192~193C. Source: REN SHEN Panax ginseng [Syn. Panax schinseng], XI

YANG SHEN Panax quinquefolium. Ref: 2, 87.
HO
OO
OH
OH
OH
OH
OH
H
OH
HO
OO
OH
OH
O
HO
O
OH
H
OO
OH
OH
O
OH
H
OH
OH
OH
HO
OH
OH
OH
OH
HO
OO
OO
OH
OH
OH
OH
OH
OH
HO
8423 Ginsenoside Rb1
OO
Sanchinoside E1; Gypenoside III [41753-43-9] C54H92O23 (1109.32). White
OH
powder (ethanol:butyl alcohol = 1:1), mp 197~198C, []D22 = +12.42 (c =
OH
OH
0.91, methanol). Pharm: Antiarrhythmic (rat arrhythmia caused by BaCl2);

inhibits fatigue; antiviral; inhibits replication of HSV-1; bidirectional action to
blood pressure (mus, first increases and then lowers blood pressure, while

OO
O O
OH
OH
OH
OH
OH
OH
OH
644.8g/mL); cAMP phosphodiesterase inhibitor (in vitro, IC50 = 137mol/L);

antihypercholesterolemic (reduces the level of cholesterol in serum); promotes
OH
H
OO
OH
OH
HO
secretion of corticosterone (ED50 = 112mol/kg); liver and nerve protectant;

reduces uterine contraction (gpg, in vitro, caused by acetylcholine);
vasodilator (dog); anti-inflammatory (modulator of cytokine network: inhibits

TNF- production in RAW264.7 and U937 cells stimulated with LPS, .mean
IC50 = 56.5mol/Land 51.3mol/L, respectively)[4416]; antinociception (i.t.
OH
OH
biosynthesis of DNA, protein and lipid (murine marrow cells); enhances

cytotoxic effects of daunomycin and vincaleucoblastine; promotes plasma
H
HO
0.3L into lateral area of rat hypothalamus, average arteriotony noticeably

rising); antioxidant (rat hepatic homogenate, caused by H2O2, IC50 =
OH
heart rate slows); calcium antagonist; increases blood pressure (injecting
injected 0.7g substance P-induced pain model, EC = 50g i.t.)[5474]; neurite

OH
outgrowth enhancer (hmn neuroblastoma SK-N-SH cells, 100mol/L, total

length of neurites = 149.3m, number of varicosity per cell = 0.93, p<0.05;
control, total length of neurites = 45.3m, number of varicosity per cell =

0.10)[4647]; hepatoprotective (inhibits activation of macrophages, inhibits
increase in sALT and sAST levels, in vivo, D-GalN/LPS-induced liver injury

in mouse, 100mg/kg ip for sALT, InRt = 33%; 100mg/kg ip for sAST, InRt =
O
OH
HO
OO
O
OH
OH
H
OH OH
OH
OH
OO
OH
OO
yixingense, JIAO GU LAN Gynostemma pentaphyllum, REN SHEN Panax
H
H
0.56%[5501]), SAN QI HUA LEI Panax pseudo-ginseng var. notoginseng [Syn.

Panax notoginseng] (flower bud: yield = 0.24%dw)[4702], SAN QI Panax
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (flower: mean

notoginseng [Syn. Panax notoginseng] (rhizome: content = 4.1%)[5508], XI
YANG SHEN Panax quinquefolium (rhizome: content = 1.9%)[5508], YU YE
OH
OH
content of 8 origins = 1.60%)[5525], SAN QI Panax pseudo-ginseng var.
OH
HO
for sAST, InRt = 97%)[4702]. Source: HUI GUO JIAO GU LAN Gynostemma
ginseng [Syn. Panax schinseng] (rhizome: content = 0.88%[5508]; content =
OH
HO
40%; control Hydrocortisone, 20mg/kg ip for sALT, InRt = 99%; 20mg/kg ip
OH
SAN QI Panax japonicus var. bipinnatifidus, ZHU JIE SAN QI Panax
429
pseudo-ginseng var. japonicus (rhizome: content = 1.7%[5508], yield =
0.025%dw[4647]). Ref: 2, 4, 87, 135, 329, 613, 900, 4139, 4416, 4647, 4702,
[68406-26-8] C53H90O23 (1095.29). White powder, mp 193~195C, []D20 =
5474, 5501, 5508, 5525.
+19.4 (c = 1, MeOH). Pharm: Neurite outgrowth enhancer (hmn

neuroblastoma SK-N-SH cells, 100mol/L, total length of neurites = 131.4m,
HO
OO
OH
OH
OO
number of varicosity per cell = 0.80, p<0.05; control, total length of neurites =
OH
OH
H
OH
OH
OH
45.3m, number of varicosity per cell = 0.10)[4647]; hepatoprotective (inhibits
activation of macrophages, inhibits increase in sALT and sAST levels, in vivo,

D-GalN/LPS-induced liver injury in mouse, 50mg/kg ip for sALT, InRt = 77%,
100mg/kg ip for sALT, InRt = 91%; 50mg/kg ip for sAST, InRt = 72%;
H
HO
OO
100mg/kg ip for sAST, InRt = 80%; control Hydrocortisone, 20mg/kg ip for
OH
sALT, InRt = 99%; 20mg/kg ip for sAST, InRt = 97%)[4702]. Source: JIAO GU
LAN Gynostemma pentaphyllum (leaf: yield = 0.007%dw)[4757], REN SHEN
OH
HO
Panax ginseng [Syn. Panax schinseng], SAN QI HUA LEI Panax
OH
OH
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (flower bud: yield

= 3.15%dw)[4702], XI YANG SHEN Panax quinquefolium, YU YE SAN QI
OH
Panax japonicus var. bipinnatifidus, ZHU JIE SAN QI Panax pseudo-ginseng

var. japonicus (underground part: yield = 0.025%dw)[4647]. Ref: 135, 451,
4647, 4702, 4757.
[11021-13-9] C53H90O22 (1079.30). White powder (ethanol:butyl alcohol =1:5),
mp 200~203C, []D22 = +3.05 (c = 0.98, methanol), []D20 = +12.3 (c = 0.92,
OH
MeOH). Pharm: Antiarrhythmic (rat arrhythmia caused by BaCl2);
O
O
OH OH
OH
antineoplastic (inhibits mus melanoma lung metastasis and prevents new
OH
vessel formation); inhibits fatigue; antiviral; inhibits replication of HSV-1;
OH
H
OH
bidirectional action to blood pressure (murine, first increases and then lowers
blood pressure, while heart rate slows); calcium antagonist; hemolytic;
inhibits kidney damage in diabetic rat; platelet aggregation inhibitor; inhibits
content of free radicals in myocardial cells (induced by xanthinoxidase);
cAMP phosphodiesterase inhibitor (in vitro, IC50 = 199mol/L);
antihypercholesterolemic (reduces the level of cholesterol in serum); promotes
biosynthesis of DNA, protein and lipid (murine marrow cells); promotes RNA
polymerase activity (promotes synthesis of rRNA and mRNA in diabetic rat);
H
OO
HO
OH
OH
HO
OH
OO
OH
OH
OH
vasodilator (dog); anti-inflammatory (modulator of cytokine network: inhibits
8426 Ginsenoside Rc
TNF- production in RAW264.7 and U937 cells stimulated with LPS, .mean
[11021-14-0] C53H90O22 (1079.30). White powder (ethanol:butyl alcohol =
IC50 = 27.5mol/L and 26.8mol/L, respectively)[4416]; antinociception (i.t.
1:5), mp 199~201C, []D20 = +1.83 (c = 0.65, methanol). Pharm:
injected 0.7g substance P-induced pain model, EC = 50g i.t.)
[5474]
. Source:
Antiarrhythmic (rat arrhythmia caused by BaCl2); inhibits fatigue ;
REN SHEN Panax ginseng [Syn. Panax schinseng] (rhizome: content =
bidirectional action to blood pressure (murine, first increases and then lowers
blood pressure, while heart rate slows); calcium antagonist; antioxidant of rat
hepatic homogenate (caused by H2O2, IC50 = (265.548.1)g/mL, by FeSO4,
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (rhizome: content
IC50 = (129.35.6)g/mL, by H2O2 + FeSO4, IC50 = (536.8142.3)g/mL);
= 0.17%)[5508], XI YANG SHEN Panax quinquefolium (rhizome: content =
cAMP phosphodiesterase inhibitor (in vitro, IC50 = 264mol/L); promotes
0.10%[5508]). Ref: 4, 87, 451, 900, 4416, 4702, 5474, 5508.
biosynthesis of DNA, protein and lipid (murine marrow cells); promotes

plasma secretion of corticosterone (ED50 = 44mol/kg); antihepatotoxin
OH
OO
OH
OH
by acetylcholine); vasodilator (dog); hepatoprotective (inhibits activation of

OH
OH
H
OO
HO
OH
OO
OH
OH
OH
H
macrophages, inhibits increase in sALT and sAST levels, in vivo,

D-GalN/LPS-induced liver injury in mouse, 50mg/kg ip for sALT, InRt =
77%, 100mg/kg ip for sALT, InRt = 89%; 50mg/kg ip for sAST, InRt = 80%;
100mg/kg ip for sAST, InRt = 87%; control Hydrocortisone, 20mg/kg ip for
sALT, InRt = 99%; 20mg/kg ip for sAST, InRt = 97%)[4702]. Source: REN
SHEN Panax ginseng [Syn. Panax schinseng] (rhizome: content =
OH
HO
(GalN-caused liver damage); reduces uterine contraction (gpg, in vitro, caused
OO
OH

OH
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng], XI YANG SHEN

Panax quinquefolium (rhizome: content = 0.13%[5508]), ZHU JIE SAN QI
430
Panax pseudo-ginseng var. japonicus (rhizome: content = 0.23%[5508], yield =
8428 Ginsenoside Re
0.0011%dw[4647]). Ref: 4, 900, 4647, 4702, 5508.
Chikusetsusaponin IVc; Ginsenoside B2 [52286-59-6] C48H82O18 (947.18).
Pharm: Analgesic (mus, 10mg/kg); inhibits fatigue; bidirectional action to
OH
OH
HO
Colorless acicular Crystals, mp 201~203C, []D20 = 1.5 (c = 0.52, MeOH).
OO
OH
OH
OH
H
OH
blood pressure (murine, first increases and then lowers blood pressure, while
heart rate slows); reduces uterine contraction (gpg in vitro, caused by

acetylcholine); hepatoprotective (inhibits activation of macrophages, inhibits
increase in sALT and sAST levels, in vivo, D-GalN/LPS-induced liver injury
H
HO
OO
in mouse, 100mg/kg ip for sALT, InRt = 92%; 100mg/kg ip for sAST, InRt =
OH
90%; control Hydrocortisone, 20mg/kg ip for sALT, InRt = 99%; 20mg/kg ip
OH
HO
for sAST, InRt = 97%)[4702]. Source: REN SHEN Panax ginseng [Syn. Panax
schinseng] (rhizome: content = 0.30%[5501]; content = 0.57%[5508]), SAN QI
OH
OH
Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (rhizome:

content = 0.50%)[5508], XI YANG SHEN Panax quinquefolium (rhizome:
OH
content = 2.0%[5508]), ZHU JIE SAN QI Panax pseudo-ginseng var. japonicus

8427 Ginsenoside Rd
(rhizome: content = 0.04%[5508], yield = 0.011%dw[4610]). Ref: 4, 87, 451, 613,
Gypenoside VIII [52705-93-8] C48H82O18 (947.18). White powder
658, 1521, 4610, 4702, 5501, 5508.
(ethanol:butyl alcohol = 1:1), mp 206~209C, []D22 = +19.38 (c = 1.03,

methanol). Pharm: Antiarrhythmic (rat arrhythmia caused by BaCl2); antiviral;
OO
HO
OH
inhibits replication of HSV-1; antioxidant (rat hepatic homogenate, caused by
OH
H2O2, IC50 = (12.00.8)g/mL,by FeSO4, IC50 = (457.515.4)g/mL);
OH
H
11--Hydroxysteroid dehydrogenase inhibitor; cAMP phosphodiesterase

inhibitor (in vitro, IC50 = 84mol/L); promotes cytotoxic effects of
OH
H
HO
daunomycin and vincaleucoblastine; promotes plasma secretion of
O
O
HO
corticosterone (ED50 = 112mol/kg); regulates kidney function and inhibits
OH
reproduction of glomerulus cells; vasodilator; antinociception (i.t. injected
OH
OH
0.7g substance P-induced pain model, EC = 50g i.t.)[5474];

hepatoprotective (inhibits activation of macrophages, inhibits increase in
sALT and sAST levels, in vivo, D-GalN/LPS-induced liver injury in mouse,

OH OH
control Hydrocortisone, 20mg/kg ip for sALT, InRt = 99%; 20mg/kg ip for
sAST, InRt = 97%)[4702]. Source: JIAO GU LAN Gynostemma pentaphyllum
8429 Ginsenoside Rf
(leaf: yield = 0.009%dw)[4757], QIN LING ZHU ZI SHEN Panax japonicus
[52286-58-5] C42H72O14 (801.03). White powder, mp 197~198C. Pharm:
var. major, REN SHEN Panax ginseng [Syn. Panax schinseng] (rhizome:
Antineoplastic; inhibits fatigue; bidirectional action to blood pressure (murine,
content = 0.16%[5508]), SAN QI HUA LEI Panax pseudo-ginseng var.
first increases and then lowers blood pressure, while heart rate slows); reduces
notoginseng [Syn. Panax notoginseng] (flower bud: yield = 0.010%dw)[4702],
uterine contraction (gpg, in vitro, caused by acetylcholine); antinociception
SAN QI Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]
(i.t. injected 0.7g substance P-induced pain model, EC = 50g i.t.)[5474].
[5508]
(rhizome: content = 1.3%)
, XI YANG SHEN Panax quinquefolium
(rhizome: content = 0.78%[5508]), ZHU JIE SAN QI Panax pseudo-ginseng var.

[4647]
japonicus (underground part: yield = 0.0018%dw)
. Ref: 4, 87, 451, 900,
Source: REN SHEN Panax ginseng [Syn. Panax schinseng] (rhizome: content
= 0.15%[5508]), XI YANG SHEN Panax quinquefolium. Ref: 4, 87, 658, 5474,
5508.
4647, 4702, 4757, 5474, 5508.

OH
OO
HO
OH
H
OH
OH
OH
OH
H
H
H
OO
HO
OH
HO
H
OH
OH
O
HO
OH
OH
OO
HO
HO
OH
OH
OH
OH
OH
431
8430 Ginsenoside Rg1
8432 20(S)-Ginsenoside Rg3
Ginsenoside A2 [22427-39-0] C42H72O14 (801.03). mp 194.0~196.5C.
Pharm: Antineoplastic; treatment of cancer of stomach; inhibits fatigue;
bidirectional action to blood pressure (murine, first increases and then

lowers blood pressure, while heart rate slows); promotes biosynthesis of
OH
DNA, protein and lipid (murine marrow cells); reduces uterine contraction
OH
H
(gpg, in vitro, caused by acetylcholine); vasodilator (animal model);

hepatoprotective (inhibits activation of macrophages, inhibits increase in
H
sALT and sAST levels, in vivo, D-GalN/LPS-induced liver injury in mouse,

HO
OH
sAST, InRt = 97%)[4702]; LD50 (mus, orl) 5000mg/kg, (mus, ip) =

[Syn. Panax schinseng] (rhizome: content = 0.46%
[5501]
HO
; content =
0.38%[5508]), SAN QI Panax pseudo-ginseng var. notoginseng [Syn. Panax
OH
control Hydrocortisone, 20mg/kg ip for sALT, InRt = 99%; 20mg/kg ip for

1600mg/kg, (mus, iv) = 396mg/kg. Source: REN SHEN Panax ginseng
OO
OO
OH
OH
OH
notoginseng] (rhizome: content = 4.7%[5508]), XI YANG SHEN Panax

quinquefolium (rhizome: content = 0.20%[5508]), ZHU JIE SAN QI Panax
pseudo-ginseng var. japonicus (rhizome: content = 0.09%[5508], yield =
0.011%dw[4610]). Ref: 4, 87, 658, 4139, 4610, 4702, 5501, 5508.

3-O--D-Glucopyranosyl 3,12,20(S),24(R)-tetrahydroxy-dammar-25-ene
20-O--D-glucopyranoside C42H72O14 (801.03). White powder. Source: REN
SHEN YE Panax ginseng [Syn. Panax schinseng]. Ref: 3517.
OO
HO
OH
OH
OH
H
OH
OH
H
HO
OO
HO
OH
H
O
HO
OH
OH
OH
OH
OO
HO
OH
OH
OH
OH
OH

Ginsenoside C C42H72O13 (785.03). Crystals, mp 187~189C, []D30 = +5.5 (c
= 1, MeOH). Source: REN SHEN Panax ginseng [Syn. Panax schinseng], XI
8434 20(R)-Ginsenoside Rh1
YANG SHEN Panax quinquefolium. Ref: 1521.

schinseng]. Ref: 2.
OH
OH
OH
H
OH
H
H
HO
H
HO
O
OH
OH
OH OO
OH OH
H
HO
O
O
HO
OH
OH
OH
432
8435 20(S)-Ginsenoside Rh1
8438 Ginsenoside Rh3
Ginsenoside Rh1 [63223-86-9] C36H62O9 (638.89). Pharm: Hepatoprotective
3,12-Dihydroxy-dammar-20(22),24-diene-3-O--D-glucopyranoside
(inhibits activation of macrophages, inhibits increase in sALT and sAST
[105558-26-7] C37H62O7 (618.90). White powder, mp 255~257C, []D27 = +7
levels, in vivo, D-GalN/LPS-induced liver injury in mouse, 100mg/kg ip for
(c = 0.778, methanol). Source: REN SHEN Panax ginseng [Syn. Panax
sALT, InRt = 93%; 100mg/kg ip for sAST, InRt = 90%; control
Hydrocortisone, 20mg/kg ip for sALT, InRt = 99%; 20mg/kg ip for sAST,
OH
H
InRt = 97%)[4702]. Source: REN SHEN Panax ginseng [Syn. Panax schinseng],
SAN QI Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng],
XI YANG SHEN Panax quinquefolium. Ref: 2, 28, 87, 4702.
H
HO
OO
OH
OH
OH
OH
H
OH

[174721-08-5] C36H60O8 (620.87). Colorless thin crystals (methanolwater),
H
HO
mp 160~161C, []D = +28.2 (c = 1, methanol). Pharm: Cytotoxic (P388, ED50
= 25mol/L, L1210, ED50 = 23mol/L). Source: REN SHEN Panax ginseng
OO
HO
[Syn. Panax schinseng]. Ref: 1149.
OH
OH
OH
H
OH
8436 20(R)-Ginsenoside-Rh2
HO
[112246-15-8] C36H62O8 (622.89). Pharm: Antineoplastic (hmn, leukemia
H
HO
HL-60, 2g/mL; mus myelocytic leukemia M1, inducing cell differentiation
OH
activity, 50mol/L, growth rate = 70%); cytotoxic (in vitro, enhances
OH
cytotoxicity for drug-resistant strain P388, IC50 = 75.6mol/L, MT-4, CC50
OH
(concentration of half cytotoxicity) = 475mol/L). Source: REN SHEN Panax
ginseng [Syn. Panax schinseng]. Ref: 2, 1615, 1616, 1617, 1618.
3,6,12,24-Tetrahydroxy-dammar-20(22),25-diene
6-O--D-glucopyranoside C36H60O9 (636.87). White powder, []D21 = +20.8
(c = 0.1, MeOH). Source: REN SHEN YE Panax ginseng [Syn. Panax
OH
OH

OH
OH
H
HO
OH
OH
HO
OH
HO
OH
8437 20(S)-Ginsenoside Rh2
OH
OH


3,6,12,20(S)-Tetrahydroxy-25-hydroperoxy-dammar-23-ene 20-O--Dglucopyranoside C36H62O11 (670.89). White powder, []D21 = +21.8 (c = 0.1,
OH
OH
H
MeOH). Source: REN SHEN YE Panax ginseng [Syn. Panax schinseng]. Ref: 3517.
OO
HO
OH
H
HO
OO
OH
OH
OH
OH
OH
OH
HO
OH
OH
433
8446 Ginsenoside Rs1
3,7,12,20(S)-Tetrahydroxy-dammar-5,24-diene
[87733-67-3A] C55H92O23 (1121.33). Source: REN SHEN Panax ginseng
20-O--D-glucopyranoside C36H60O9 (636.87). White powder, []D21 = +30.1
(c = 0.1, MeOH). Source: REN SHEN YE Panax ginseng [Syn. Panax

OH
OO
OH
OO
HO
OH
OH
H
OO
OH
OH
OH
HO
OO
OH

3,6,20(S)-Trihydroxy-dammar-24-ene-12-one 20-O--D-glucopyranoside
OH
OH
C36H60O9 (636.87). White powder. Source: REN SHEN YE Panax ginseng

8447 Ginsenoside Rs2

OO
HO
OH
OH
HO
OH
H
OH
OH
OH
OH
OO
OH
OH
OH
OH
HO
OH
O
OO
OH
20-O--D-glucopyranoside C36H60O9 (636.87). White powder. Source: REN

SHEN YE Panax ginseng [Syn. Panax schinseng]. Ref: 3517.

3,6,20(S)-Trihydroxy-12,23-epoxy-dammar-24-ene
OH
H
OH
OH
OH
HO
OO
OH
OH
HO
OH
OH
O
OH
8448 Ginsenoyne A
H
O
HO
OH
HO
HO
OH
OH
OH
O
8445 Ginsenoside Ro
Panax schinseng] (rhizome: content = 1.8%[5508]), XI YANG SHEN Panax
quinquefolium (rhizome: content = 0.65%[5508]), ZHU JIE SAN QI Panax
pseudo-ginseng var. japonicus (rhizome: content = 2.7%)[5508]. Ref: 2, 5508.
8449 Ginsenoyne B
[139035-29-3] C17H23ClO2 (294.82). Source: REN SHEN Panax ginseng [Syn.
HO
H
OH
OO
OH
HO
OO
OH
OH
OH
OO
HO
OH
Cl
8450 Ginsenoyne C
OH
HO
OH
OH
OH
OH
OH
434
8451 Ginsenoyne D
8456 Girinimbine
[23095-44-5] C18H17NO (263.34). Pharm: Antibacterial (Staphylococcus
schinseng]. Ref: 2.
aureus, MIC = 3.13g/mL, MIC =0.012mol/L, control Kanamycin, MIC =
HO
3.13g/mL; Bacillus subtilis, MIC = 25g/mL, MIC =0.095mol/L,

Kanamycin, MIC = 6.25g/mL; Escherichia coli, MIC = 50g/mL, MIC
=0.190mol/L, Kanamycin, MIC = 12.5g/mL; Proteus vulgaris, MIC =
12.5g/mL, MIC =0.047mol/L, Kanamycin, MIC = 12.5g/mL)[5299];

8452 Ginsenoyne E
antifungal (Aspergillus niger, MIC = 25g/mL, MIC =0.095mol/L; Candida
3-Oxopanaxydol; PQ-3 [126146-63-2] C17H22O2 (258.36). Oil, []D = 36.9C
albicans, MIC = 100g/mL, MIC =0.302mol/L, control Fluconazole, MIC =
(c = 0.68, MeOH). Pharm: Cytotoxic (L1210, 0.5-1.0g/mL, InRt = 100%).
25g/mL, MIC = 0.082mol/L)[5299]. Source: NEN YE JIU LI XIANG
Source: REN SHEN Panax ginseng [Syn. Panax schinseng], XI YANG SHEN
Murraya microphylla, YUAN DONG JIU LI XIANG Murraya siamensis,
Panax quinquefolium. Ref: 2, 1017, 1521.
YIN DU JIU LI XIANG Murraya koenigii (stem cortex). Ref: 11, 5299.
O
O
8453 Ginsinsene
NH
(1R*,6R*,7R*)-3,7,10,10-Tetramethyltricyclo[4.3.2.02,6]undec-2-ene C15H24
(204.36). Source: REN SHEN Panax ginseng [Syn. Panax schinseng]. Ref:
5330.
8457 Gitogenin
[511-96-6] C27H44O4 (432.65). mp 271~272C. Source: DA YU BIAO HUA
Hosta sieboldiana, FAN MA Agave americana, HU LU BA Trigonella
foenum-graecum, JI LI GEN Tribulus terrestris. Ref: 6, 10.
8454 Giraldine G
C40H57N3O11 (755.91). White amorphous powder, mp 108~110 C, []D20 =
+35.4 (c = 0.42, CHCl3). Source: QIN LING CUI QUE HUA Delphinium
O
giraldii (root). Ref: 4278.

H
HO
H O
O
OH
H
O
H
N
8458 F-Gitonin
OH
O
O
HO
H
O
Gitogenin -lycotetraoside [28591-01-7] C50H82O23 (1051.20). Micro needles

from MeOH, mp 260~263C, []D24 = 51.6 (c = 0.21, pyridine). Pharm:
Antineoplastic (HeLa, inhibits 32P combines with phospholipid in HeLa cells,
NH2
O
50g/mL, InRt = 23.1%); antiviral (reduces titer of tobacco masaic virus by

2~3 times). Source: CI JI LI Tribulus terrestris. Ref: 706, 1636, 1637, 1638.
8455 Giraldine H
20
C41H59N3O11 (769.94). White amorphous powder, mp 122~124 C, []D =

O
+34.6 (c = 0.35, CHCl3). Source: QIN LING CUI QUE HUA Delphinium
giraldii (root). Ref: 4278.
O
H
HO
H O
O
H
H
N
O
OH
H
O
H
N
O
O
OH
OH
OH
O
OH
OH
OH
OH
HO
O
OH
NH2
O
HO
HO
OH
OH
H
H
435
8459 Gitonin
8463 Glabcensin B
Capsicosin D1 [39937-47-8] C50H82O23 (1051.20). Acicular Crystals (MeOH),
mp 250~253C, []D19 = 40 (c = 1, pyridine). Source: CI JI LI Tribulus
Source: MAO GENG XIA YE XIANG CHA CAI Isodon angustifolius var.
terrestris. Ref: 706.
glabrescens. Ref: 4067.

O
O
O
HO
HO
O
OH
OH
HO
HO
OH
OH
HO
OO
HO
OH
OH
O
O
OH
8464 Glabcensin C
OH
8460 Gitoxigenin
[545-26-6] C23H34O5 (390.52). mp 220~225C. Source: JIA ZHU TAO
Nerium indicum. Ref: 6.
O
O
OH
HO
O
H
H
HO
OH
O
OH
O
O
8461 Gitoxin
[4562-36-1] C41H64O14 (780.96). Pharm: Cardiotonic; toxin (vertebrate). Source:
[5508]
MAO DI HUANG Digitalis purpurea (dried leaf: content = 0.0140%
), MAO
HUA MAO DI HUANG Digitalis lanata. Ref: 658, 5508.
8465 Glabcensin D
OH OH
O
O
H
O OH
OH
O
H
OH
HO
OO
O
OH
O
O
OH
8462 Glabcensin A
C28H38O10 (534.61). Amorphous powder, mp 198~199C, []D22 = 74.9 (c =
8466 Glabcensin E
0.57, MeOH). Source: MAO GENG XIA YE XIANG CHA CAI Isodon
angustifolius var. glabrescens. Ref: 4067.
O
HO
O
HO
HO
O
O
H
H
O
O
O
O
O
O
O
436
8467 Glabcensin F
8472 Glabcensin K
HO
HO
HO
H
HO
O
OH
OH
O
8473 Glabcensin L
8468 Glabcensin G

O
HO
HO
H
O
O
H
O
OH
OH
O
OH
8474 Glabcensin M
8469 Glabcensin H
22

O
HO
HO
HO
H
O
O
H
HO
O
OH
O
O
8475 Glabcensin N


O
O
HO
HO
H
O
H
O
O
OH
OH
O
8476 Glabcensin O
22


O
HO
HO
H
H
8471 Glabcensin J
HO
8470 Glabcensin I
OH
O
H
O
O
O
O
OH
437
8477 Glabcensin P
8481 Glabcensin T
O
HO
H
O
O
H
O
OH
OH
OH
O
8482 Glabcensin U
8478 Glabcensin Q

O
OH
O
H
HO
H
O
O
O
OH
O
8483 Glabcensin V
Gesneroidin F C24H34O7 (434.53). Amorphous powder, []D22 = 7.32 (c =
8479 Glabcensin R
0.48, CHCl3); []D25.6 = 22.0 (c = 0.25.0, MeOH). Pharm: Cytotoxic (hmn

tumor K562 cells, IC50 = 0.4g/mL, control cis-Platin IC50 = 1.1g/mL)[4955].
glabrescens, DONG LING CAO Rabdosia rubescens (leaf). Ref: 1869,
4067, 4955.
O
O
OH
HO
O
H
O
O
O
H
O
O
OH
O
O
8480 Glabcensin S
8484 Glabcensin W
C28H38O9 (518.61). Amorphous powder, []D22 = 59.98, (c = 0.42, MeOH).
glabrescens. Ref: 1869, 4067.
OH
O
H
O
O
O
O
O
H
O
O
O
O
O
438
8485 Glabcensin X
8490 Glabrene
aureus ATCC13709 and Mycobacterium smegmatis ATCC607, MIC =
25g/mL). Source: GUANG GUO GAN CAO Glycyrrhiza glabra. Ref: 2,
658, 660.
HO
H
HO
O
O
OH
O
O
8491 Glabrephinine
8486 Glabcensin Y
C24H34O7 (434.53). Amorphous powder, []D = 13.0(c = 0.54, CHCl3).
[132160-37-3] C22H33NO6 (407.51). White acicular Crystals, mp 201~203C.
Source: ZHAN MAO CUI QUE HUA Delphinium kamaonense var.
22
OH
H
HO
O
O
OH
OH
OH
OH OH
8492 Glabrescin
8487 Glabranin
[41983-91-9] C20H20O4 (324.38). Pharm: Antimicrobial (broad spectrum);
C48H78O9 (799.15). Orange oil, []D24 = +82 (c = 0.35, CHCl3). Source:
promotes estrogenic activity. Source: MEI ZHOU GAN CAO Glycyrrhiza
Neoboutonia glabrescens. Ref: 3441.
lepidota, GUANG GUO GAN CAO Glycyrrhiza glabra, GUANG GUO GAN
CAO Glycyrrhiza glabra (leaf)[4685]. Ref: 2, 658, 660, 4685.
H
H
O
H
O
HO
O
O
OH
OH OH
O
O
8493 Glabridin
8488 Glabratine
C20H20O4 (324.38). Pharm: Antibacterial (Staphylococcus aureus ATCC13709,
C27H34N2O9 (530.58). Source: CHANG HUA GOU TENG Uncaria longiflora,
MIC = 6.25g/mL; Mycobacterium smegmatis); antifungal (Candida albicans
MIAN MAO GOU TENG Uncaria lanosa. Ref: 5341.
ATCC1023, MIC = 25g/mL). Source: GUANG GUO GAN CAO
HO
Glycyrrhiza glabra. Ref: 2, 658, 660.
O
OH
OH
OH
N
H H
OH
O
H
OH
OH
8489 Glabratolide
8494 Glabrin C
[75744-65-9] C19H24O5 (332.40). Amorphous gum. Pharm: Cytotoxic (KB in
Cyclo-(prolyl-glycyl-tyrosyl-valy-leucyl-alanyl-leucyl-valyl) C41H64N8O9
vitro, ED50 = 2.3g/mL). Source: GUANG CI BAO JU Acanthospermum
(813.02). Amorphous powder, mp153, []D29 = 35.11 (c = 0.235, MeOH).
glabratum. Ref: 658, 661, 1521.
Source: YUAN HUA FAN LI ZHI Annona glabra. Ref: 1858.

N
H
O
N
O
H
H
N
OH
NH
HN
N
H
O
N
H
NH
439
8495 Glabrin D
8500 Glabrolide
Cyclo-(prolyl-prolyl-valyl-tyrosyl-glycyl-prolyl-glutamyl) C36H49N7O10
[10401-33-9] C30H44O4 (468.68). Source: CU MAO GAN CAO Glycyrrhiza
(739.83). Amorphous powder, mp219, []D29 = 53.54 (c = 0.551 MeOH).
aspera, GAN CAO Glycyrrhiza uralensis, GUANG GUO GAN CAO
Source: YUAN HUA FAN LI ZHI Annona glabra. Ref: 1858.
Glycyrrhiza glabra. Ref: 1521.

O
N
N
H
N
O
HN
HO
NH
O
N
H
H
HO
OH
8496 Glabrocoumarin
C20H16O5 (336.35). Slightly yellow needles (benzeneacetone), mp
8501 Glabrone
254~256C. Source: GUANG GUO GAN CAO Glycyrrhiza glabra (root).
Eurycarpin B; 7,2'-Dihydroxy-6'',6''-dimethylpyrano-(2'',3'':4',3')isoflavone
Ref: 4486.
[60008-02-8] C20H16O5 (336.35). Yellowish acicular Crystals, mp 227~229C.

Pharm: Antioxidant (in vitro, 8g/mL, oxygen clearance = 28.6%, 10g/mL,
HO
hemolytic InRt induced by H 2O2 = 94.2%). Source: GUANG GUO GAN CAO
Glycyrrhiza glabra, HUANG GAN CAO Glycyrrhiza kansuensis, ZHANG

GUO GAN CAO Glycyrrhiza inflata. Ref: 2, 379, 660, 1753.
OH
8497 Glabroisoflavanone A
C20H18O5 (338.36). Colorless prisms (MeOHH2O), mp 113~116C, []D25 =
HO
0 (c = 0.073, MeOH). Source: GUANG GUO GAN CAO Glycyrrhiza glabra

(root). Ref: 4486.
O
O
HO
OH
8502 Glanduliforol
OH
C15H24BrClO (335.71). Source: XIAO XIAN AO DING ZAO Laurencia
8498 Glabroisoflavanone B
C21H20O5 (352.39). Colorless prisms (MeOHH2O), mp 161~162C, []D =
glandulifera (in 1974, the compound was isolated from the plant by M.Suzuki
0 (c = 0.036, MeOH). Source: GUANG GUO GAN CAO Glycyrrhiza glabra
et al.). Ref: 5505.
25
(root). Ref: 4486.

HO
Cl
O
OH
Br
8499 Glabrol
8503 Glandulone C
aureus ATCC13709, MIC = 1.56g/mL; Mycobacterium smegmatis ATCC607,
C15H20O3 (248.32). Brown oil, []D25 = +23.6 (c = 0.12, methanol). Source:
MIC = 1.56g/mL). Source: GUANG GUO GAN CAO Glycyrrhiza glabra,
XIANG RI KUI YE Helianthus annuus. Ref: 1521, 1556.
HUANG GAN CAO Glycyrrhiza kansuensis. Ref: 2, 591, 658, 660.

OH
OH
HO
O
O
440
8504 Glansrin A
8507 Glaocogenin C mono-D-thevetoside
C48H32O31 (1104.77). Off-white amorphous powder, []D23 = 11 (c = 0.3,
Glaucogenin C 3-O--D-thevetopyranoside C28H40O9 (520.63). Colorless fine
MeOH). Pharm: Antioxidant (SOD-like activity, EC50 = 190mol/L, control
needles, mp 185~187C, []D25 = +26.10 (c = 0.991, MeOH). Pharm:
Gallic acid, EC50 = 31.7mol/L, L-Ascorbic acid, EC50 = 34.6mol/L);
Anti-inflammatory inactive (no significant inhibitory effects on mast cells and
antioxidant (DPPH free radical scavenger, EC50 = 0.36mol/L, control Gallic
neutrophils stimulated with various inducers; no significant inhibitory effects
acid, EC50 = 5.88mol/L, L-Ascorbic acid, EC50 = 6.25mol/L). Source: HU
on TNF- formation from RAW264.7 stimulated with LPS and N9
TAO REN Juglans regia. Ref: 3408.
microglial cells stimulated with LPS/INF-)[3054]; vasodilator inactive (in vitro,

rat isolated aortic rings with endothelium, pre-contracted by 0.1mol/L
OH
OH
OO
HO
O
Phenylephrine or 100mmol/L KCl)[4077]. Source: BAI WEI Cynanchum
OH
HO
HO
OH
atratum (root), LIU YE BAI QIAN Cynanchum stauntonii. Ref: 3054, 4077.
O
H
OH
O
O
O
OH
OH
OH HO
HO
OO
OH
OH OH OH
HO
8505 Glansrin B
OH
C40H26O25 (906.64). Off-brown amorphous powder, []D23 = +90 (c = 0.1,
OH
MeOH). Pharm: Antioxidant (SOD-like activity, EC50 = 41.9mol/L, control
8508 Glaucacyclopeptide A
C28H47N7O7 (593.73). Colorless solid, mp 174~175C, [] D22 = 57 (c = 0.2,
MeOH). Pharm: Cytotoxic (in vitro, KB cells, IC50 = 0.73mol/L, control
Doxorubicin, IC50 = 0.02mol/L). Source: ROU MAO FAN LI ZHI Annona
glauca (seed). Ref: 5282.

O
OH
OH
HO
HO
O
O OH
HO
HO
N
H
O
H
N
NH
NH
H
N
O
O
H
N
H
OH
OH
HO
8509 Glaucarubinone
OH OH OH
HO
[1259-86-5] C25H34O10 (494.54). mp 228~230C, []D20 = +50 (c = 0.27,

methanol). Pharm: Antiamebic; antineoplastic (P388, Lewis lung cancer and
8506 Glansrin C
C41H26O26 (934.65). Off-brown amorphous powder, []D = +79 (c = 0.1,
B16 melanoma, 0.12~0.5mg/kg); antimalarial (ED = 0.006g/mL); cytotoxic
MeOH). Pharm: Antioxidant (SOD-like activity, EC50 = 21.4mol/L, control
(KB, ED50 = 0.025g/mL); pesticide. Source: GAO CHU Ailanthus excelsa.
Ref: 661.
23
OH
HO
OH

OH
O
OH
OH
HO
OH
8510 Glaucarubolone
O
O
HO
HO
OH
O
C20H26O8 (394.43). Source: Eurycoma harmandiana (root). Ref: 5164.

OH
O
O
OH
O
HO
OH
OH
OH
HO
HO
OH
OH
OH OH
H
H
H
H
441
8511 Glaucedine
8515 Glaucocalyxin A
C30H49NO8 (551.73). Source: HEI SHUI CUI QUE HUA BIAN ZHONG
Leukamenin F C20H28O4 (332.44). mp 220~222C, []D20 = 182.9 (c = 0.25,
Delphinium potaninii var. jiufengshanense (root). Ref: 4227.
CHCl3). Source: LAN E XIANG CHA CAI Isodon japonica var. glaucocalyx.
Ref: 4067.
O
O
N
OH
H
O
OH
H
H
OH
O
OH
8512 Glaucin A
[88848-59-3] C26H30O10 (502.52). Source: WU ZHU YU Evodia rutaecarpa.
Ref: 482.
8516 Glaucocalyxin B
C22H30O5 (374.48). mp 190~192C, []D20 = 127.9 (c = 0.203, CHCl3).
Source: LAN E XIANG CHA CAI Isodon japonica var. glaucocalyx. Ref:
4067.
O
OH
O
O
OH
O
O
OH
8513 Glaucine
8517 Glaucocalyxin C
[475-81-0] C21H25NO4 (355.44). mp 120C. Pharm: Treatment of amebic
C20H30O4 (334.46). mp 272~273C, []D29 = 109 (c = 0.1, MeOH). Source:
dysentery. Source: BEI JIA ER TANG SONG CAO Thalictrum baicalense,
LAN E XIANG CHA CAI Isodon japonica var. glaucocalyx. Ref: 4067.
DONG BEI YAN HU SUO Corydalis ambigua var. amurensis [Syn.

Corydalis ambigua] (rhizome: mean content of 3 origins = 0.114%[5508]),
HUANG HUA HAI YING SU Glaucium davum, SHAN YAN HU SUO
Corydalis bulbosa [Syn. Corydalis solida], SUI MAO HE BAO MU DAN
Dicentra eximia, XIANG TANG SONG CAO Thalictrum foetidum, XIAO
H
O
GUO TANG SONG CAO Thalictrum microgynum (root: content =
OH
OH
OH
0.093%)[5508], YAN HU SUO Corydalis yanhusuo [Syn. Corydalis

turtschaninovii f. Yanhusuo] (rhizome: mean content of 2 origins =
0.078%[5508]), YING SU Papaver somniferum. Ref: 4, 56, 658, 660, 5508.
8518 Glaucocalyxin D
C22H30O5 (374.48). mp 130~132C, []D19 = 161.5 (c = 0.15, MeOH).
4067.
O
O
O
O
OH
8514 Glaucocalactone
O
O
C22H26O7 (402.45). mp 318~320C, []D25 = +55 (c = 0.30, CHCl3). Source:

LAN E XIANG CHA CAI Isodon japonica var. glaucocalyx. Ref: 4067.
C20H30O4 (334.46). mp 228~230C, []D20 = 142.5 (c = 0.15, MeOH).
O
O
O
8519 Glaucocalyxin E
4067.
H
O
H
O
OH
O
OH
442
8520 Glaucogenin C 3-O--D-cymaropyranosyl-(14)--L-diginopy-
8524 Glaziovine
ranosyl-(14)--D-thevetopyranoside
[6808-72-6] C18H19NO3 (297.36). Colorless lamellar Crystals (benzene), mp
C42H64O15 (808.97). Pharm: Anti-inflammatory (in vitro, inhibits TNF-
223C, []D = 45.74 (c = 0.26, methanol). Pharm: Antineoplastic
formation, 30mol/L: RAW264.7 cell lines LPS-stimulated, InRt = (33.76.2)%;
(nasopharyngeal carcinoma cells, ED50 = 2.6g/mL); antiulcerative (rat and
N9 microglial cell lines, LPS/IFN--stimulated, InRt = (30.94.3)%; no significant
gpg, 5mg/kg iv); CNS depressant (animal, relieves anxiety); antihypertensive
inhibitory effects on mast cells and neutrophils stimulated with various inducers);
(rat, 5~15mg iv, 1~3h blood pressure reduced by (50~70)%); anxiolytic and
cytotoxic (in vitro, 212 cells, ED50 = 0.96g/mL, significant activity). Source: BAI
antidepressant, treatment of terror, anxiety and melancholy. Source: SAN
WEI Cynanchum atratum (root). Ref: 3054.
HUA BA DOU Croton sparsiflorus, WEI ER SHI LV RONG HAO

Meconopsis cambrica, ZI FAN LI ZHI Annona purpurea. Ref: 658, 661.
O
O
H
O
O
O
HO
O
OO
O
OO
O O
O
OH
HO
8525 Glechomanolide

8521 Glaucopine A
14-Hydroxy-13-methoxy-8-oxocyatha-3,11-diene-12-carbaldehyde
C21H30O4 (346.47). Colorless resin, []D31 = 30.8 (c = 0.42, CHCl3). Pharm:
Anti-inflammatory (in vivo, mouse ear edema induced by croton oil,

1.0mol/cm2, edema reduction = 62%, control Indomethacin, 0.3mol/cm2,
edema reduction = 61%). Source: CANG BAI BING ROU CHI JUN
Sarcodon glaucopus. Ref: 5063.
O
OH
8526 Gleditsiasaponin B
C94H148O44 (1982.20). []D25 = 20 (c = 0.10, MeOH). Pharm: Cytotoxic
(HL-60, IC50 = (1.00.2)mol/L, control Taxol, IC50 = (4.1E-41.1E-4)mol/L;
8522 Glaucopine B
MCF7, IC50 = (24.51.2)mol/L, Taxol, IC50 = (15.32.6)mol/L; Bel7402,
14-Hydroxy-11-methoxy-8-oxocyatha-3,12-diene-12-carbaldehyde C21H30O4
IC50 = (42.64.2)mol/L, Taxol, IC50 = (0.30.1)mol/L; BGC823, IC50 =
(346.47). Colorless resin, []D31 = 98.0 (c = 0.73, CHCl3). Pharm:

Anti-inflammatory (in vivo, mouse ear edema induced by croton oil, 1.0mol/cm2,
edema reduction = 55%, control Indomethacin, 0.3mol/cm2, edema reduction = 61%).
Source: CANG BAI BING ROU CHI JUN Sarcodon glaucopus. Ref: 5063.
O
(60.62.8)mol/L; HeLa, IC50 = (50.60.4)mol/L, Taxol, IC50 =

(33.06.1)mol/L; KB, IC50 = (44.74.0)mol/L, Taxol, IC50 > 100mol/L);
apoptosis inducer (HL-60 cells, 15mol/L, sub-G1 population = (59.12.8)%,
control sub-G1 population = (5.43.2)%, positive control Taxol, sub-G1
population = (40.50.2)%). Source: ZAO JIA Gleditsia sinensis [Syn.
Gleditsia horrida] (fruit). Ref: 5015.
OH
OH
8523 Glaudine
[5140-40-9] C22H25NO6 (399.45). mp 103~105C. Source: YA PIAN Papaver
OH O O
OO
OH
OH
OH
somniferum. Ref: 6.
OH
OH
OH
OH
OH
H O
O
OH
OH
OO
N H
O
OO
H
OO
OO
OH
OH
O OH OH OH
OH
OO
OH
OH
HO
OO
OH
OH
443
8527 Gleditsiasaponin C
8529 Gleditsiasaponin E'
C69H112O34 (1485.64). White amorphous solid, mp 232~233C(dec), []D21 =
33 (c = 0.10, MeOH). Source: ZAO JIA Gleditsia sinensis [Syn. Gleditsia
horrida]. Ref: 2375.

H
OH
OO
OH
OO
OH O O
OO
OH
OH
OH
OH
OH OH OH
O
OH
OO
OH
OO
OH
OH
OH
OH OH
OH
O
OH
O OH OH OH
OH
OO
OH
OO
OO
O O
OH
OH
OH
OH
OH
OO
O
OH
OH
OH
H OH OO
OH
OH
OH
OH
OH
HO
OH
8530 Gleditsioside A
OH
(HL-60, IC50 = (16.70.8)mol/L, control Taxol, IC50 =
8528 Gleditsiasaponin C'

3-O--D-Xylopyranosyl(12)--L-arabinopyranosyl(16)--D-glucopyrano
syl-28-O--D-Xylopyranosyl(13)--D-Xylopyranosyl(14)--L-rhamnopy
ranosyl(12)-[-L-rhamnopyranosyl(16)]--D-glucopyranosyl
echinocystic acid C74H120O38 (1617.76). White amorphous solid, mp
21
234~235C(dec), []D = 18 (c = 0.10, MeOH). Pharm: Cytotoxic (HL-60,

IC50 = (100.05.2)mol/L, control Taxol, IC50 = (4.1E-41.1E-4)mol/L;
IC50 > 100mol/L, Taxol, IC50 = (0.30.1)mol/L; BGC823, IC50 =
(1003.7)mol/L; HeLa, IC50 = (54.01.7)mol/L, Taxol, IC50 =
(4.1E-41.1E-4)mol/L; MCF7, IC50 = (12.91.1)mol/L, Taxol, IC50 =

(15.32.6)mol/L; Bel7402, IC50 = (34.60.8)mol/L, Taxol, IC50 =
(0.30.1)mol/L; BGC823, IC50 = (37.52.5)mol/L; HeLa, IC50 =
(35.81.2)mol/L, Taxol, IC50 = 33.06.1)mol/L; KB, IC50 =
(44.53.0)mol/L, Taxol, IC50 > 100mol/L); apoptosis inducer (HL-60
cells, 15mol/L, sub-G1 population = (8.31.7)%, control sub-G1
population = (5.43.2)%, positive control Taxol, sub-G1 population =
(40.50.2)%). Source: ZAO JIA Gleditsia sinensis [Syn. Gleditsia horrida]
(fruit). Ref: 5015.
(33.06.1)mol/L; KB, IC50 > 100mol/L, Taxol, IC50 > 100mol/L)[5015];

population = (40.50.2)%)[5015]. Source: YUN NAN ZAO JIA Gleditsia
H
delavayi, ZAO JIA Gleditsia sinensis [Syn. Gleditsia horrida]. Ref: 2257,
2375, 5015.
OO
OO
OH
OO
H
OH
OO
OH
OO
OO
OH
OH
OH OH OH
OO
O O
O
OH
O
OH
OH
OH
OH
OH OH
HO
O
O
OH
O
OH
OH
OH
OH
OH
OO
OH
OH
OH
OH
OO
OH
OH
OH
OH
OH
OH
OO
OH
OH
O
OH OH
OH OH OH
444
8531 Gleditsioside B
8533 Gleditsioside D
(4.1E-41.1E-4)mol/L; MCF7, IC50 = (17.50.8)mol/L, Taxol, IC50 =
(35.91.7)mol/L, Taxol, IC50 = (33.06.1)mol/L; KB, IC50 =
(fruit). Ref: 5015.
H
H
H
OH
OO
OO
OH
OO
HO
O
OH
OH
OH
O
O
OH
OH
HO
OH
OH
OO
OO
OH
OH
OH
O
OH
O
O
OH
OH OH
OO
OO
O
OH OH
OH
OO
OH
OH
H
OH O O
OO
OH
OH
OH
OH
OH
OH
OH OH
HO
OH OH OH
OH OH
HO
OH
8532 Gleditsioside C
OH

8534 Gleditsioside E
(Bel7402 cancer cell, IC50 = (3.12.8)mol/L, control Paclitaxel, IC50 =
(5.03.4)mol/L, Paclitaxel, IC50 = (33.06.1)mol/L; HL-60, IC50 =
(3.01.3)mol/L, Paclitaxel, IC50 = (4.1E-41.1E-4)mol/L; KB, IC50 =
(34.34.5)mol/L; MCF7, IC50 = (6.62.3)mol/L, Paclitaxel, IC50 =
(15.32.6)mol/L)[5410]. Source: ZAO JIA Gleditsia sinensis [Syn. Gleditsia

horrida] (fruit). Ref: 5015, 5410.
OH
OO
OO
OH
OO
OH
OH
OH
O
OH
OH
OH
OO
OO
O
OH OH
OH
HO
HO
OH
OH
OH
OO
OH
OH
OO
OO
O
OH
OH
OH OH
OO
OO
OO
OH
OH
OH
OH
OH
HO
OH
OO
OH
O OH OH OH
OH
OH
O O
OH
OH
HO
OH
OH
OH
OH
OH
OH
OH
445
8535 Gleditsioside F
8537 Gleditsioside H
(4.11041.1104)mol/L; MCF7, IC50 = (23.63.2)mol/L, Taxol, IC50 =

H
O

H
OH
OO
OH
(fruit). Ref: 5015.
OO
OH
OH
OO
OH
OH
OH
OO
OO
OH
OH
OH OH
OH
OH

OH
O OH OH OH
OH
OO
OH
OO
OO
O
OH
OH
OH
8538 Gleditsioside I
OH
OO
OH
OH
OO
OH
OH
OH OH OH
OO
O O
O
OH
OH
OH
OO
OH
OH
OO
OH
OO
OH
OH
HO
OH
OH
O
8536 Gleditsioside G
H
OH
OH

OO
OO
HO
OO
OH
OH
OH
OH
O
OH
OH
OH
OO
O O
OH
OH
OH
O
OH
OH OH
OH
OH
8539 Gleditsioside J
(fruit). Ref: 5015.
H
OH
OO
OH
OH
OO
OH
O
OH
OO
OH
OO
OH
OH
OH
OH
OH
OO
OO
OH
O OH OH OH
OH
OH
HO
OH
OH
HO
OH O O
OO
OH
OH
OO
OO
OH
O
H
OH
OH
O O
OH
O
OH
OH
OH
OH
OH
O
O
OH
OH
OO
OH OH
HO
HO
OH
OH
OO
OH
OH
446
8540 Gleditsioside K
8542 Gleditsioside O
(4.11041.1104)mol/L); apoptosis inducer (HL-60 cells, 15mol/L,

sub-G1 population = (7.82.5)%, control sub-G1 population = (5.43.2)%,
positive control Taxol, sub-G1 population = (40.50.2)%). Source: ZAO JIA
Gleditsia sinensis [Syn. Gleditsia horrida] (fruit). Ref: 5015.
O
H
H
OH
OO
OH
OH
OO
OH
OH
O O
OH
OO
OH
OH
OH
OHO
O
OH
HO
OO
OH
OH
OH
OH
OH
O
O
OH
OO
OH
OH
OH
O
OH
OH
OH
O
HO
OH
OH
OH
OH
OO
OO
OH
HO
OH
OO
O
OH
OH
8541 Gleditsioside N
O
OH
OH OH OH
OH
C88H138 O38 (1804.06). []D25 = 18 (c = 0.10, MeOH). Pharm: Cytotoxic

8543 Gleditsioside P
(4.11041.110 4)mol/L; MCF7, IC50 = (58.14.2)mol/L, Taxol, IC50
C103H160 O43 (2086.40). []D25 = 20 (c = 0.10, MeOH). Pharm: Cytotoxic
= (15.32.6)mol/L; Bel7402, IC50 = (49.35.8)mol/L, Taxol, IC50 =
(4.11041.110 4)mol/L; MCF7, IC50 = (23.12.0)mol/L, Taxol, IC50
= (15.32.6)mol/L; Bel7402, IC50 = (40.02.3)mol/L, Taxol, IC50 =
60.63.5)mol/L, Taxol, IC50 > 100mol/L); apoptosis inducer (HL-60
36.74.3)mol/L, Taxol, IC50 > 100mol/L); apoptosis inducer (HL-60
(40.50.2)%). Source: ZAO JIA Gleditsia sinensis [Syn. Gleditsia
horrida] (fruit). Ref: 5015.

(40.50.2)%). Source: ZAO JIA Gleditsia sinensis [Syn. Gleditsia
horrida] (fruit). Ref: 5015.
H
H
OH
OO
OO
OH
OH
OH
OO
OH
OH
HO
O
O
HO
OH
O
O
OH
OH
OH
OO
O
OH
OH
OH
OO
O
OH
OH
OH
OH
OH
OH OH OH
OH
H
OO
OO
OO
OH
HO
HO
OH
OH
OH
O
O HO
O
OO
OH
OO
O
OH
OH
OH
OH
OH OH OH
447
8544 Gleditsioside Q
8547 Glehlinoside C
C26H32O13 (552.54). Off-white amorphous solid, []D = 34.3 (c = 0.087,
MeOH). Pharm: Antioxidant (DPPH scavenger, EC50 > 50g/mL, 50g/mL
InRt = 18%, control Ascorbic acid, EC50 = 1.6g/mL = 9.1mol/L). Source:
BEI SHA SHEN Glehnia littoralis (underground part). Ref: 4154.
HO
OH
H
O
O

(fruit). Ref: 5015.
HO
O
OO
HO
OH
OH
OH
8548 Glepidotin A
H
H
OH
OO
OO
OO
HO
OH
OH
OH
OO
OH
OH
O
O
OH
OH

aureus, Mycobacterium smegmatis and Klebsiella pneumoniae); antifungal
(Candida albicans). Source: MEI ZHOU GAN CAO Glycyrrhiza lepidota.
OH
OH
OH
Ref: 1521.
OH
OH
OH
OH
OO
HO
OH
OH OH
OH OH OH
8549 Glepidotin B
[87440-56-0] C20H20O5 (340.38). Pharm: Antimicrobial (broad spectrum).
8545 Glehlinoside A
Source: MEI ZHOU GAN CAO Glycyrrhiza lepidota. Ref: 1521.
C34H43O14 (674.71). Colorless amorphous solid, []D = 158.3 (c = 0.08,

MeOH). Pharm: Antioxidant (DPPH scavenger, EC50 = 18.9g/mL =
HO
28.0mol/L, control Ascorbic acid, EC50 = 1.6g/mL = 9.1mol/L)[4154].
Source: BEI SHA SHEN Glehnia littoralis (underground part). Ref: 4154.
OH
OH
8550 Glepidotin C
OO
[126026-25-3] C19H22O3 (298.39). Pharm: Antimicrobial. Source: MEI ZHOU
OH
HO
OH
OH
OH
GAN CAO Glycyrrhiza lepidota. Ref: 658.

OH
OH
HO
OH
OH
8546 Glehlinoside B
C35H44O15 (704.73). Colorless amorphous solid, []D = 54.5 (c = 0.107,
8551 Glepidotin D
MeOH). Pharm: Antioxidant (DPPH scavenger, EC50 > 50g/mL, 50g/mL
2-(3-Methyl-2-butenyl)-3-O-(3-methyl-2-butenyl)-5-[2-(3-hydroxyphenyl)eth
InRt = 37%, control Ascorbic acid, EC50 = 1.6g/mL = 9.1mol/L)[4154].
yl]-1,3-benzenediol C24H30O3 (366.50). Pharm: Anti-HIV (IC50 = 5.0g/mL,
Source: BEI SHA SHEN Glehnia littoralis (underground part). Ref: 4154.
EC50 = 2.0g/mL)[5180]. Source: MEI ZHOU GAN CAO Glycyrrhiza lepidota

O
O
OH
OO
OH
HO
O
OH
OH
OH
OH
OH
O
HO
O
448
8552 Glicoricone
8557 Globulixanthone E
C37H30O9 (618.65). Pale yellow amorphous powder, mp 228C. Pharm:

Antimicrobial (in vitro, significant activity against a range of microorganisms).
HO
Source: KA MAI LONG XIN FO NI A Symphonia globulifera. Ref: 2029.

OH
O
HO
OH
OH
HO
8553 Glisoflavanone
O
O
C25H28O6 (424.50). Pale yellow acicular Crystals, mp 131C, []D = 0 (c = 1,
acetone). Source: GAN CAO Glycyrrhiza uralensis. Ref: 748.

O
HO
OH
O
HO
OH
8558 Globuxanthone
[13586-28-2] C18H16O5 (312.33). Source: KA MAI LONG XIN FO NI A
Symphonia globulifera, Garcinia vilersiana (bark). Ref: 1521, 3902.
8554 Globoidnan A
C26H20O10 (492.44). Brown oil, []D = +14.4 (c = 0.118, MeOH). Pharm: HIV
integrase Inhibitor (IC50 = 0.64mol/L). Source: Eucalyptus globoidea (bud).
OH
OH
Ref: 3894.
O
OH
O
OH
HO
8559 Glochidacuminoside A
HO

OH
OH
OH
Source: JIAN JIAN SUAN PAN ZI Glochidion acuminatum (leaf). Ref: 4286.
OH
8555 Globulixanthone C
1,7,8-Trihydroxy-2,2-dimethylpyrano[5',6': 3,4]xanthone C18H14O6 (326.31).
Yellow needles, mp 285C. Pharm: Antimicrobial (in vitro, significant activity
against a range of microorganisms). Source: KA MAI LONG XIN FO NI A
HO
O
OH
Symphonia globulifera. Ref: 2029.

OH
OH
OH
OH
8560 Glochidacuminoside B
HO

O
8556 Globulixanthone D
(326.35). Yellow Crystals, mp 120C. Pharm: Antimicrobial (in vitro,
significant activity against a range of microorganisms); cytotoxic (P 388 ED50 =
OO
1,6-Dihydroxy-5-methoxy-7-(3-methylbut-2-enyl)xanthone C19H18O5
HO
OH
OH
OH
OH
0.42g/mL, control Mithramycin ED50 = 0.06g/mL, HT29 ED50 =

0.98g/mL, control Mithramycin ED50 = 0.08g/mL)[4094]. Source: KA MAI
8561 Glochidacuminoside C
LONG XIN FO NI A Symphonia globulifera, TAI WAN LV DAO TENG
HUANG Garcinia linii. Ref: 2029, 4094.
OH
OO
O
HO
O
O
HO
OH
OH
O
OH
OH
449
8562 Glochidacuminoside D
8566 Glochidionionoside B
C21H21NO11 (463.40). Amorphous powder, []D28 = 72.8 (c = 0.67, MeOH).
(6R,9S)-Megastigman-3-on-4-ene-9,13-diol C19H32O8 (388.46). Amorphous
powder, []D28 = +7.4 (c = 1.22, MeOH); []D25 = +7.5 (c = 0.53, MeOH).

Source: CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (leaf), LV BEI
OO
HO
GUI HUA Excoecaria cochinchinensis var. viridis. Ref: 4323, 4543.
OH
OH
OH
O
O
H
O
OH
OO
HO
HO
OH
OH
OH
OH
OH
8563 Glochidiol
C30H50O2 (442.73). mp 260~262C, []D23 = +19 (c = 0.98, CHCl3); mp
20
265~267C (hexane), []D = +18.3 (c = 0.05g/mL, CHCl3). Pharm:

Antineoplastic (EBV-EA induced by TPA, IC50 = 290 (mol ratio/32pmol TPA,
8567 Glochidionionoside C
(6R,7E,9S)-Megastigman-3-one-4,7-diene-9,13-diol 13-O-D-glucopyranoside C19H30O8 (386.45). Amorphous powder, []D28 = +112.1 (c = 1.42,
control Curcumin IC50 = 343 (mol ratio/32pmol TPA)[4099]; cytotoxic
MeOH). Source: CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (leaf).
(inhibition growth of hmn tumor cell lines, MCF7 (breast), GI50 =
Ref: 4323.
OH
(6.60.7)mol/L, control Doxorubicin, GI50 = (42.88.2)mol/L;

NCI-H460 (lung), GI50 = (7.50.5)mol/L, Doxorubicin, GI50 =
(94.08.7)mol/L; SF268(CNS), GI50 = (9.70.3)mol/L, Doxorubicin,
GI50 = (93.07.0)mol/L)[5065]. Source: CHUI ZHU SUAN PAN ZI
H
O
OO
HO
Glochidion zeylanicum (stem cortex), MAO GUO SUAN PAN ZI Glochidion
OH
eriocarpum (root and stem wood), YUAN GUO SUAN PAN ZI Glochidion
OH
sphaerogynum (root and stem wood). Ref: 4099, 5065.
OH
8568 Glochidionionoside D
H
Source: CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (leaf). Ref: 4323.
OH
HO
OO
HO
OH
8564 Glochidiolide
OH
C16H16O6 (304.30). Colorless rods, mp 210~213C, []D25 = 69.8 (c = 0.49, DMSO).

O
OH
OH
8569 Glochidone
C30H46O (422.70). mp 165~167C, []D23 = +42 (c = 0.46, CHCl3); mp
163~164C (EtOH), []D20 = +70.6 (c = 7mg/mL, CHCl3). Pharm:
OO
control Curcumin IC50 = 343 (mol ratio/32pmol TPA)[4099]; cytotoxic

(inhibition growth of hmn tumor cell lines, MCF7 (breast), GI50
HO
HO
>100mol/L, control Doxorubicin, GI50 = (42.88.2)mol/L; NCI-H460
8565 Glochidionionoside A
(lung), GI50 >100mol/L, Doxorubicin, GI50 = (94.08.7)mol/L;
(6S,7E,9S)-Megastigman-3-one-4,7-diene-6,9,13-triol 13-O--D-glucopyranoside
SF268(CNS), GI50 >100mol/L, Doxorubicin, GI50 =
C19H30O9 (402.45). Amorphous powder, []D28 = +29.1
(c = 1.48, MeOH). Source:
CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (leaf). Ref: 4323.

OH
(93.07.0)mol/L)[5065]. Source: CHUI ZHU SUAN PAN ZI Glochidion

zeylanicum (stem cortex), MAO GUO SUAN PAN ZI Glochidion
eriocarpum (root and stem wood). Ref: 4099, 5065.
OH
O
O
HO
O
OH
OH
OH
450
8570 Glochidonol
8574 Glochiflavanoside D
C30H48O2 (440.72). mp 225~227C, []D23 = +23 (c = 0.95, CHCl3); mp
C23H28O11 (480.47). Amorphous powder. Source: CHUI ZHU SUAN PAN ZI
228~230C (hexane), []D20 = +50.7 (c = 0.5g/100mL, CHCl3). Pharm:
Glochidion zeylanicum (leaf). Ref: 4103.
control Curcumin IC50 = 343(mol ratio/32pmol TPA)[4099]; cytotoxic (inhibition

growth of hmn tumor cell lines, MCF7 (breast), GI50 = (9.03.7)mol/L,
control Doxorubicin, GI 50 = (42.88.2)mol/L; NCI-H460 (lung), GI50 =
OH
O
HO
(4.90.2)mol/L, Doxorubicin, GI50 = (94.08.7)mol/L; SF268(CNS),

GI50 = (9.80.5)mol/L, Doxorubicin, GI50 = (93.07.0)mol/L)[5065].
HO
OH
Source: CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (stem cortex),

MAO GUO SUAN PAN ZI Glochidion eriocarpum (root and stem wood),
OH
YUAN GUO SUAN PAN ZI Glochidion sphaerogynum (root and stem
OH
8575 Gloeophyllic acid A dimethylacetal
wood). Ref: 4099, 5065.
4,4,14-Trimethyl-24-oxo-5-chol-8-en-21-oic acid dimethylacetal C29H48O5

(476.70). Amorphous yellow powder, mp 205~210C. Source: Gloeophyllum
odoratum. Ref: 3972.
H
OH
O
O
HO
H
8571 Glochiflavanoside A
HO
Source: CHUI ZHU SUAN PAN ZI Glochidion zeylanicum (leaf). Ref: 4103.
8576 Gloeophyllol A
C15H20O2 (232.23). Colorless oil, [] D = 33 (c = 0.2, CHCl3:CH3OH =
O
OH
O
OO
HO
inactive (Mucor miehei, Paecilomyces notatum, Paecilomyces variotii,
OH
OH
Nematospora coryli, 100g/filter disc); cytotoxic inactive (HeLa-S3, HL-60,
OH
OH
19:1). Pharm: Antibacterial inactive (Bacillus brevis, Bacillus subtilis,

Enterobacter dissolvens, Micrococcus luteus, 100g/filter disc); antifungal
COS-7). Source: Gloeophyllum sp. Ref: 3968.
8572 Glochiflavanoside B
OH
C24H30O12 (510.50). Colorless needles(MeOH), mp 222~224C, []D22 =

61.4 (c = 0.57, MeOH). Source: CHUI ZHU SUAN PAN ZI Glochidion
zeylanicum (leaf). Ref: 4103.
OH
8577 Gloeophyllol B
O
OH
O
OO
HO
OH
Penicillium notatum, 50g/filter disc, weak activity); cytotoxic inactive

(HeLa-S3, HL-60, COS-7). Source: Gloeophyllum sp. Ref: 3968.
OH
C16H22O2 (246.35). Colorless oil. Pharm: Antifungal (Mucor miehei,
OH
OH
8573 Glochiflavanoside C
C24H30O12 (510.50). Colorless needles(MeOH), mp 260~262C, []D25 = 5.7
(c = 0.35, MeOH). Source: CHUI ZHU SUAN PAN ZI Glochidion
zeylanicum (leaf). Ref: 4103.
OH
8578 Gloeophyllol C
C15H20O3 (248.32). Colorless oil, with no optical activity (c = 0.6, CHCl3). Pharm:
Antifungal inactive (Mucor miehei, Penicillium notatum, 50g/filter disc);
cytotoxic inactive (HeLa-S3, HL-60, COS-7). Source: Gloeophyllum sp. Ref: 3968.
O
O
O
HO
O
OH
HO
O
OH
OH
OH
OH
HO
OH
451
8579 Gloeophyllol D
8584 Glomeratose C
C15H22O4 (266.34). Colorless oil, with no optical activity (c = 0.4, CHCl 3).
C33H40O17 (708.68). []D = 71.2. Source: DA JIN NIU CAO Polygala
Pharm: Antibacterial inactive (Bacillus brevis, Bacillus subtilis,
chinensis [Syn. Polygala glomerata]. Ref: 2184.
Enterobacter dissolvens, 100g/filter disc); antifungal (Mucor miehei,
Paecilomyces notatum, Paecilomyces variotii, Nematospora coryli,

100g/filter disc); cytotoxic inactive (HeLa-S3, HL-60, COS-7). Source:
Gloeophyllum sp. Ref: 3968.
OH
OOH O
O
HO
OH
HO
O
OH
HO
O
OH OH
HO
8585 Glomeratose D
OH
8580 Gloeophyllone
C15H20O3 (248.32). Colorless oil, [] D = 140 (c = 0.3, CHCl3). Pharm:
Antibacterial inactive (Bacillus brevis, Bacillus subtilis, Enterobacter

O
O
dissolvens, 100g/filter disc); antifungal inactive (Mucor miehei,

Paecilomyces notatum, Paecilomyces variotii, Nematospora coryli,
O
OH
OH
100g/filter disc); cytotoxic inactive (HeLa-S3, HL-60, COS-7). Source:
HO
Gloeophyllum sp. Ref: 3968.

HO
O
O
OOH O
O
O
OH OH
8586 Glomeratose E
HO
8581 Gloeosteretriol
C15H26 O3 (254.37). Colorless prismatic Crystals, mp 205~206C, []D22 =
+5.6 (c= 0.115, methanol). Source: YU ER Gloeostereum incarnatum.

HO
Ref: 214.
OH
HO
OH
HO
OH
O
O OH
O
OH
OH
HO
H
O
OH
8587 Glomeratose F
8582 Glomeratose A
C24H34O15 (562.53). []D = +5.7. Source: DA JIN NIU CAO Polygala
O
O
HO
OH
HO
OO
OH
OH
OH
HO
HO
OH
8583 Glomeratose B
O OH O
O
OH OHO
O
O
8588 Gloriogenin
sisalana. Ref: 2503.
OH
OHHO
O
OH
[38676-82-3] C27H42O4 (430.63). mp 166C. Source: JIAN MA Agave
O
O
OH
OH
OH OHO
HO
HO
O
HO
OH
O OH O
O
OH
H
HO
452
8589 Glucobrassicin
8593 Glucoconvallasaponin B
[4356-52-9] C16H20N2O9S2 (448.47). Source: BAO ZI GAN LAN Brassica
[16939-88-1] C38H62O15 (758.91). Source: LING LAN Convallaria keiskei
oleracea var. gemmifera, DA QING YE Isatis indigotica, GAN LAN Brassica
[Syn. Convallaria majalis]. Ref: 6.
oleracea var. capitata, LAI FU ZI Raphanus sativus, OU ZHOU YOU CAI
Brassica napus. Ref: 2, 1521.

O
OH
H
OH
O S O
O
N
HO
OS
HO
OH
O
O
OH
OH
OH
OH
OO
OH
OH
OH
N
OH H
OH
8590 Glucobrassicin-1-Sulfonate
C16H20N2O12S3 (528.54). Source: DA QING YE Isatis indigotica. Ref: 2, 6.
8594 Glucodichotomine B
OH
O S O
HO
Pharm: -Hexosaminidase inhibitor inactive (RBL-2H3 cells, 100mol/L,
InRt = (3.21.1)%, control Ketotifen fumarate, InRt = (19.11.3)%)[2571].
OS
Source: YIN CHAI HU Stellaria dichotoma var. lanceolata (root: yield =
OH
OH
0.0014%). Ref: 2571.

OH N
O S OH
OH
OH
OH
H
N
8591 Glucocheirolin
[554-86-9] C11H20NO11S3 (438.47). Monohydrate, acicular crystals (90%
OH
Source: GUI ZHU XIANG Cheiranthus cheiri, HUA YE CAI Brassica

oleracea var. botrytis, LA GEN Armoracia lapathifolia, WU JING GAN LAN
Brassica napus var. napobrassica. Ref: 661.
OH
HO
ethanol), mp 158~160C, []D27 = 21.56 (water). Pharm: Antibacterial.

O
8595 Glucoerucin
[21973-56-8] C12H22NO9S3 (420.50). Source: BAO ZI GAN LAN Brassica
oleracea var. gemmifera, GAN LAN Brassica oleracea var. capitata, WU
JING GAN LAN Brassica napus var. napobrassica, ZHI MA CAI Eruca
O S O
N
sativa. Ref: 658.
O
S
HO
OS
OH
OH
O S O
N
O
S
OH
HO
OS
OH
8592 Glucoconvallasaponin A
[19316-99-5] C38H62O14 (742.91). Source: LING LAN Convallaria keiskei
OH
OH
[Syn. Convallaria majalis]. Ref: 6.

8596 Glucoerysolin
O
[74542-16-8] C12H22NO11S3 (452.50). Pharm: Antibacterial (using its ligand

erysoline); antifungal (using its ligand erysoline); cytotoxic (animal, using its
OH
H
H
OH
OO
OH
ligand erysoline). Source: WU JING GAN LAN Brassica napus var.
napobrassica, A FU HAN TANG JIE Erysimum perofskianum. Ref: 658.
H
O
OH
O S O
N
OO
HO
OH
O
S
HO
OS
OH
OH
OH
OH
OH
453
8597 1-O-Gluco-2-O-gadoleic-glyceride
8601 5''-O--D-Glucopyranosylamarogentin
C29H54O9 (546.75). White lamellar solid, mp 177~179C. Source: CAO SU
C35H40O18 (748.70). Source: RI BEN ZHANG YA CAI Swertia japonica. Ref: 2573.
Phlomis umbrosa. Ref: 823.
OH
HO
HO
OH
OO
HO
OH
H
OO
OH
OH
OH
O
HO
8598 Glucoiberin
OH
Source: BAO ZI GAN LAN Brassica oleracea var. gemmifera, GAN LAN
Brassica oleracea var. capitata, HUA YE CAI Brassica oleracea var. botrytis,
LA GEN Armoracia lapathifolia, PIE LAN Brassica oleracea var. gongylodes,
QU QU HUA Iberis amara, YU YI GAN LAN Brassica oleracea var.
sabauda. Ref: 658.
OH

O
OH
H
OO
HO
OH
S O
OS
OH
OH
8602 5''-O--D-Glucopyranosylamaroswerin
O S O
HO
O
OH
[554-88-1] C11H20NO10S3 (422.47). Pharm: Cytotoxic (animal model).
HO
OH
OH
OH
O
HO
HO
OH
8599 Gluconasturtiin
OH
2-Phenylethyl glucosinolate [499-30-9] C15H21NO9S2 (423.46). Off-white
OH
20
crystals (MeOHEtOH, as K salt), mp 171C (K salt), []D = 20.7 (c = 1.0,

H2O). Pharm: Cytotoxic (animal model). Source: BAI JIE ZI Sinapis alba
[Syn. Brassica alba; Brassica hirta], DOU BAN CAI Nasturtium officinale,
HEI JIE Brassica nigra, JIE CAI Brassica juncea, JIE ZI Brassica juncea,
JIA DU XING CAI Lepidium sativum, OU ZHOU SHAN JIE Barbarea
8603 1-O--D-Glucopyranosylamplexin
[157464-32-9] C16H26O9 (362.38). Source: BAI HUA LONG DAN Gentiana
algida[704], LONG DAN Gentiana scabra (dried rhizome and root)[3097], RI
BEN ZHANG YA CAI Swertia japonica[2528]. Ref: 704, 2528, 3097.
O
vulgaris. Ref: 658, 1521, 3196.

HO
OS
OH
OH
O
O S O
OH
OH
OH
OH
OO
OH
HO
H
OH
8604 3-O-[-D-Glucopyranosyl-(13)][-L-arabinopyranosyl-(12)]-L-arabinopyranosyl-pseudojujubogenin
C46H74O17 (899.09). Source: JIA MA CHI XIAN Bacopa monniera (whole
8600 Gluconic acid
herb: yield = 0.019%fw). Ref: 4664.
D-Gluconic acid C6H12O7 (196.16). mp 125~126C. Source: HE YE Nelumbo

nucifera. Ref: 6.
HO
O
H
HO
OH
OH
O
OH
OH
OH
OH
HO
HO
HO
OO
O O
OH
O
OH
O
HO
OH
454
8605 3-O--D-Glucopyranosyl-20-O-[-L-arabinopyranosyl(12)-
8608 3-[(O--D-Glucopyranosyl-(13)--L-arabinopyranosyl)oxy]-23-
-D-glucopyranosyl]3,12,20(S)-trihydroxydammar-24-ene
hydroxyolean-12-en-28-oic acid O--L-rhamnopyranosyl-(14)-O--D-
glucopyranosyl-(16)--D-glucopyranosyl ester
+34.5 (c = 0.08, MeOH). Pharm: Inhibits zoospore motility (Aphanomyces
C59H96O27 (1237.41). Source: SAN YE MU TONG Akebia trifoliata (stem).
cochlioide, a causative fungus of spinach root rot). Source: SAN QI Panax
Ref: 4545.
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]. Ref: 2387.

HO
OO
OH
OH
HO
OH
OO
OH
H
OH O O
O O
HO
OH
HO
OH
OO
OH
OH
OH
OO
OH
8606 3-O--D-Glucopyranosyl-(14)--L-arabinopyranosyl
OO
OO
OH
OH
OH
OH
OH
H
HO
OH
OH
OH
OH
OH OH
hederagenin 28-O--L-rhamnopyranosyl ester

C47H76O17 (913.12). Colorless plate crystals (MeOH), mp 237~242C, []D25 =
+33.3 (c = 0.1, MeOH). Pharm: Antifungal (Penicillium avellaneum, MIA =
8g/disc, control Amphotericin B, MIA = 0.04g/disc; Candida albicans, MIA =
50g/disc, control Amphotericin B, MIA = 0.4g/disc; Candida glabrata, MIA =
8609 5-O-(-D-Glucopyranosyl)-10-benzoyltaxacustone
C37H48O14 (716.79). mp 178~180C, []D = 92.6 (CHCl3). Source: ZI SHAN
Taxus cuspidata. Ref: 662.
20g/disc, Amphotericin B, MIA = 0.8g/disc; Saccharomyles cerevisiae, MIA

O
= 5g/disc, Amphotericin B, MIA = 3.2g/disc; Cryptococcus neoformans, MIA

= 50g/disc, Amphotericin B, MIA = 0.0.8g/disc; T. beigelii, MIA = 10g/disc,
Amphotericin B, MIA = 0.8g/disc; P. oryzae, MIA = 10g/disc, Amphotericin

B, MIA = 0.08g/disc). Source: GAN QING TIE XIAN LIAN Clematis
tangutica. Ref: 5413.

HO
H
O
OO
HO
OH
OH
O
OH
OO
HO
OH
OH
OO
OO
8610 26-O--D-Glucopyranosyl-3,26-dihydroxy-5-choleslen-16,22-
HO
dioxo-3-O--L-rhamnopyranosyl-(12)--D-glucopyranoside
OH OH
C45H72O18 (901.06). White powder (MeOH), mp 225~226C, mp 208~209C
OH
OH
OH
Source: BAI HE Lilium brownii var. viridulum [Syn. Lilium brownii var.
colchesteri]. Ref: 418, 441.
OH
8607 3-O--D-Glucopyranosyl(13)--L-arabinopyranosyl oleanolic acid

C41H66O12 (750.98). White powder (CHCl3/MeOH), mp 224~226C. Source:
HUANG HUA BAI JIANG Patrinia scabiosaefolia. Ref: 2455.

H
H
HO
H
H
OH O O
HO
O O
OH
OH
OH
OH
OH O O
OH OH
OH
OH
OO
OH
O
O
HO
O
OH
OH
OH
455
8611 3-O--D-Glucopyranosyl betulinic acid-28-O--D-glucopyranosyl-
8616 7-O--D-Glucopyranosyl-3,4'-dihydroxy-3'-(4''-acetoxyl-3''-meth-
ylbutyl)-5,6-dimethoxyflavone
Cirensenoside P C48H78O18 (943.15). White powder, mp 204~206C, []D20 =
C30H36O14 (620.61). Yellowish gummy solid, []D24 = +14.2 (c = 0.07,
16.9 (c = 0.5, methanol). Source: DONG BEI CI REN SHEN Oplopanax
MeOH). Pharm: -Glucosidase inhibitor inactive. Source: JIA LIAN QIAO
elatus. Ref: 370.
YE Duranta repens. Ref: 4050.
HO
H
H
OO
OH
OH
OH
OH
OH
OH
OH
OH
O
OH
8612 1-O-(3'-O--D-Glucopyranosyl)-(E)-caffeoyl--D-glucopyranose
MeOH). Source: GE XUN Balanophora japonica (underground part: yield =
0.0026%). Ref: 4101.
O
O
OH
OO
OO
HO
OH
OH
O
OH
H
HO
O
OH
8617 7-O--D-Glucopyranosyl-3,5-dihydroxy-3'-(4''-acetoxyl-3''-methylbutyl)-6,4'-dimethoxyflavone
C30H36O14 (620.61). Yellowish gummy solid, []D24 = +27 (c = 0.1, MeOH).
Pharm: -Glucosidase inhibitor (IC50 = (65.52.5)mol/L, control Deoxynojirimycin, IC50 = (425.68.1)mol/L). Source: JIA LIAN QIAO YE Duranta
repens. Ref: 4050.
OH
OO
HO
OH
OH
HO
HO
OH
OH
OH
OH
OH
OH
8613 3'-O--D-Glucopyranosyl-catalpol
Source: CHA RU SHI WAN CUO Asystasia intrusa. Ref: 2589.
HO
HO
HO
HO
OH
OH
OH
O
OH
OO
OH
8618 6-C-Glucopyranosyl-5,7-dihydroxy-2-isopropylchromone
O
H
HO
OH
0.51, MeOH). Source: GANG SONG Baeckea frutescens. Ref: 1895.
O
HO
OH
OH
OH
OH
8619 8-C-Glucopyranosyl-5,7-dihydroxy-2-isopropylchromone
OH
OH
8614 4-O--D-Glucopyranosyl-1-deoxynojirimycin
1.05, MeOH). Source: GANG SONG Baeckea frutescens. Ref: 1895.
C12H23NO9 (325.32). Source: Morus sp. Ref: 2513.

OH
H
N
HO
OH
OO
HO
OH
OH
O
HO
O
OH
OH
OH
OH
OH
OH
8615 15-O--D-Glucopyranosyl-11,13-dihydrourospermal A
C21H30O10 (442.47). Oil. Source: XU DUAN JU Sonchus asper [Syn. Sonchus
8620 C--D-Glucopyranosyl-2,6-dihydroxyl benzene
oleraceus var. asper] (root). Ref: 3923.
C12H16O7 (272.26). Source: NANG ZHUANG ZI TAN Pterocarpus

marsupium (heartwood). Ref: 3789.
OO
HO
OH
OH
OH
OH
HO
HO
O
OH
OH
OH
OH
456
8621 28-O--D-Glucopyranosyl-2-3-dihydroxyolean-12-ene-24,28-
8625 2-O-(2)--D-Glucopyranosyl-4,6-dimethoxy phenylenthanone
dioic acid
C16H22O9 (358.35). White powder. Source: YAN SHENG JIA MU ZEI
C36H56O11 (664.84). Pharm: Tissue factor inhibitor (IC50 =0.036mmol/L/Unit
Anabasis salsa, DUAN YE JIA MU ZEI Anabasis brevifolia. Ref: 4861.

O
of TF). Source: MU GUA Chaenomeles sinensis. Ref: 5387.

O
O
O
HO
O
H
O
HO
HO
O
OH
HO
OH
8626 3-O--D-Glucopyranosyl-(14)--D-fucopyranosyl (22S,24Z)-
cycloart-24-en-3,22,26-triol 26-O--L-arabinopyranosyl-(16)--D-
OH
OH
OH
OH
glucopyranoside
OH
8622 1-(3-O--D-Glucopyranosyl-4,5-dihydroxyphenyl)-ethanone
HUA DONG TANG SONG CAO Thalictrum fortunei (aerial parts: yield =
0.0040%dw). Ref: 911.
OH
OH
HO
OO
OH
OH
OH
OH
OH
HO
O O
OH
8623 26-O--D-Glucopyranosyl-3,26-dihydroxy-20,22-seco-25(R)-furost-5-en-20,22-dione-3-O--L-rhamnopyranosyl-(14)--L-rhamnopy-
OH
OH
OH
OO
OH
OH
OH
OH
OH
OH
ranosyl-(14)-[-L-rhamnopyranosyl-(12)]--D-glucopyranoside
C57H92O27 (1209.35). White amorphous powder. Pharm: Antifungal inactive
cycloart-24-en-3,22,26-triol 26-O--D-glucopyranoside
(Candida albicans, Candida glabrata, Candida tropicalis, MIC > 200g/mL).
Source: YUAN SHU YU Dioscorea rotundata [Syn. Dioscorea cayenensis].
Ref: 2560.
0.0048%dw). Ref: 911.

OH
OO
O
O
H
H
HO
H
H
HO
OH
OH
HO
OH
HO
OO
OH
O OOH
OH O O
OH OH
OH OH
O O
OO
OH
OH
OH
OH
OH
OH
OH
OH
8628 3-O--D-Glucopyranosyl-(14)--D-fucopyranosyl (22S,24Z)OH OH
cycloart-24-en-3,22,26-triol 26-O--D-quinovopyranosyl-(16)--Dglucopyranoside
8624 3-O-(-D-Glucopyranosyl)-1-(3',5'-dimethoxy-4'-hydroxyphenyl)-
1-propanone
0.0025%dw). Ref: 911.

OH
H
O
OH
OO
HO
OH
O
O
OH
OH
OO
OH
HO
O O
OH
OH
OH
OO
OH
OH
OH
OH
OH
OH
OH
457
8633 26-O--D-Glucopyranosyl(25R)-5-furostane-12-one-3,22,26-
cycloart-24-en-3,22,26-triol 26-O--D-xylopyranosyl-(16)--D-gluco-
triol-3-O--D-glucopyranosyl-(12)--D-galactopyranoside
pyranoside
C45H74O20 (935.08). White powder, []D15 = 15 (c = 0.2, pyridine). Pharm:
Enhances sex drive; inhibits onset of senility; treatment of angiocardiopathy.
Source: CI JI LI Tribulus terrestris. Ref: 688.
0.0017%dw). Ref: 911.
OH
OH
O
O
OO
OH
HO
O O
OO
OH
OH
OH
O
OH
OH
OH
OH
Dracaena cochinchinensis. Ref: 2114.
8634 26-O--D-Glucopyranosyl(25R,S)-5-furostane-12-one-20(22)en-3,26-diol-3-O--D-glucopyranosyl-(14)--D-galactopyranoside
Source: CI JI LI Tribulus terrestris. Ref: 688.
HO
O
OO
OH
OH
OH
OH
O
OH
OH
OH
OH
C22H30O14 (518.48). Source: LONG DAN Gentiana scabra (dried rhizome
OO
and root). Ref: 3097.
OH
OH
OO
OH
H HO
8635 4'-O--D-Glucopyranosylgentiopicroside
OH
O HO
H
HO
O O
HO
MEN Asparagus gobicus (root). Ref: 4975.
O
OH
C39H66O14 (758.95). []D21 = 48.0 (c = 1.00, MeOH). Source: GE BI TIAN
OH
OH
OH
OH
Enhances sex drive; inhibits onset of senility; treatment of angiocardiopathy.
OH
OO
OH
OO
OH
8631 26-O--D-Glucopyranosylfurostane-3,26-diol-3-O--D-glucopyranoside
HO
O
H
H
OH
HO
C45H72O19 (917.06). White powder, []D15 = +5 (c = 0.2, pyridine). Pharm:
OH
O
OH
OH
C38H60O14 (740.89). White powder. Source: JIAN YE LONG XUE SHU
H HO
OH
HO
tetrahydroxy-1-O--L-arabinopyranoside
OH
OO
OH
OH
OH
HO
OH
8630 26-O--D-Glucopyranosyl-furostan-5,25(27)-diene-1,3,22,26-
OH
HO
OH
OO
HO
OH
8632 26-O--D-Glucopyranosylfurostane-3,26-diol-3-O--D-xylopyranosyl(14)--D-glucopyranoside
OO
HO
OH
C44H74O18 (891.07). []D21 = 29.5 (c = 0.75, MeOH). Pharm: Cytotoxic (in

vitro, HO-8910, IC50 > 226mol/L, Vincristine, IC50 = (25.11.9)mol/L;
OH
Bel7405, IC50 > 226mol/L, Vincristine, IC50 = (31.43.4)mol/L). Source:

GE BI TIAN MEN Asparagus gobicus (root). Ref: 4975.
OH
OH
8636 6'-O--D-Glucopyranosylgentiopicroside
[115713-06-9] C22H30O14 (518.48). Source: LONG DAN Gentiana scabra
OH
O HO
H
H
HO
OO
OH
OO
OH
H
H
OO
OH
(dried rhizome and root)[3097], QIN JIAO Gentiana macrophylla, RI BEN

ZHANG YA CAI Swertia japonica. Ref: 707, 2573, 3097.
O
OH
H
O
OH
OO
HO
OH
OH
OH
OH
OH
OO
OH
OH
OH
OH
458
8637 3-O--D-Glucopyranosyl-(16)--D-glucopyranoside of ethyl
8641 -D-Glucopyranosyl-(12)--D-glucopyranosyl-15,16-epoxy-12-
3-hydroxyoctanoate
oxo-8(17),13(16)-14-ent-labdatrien-19-oate
C22H40O13 (512.56). Source: DENG LONG CAO Physalis peruviana. Ref: 1997.
O
HO
OO
OO
OH
OH
C32H46O14 (654.72). Yellow gum, []D25 = 2.0 (c = 0.25, CH3OH). Source:

BI CHI YAN ZI CAI Potamogeton pectinatus. Ref: 3849.
O
OH
OH
OH
OH
8638 3-O-[-D-Glucopyranosyl-(13)]-[-D-glucopyranosyl-(12)]--
HO
L-arabinopyranosyl echinocystic acid

Source: Dizygotheca kerchoveana (stem and leaf of branch). Ref: 3885.
OO
OH
OH
HO
OH
OH
OH
8642 28-O--D-Glucopyranosyl-(16)--D-glucopyranosyl ester of 3-OOH
H
OH O
OH
HO
yl-(13)--L-rhamnopyranosyl-(12)--arabinopyranosyl-hederagenin
C71H116O36 (1545.69). White powder, mp 224~227C, []D21 = 17.4 (c =
OO
[-D-glucopyranosyl-(14)][-L-rhamnopyranosyl-(13)]--D-glucopyranos
0.25, MeOH). Source: CHUAN XU DUAN Dipsacus asperoides. Ref: 265.
OH
OO
HO
OH
OH
OH
OH
OH
H
8639 3-O-[-D-Glucopyranosyl-(13)]-[-D-glucopyranosyl-(12)]-
OH
-L-arabinopyranosyl echinocystic acid 28-O-[-L-rhamnopyranosyl-
OO
HO
OH
OH
(14)--D-glucopyranosyl-(16)--D-glucopyranosyl] ester
OO
HO
OO
HO
OH
HO
H
OO
OH
OH
OH
HO
OH
OO
OO
OH
OH
OO
OH
OH
HO
OH
OH
OH
OH
O O OH
O
O
OH O
OH
OH
OH
OO
OH
OH
OH
HO
H
O
OH
OH
OH
Source: Dizygotheca kerchoveana (stem and leaf of branch). Ref: 3885.
OH
OH OH
8643 28-O--D-Glucopyranosyl-(16)--D-glucopyranosyl ester of 3-OOH
[-D-xylopyranosyl-(14)--D-glucopyranosyl-(14)][-L-rhamnopyran
osyl-(13)]--D-glucopyranosyl-(13)--L-rhamnopyranosyl-(12)--a
rabinopyranosyl-hederagenin
OH OH
8640 3-[(O--D-Glucopyranosyl-(12)-O-[-D-glucopyranosyl-
C76H124O40 (1677.81). White powder, mp 236~240C (methanolacetic ester),
(13)]--L-arabinopyranosyl)oxy]olean-12-en-28-oic acid
[]D21 = 21.8 (c = 0.24, methanol). Source: CHUAN XU DUAN Dipsacus
asperoides. Ref: 249.

OH
OH
H
OH
O
HO
OO
OH
OH
HO
OH
OH
OO
OH
OH
OH
O O OH
O
OH
OO
OH
OH
OH
O
OH
OH
H
H
HO
OO
HO
OO
OH
OH
OH
OH OH
H
HO
OO
OH
O
O
OH
OH
OH
OH
OH
459
8644 1-[(-D-Glucopyranosyl-(16)-O--D-glucopyranosyl-(13)-O-
8648 3-O--D-Glucopyranosyl-(16)--D-glucopyranosyl oleanolic acid
-D-glucopyranosyl-(16)-O--D-glucopyranosyl)oxy]-8-hydroxy-3-
28--D-glucopyranosyl-(16)--D-glucopyranosyl ester
methyl-9,10-anthraquinone
C39H50O24 (902.82). Source: JUE MING ZI Cassia tora. Ref: 2.
0.12, MeOH). Source: CHI GENG TENG Gymnema sylvestre. Ref: 766.
HO
HO
OO
OH
OH
OH
OH
OH
O
OH
OH
OH
OO
OO
H
OH
OH
HO
OH
OO
OO
OH
OH
8645 1-[(-D-Glucopyranosyl-(13)-O--D-glucopyranosyl-(16)-
H
HO
OH
OH
OH
OH
OH
OH
OH
O--D-glucopyranosyl)oxy]-8-hydroxy-3-methyl-9,10-anthraquinone
OO
O
OH
OH
OH
OH
C33H40O19 (740.68). Source: JUE MING ZI Cassia tora. Ref: 2.

O
8649 9-[(-D-Glucopyranosyl-(16)-O--D-glucopyranosyl)oxy]-10hydroxy-7-methoxy-3-methyl-1H-naphthol[2,3-c]pyran-1-one
HO
HO
O
OH
OH
OH
O
OH
Cassiaside C; Toralactone 9-gentiobioside [119170-52-4] C27H32O15 (596.55).
OO
OO
OH
Source: DUN YE JUE MING Cassia obtusifolia, JUE MING ZI Cassia tora.
Ref: 2, 2081.
OH
OH
OH
OH
8646 3-O-[-D-Glucopyranosyl(16)--D-glucopyranosyl]-20-O--Dglucopyranosyl-3,12,20(S)-trihydroxydammar-24-ene
+13.2(c = 0.45, MeOH). Pharm: Inhibits zoospore motility (Aphanomyces
cochlioide, a causative fungus of spinach root rot)[2387]. Source: SAN QI
OO
OH
OH
Panax pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]. Ref: 2387.

HO
OH
O
HO
OH
OH
OH
OH
OO
OH
OH
8650 (25S)-26-[(O--D-Glucopyranosyl-(16)--D-glucopyranosyl)
OH OH
oxy]-22-methoxyfurost-5-en-3-yl O--L-rhamnopyranosyl-(12)-O[O--D-glucopyranosyl-(14)--L-rhamnopyranosyl-(13)]--D-glucopyranoside
HO
OH
OH
OH
C64H106O32 (1387.54). Amorphous solid, []D25 = 54.0 (c = 0.10, CHCl3
OO
OO
MeOH = 1:1). Source: JIAN GEN SHU Tacca chantrieri [Syn. Tacca minor;
OH
OH
OH
Tacca esquirolii] (rhizome: yield = 0.00090%dw). Ref: 4648.
8647 3-O--D-Glucopyranosyl-(16)--D-glucopyranosyl oleanolic
HO
HO
HO
acid 28-O--D-glucopyranosyl ester
OO
OH HO
HO
OH
0.11, MeOH). Source: CHI GENG TENG Gymnema sylvestre. Ref: 766.
O
H
H
H
H
OO
HO
OH
OH
OO
OH
OH
OH
OH
HO
HO
OO
HO
OH
OH
HO
HO
OO
OH
OH
OH
HO
HO
OH
O
OH
OH
H
H
460
8651 6-O--D-Glucopyranosyl-20-O--D-glucopyranosyl-3,6,12,
8654 (25R)-3-[(O--D-Glucopyranosyl-(13)-O--D-glucopyranosyl-
20(S),25-pentahydroxydammar-23-ene
(12)-O-[O--L-rhamnopyranosyl-(14)--D-glucopyranosyl-(13)]-
O--D-glucopyranosyl-(14)--D-galactopyranosyl)oxy]-15-hydroxy-
+31.2 (c = 0.25, MeOH). Pharm: Inhibits zoospore motility (Aphanomyces
5-spirostan-12-one
cochlioide, a causative fungus of spinach root rot). Source: SAN QI Panax
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]. Ref: 2387.
Pharm: Cytotoxic (hmn oral squamous cell HSC-2, LD50 = 35g/mL; normal
hmn gingival fibroblast HGF cell, LD50 = 34g/mL). Source: Camassia
OO
HO
leichtlinii (bulb). Ref: 3535.
OH
OH
OH
OH
O
OH
HO
H
O
O
HO
OO
HO
OH
OH
OH
OO
HO
OH
HO
8652 3-O-[-D-Glucopyranosyl-(13)--D-glucopyranosyl]
phytolaccagenic acid 28-O--D-glucopyranosyl ester
C49H78O21 (1003.16). mp 214~218C, []D25 = +48.3 (c = 0.65, MeOH).
Source: CANG BAI CHENG GOU FENG Diploclisia glaucescens. Ref:
2054.
O
O
OH
OH
OH
OH
OH
OO
OH
O
OH
O
HO
OH OH
O
O
OH
OH
OH
OH
OH
(12)-O-[O--L-rhamnopyranosyl-(14)--D-glucopyranosyl-(13)]-
H
HO
HO
O
OH
OH
OH
O--D-glucopyranosyl-(14)--D-galactopyranosyl)oxy]-22-methoxy-
OO
HO
OO
5-furostan-26-yl -D-glucopyranoside
OH
OH
OH
OH
OH
Pharm: Cytotoxic (hmn oral squamous cell HSC-2, LD50 = 4.7g/mL; normal
OH
(12)-O-[O--L-rhamnopyranosyl-(14)--D-glucopyranosyl-(13)]O--D-glucopyranosyl-(14)--D-galactopyranosyl)oxy]-5-spirostanOH
C63H102O33 (1387.50). Pharm: Cytotoxic (hmn oral squamous cell HSC-2,
OH
LD50 = 2.2g/mL; normal hmn gingival fibroblast HGF cell, LD50 =
OH
H
2.4g/mL). Source: Camassia leichtlinii (bulb). Ref: 3535.

H
O
O
H
OO
HO
OH
HO
O
OH
OO
OH OH
OH
OH
OH
OH
OO
HO
OH
O
O
OH
OH
OH
OH
OH
OO
HO
HO
OH
OH O O
OO
HO
OO
HO
OH
OO
HO
12-one
OH
OH
OH
OO
HO
OH OH
O O
OH
OH OH
OH
OH
OH
O
O
461
8656 3-O-[-D-Glucopyranosyl(12)--D-glucopyranosyl]-(25S)-5-
8659 3-[(O--D-Glucopyranosyl-(13)-O--D-glucopyranosyl-(12)-
spirostan-3-ol
O-[-D-xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--D-galacto-
C39H64O13 (740.94). []D21 = 60.9 (c = 1.00, C5H5N). Pharm: Cytotoxic (in
pyranosyl)oxy]-16-[[(4R)-5-(-D-glucopyranosyloxy)-4-methyl-1-oxo-
vitro, HO-8910, IC50 = (5.80.4)mol/L, Vincristine, IC50 = (25.11.9)mol/L;
pentyl]oxy]-2-hydroxypregn-5-en-20-one
Bel7405, IC50 = (5.90.4)mol/L, Vincristine, IC50 = (31.43.4)mol/L).
Source: GE BI TIAN MEN Asparagus gobicus (root). Ref: 4975.
Pharm: Cytotoxic (in vitro, HSC-2, LD50 > 300g/mL; control Doxorubicin,
LD50 = 2.5g/mL). Source: YE XIANG SHU Cestrum nocturnum (leaf: yield
= 0.0026%fw). Ref: 4667.
H
H
HO
OO
H
H
HO
OH
OH
HO
HO
HO
HO
HO
O HO
O
HO HO
OH
OH O HO
O
HO
OO
OH
OO
OH
HO
HO
HO
OH
OH
OH
OH
OH
OH
pyranosyl)oxy]-2-hydroxypregna-5,16-dien-20-one
pyranosyl)-oxy]-2,16-dihydroxypregn-5-ene-20-carboxylic acid -lac-
tone
Pharm: Cytotoxic (in vitro, HSC-2, LD50 = 192g/mL; control Doxorubicin,


= 0.0082%fw). Ref: 4667.
= 0.0014%fw). Ref: 4667.

O
O
HO HO
OH
HO
HO
HO
OH
O
O HO
O
O HO
O
HO
O
OH O HO
O
OH
OO
OH
H
OH
HO
OO
O
HO
OH O
O
HO
HO
HO
O HO
O
HO HO
HO
HO
OH
OO
OH
OH
OH
OH
OH
8661 (25R)-3-[(O--D-Glucopyranosyl-(13)--D-glucopyranosyl8658 (25R)-3-[(O--D-Glucopyranosyl-(13)-O--D-glucopyranosyl-
(12)-O-[-D-xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--
(12)-O-[-D-xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--D-
D-galactopyranosyl)oxy]-5-spirostan-12-one
galactopyranosyl)-oxy]-26-[(-D-glucopyranosyl)oxy]-2-hydroxycholes-
ta-5,17-diene-16,22-dione
Pharm: Cytotoxic (in vitro, HL-60, IC50 = 5.9g/mL; HSC-2, IC50 = 1.5g/mL;
control Etoposide: HL-60, IC50 = 0.3g/mL; HSC-2, IC50 = 24.4g/mL).
Pharm: Cytotoxic (in vitro, HSC-2, LD50 = 281g/mL; control Doxorubicin,
Source: WAN XIANG YU Polianthes tuberosa (underground part: yield =
0.0065%dw). Ref: 4651.
= 0.0088%fw). Ref: 4667.
O
O
HO HO
OH
HO
HO
HO
O HO O
HO O
O
OH O HO
O
OH
OH
OH
OO
OH
HO
HO
HO
HO
HO
HO
HO
HO
O
OH
HO
HO
HO
HO
HO
O O
HO
O O
O HO
O
OH
HO
OH
OO
OH
OH
H
H
462
8662 3-O-(-Glucopyranosyl-(12)--glucopyranosyl(13)--xylo-
8665 6-O--D-Glucopyranosyl-5-hydroxyangelicin
pyranosyl)-16-hydroxyolean-12-en-28-O-(-galactopyranosyl) ester-
C17H16O10 (380.31). Light yellow amorphous powder, []D20 = 40.0 (c =
30-oic acid
0.04, pyridine). Pharm: Antiproliferation inactive (hmn mononuclear cells
C53H84O25 (1121.25). White amorphous powder, []D25 = +18 (c = 1,
MeOH). Pharm: Antiproliferative (in vitro, J774 cell line, IC50 = 0.20mol/L,
peripheral blood, 100mol/L; control Cyclosporine, IC50 = 12nmol/L). Source:
control 6-Mercaptopurine, IC50 = 0.003mol/L; HEK-293, IC50 =
LAN YU LUO YE RONG Ficus ruficaulis var. antaoensis (leaf: yield =
0.15mol/L, 6-Mercaptopurine, IC50 = 0.007mol/L; WEHI-164, IC50 =
0.0012%fw). Ref: 4794.
0.24mol/L, 6-Mercaptopurine, IC50 = 0.017mol/L). Source: Schefflera

fagueti. Ref: 5436.
OH
HO
HO
HO
HO
HO
OO
HO
O
OH
OH
OH
HO
OH
O
O
OH
OH
OH
8666 (2R)-2-O--D-Glucopyranosyl-5-hydroxy-2H-1,4-benzoxazin3(4H)-one
C14H17NO9 (343.29). Amorphous powder, []D26 = +95.0 (c = 0.40, DMSO).
OH
Source: LAO SHU LE Acanthus ilicifolius (aerial parts). Ref: 5204.
OH
OH
OO
OH
OH
HO
O
OH
OH
OH
8663 3-O-[-D-Glucopyranosyl-(13)-O--D-glucuronopyranosyl]-15-hydroxyolean-12-en-16-one
C42H66O14 (794.99). White amorphous powder, mp 248~250C. Source: YUN
8667 20-O--Glucopyranosyl 18-hydroxycamptothecin
NAN GE TENG Pueraria peduncularis. Ref: 853.
C26H26N2O10 (526.50). Source: XI SHU Camptotheca acuminata. Ref: 4097.
H
HO
O
OO
O
HO
OH
OH
OH
OH
OH
HO
OH
OH
OH
O
O O
OH
OH
8664 5-O--D-Glucopyranosyl-6-hydroxyangelicin
8668 1-O--D-Glucopyranosyl-(2S,3R,4E,8Z)-2-N-(2'-hydroxydocosano-
C17H16O10 (380.31). Light yellow amorphous powder, []D20 = +4.1 (c = 0.15,
yl) eicosasphinga-4,8-dienine
pyridine). Pharm: Anti-inflammatory (antiproliferation, hmn mononuclear
C48H91NO9 (826.26). White powder. Source: XIAO YE GUAN ZHONG
cells involving T lymphocytes, B lymphocytes, and macrophages isolated
Matteuccia struthiopteris (rhizome). Ref: 4862.
from peripheral blood, IC50 = 33.4mol/L; control Cyclosporine, IC50 =

12nmol/L). Source: LAN YU LUO YE RONG Ficus ruficaulis var.
OH
antaoensis (leaf: yield = 0.00454%fw). Ref: 4794.
O
NH
OO
HO
OH
HO
HO
HO
HO
OH
OH
OO
OH
OH
463
8669 (25R)-26-O--D-Glucopyranosyl-22-hydroxy-5-furostane-3,26-
8672 1-O--D-Glucopyranosyl-(2S,3R,4E,11E)-2-(2'R-hydroxyhexadece-
diol 3-O--D-glucopyranosyl-(12)-O--D-galactopyranoside
noylamino)-4,11-octadecadiene-1,3-diol
C45H76O19 (921.10). White powder, mp 194~196C []D25 = 31.5 (c = 0.001,
C40H75NO9 (714.05). White amorphous powder, mp 136~138C, []D25 =
H2O). Pharm: Cytotoxic (SF268 and NCI-H460 cancer cells, EC = 25g/mL;
6.0 (c = 0.5, MeOH). Pharm: Antibacterial (Bacillus subtilis, MIC =
HepG2 cells, inactive). Source: XIE BAI Allium macrostemon. Ref: 4897.
20g/mL, control Penicillin G, MIC = 0.80g/mL; Staphylococcus aureus,

MIC = 50g/mL, control Penicillin G, MIC = 0.34g/mL)[3472]; antifungal
(Aspergillus niger, MIC = 30g/mL, control Ketoconazole, MIC = 0.90g/mL;
OH
Candida albicans, MIC = 10g/mL, control Ketoconazole, MIC =

0.65g/mL). Source: BAN XIA Pinellia ternata. Ref: 3472.
O
H
HO
HO
OO
H
O
HO
OH
OH
HN
OH
OH
OH
HO
OO
HO
OH
OO
OH
OH
OH
OH
OH
OH
8673 8-O--D-Glucopyranosyl-6-hydroxy-2-methyl-4H-1-benzopyran-
8670 (25S)-26-O--D-Glucopyranosyl-22-hydroxy-5-furostane-
4-one
3,26-diol 3-O--D-glucopyranosyl-(12)-O--D-galactopyranoside
C45H76O19 (921.10). Pharm: Cytotoxic (SF268 and NCI-H460 cancer cells,
Tyrosinase inhibitor (IC50 = (256.970.96)mol/L, control Kojic acid, IC 50 =
EC = 25g/mL; HepG2 cells, inactive). Source: ZHI MU Anemarrhena
(16.670.52)mol/L, L-Mimosine, IC50 = (3.680.02)mol/L). Source: A FU
asphodeloides. Ref: 2.
HAN DU JUAN HUA Rhododendron collettianum. Ref: 2544.

OH
HO
OH
O
H
HO
HO
OO
OH
H
HO
8674 1-O-(-D-Glucopyranosyl)-(2S,3R,4E,8E)-2-[(2'R)-2'-hydroxynonadecanoylamino]-9-methyl-4,8-octadecadiene-1,3-diol
OH
C44H83NO9 (770.15). Colorless solid, mp 218~220C, [] D28 = 13.2 (c =
OO
0.05, CHCl3). Source: Lobophytum sp. Ref: 4432.
OH
OH
OH
HO
HO
OH
O
OH
OH
OH
OH
8671 (25R)-26-O--D-Glucopyranosyl-22-hydroxy-furost-5(6)-ene3,26-diol-3-O--D-glucopyranosyl(12)[-D-glucopyranosyl(13)]-
NH
HO
-D-glucopyranosyl(14)--D-galactopyranoside
OO
OH
C57H94O29 (1243.37). White powder, mp 223~225C []D27 = 32.7 (c =

0.098, H2O). Pharm: Cytotoxic (SF268 cells, EC = 25g/mL, NCI-H460 cells,
OH
OH
OH
EC = 25g/mL, HepG2 cells, inactive). Source: XIE BAI Allium
8675 (2S)-2-O--D-Glucopyranosyl-2-hydroxyphenylacetic acid
macrostemon. Ref: 4897.
C14H18O8 (314.29). Colorless oil, []D = +6. Pharm: Plant growth stimulatory
or inhibitory activity (radicle length: Lactuca sativa, 1mol/L, StRt or InRt <
OH
10%, 10mol/L, StRt or InRt < 10%, 100mol/L, StRt or InRt < 10%,
1mmol/L, StRt or InRt < 10%; Raphanus sativus, 1mol/L, InRt = (10~30)%,
O
OO
HO
OH
HO
OH
OH
OH
OO
OO
HO
OH
OH
OH
O OH
OH
OH
10mol/L, InRt = (10~30)%, 100mol/L, InRt = (10~30)%, 1mmol/L, InRt =

(10~30)%; Allium cepa, 1mol/L, InRt = (10~30)%, 10mol/L, InRt =
OH
OH
(10~30)%, 100mol/L, InRt = (10~30)%, 1mmol/L, InRt = (31~60)%).

Source: XI YANG JIE GU MU Sambucus nigra. Ref: 5217.
OH
OO
HO
OH
OH
OH
OH
H
HO
OH
464
8676 1-O--D-Glucopyranosyl-2-(3-hydroxyphenyl)-ethanol
8680 -D-Glucopyranosyl-8(17),13-ent-labdadien-16,15-olid-18-oate
C14H20O7 (300.31). Colorless oil. Pharm: Plant growth stimulatory or
C26H38O9 (494.59). Yellow gum, []D25 = 18.1 (c = 0.73, CH3OH). Source:
inhibitory activity (radicle length: Lactuca sativa, 1mol/L, StRt or InRt <
GUANG YE YAN ZI CAI Potamogeton lucens (whole herb). Ref: 3795.
10%, 10mol/L, StRt or InRt < 10%, 100mol/L, StRt = (31~60)%, 1mmol/L,
StRt = (31~60)%; Raphanus sativus, 1mol/L, StRt or InRt < 10%, 10mol/L,
InRt = (10~30)%, 100mol/L, InRt = (10~30)%, 1mmol/L, InRt = (10~30)%;
Allium cepa, 1mol/L, InRt = (10~30)%, 10mol/L, StRt or InRt < 10%,
100mol/L, InRt = (10~30)%, 1mmol/L, InRt = (10~30)%). Source: XI
YANG JIE GU MU Sambucus nigra. Ref: 5217.
O
OO
HO
OH
OH
OO
HO
OH
OH
OH
OH
OH
8681 (1S,2R)-1-(4'-O--D-Glucopyranosyl-3'-methoxyphenyl)-2-(4''-
8677 5-O--D-Glucopyranosyl-8-hydroxypsoralen
hydroxy-3''-methoxyphenyl)-1,3-propanediol
C17H16O10 (380.31). Pharm: Antiproliferation inactive (hmn mononuclear
cells involving T lymphocytes, B lymphocytes, and macrophages isolated
MeOH). Source: SHAN FAN GEN Symplocos caudata. Ref: 2535.
from peripheral blood, 100mol/L; control Cyclosporine, IC50 = 12nmol/L).

O
Source: LAN YU LUO YE RONG Ficus ruficaulis var. antaoensis (leaf: yield
= 0.00065%fw). Ref: 4794.
O
OH
O
OH
OH
HO
HO
OO
OH
HO
HO
HO
OH
OH
OH
8682 4-O--D-Glucopyranosyl methyl gallate

8678 8-O--D-Glucopyranosyl-5-hydroxypsoralen
C14H18O10 (346.29). Yellowish powder, mp 169~170C. Source: JUAN MAO
C17H16O10 (380.31). Light yellow amorphous powder, []D20 = 28.8 (c =
QIANG WEI Rosa sericea. Ref: 676.
0.07, pyridine). Pharm: Antiproliferation inactive (hmn mononuclear cells

O
peripheral blood, 100mol/L; control Cyclosporine, IC50 = 12nmol/L). Source:

HO
LAN YU LUO YE RONG Ficus ruficaulis var. antaoensis (leaf: yield =

0.00075%fw). Ref: 4794.
OO
HO
HO
HO
HO
O
O
OH
OH
OH
OH
OH
8683 3-O-[-D-Glucopyranosyl (13)--D-6-O-methyl-glucoronopyra-
OH
8679 3-O--D-Glucopyranosyl-23-hydroxyursolic acid

C36H58O9 (634.86). White amorphous powder (MeOH/CH2Cl2), 280~281C,
[]D31 = +43.4 (c = 0.046, MeOH). Pharm: Anti-inflammatory (in vitro,
murine macrophage RAW264.7 Cells, inhibits LPS-induced NO and PGE2
nosyl]-3,15,23-trihydroxy-olean-12-en-16-one
MeOH). Pharm: Antifungal (Aspergillus niger). Source: YUN NAN GE
TENG Pueraria peduncularis. Ref: 2159.
release). Source: Cussonia bancoensis. Ref: 5016.
H
O
OH
HO
OO
OH
OH
H
OH
OH
O
OO
HO
O
OH
OH
O
OH
OH
H
H
OH
OH
O
OH
465
8684 4'-O--Glucopyranosyl-5-O-methylvisamminol
8688 (25S)-26-[(-D-Glucopyranosyl)oxy]furosta-5,20(22)-dien-3-yl
C22H28O10 (452.46). Source: FANG FENG Saposhnikovia divaricata [Syn.
O--L-rhamnopyranosyl-(12)-O-[O--D-glucopyranosyl-(14)--L-
Ledebouriella seseloides]. Ref: 2.
rhamnopyranosyl-(13)]--D-glucopyranoside
C57H92O26 (1193.35). Amorphous solid, []D25 = 60.0 (c = 0.10,
CHCl3:MeOH = 1:1). Source: JIAN GEN SHU Tacca chantrieri [Syn. Tacca
minor; Tacca esquirolii] (rhizome: yield = 0.0018%dw). Ref: 4648.

HO
HO
OO
OH
OH
HO
O
HO
OH
O
H
8685 6'-O--D-Glucopyranosylmorroniside
H
HO

HO
MeOH). Source: RI BEN SHUANG HU DIE Tripterospermum japonicum.

Ref: 3533.
HO
O
O
OH OH
8689 (3R,5R)-3-(-D-Glucopyranosyloxy)-5-hexanolide
C12H20O8 (292.29). Oil, []D22 = 21.8 (c = 1.62, MeOH). Source: MO JUE
HO
O
Hymenophyllum barbatum. Ref: 4151.
O
OO
OO
OO
HO
OH
OH
OH
OH
OO
HO
OH
OH
OH
OO
HO
HO
HO
OH
OH
OH
OH
OH
O
OH
8690 (24S,25R)-1-[(-D-Glucopyranosyl) oxy]-6-hydroxy-3,5-cyclo8686 (Z)-8--D-Glucopyranosyloxycinnamic acid
spirostan-24-yl -D-glucopyranoside
C15H18 O8 (326.31). Source: LV DOU Onobrychis viciifolia (leaf). Ref:
C39H62O15 (770.92). Amorphous solid, []D26 = 42.0 (c = 0.10, MeOH). Source:
5084.
DUO ZHI LONG XUE SHU Dracaena surculosa (whole herb). Ref: 4216.
HO
O O
OH
OH
OO
HO
OH
OH
OH
O
HO
H
H
O
OH
OH
OH
OH
OH
OH
8687 16-[(-D-Glucopyranosyl)-oxy]-3,7-dihydroxycholest-5-en23-one
C33H54O9 (594.79). Pharm: Cytotoxic (hmn oral squamous cell HSC-2, LD50
= 68g/mL; normal hmn gingival fibroblast HGF cell, LD50 = 83g/mL).
Source: Camassia leichtlinii (bulb). Ref: 3535.
8691 3-[(-D-Glucopyranosyl)oxy]-17-hydroxy-16-[(O-(2-O-3,4dimethoxybenzoyl--D-xylopyranosyl)-(12)-2-O-acetyl--L-arabinopyranosyl)oxy]cholest-5-en-22-one
Cytotoxic (HL-60 cells, IC50 = 0.00048mol/L, control Etoposide, IC50 =
0.025mol/L). Source: XIA FENG XIN ZI Galtonia candicans (bulb). Ref: 4116.
O
O
H
H
HO
H
H
OH
O
HO
O
OH
OH
H
HO
OH
OH
OO
OH
O
OH
OH
OH
O
OH
O
OH
O
O
O
466
8692 1-D-Glucopyranosyloxy-6-hydroxyeudesman-4(15)-ene
8696 2-(-D-Glucopyranosyloxy)-8-hydroxy-1-methoxy-3-methyl-9,10-
C21H36O7 (400.52). Colorless oil, []D17 = 14 (c = 1.90, CHCl3). Pharm:
anthraquinone
Cytotoxic (inhibits growth of Bel7402 cell, 0.0001mol/L, InRt = 30.1%,
Obtusifolin-2-O--D-glucoside C22H22O10 (446.41). Pharm: Platelet
control Etoposide, InRt = 96.0%). Source: YI NIAN PENG Erigeron annuus
aggregation inhibitor (rat). Source: DUN YE JUE MING Cassia obtusifolia,
JUE MING ZI Cassia tora. Ref: 2, 658, 660.
HO
O
OH
OH
OH
HO
OO
OH
OH
OH
OH
8693 (25R)-26-[(-D-Glucopyranosyl)oxy]-2-hydroxyfurosta-5,20(22)- dien-3-yl
OH
O--D-glucopyranosyl-(13)-O--D-glucopyranosyl-(12)-O-[-D-xylopyranosyl-
8697 2--D-Glucopyranosyloxy-5-hydroxyphenylacetic acid methyl
(13)]-O--D-glucopyranosyl-(14)--D-galactopyranoside
ester


RI BEN LU TI CAO Pyrola japonica (whole herb). Ref: 4294.
= 0.0033%fw). Ref: 4667.
HO
OO
OH
OO
OH
O O HO
OH
HO
HO
HO
HO
HO
O HO
O
HO HO
HO
HO
O
OH
OH
HO
HO
HO
OH
OH
OO
OH
OH
OH
8698 (24S,25S)-24-[(-D-Glucopyranosyl)oxy]-2-hydroxyspirost-5en-3-yl O--D-glucopyranosyl-(13)-O--D-glucopyranosyl-(12)-O[-D-xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--D-galacto-
8694 (25S)-1-[(-D-Glucopyranosyl)oxy]-6-hydroxy-22-methoxy-
pyranoside
3,5-cyclofurostan-26-yl -D-glucopyranoside
C40H66O15 (786.96). Amorphous solid, []D26 = 42.0 (c
= 0.10, MeOH). Source:
DUO ZHI LONG XUE SHU Dracaena surculosa (whole herb). Ref: 4216.
O
HO
LD50 = 2.5g/mL)[4667]. Source: YE XIANG SHU Cestrum nocturnum (leaf:

yield = 0.0060%fw). Ref: 4667.
OH
OH
HO
O O
OH O
OH
OH
O
H
OH
OH
O
O
O HO
HO HO
H
HO
HO
HO
OH
8695 (25R)-26-[(-D-Glucopyranosyl)oxy]-2-hydroxy-22-methoxyfurost-5-
OH
HO
OO
HO
HO
HO
OH
O
O
OH
OO
H
H
OH
HO
HO
OH
OH
OH
en-3-yl-O--D-glucopyranosyl-(13)-O--D-glucopyranosyl-(12)-O-[-D-
8699 3-[(-D-Glucopyranosyl)oxy]-17-hydroxy-16-[(O--D-xylopy-
xylopyranosyl-(13)]-O--D-glucopyranosyl-(14)--D-galactopyranoside
ranosyl-(12)-2-O-acetyl--L-arabinopyranosyl)oxy]cholest-5-en-22-one
C63H104O34 (1405.51). Amorphous powder, []D27 = 60.0 (c = 0.10, MeOH). Pharm:
Cytotoxic (in vitro, HSC-2, LD50 = 6.1g/mL; control Doxorubicin, LD50 = 2.5g/mL).
Cytotoxic (HL-60 cells, IC50 = 0.0024mol/L, control Etoposide, IC50 =
Source: YE XIANG SHU Cestrum nocturnum (leaf: yield = 0.0264%fw). Ref: 4667.
0.025mol/L). Source: XIA FENG XIN ZI Galtonia candicans (bulb). Ref: 4116.
O
O
O
HO HO
HO
HO
HO
O HO
O
OH
HO
OO
OH
HO
HO
OH
O O HO
OH
OH
OO
OH
OH
HO
HO
HO
H
O
OH
HO
O
OO
OH
OH
OH
H
OH
OH
OH
O
OH
467
8700 18--D-Glucopyranosyloxy-8(17),13-ent-labdadien-16,15-olide
8703 (25S)-26-[(-D-Glucopyranosyl)oxy]-22-methoxyfurost-5-en-3-yl
C26H40 O8 (480.60). Yellow oil, []D25 = 37.8 (c = 0.87, CH3OH).
O--L-rhamnopyranosyl-(12)-O-[O--D-glucopyranosyl-(14)--L-rha
Source: GUANG YE YAN ZI CAI Potamogeton lucens (whole herb). Ref:
mnopyranosyl-(13)]-6-O-acetyl--D-glucopyranoside
3795.

O
HO
HO
HO
OH
HO
OH
OH
H
O
OH
O
HO
8701
7-O-(4--D-Glucopyranosyloxy-3-methoxybenzoyl) secolo-
ganolic acid
26
C30H40 O18 (688.64). Amorphous powder, []D = 96.4 (c = 0.149,
HO
HO
HO
OO
O
O
HO
OH
OH
OH
OO
O
OH OH
MeOH). Source: JIN YIN HUA Lonicera japonica (stem and leaf). Ref:
8704 (25S)-26-[(-D-Glucopyranosyl)oxy]-22-methoxyfurost-5-en-3-yl
4220.
O--L-rhamnopyranosyl-(12)-O-[O--D-glucopyranosyl-(14)--L-rha
mnopyranosyl-(13)]--D-glucopyranoside
OO
HO
OH
OH
OH
OH
HO
HO
O
OH
H
OO
HO
OH
OH
HO
O
H
OH
H
HO
8702 (25S)-26-[(-D-Glucopyranosyl)oxy]-22-methoxyfurosta-5,20(22)-
HO
dien-3-yl O--L-rhamnopyranosyl-(12)-O-[O--D-glucopyranosyl(14)--L-rhamnopyranosyl-(13)]-6-O-acetyl--D-glucopyranoside
25
C59H94O27 (1235.39). Amorphous solid, []D = 42.0 (c = 0.10,
HO
OO
HO
HO
OH
OH
O
O
HO
OH
O
O
OH OH
8705 (25R)-26-(-D-Glucopyranosyloxy)-22-methoxyfurost-5-en-3-yl-
O--L-rhamnopyranosyl-(12)-O-[-D-glucopyranosyl-(16)]--D-glucopyranoside
HO
HO
O
HO
OH
[244160-64-3] C52H86O23 (1079.25). Amorphous solid, []D29 = 69.0 (c =

0.29, MeOH). Source: QING LIANG BAI HE Lilium candidum. Ref: 2303.
H
O
O
H
O
H
O
HO
HO
HO
HO
OH
OH
HO
O
H
OO
HO
OO
OO
OH
OH
OH
O
OH
OO
OH
OH
OH OH
OO
OH
OH OH
HO
OO
OH
OH
OH
468
8706 2-(-D-glucopyranosyloxy)-8-(4''-methoxyphenylacetoxy)-guaia-
8710 26-O--D-Glucopyranosyl-(25S)-3,5,6,22,26-pentahydroxyl-
4(15),10(14),11(13)-trien-1,5,6,7H-12,6-olide
5-furostane 3-O--L-rhamnopyranosyl-(14)--D-glucopyranoside
C30H36O11 (572.61). Source: NAN XI BAN YA HUAN YANG SHEN Crepis
C45H76O20 (937.10). Amorphous powder, []D29 = 53.2 (c = 0.20, pyridine).
tingitana. Ref: 1859.
Source: JIU ZI Allium tuberosum. Ref: 4262.
H
HO
OH
H
OH
OO
OH
O O
HO
OH
OH
HO OH
8707 16-[[(4S)-5-(-D-Glucopyranosyloxy)-4-methyl-1-oxopentyl]oxy]-
3-[(O--L-rhamnopyranosyl-(12)-O-[O--D-glucopyranosyl-(14)-C57H92O28 (1225.35). Amorphous solid, []D25 = 22.0 (c = 0.10,
OO
HO
OH O O
OH
HO
HO
HO
O
OH
OH
OH
L-rhamnopyranosyl-(13)]--D-glucopyranosyl)oxy]pregn-5-en-20-one
OH
OH OH
O
H
H
HO
HO
HO
OO
HO
HO
OH
H
H
3-O--D-Glucopyranosyl-2,3,16,23,24-pentahydroxyolean-12-ene-28-oic
acid C36H58O12 (682.86). White amorphous powder. Source: JIE GENG
OO
Platycodon grandiflorum. Ref: 4900.
O
HO
OH OH
8711 3-O--D-Glucopyranosyl platycodigenin
O
O
OH OH
H
O
HO
8708 5-[3''-(-D-Glucopyranosyloxy)propyl]-7-methoxy-2-(3',4'-dimethoxyphenyl)benzofuran
C26H32O10 (504.54). White powder, []D25 = 22.23 (c = 0.8, CH3OH). Pharm:
Antibacterial (Staphylococcus aureus, MIC = 20g/mL; control
OH
OH
OO
HO
OH
HO
OH
Chloramphenicol, MIC = 5g/mL); antifungal (Candida albicans, MIC =
OH
OH
20g/mL, control Chloramphenicol, MIC = 5g/mL; Cladosporium

sphaerospermum, inactive at 20g). Source: XIU SE AN XI XIANG Styrax
ferrugineus (leaf). Ref: 5100.
C17H22O10 (386.36). Amorphous powder. Source: BAI HUA DAN Plumbago

zeylanica. Ref: 2047.
OO
HO
OH
OH
OH
8712 3'-O--Glucopyranosyl plumbagic acid
OH
HO
OO
OH
OH
8709 5-[3''--D-Glucopyranosyloxy)propyl]-7-methoxy-2-(3',4'-methylenedioxyphenyl)benzofuran
C25H28O10 (488.50). White powder. Pharm: Antibacterial (Staphylococcus
aureus, MIC = 15g/mL; control Chloramphenicol, MIC = 5g/mL);
antifungal (Candida albicans, MIC = 15g/mL, control Chloramphenicol,
MIC = 5g/mL; Cladosporium sphaerospermum, inactive at 20g). Source:
OH
OH
8713 3'-O--Glucopyranosyl plumbagic acid methyl ester

C18H24O10 (400.39). []D27 = 37 (c = 0.35, MeOH). Source: BAI HUA DAN
Plumbago zeylanica. Ref: 2047.
XIU SE AN XI XIANG Styrax ferrugineus (leaf). Ref: 5100.

OH
HO
OO
HO
OH
OH
O
OH
OH
OH
OO
O
H
OH
469
8714 3-O--D-glucopyranosyl-(12)--D-quinovopyranosyl quinovic

acid
C42H66O14 (794.99). Colorless crystalline solid, mp 220~222 C (H2O), []D22
= +43 (c = 0.6, MeOH). Source: WU BING XIN WU TAN Neonauclea

OH O O
OH
sessilifolia [Syn. Nauclea sessilifolia; Adina sessilifolia](root). Ref: 4405.
HO
OH
OH O O HO
HO
OO
OH
OO
OH
OH
OH
HO
OH
8717 3-O-(-Glucopyranosyl-(13)--rhamnopyranosyl-(12)--
OH
HO
O O OH
OH
OH
OH
HO
OH
arabinopyranosyl)-23-hydroxylup-12-en-28-O-(-rhamnopyranosylOO
(14)--glucopyranosyl-(16)--galactopyranosyl) ester
OH
C65H106O31 (1383.55). White amorphous powder, []D25 = +120 (c = 1, MeOH).
OH
Pharm: Antiproliferative (in vitro, J774 cell line, IC50 = 0.46mol/L, control
OH
6-Mercaptopurine, IC50 = 0.003mol/L; WEHI-164, IC50 = 1.9mol/L,

6-Mercaptopurine, IC50 = 0.017mol/L). Source: Schefflera fagueti. Ref: 5436.
8715 3-O-(-D-Glucopyranosyl-(13)--L-rhamnopyranosyl(12)--L-arabinopyranosyl)-hederagenin-28-O--D-glucopyranosyl ester
C53H86O22 (1075.26). White powder, []D25 = +47, (c = 1, MeOH). Pharm:
OH
Cytotoxic (antiproliferative in vitro: J774.A1 cell line, IC50 = 0.51mol/L,
OO
OH
HEK-293 cell line, IC50 = 1.8mol/L, WEHI-164 cell line, IC50 = 1.74mol/L;
control 6-Mercaptopurine, J774.A1 cell line, IC50 = 0.003mol/L, HEK-293
OH
OO
cell line, IC50 = 0.007mol/L, WEHI-164 cell line, IC50 = 0.015mol/L).
OO
OH
OO
OH
OH
O O OH
HO
Ref: 5036.
OH
OH
Source: YUAN YE E ZHANG CHAI Schefflera rotundifolia (aerial parts).
O O HO
HO
HO
OH
OH OH
OH
OH
O
8718 3-O-(-Glucopyranosyl-(13)--rhamnopyranosyl-(12)-arabinopyranosyl)-lup-12-en-28-O-(-rhamnopyranosyl-(14)--glu-
OH
OO
OH
OH
HO
OO
HO
OH
C65H106O30 (1367.55). White amorphous powder, []D25 = +139 (c = 1,

MeOH). Pharm: Antiproliferative (in vitro, J774 cell line, IC50 = 0.19mol/L,
OH
OO
copyranosyl-(16)--galactopyranosyl) ester
OH
control 6-Mercaptopurine, IC50 = 0.003mol/L; WEHI-164, IC50 =

0.56mol/L, 6-Mercaptopurine, IC50 = 0.017mol/L). Source: Schefflera
O O OH
HO
fagueti. Ref: 5436.
OH
OH
OH
O
8716 3-O-(-D-Glucopyranosyl-(13)--L-rhamnopyranosyl-
OH
(12)--L-arabinopyranosyl)-hederagenin-28-O-(-D-glucopyra-
OO
OH
nosyl-(14)--D-glucopyranosyl)ester
C59H96O27 (1237.41). White powder, []D25 = +29, (c = 1, MeOH). Pharm:
OH
Cytotoxic (antiproliferative, in vitro: J774.A1 cell line, IC50 = 1.63mol/L,

WEHI-164 cell line, IC50 = 0.64mol/L; control 6-Mercaptopurine, J774.A1
cell line, IC50 = 0.003mol/L, WEHI-164 cell line, IC50 = 0.015mol/L).
Source: YUAN YE E ZHANG CHAI Schefflera rotundifolia (aerial parts).
Ref: 5036.
OH
OH
OO
O O OH
HO
OH
OH OH
OH
OH
O O HO
HO
OO
OO
OH
OH
OH
470
8719 3-O--L-Glucopyranosyl-(13)--L-rhamnopyranosyl-(12)--L-
8722 (25R)-3-[(O--D-Glucopyranosyl-(12)-O-[O--L-rhamnopyra-
arabinopyranosyloleanclic acid
nosyl-(14)--D-glucopyranosyl-(13)]-O--D-glucopyranosyl-(14)-
C47H76O16 (897.12). Source: SAN YE MU TONG Akebia trifoliata (stem),
-D-galactopyranosyl)oxy]-5-spirostane
HUANG HUA BAI JIANG Patrinia scabiosaefolia. Ref: 660, 4545.
C57H94O27 (1211.37). Pharm: Cytotoxic (hmn oral squamous cell HSC-2,

LD50 = 1.9g/mL; normal hmn gingival fibroblast HGF cell, LD50 =
20g/mL). Source: Camassia leichtlinii (bulb). Ref: 3535.
O
OH
O
O
OH
OH
H
H
OO
HO
O
O
OH
OO OH
OH
OH
OO
OH
HO
OH
OO
HO
OH O O
HO
OH
OH
HO
O
OH OH
OH
OH
OH OH
OH
8720 3-[(O--D-Glucopyranosyl-(13)-O-[-L-rhamnopyranosyl-(12)]-L-arabinopyranosyl)oxy]olean-12-en-28-oic acid O--L-rhamnopyranos-
8723 3-O-[-D-Glucopyranosyl-(14)][-L-rhamnopyranosyl-(13)]-
yl-(14)-O--D-glucopyranosyl-(16)--D-glucopyranosyl ester
-D-glucopyranosyl-(13)--L-rhamnopyranosyl-(12)--arabinoyra-
nosyl-hederagenin
MeOH). Source: CHUAN XU DUAN Dipsacus asperoides. Ref: 265.
H
H
OH
HO
H
HO
O
OH
OH
OH
OO
OH
OH OH
OO
OH
OO
OO
OH
OH
OH
OO
OH
OH
OH
OH
OH
OH OH
HO
nosyl-(14)--D-glucopyranosyl-(13)]-O--D-glucopyranosyl-(14)-
HO
OH
-D-galactopyranosyl)oxy]-5-spirostan-12-one
OH

O
O
H
OH
OO
O O
OH O
OH
OH
Pharm: Cytotoxic (hmn oral squamous cell HSC-2, LD50 = 2.4g/mL; normal
OH
O O OH
O
8721 (25R)-3-[(O--D-Glucopyranosyl-(12)-O-[O--L-rhamnopyra-
OH OH
8724 3-O--D-Glucopyranosyl-(12)-[-L-rhamnopyranosyl-(14)]-D-glucuronopyranosyl-22-O-angeloyl-barrigenol R1
MeOH). Source: TIAN YE CI QIN Eryngium campestre (root). Ref: 4518.
H
H
OO
HO
OH
HO
O
OH
OH
OO
OH OH
HO
OH
OO
OO
HO
H
O
OH
OH OH OH
OH
OH
OH
OO
OH
OH
O
OH
OH
HO
OH
OO
HO
OO
OH
OH
O
OH
OH
471
8725 3-O--D-Glucopyranosyl-(12)-[-L-rhamnopyranosyl-(14)]-
8728 3-[(O--D-Glucopyranosyl-(14)-O--D-ribopyranosyl-(13)-
-D-glucuronopyranosyl-22-O-,-dimethylacryloyl-barrigenol A1
O--L-rhamnopyranosyl-(12)--L-arabinopyranosyl)oxy]olean-12-en-
28-oic acid O--D-glucopyranosyl ester
MeOH). Source: TIAN YE CI QIN Eryngium campestre (root). Ref: 4518.
C58H94 O25 (1191.38). Amorphous solid, []D25 = 38.0 (c = 0.10, MeOH).

Source: WEI LING XIAN Clematis chinensis (root: yield = 0.00028%).
Ref: 4763.
O
O
H
HO
O
OO
OH
H
O
OH
OH
OH
OH
OH
OO
HO
OO
HO
OO
OH
OH
HO
8726 3-O--D-Glucopyranosyl-(13)--L-rhamnopyranosyl-(12)-
OH
OH
-D-xylopyranosyl oleanolic acid
OH
O O OH
OO
HO
HO
O O
HO
OH OH OH
HO
HO
HO
OH
C47H76O16 (897.12). White powder (acetone), mp 234~238C (dec). Source:

HUANG HUA BAI JIANG Patrinia scabiosaefolia. Ref: 776.
8729 3-[(O--D-Glucopyranosyl-(14)-O--D-ribopyranosyl-(13)O--L-rhamnopyranosyl-(12)--L-arabinopyranosyl)oxy]olean-12-en28-oic acid O--L-rhamnopyranosyl-(14)-O--D-glucopyranosyl(16)--D-glucopyranosyl ester
OH
OH
OH
yield = 0.0125%). Ref: 4763.
OH
H
OO
C70H114O34 (1499.67). Source: WEI LING XIAN Clematis chinensis (root:
O
O
H
OH
HO
O O OH
OO
HO
OH
OH
O
O
HO
OH
8727 3-[(O--D-Glucopyranosyl-(14)-O--D-ribopyranosyl-(13)-
O O
HO
HO
HO
OO
HO
O
HO
HO
OH
OH
OH
OO
OH
HO
HO
O O
OH
OH
OH
OH
O--L-rhamnopyranosyl-(12)--L-arabinopyranosyl)oxy]-21-hydroxy
olean-12-en-28-oic acid O--L-rhamnopyranosyl-(14)-O--D-glucopyranosyl-(16)--D-glucopyranosyl ester
C70H114 O35 (1515.67). Amorphous solid, []D25 = 108.0 (c = 0.25,
MeOH). Source: WEI LING XIAN Clematis chinensis (root: yield =
8730 2"-O--D-glucopyranosyl saikosaponin b2

C48H78O18 (943.15). Source: WEN CHUAN CHAI HU Bupleurum
wenchuanense. Ref: 2247.
0.0024%). Ref: 4763.

OH
H
OH
O
OH
OH
H
O
HO
HO
HO
HO
O O
OH
HO
O
HO
HO
O O OH
OH
OH
HO
O
OH OH
HO
OO
O O
HO
HO
OO
OH HO
HO
OH
OH
OH
OH OH
OH
OH
OH
472
8731 2'-O--D-Glucopyranosylsalicin
8735 4'-O--D-Glucopyranosylswertiamarin
C19H28O12 (448.43). []D22 = 33 (c = 0.35, MeOH). Source: BA JIAO FENG
Alangium chinense (leaf). Ref: 4131.

O
OO
HO
OH
OH
O
OH
OO
HO
OH
HO
OH
OH
H
O
OH
OH
HO
OO
OH
OH
OH
8732 3-O--D-Glucopyranosyl--sitosterol
C35H60O6 (576.86). Crystals, mp 287~289C. Source: Zygophyllum
atriplicoides (whole herb). Ref: 4504.
OH
C22H32 O15 (536.49). Source: RI BEN ZHANG YA CAI Swertia japonica.
Ref: 2573.
O
OH
O
H
H
HO
OO
HO
OH
OH
OH
OH
OO
OH
OH OH
OH
OH
8737 3'-O--D-Glucopyranosylsyringopicroside
8733 3'-O--Glucopyranosyl-stilbericoside
Source: TAI GUO SHAN QIAN NIU Thunbergia laurifolia. Ref: 1968.
OH
H
OH
O
H
OO
HO
HO
OH
OH
amurensis] (leaf). Ref: 4175.
H
O
O
HO
O
OH
HO
OH OH
O
OH
OH
OH
OH
OH
OH

O
OH
OH
O
HO
H
HO
O O
HO
O
HO
OH
OH
OH
OH
OO
OH
OH
OH
OH
H
OO
OH
OH
473
8743 4-C--D-Glucopyranosyl-1,3,6-trihydroxy-7-methoxyxanthone
C20H20O11 (436.38). Yellow powder, mp 182~186C. Source: YUAN ZHI
Polygala tenuifolia. Ref: 2433.

O
O
OH
H
OH
HO
OO
OH
OH
HO
OH
HO
H
OO
OH
O
OH
OH
OH
OH
OH
OH
8744 3-O--D-Glucopyranosyl-5,9,4'-trihydroxy-8-methoxyflavone
8740 5-O--D-Glucopyranosyl-1,3,8-trihydroxyanthone
C22H22O11 (462.41). Source: MA HUANG Ephedra sinica. Ref: 2.
C19H18O11 (422.35). Yellow amorphous powder, mp 280~282C. Source:

CHUAN DONG ZHANG YA CAI Swertia davidii (whole herb). Ref: 4839.
OH
O
O
OH
OH
O
OH
OH
OH
OH
OO
HO
HO
OH
OH
OH
OH
8745 21-O--D-Glucopyranosyl-3,21,30-trihydroxyolean-13(18)-en24-oic acid
8741 4-O--D-Glucopyranosyl-2,6,4'-trihydroxybenzophenone
C36H58O10 (650.86). Amorphous white powder (MeOH), mp 270~272C,
C19H20O10 (408.37). Source: KUO YE GU SUI BU Davallia solida. Ref:
[]D25 = 11.7 (c = 0.41, MeOH). Source: SI CHI SI LENG CAO Schnabelia
5150.
tetradonta (aerial parts: yield = 0.00010%dw). Ref: 4665.

OH
OO
HO
OH
OH
OH
OH
HO
OH
OH
OO
HO
OH
OH
8742 26-O--D-Glucopyranosyl-(25R)-3,22,26-trihydroxyl-5-furostane 3-O--chacotrioside

C51H86O22 (1051.24). Amorphous powder, []D29 = 45.4 (c = 0.17, pyridine).
HO
Source: JIU ZI Allium tuberosum. Ref: 4262.
HO
O O
OH
OH
OH
8746 N,-D-Glucopyranosyl vincosamide

C32H40N2O13 (660.68). Yellow amorphous powder. Source: PING HUA GUO
OH
JIU JE Psychotria leiocarpa (shoot). Ref: 3769.
OH
H
H
OO
HO
OH
OH
OO
N
HO
O
OH
OH
OH
OO
OO
OH HO
OH
OH
OH OH
OH OH
OH
474
8747 3-[(O--D-Glucopyranosyl-(13)-O-[-D-xylopyranosyl-(12)]-
8750 3-O-[-D-Glucopyranosyl-(12)--D-xylopyranosyl]phytolaccinic
-L-arabinopyranosyl)oxy]olean-12-en-28-oic acid O--L-rhamnopyra-
Acid
nosyl-(14)-O--D-glucopyranosyl-(16)--D-glucopyranosyl ester
C42H66O15 (810.99). Amorphous powder, []D21.8 = +46.1 (c = 0.74, MeOH).
C64H104O30 (1353.52). Source: SAN YE MU TONG Akebia trifoliata (stem).
Source: MEI SHANG LU Phytolacca americana [Syn. Phytolacca decandra].
Ref: 4545.
Ref: 2443.
O
HO
OO
H
HO
OH
OH
OH
OH OH
OH
OH
OO
HO
OO
OO
OO
OO
OH
OH
OH
OH
OH
OH
OH
OHOH
OH
OH
OH
OO
OH
H
OH
OH
8748 (25R)-3-[(O--D-Glucopyranosyl-(12)-O-[-D-xylopyranosyl-
8751 2'-O--D-Glucopyranosyl-6'-O--D-xylopyranosylsalicin
(13)]-O--D-glucopyranosyl-(14)--D-galactopyranosyl)oxy]-26-[(-
C24H36O16 (580.54). []D19 = 31 (c = 0.27, MeOH). Source: BA JIAO FENG
D-glucopyranosyl)oxy]-2-hydroxycholesta-5,17-diene-16,22-dione
Alangium chinense (leaf). Ref: 4131.

OO
OH
= 0.0040%fw). Ref: 4667.
OO
OH
OH
OH
OH
HO
OO
OH
OH
O
HO
O HO
HO H O
OH
HOHO
OH
O O HO
HO
H
OH
OO
OH
OH
8752 Glucoraphanin
[21414-41-5] C12H22NO10S3 (436.50). Pharm: Antifungal; antimicrobial.
H
HO
HO
HO
OH
OH
Source: BAO ZI GAN LAN Brassica oleracea var. gemmifera, GAN LAN
OO
Brassica oleracea var. capitata, JU SAN HUA YE CAI Brassica oleracea var.
botrytis subvar. cymosa, LAI FU ZI Raphanus sativus. Ref: 658.
OH
O
O S O
N
8749 3-O-(-Glucopyranosyl-(13)--xylopyranosyl)-16-hydroxyolean-12-ene-28,30-dioic acid 28-O-(-galactopyranosyl) ester
S
HO
C47H74 O20 (959.10). White amorphous powder, []D25 = +11 (c = 1,

MeOH). Pharm: Antiproliferative (in vitro, J774 cell line, IC50 =
OS
OH
OH
3.6mol/L, control 6-Mercaptopurine, IC50 = 0.003mol/L; HEK-293,
OH
IC50 = 0.50mol/L, 6-Mercaptopurine, IC50 = 0.007mol/L; WEHI-164,

IC50 = 0.18mol/L, 6-Mercaptopurine, IC50 = 0.017mol/L). Source:
8753 Glucosamine
Schefflera fagueti. Ref: 5436.
[3416-24-8] C6H13NO5 (179.17). mp () 88C, () 110C (dec). Pharm:

Antiarthritic (approved by clinical trial). Source: BAI FAN DOU Phaseolus
O
vulgaris, GAN DI HUANG Rehmannia glutinosa [Syn. Rehmannia glutinosa

OH
f. Huechingensis], HAI SHEN CHANG Stichopus japonicus, LU RONG

Cervus nippon; Cervus elaphus, NIU NAO Bos taurus domesticus; Bubalus
bubalis, YE JU Chrysanthemum indicum, ZI ZHI Ganoderma japonicum [Syn.

Ganoderma sinense]. Ref: 2, 658, 660.
OH
OO
HO
O
OH
OH
OH
OH
HO
HO
OO
OH
HO
O
OH
OH
OH
OH
OH
NH2
475
8754 4'-O--D-Glucosyl-9-O-(6''-deoxysaccharosyl)olivil
8758 3'''-O-Glucosylsenburiside II
C38H54O22 (862.84). []D21 = 27 (c = 0.05, DMSO). Pharm: Adenosine A1
Senburiside IV C36H42O19 (778.72). Amorphous, []D26 = 83.4 (c = 0.69,
receptor partial agonist (rat and hmn adenosine A1 receptor, the first
MeOH); White amorphous powder (MeOHH2O), []D25 = 60.2 (c = 1.14,
non-nucleoside adenosine receptor agonist not structurally related to
MeOH). Source: LIU QIU SHE GEN CAO Ophiorrhiza liukiuensis (whole
adenosine). Source: XIE CAO Valeriana officinalis (root: yield = 0.021%dw).
herb), BAO JING ZHANG YA CAI Swertia franchetiana (whole herb). Ref:
Ref: 4656.
4527, 4469.
O
O
HO
HO
O O
HO
HO
OH
H
OH
HO
O
OH
OH
OH
OH
OH
OH
OO
HO
OH
schinseng], ZHU JIE SAN QI Panax pseudo-ginseng var. japonicus
OH
(underground part: yield = 0.010%dw). Ref: 2, 4610.
[33228-65-8] C15H20O10 (360.32). Amorphous powder, mp 204~207C, mp
OH
H
215~217C. Source: LIU CHUAN YU Linaria vulgaris, NAO YANG HUA
OH
Rhododendron molle, QUE MEI TENG Sageretia theezans [Syn. Sageretia

thea]. Ref: 515, 4237, 5396.
H
HO
OH
8759 Glucosyringic acid
OO
OH
OH
O
H
HO
OO
OH
OH
8755 20-Glucosylginsenoside Rf
HO
H
O
HO
O
O
OH
OH
HO
HO
O
O
OO
OH
OH
O
OH
8760 Glucotropaeolin
8756 p-Glucosyloxymandelonitrile
C14H17NO7 (311.29). Pharm: Toxin. Source: NAN TIAN ZHU ZI Nandina
domestica. Ref: 658.
HO
[499-26-3] C14H19NO9S2 (409.44). Acicular Crystals (ethanol),

tetramethylammonium, mp 188.0~189.2C, []D21 = 16.7 (water). Pharm:
Antibacterial; antifungal. Source: HAN LIAN HUA Tropaeolum majus, LA
GEN Armoracia lapathifolia, FAN MU GUA Carica papaya. Ref: 6, 661.
O
OO
O S OH
OH
OH
OH
OH
OH
OH
OH
OH
HO
C16H22O9 (358.35). mp 168~169C (Me2CO), []D22 = 80 (c = 1.610,

MeOH). Source: DUO TOU GE NI DI MU Gnidia polycephala (stem). Ref:
3502.
OS
OH
OH
8757 2-O--D-Glucosyloxy-4-methoxybenzenepropanoic acid
OH
8761 Glucuronic acid

Glycuronic acid C6H10O7 (194.14). Pharm: Antidote. Source: HUANG QI
Astragalus membranaceus, LU HUI Aloe vera [Syn. Aloe barbadensis], REN
SHEN Panax ginseng [Syn. Panax schinseng]. Ref: 2, 658.
OH
O
OO
HO
HO
O
O
OH
OH
OH
H
O
OH
OH
OH
OH
OH
OH
476
8762 7-O--D-Glucuronopyranosyl-4'-O-[2'-O-p-E-coumaroyl-O--D-
8765 3-O--D-Glucuronopyranosyl gypsogenin
glucuronopyranosyl(12)-O--D-glucuronopyranoside]apigenin
C36H54O10 (646.83). White lamellar Crystals, mp 238~240C. Source: SHAN
C 42 H 40 O 25 (944.77). Amorphous powder, mp 197~198C, [] D 20 =
KU GUA Momordica dioica. Ref: 645.
52.45 (c = 0.1, MeOH). Source: MU XU Medicago sativa (aerial

parts). Ref: 5167.
HO
HO
HO
OO
OH
OH
OH
O
HO
OH
O
O
OH
8766 3-[(O--D-Glucuronopyranosyl-(13)-O-[-L-rhamnopyranosyl-
OH
HO
OH
OH
OO
O
OH
OH
OH
(12)]--L-arabinopyranosyl)oxy]olean-12-en-28-oic acid
OH
8763 7-O--D-Glucuronopyranosyl-4'-O-[2'-O-E-feruloyl-O--D-glucuronopyranosyl(12)-O--D-glucuronopyranoside]apigenin
OH
Ref: 5167.
OO
OH
OH
O
O
HO
OO
OH
O O OH
OH
OH
OH
O
HO
OH
O
O
OH
OH
OH
HO
OH
O
OO
HO
OH
OH
10.23 (c = 0.1, MeOH). Source: MU XU Medicago sativa (aerial parts).
HO
C43H42 O26 (974.80). Amorphous yellow powder, mp 197~198C, []D20 =
OH
8767 3-O--D-Glucuronopyranosyl-2,3,16-trihydroxy-28-norolean12-en-15-on-23-oic acid
C35H52O12 (664.8). White needles (MeOH), mp >350C, []D25 = +54.5 (c =
0.44, MeOH). Source: SI CHI SI LENG CAO Schnabelia tetradonta (aerial

parts: yield = 0.00026%dw). Ref: 4665.
8764 3-O-[-D-Glucuronopyranosyl-(12)-O--D-glucuronopyranosyl]-24-hydroxyglabrolide
C43H62O17 (850.96). White powder, []D25 = +3.5 (c = 0.002, CHCl3:CH3OH =

1:5). Source: GAN CAO Glycyrrhiza uralensis. Ref: 2085, 2445.
O
OH
O
H
OH
O
O
OH
OH
O
OH
O
O
OH
8768 Gluroside
C15H24O8 (332.35). Source: ROU CONG RONG Cistanche deserticola. Ref:
2448.
H
OH
HO
HO
OH OH
OH
OH
OO
HOHO
O
HO
OH
OH
OH
477
8769 L-Glutamic acid--methylamide
8775 -L-Glutamyl-glycine
C6H10N2O5 (190.16). Source: CHA ZI XIN Camellia oleifera, YOU CHA
C7H12N2O5 (204.18). Source: NIU NAO Bos taurus domesticus; Bubalus
GEN PI Camellia oleifera. Ref: 6.
bubalis. Ref: 6.
O
NH2
NH2
HO
OH
N
H
HO
NH2
OH
8770 -Glutamyl-alanine
8776 L--Glutamyl-L-hypoglycin
[5875-41-2] C8H14N2O5 (218.21). mp 194~195C (dec) , []D = 28 (c = 2,
C12H18N2O5 (270.29). Pharm: Supertoxic agent. Source: XI FEI LI ZHI GUO
H2O). Source: NIU NAO Bos taurus domesticus; Bubalus bubalis. Ref: 6,
Blighia sapida. Ref: 658.
1521.
O
H2N
OH
H O O
OH
NH2
H
N
O
OH
OH
8777 -L-Glutamyl-petiveriin A
8771 -L-Glutamyl-L--aminoisobutyric acid
(SC2RC7RS)--Glutamyl-S-benzylcysteine sulfoxide C15H20N2O6S (356.40).
White hygroscopic solid, mp 126~129C, []D22 = +3.2 (c = 0.06, H2O).
bubalis. Ref: 6.
Source: SUAN CHOU MU JI CAO Petiveria alliacea (root). Ref: 5322.

NH2
H
N
HO
O
OH
O
OH
O
OH
N
H
NH2
8772 (SC2RC7)--Glutamyl-S-benzylcysteine
C15H20N2O5S (340.40). White hygroscopic solid, mp 152~155C, []D22 =
14.7 (c = 0.03, H2O). Source: SUAN CHOU MU JI CAO Petiveria alliacea
8778 -L-Glutamyl-petiveriin B
(root). Ref: 5322.
(SC2RC7SS)--Glutamyl-S-benzylcysteine sulfoxide C15H20N2O6S (356.40).
HO
S
White hygroscopic solid, mp 138~140C, []D22 = 26.2 (c = 0.06, H2O).

O
Source: SUAN CHOU MU JI CAO Petiveria alliacea (root). Ref: 5322.
OH
N
H
NH2
OH
O
OH
N
H
NH2
8773 -L-Glutamyl-L-glutamic acid

[1116-22-9] C10H16N2O7 (276.25). mp 191~192C, []D16 = +6.6 (c = 1,
1mol/L HCl). Source: NIU NAO Bos taurus domesticus; Bubalus bubalis. Ref:
6, 1521.
O
H2N
8779 -L-Glutamyl-L-phenylalanine
C14H18N2O5 (294.31). mp 164~174C (dec). Source: DI YANG QUE Lotus
corniculatus. Ref: 6, 1521.
OH
OH
H O O
N
OH
H2N
H O
H O
OH
N
H
OH
8774 -L-Glutamyl-glutamine
C10H17N3O6 (275.26). mp 191~192C, []D16 = +11 (c = 1, 1mol/L HCl).
Source: NIU NAO Bos taurus domesticus; Bubalus bubalis. Ref: 6, 1521.
8780 -L-Glutamyl-S-(prop-1-enyl)cystein sulfoxide
O
H2N
C11H18N2O6S (306.34). Source: TAN XIANG Santalum album. Ref: 6.
OH
H O O
N
H
OH
HO
H O
NH2
S
O
NH2
H
N
OH
O
478
8781 -Glutamyl-serine
8786 -Glutenol
Glut-5-en-3-ol C30H50O (426.73). mp 203~205C. Source: BA WANG BIAN
bubalis. Ref: 6.
Euphorbia royleana, XI YE DA JI Euphorbia esula var. cyparissoides. Ref: 6,

1521.
OH
HO
OH
N
H
NH2
O
H
8782 -L-Glutamyl-L-tyrosine
[6720-09-8] C14H18N2O6 (310.31). mp 221~222C (dec) , []D31 = +26.6 (c =
HO
4). Source: DI YANG QUE Lotus corniculatus. Ref: 6, 1521.

O
8787 Glutinic acid
OH
C20H30O4 (334.46). White acicular Crystals, mp 119~120C, easy soluble in
OH
H O O
H2N
N
H
acetone and pyridine. Source: NIAN YE YOU(2) Caryopteris glutinosa. Ref:
248.
OH
8783 -Glutamyl-valine
OH
[2746-34-1] C10H18N2O5 (246.27). mp 207C, []D = 0 (c = 2.4, H2O). Source:

NIU NAO Bos taurus domesticus; Bubalus bubalis. Ref: 6, 1521.
O
OH
OH
H2N
8788 -Glutinol
OH
H O O
N
H
Glutin-5-en-3-ol C30H50O (426.73). White amorphous material, mp 211C,
mp 212C, []D25 = 63.3 (c = 0.71, CHCl3). Pharm: Anti-inflammatory

(modified assay of Tan and Berridge, 400g/mL, InRt = 11.44%, control
Aspirin, InRt = 70.45%)[5316]; cell viability (hmn isolated neutrophils,
12.5g/mL, cell viability = 100%, 100g/mL, cell viability = 100%,
8784 Glutaric acid

Pentanedioic acid [110-94-1] C5H8O4 (132.12). mp 97~98C, bp 302~304C.
200g/mL, cell viability = 72.29%)[5316]. Source: BA WANG BIAN
Pharm: Toxin. Source: TIAN CAI Beta vulgaris, NING MENG AN YE
Euphorbia royleana, CHI YANG Alnus japonica, MENG GU LI Quercus
Eucalyptus citriodora. Ref: 6, 658.
mongolica, SONG LUO Usnea longissima, TAI WAN XIU XIAN JU Spiraea
formosana. Ref: 6, 611, 2575, 5316.
HO
OH
O
8785 Glutathione
-L-Glutamyl-L-cysteinylglycine; Glutamid; Glutinal; Triptide; Tathion

[70-18-8] C10H17N3O6S (307.33). mp 195C (50% ethanol), []D25 = 18.9 (c
HO
= 4.653, water), []D27 = 21 (c = 2.74), easily soluble in water, diluted

ethanol, liquid ammonia, dimethylformamide.[5507] Pharm: Has an important
role in normal metabolic processes; antidote (from poisoning by sulfydryl
enzyme). Source: MU LI ROU Ostrea rivularis; Ostrea talienwhanensis;
Ostrea gigas, XIAO BAI BU Asparagus officinalis. Ref: 6, 658, 1521, 5507.
O
H2N
OH
H O O
N
H
H
N
8789 Glutinone
[508-09-8] C30H48O (424.72). mp 245~246C. Source: LONG XU CAO Poa
sphondylodes. Ref: 6.
O
OH
H
SH
479
8790 Glutinoside
8796 Glyasperin A
[103744-80-5] C14H21ClO11 (400.70). Source: GAN DI HUANG Rehmannia
C25H26O6 (422.48). Source: CU MAO GAN CAO Glycyrrhiza aspera. Ref:
glutinosa [Syn. Rehmannia glutinosa f. Huechingensis]. Ref: 2.
2431.
OH
OH
H
Cl
HO
HO
HO
OH
OO
OH
OH
OH
8797 Glyasperin B
OH
8791 Glutinosin
2431.
O
JIAO NIAN XIANG CHA CAI Isodon glutinosa. Ref: 4067.
OH
OH
OH
OH
OH
8798 Glyasperin C
2431.
8792 Glutinosin A
HO
C20H34O2 (306.49). mp 190C. Source: JIAO NIAN XIANG CHA CAI Isodon
OH
glutinosa. Ref: 4067.

OH
OH
OH
8799 Glyasperin D
2431.
8793 Glutinosin B
C20H34O2 (306.49). []D = +59.6. Source: JIAO NIAN XIANG CHA CAI
OH
Isodon glutinosa. Ref: 4067.

O
OH
OH
OH
8800 Glyasperin E
2431.
OH
8794 Glutinosone
[55051-94-0] C14H20O2 (220.31). Pharm: Antifungal. Source: JIAO YAN
OH
CAO Nicotiana glutinosa. Ref: 658.
O
HO
OH
8795 Glyarallin B
8801 Glyasperin F

2431.
HO
OH
HO
OH
OH
OH
OH
480
8802 Glyasperin K
8808 Glycerol
[56-81-5] C3H8O3 (92.10). mp 17.8C, bp 290C (dec). Pharm: Vasodilator.
2431.
Source: BAI YAO ZI Stephania cepharantha, JIU Liquor, SHI LI ZI Aleurites

moluccana, SHI LIU GEN Punica granatum, SHI LUO ZI Anethum
OH
graveolens (fruit). Ref: 6, 4177.

H
8803 Glyasperin M
8809 Glycerol-,-dilinolenate-'-rhamno-rhamnoside
2431.
C51H84O13 (905.23). White powder. Source: SU MI Setaria italica. Ref: 2120.

O
HO
OH
OH
OO
OO
O
O O
OH OH OH OH
8804 Glybomine B
C19H21NO2 (295.38). Pharm: Anti-HIV (CC50 = 13.62g/mL, IC50 =

9.73g/mL, SI = 1.40; control AZT, CC50 = 794.2g/mL, IC50 = 0.131g/mL,
8810 Glycerol 2-O--L-fucopyranoside
SI = 6100). Source: MENG DA NA SHAN XIAO JU Glycosmis montana
(twig and leaf). Ref: 5266.
4177.
HO
O
OH
O
OH
O
N
H
OH
OH
OH
8811 Glycerol sinapate

C36H38O15 (710.70). Source: LAI FU ZI Raphanus sativus. Ref: 6.
8805 Glyceollin IV
[69393-94-8] C21H22O5 (354.41). Not crystalline. Pharm: Antifungal. Source:
OH
HEI DA DOU Glycine max. Ref: 661.
OH
O O
OH
OO
O
OH
H
OH
8806 D-Glyceric acid

[600-19-1] C3H6O4 (106.08). Pharm: Diuretic (rbt). Source: CAN DOU Vicia
8812 Glyceryl-1-eicosanoate
faba, CAN DOU JIA KE Vicia faba, CAN DOU JING Vicia faba, CAN DOU
C23H46O4 (386.62). White amorphous powder. Source: DUO CI HUANG
(2)
YE Vicia faba, PU
TAO Vitis vinifera, PU TAO TENG YE Vitis vinifera, YI
HUA REN Sida spinosa. Ref: 2043.
ZHU QIAN MA Urtica dioica. Ref: 6, 658, 660.
O
HO
OH
HO
OH
OH
8807 Glyceride-1,3-dipalmito-2-sorbate
8813 (2R)-1-O-Glyceryl--D-galactoside
C41H74O6 (663.04). Colorless acicular crystals, mp 62.0~62.5C (petroleum
C9H18O8 (254.24). Amorphous white powder, []D = 7.5 (c = 0.90, H2O).
spiritacetic ester). Source: DI SHAO GUA Cynanchum thesioides. Ref: 236.
Source: FEI YUE GUO Feijoa sellowiana (leaf). Ref: 3878.
O
O
OH
HO
HO
OO
OH
O
O
OH
OH
481
8814 Glyceryl linolenate I
8818 Glycitein
1-O-(9Z,12Z-Octadecadienoyl) glycerol C21H38O4 (354.53). []D20 = +0.1 (c
[40957-83-3] C16H12O5 (284.27). mp 311~313C (90% ethanol). Pharm:
= 0.5, CHCl3), mp () 15.7C, (') 13.5C. Pharm: COX-1 inhibitor (IC50 =
Antihemolytic; lipoxygenase inhibitor; anti-inflammatory (NO production
13.3g/mL, control trans-Resveratrol, IC50 = 0.25g/mL)[5030]; COX-2
inhibitor)[4415]. Source: DA DOU Glycine max (Soybean phytochemical

concentrate: yield = 0.0025%dw)[4630], HEI DA DOU Glycine max. Ref: 661,
inhibitor (IC50 = 0.18g/mL, control trans-Resveratrol, IC50 =

0.30g/mL)
[5030];
[4607]
cytotoxic inactive (in vitro, LNCaP, IC50 > 100mol/L)
4415, 4630.
Source: LANG DANG ZI Hyoscyamus niger (seed: yield = 0.004%dw),

LIAN YE TONG Hernandia Sonora [Syn. Hernandia ovigera] (seed), YU
HO
ZHI ZI Akebia quinata. Ref: 6, 4607, 5030.

O
O
OH
O
OH
8819 Glycitin
Glycitein-7-O--D-glucoside [40246-10-4] C22H22O10 (446.41). Source: DA
OH
8815 Glyceryl linolenate II
DOU Glycine max (Soybean phytochemical concentrate: yield = 0.0020%dw).
Dilinolenin C39H68O5 (616.97). mp 12.3C. Source: YU ZHI ZI Akebia
Ref: 4630.
quinata. Ref: 6.
HO
HO
HO
OH O
O
OH
8820 Glycobismine F
OH
C38H32N2O9 (660.69). Yellow oil, []D = 0 (c = 0.174, CHCl3). Source:
SHAN XIAO JU Glycosmis citrifolia (root). Ref: 4270.
OH
8816 Glyceryl linolenate III

Trilinoleyl glyceride [537-40-6] C57H98O6 (879.41). Source: BAI SU ZI
O
Perilla frutescens, YU ZHI ZI Akebia quinata, ZANG SAN QI Panax
N
O
pseudo-ginseng. Ref: 6, 743.
OH
HO
O
O O
OH
8821 Glycobismine G
C38H32N2O9 (660.69). Yellow oil, []D = 0 (c = 0.13, CHCl3). Source: SHAN

XIAO JU Glycosmis citrifolia (root). Ref: 4270.
8817 Glycine
Aminoethanoic acid [56-40-6] C2H5NO2 (75.07). mp 262C (dec). Pharm:
Metabolic intermediate. Source: BAN XIA Pinellia ternata (dried tuber:
OH
content scope of 4 origins = 0.72%~1.05%, mean content = 0.91%)[5521],

CHUAN DANG SHEN Codonopsis tangshen, DANG SHEN Codonopsis
HO
pilosula, GOU QI ZI Lycium chinense, LONG KUI Solanum nigrum, MU
XIANG Saussurea lappa [Syn. Aucklandia lappa], QIU HUA DANG SHEN
Codonopsis subglobosa, SU HUA DANG SHEN Codonopsis pilosula var.
OH
O
modesta [Syn. Codonopsis modesta]. Ref: 6, 658, 660, 5521.

OH
O
H2N
OH
482
8822 Glycoborinine
8827 Glycolic acid
C18H17NO2 (279.34). Pharm: Anti-HIV (CC50 = 20.69g/mL, IC50 =
Hydroxyacetic acid [79-14-1] C2H4O3 (76.05). mp 80C. Pharm: Irritant (to
4.47g/mL, SI = 4.63; control AZT, CC50 = 794.2g/mL, IC50 = 0.131g/mL,
skin and mucosa). Source: GAN ZHE Saccharum sinensis, HAN QIN Apium
SI = 6100). Source: MENG DA NA SHAN XIAO JU Glycosmis montana
graveolens, MENG GU SHAN LUO BO Scabiosa comosa. Ref: 6, 658.
(twig and leaf). Ref: 5266.

OH
OH
O
O
N
H
OH
8828 Glycoside E
8823 Glycocholic acid
C27H44O6 (464.65). mp 239~240C. Source: XIANG JIA PI Periploca sepium.
[475-31-0] C26H43NO6 (465.64). mp 165~168C (anhydrous), mp 230~240C
Ref: 6.
(sodium salt). Source: NIU DAN Bos taurus domesticus; Bubalus bubalis,
NIU HUANG Bos taurus domesticus; Bubalus bubalis (gallstone: mean
HO
OH
O
O
OH
H
OH
content = 0.26%). Ref: 6, 5508.

H
N
H
OH
O
HO
H
H
HO
H
OH
8829 Glycoside H1
3-O-[4-O-Acetyl-3-O-methyl--D-fucopyranosyl-(14)-2,6-dideoxy-3-O-me
thyl--D-ribo-hexopyranoside] 20-O-[-D-glucopyranosyl-(16)--D-gluco-
8824 Glycocitridine
pyranosyl-(12)-3-O-methyl--D-fucopyranoside] [37074-77-4] C56H92O24
(1149.34). mp 182C. Source: XIANG JIA PI Periploca sepium. Ref: 6.

Mithramycin, ED50 = 0.07g/mL; A549, ED50= 0.52g/mL, Mithramycin,
N
H
H
HO
O
O
O
Severinia buxifolia] (root cortex). Ref: 3075.
OO
O
HO
O
OO
OO
OH
OH
OH
OH
8825 Glycocitrine I
C20H21NO4 (339.39). Source: DONG FENG JU GEN Atalantia buxifolia [Syn.
OO
OH
OH
OH
8830 Glycoside H2
C54H88O25 (1137.29). mp 191~192C, []D = 25.9. Source: XIANG JIA PI
Periploca sepium. Ref: 2498.
OH
HO
OO
GUA Citrullus vulgaris [Syn. Citrullus lanatus]. Ref: 6.

OH
HO
OO
HO
Ethanediol [107-21-1] C2H6O2 (62.07). mp 11.5C, bp 197C. Source: XI
OH
O
OH
HO
OH O
O
HO
OO
8826 Glycol
OH
OH
OO
OH
OH
OH
OH
483
8831 Glycoside K (Periplocae)
8836 Glycyrdione B
C40H66O16 (802.96). mp 240~241C. Source: XIANG JIA PI Periploca sepium.
C25H26O5 (406.48). Source: ZHANG GUO GAN CAO Glycyrrhiza inflata.
Ref: 6.
Ref: 2431.
H
O
H
HO
O
O
HO
HO
OO
OO
OH
OH
OH
OH
OH
HO
8837 Glycyrdione D
OH
OH
8832 Glycozolidal
2,6-Dimethoxy-9H-Carbazole-3-carboxaldehyde; 2,6-Dimethoxy-3-formyl-
carbazole; O-Methyllansine. [51971-09-6] C15H13NO3 (255.28). Source:

SHAN HUANG PI Clausena excavata. Ref: 703.
OH
8838 Glycyrin
Ref: 2.
N
H
OH
HO
8833 Glycycoumarin
[94805-82-0] C21H20O6 (368.39). Pharm: Antibacterial (mutational
Streptococcus, MIC = 12.5g/mL; Staphylococcus aureus, MIC = 3.13g/mL;
Bacillus subtilis, MIC = 6.25g/mL;); antifungal (Candida sp., MIC =

50g/mL; Saccharomyces cerevisiae, MIC = 25g/mL); cAMP
phosphodiesterase inhibitor (IC50 = 7mol/L); free radical scavenger (IC50 =
41mol/L); anti-HIV. Source: GAN CAO Glycyrrhiza uralensis. Ref: 2, 1678,
1680, 1701, 1702.
Neoglycyrol [23013-84-5] C21H18O6 (366.37). Yellowish acicular crystals, mp

263~265C; mp 243.5~245.0C. Source: CU MAO GAN CAO Glycyrrhiza
aspera, GAN CAO Glycyrrhiza uralensis. Ref: 2, 6, 181, 660, 1521.
OH
HO
8839 Glycyrol
OH
O
8834 Glycyphyllin
HO
[19253-17-9] C21H24O9 (420.42). Pharm: Bitter-sweet taste. Source: Smilax sp.
8840 Glycyroside
Ref: 658.
OH
HO
OH
[125310-04-5] C27H30O13 (562.53). Yellowish powder, mp 126~128C. Source:

HUANG GAN CAO Glycyrrhiza kansuensis. Ref: 133.
OH
HO
OO
OH
OH
OO
HO
OH
O
O
OH OH
OH OH
8835 Glycyrdione A
C25H28O5 (408.50). Source: ZHANG GUO GAN CAO Glycyrrhiza inflata.
Ref: 2431.
8841 Glycyrrhetinic acid

[471-53-4] C30H46O4 (470.70). mp 297~298C. Pharm: Adrenal cortex
hormoneoid (desoxycortoneoid action); antiallergic; antibacterial (cooperates
with berberine to inhibit Staphylococcus aureus, in vitro); antineoplastic (rat,
transplanting Oberling-Guerin myeloma); anti-inflammatory (rat, tampon
OH
HO
granuloma model, formaldehyde edema model, tuberculin reaction model,

subcutaneous granuloma model, and swollen foot model caused by
OH
carrageenan); antiulcerative (pylorus-ligated rat); reduces serum bilirubin and
484
enhances output of bilirubin in urine (choledoch-ligated rat and rbt); toxin
8845 Glycyrrhiza-flavonol A
(gpg, inhibits thyroid function and reduces basal metabolism). Source: CU
[197304-01-1] C20H18O7 (370.36). Yellow acicular crystals (methanol), mp
MAO GAN CAO Glycyrrhiza aspera (root and rhizome: content = 0.72%)[15],
163C, []D = 0 (c = 1, methanol). Pharm: DPPH scavenger (EC50 =
GAN CAO Glycyrrhiza uralensis (root and rhizome: mean content of 3
37mol/L). Source: GAN CAO Glycyrrhiza uralensis. Ref: 1001.
origins = 4.93%)
[15]
, GUANG GUO GAN CAO Glycyrrhiza glabra (root and

[15]
rhizome: content = 3.40%)
, HUANG GAN CAO Glycyrrhiza kansuensis
HO
OH
(root and rhizome: content = 4.16%)[15], YUN NAN GAN CAO Glycyrrhiza
yunnanensis (root and rhizome: content = 2.52%)
[15]
, ZHANG GUO GAN
OH
OH
CAO Glycyrrhiza inflata (root and rhizome: content = 3.72%)[15]. Ref: 4, 15,
658, 5501.
8846 Glycyrrhizic acid

Glycyrrhizin; Glycyrrhetinic acid glycyside; Glycyrrhizinic acid [1405-86-3]
O
OH
O
C42H62O16 (822.95). White acicular crystals, mp 220C (dec), []D17 = +46.2

(ethanol), easily soluble in water, ethanol, insoluble in ether.[5507] Pharm:
Adrenal cortex hormoneoid; antiallergic; antineoplastic; anti-HIV
(0.5mg/mLInRt = 98%, 0.125mg/mL InRt = 50%); anti-inflammatory;
H
HO
antiviral (chickenpox virus, herpes zoster virus); antihepatotoxin (rat with

CCl4 poisoning, reduces excess SGPT); reduces accumulation of trilaurin in
liver; reduces serum bilirubin and increases output of bilirubin in urine (rbt
and rat, ligated in common bile duct); antihypercholesterolemic (reduces the
8842 Glycyrrhetol
C30H48O3 (456.72). Source: GAN CAO Glycyrrhiza uralensis. Ref: 2.
level of cholesterol in serum); antihypertensive; smooth muscle relaxant (in

vitro ileum in rbt and trachea in gpg, caused by histamine, acetylcholine and
SRSA). Source: CU MAO GAN CAO Glycyrrhiza aspera, GAN CAO
Glycyrrhiza uralensis (root and rhizome: content scope of 14 origins =
OH
Glycyrrhiza glabra (root and rhizome: mean content = 4.22%[5508]), HUANG
O
H
GAN CAO Glycyrrhiza kansuensis, XIANG SI ZI Abrus precatorius,

ZHANG GUO GAN CAO Glycyrrhiza inflata (root and rhizome: mean
H
HO
2.60%~8.44%, mean content = 5.92%[15, 5508]), GUANG GUO GAN CAO
content = 4.59%)[15, 5508]. Ref: 4, 15, 658, 660, 5501, 5507, 5508.
OH
OH
O
O
OH
OH
OH
Ref: 2.
O
HO
HO
OH
8843 Glycyrrhisoflavanone
OH
8847 Glyeurysaponin
OH
3-Hydroxy-11-oxo-olean-12-en-30-oic acid-3-O--D-glucoronopyranosyl(14)--D-glucuronopyranoside [137476-70-1] C42H62O16 (822.95). White
8844 Glycyrrhisoflavone
[116709-70-7] C20H18O6 (354.36). Pharm: Anti-HIV (20g/mL, inhibits
formation of giant-cell); free radical scavenger (EC50 = 38mol/L);
powder, mp 288C, []D18 = +22.5 (c = 0.062, methanol). Source: HUANG

GAN CAO Glycyrrhiza kansuensis. Ref: 195.
O
xanthinoxidase inhibitor (IC50 = 53mol/L); monoamine oxidase inhibitor
OH
(IC50 = 95mol/L). Source: GAN CAO Glycyrrhiza uralensis. Ref: 2, 1679,

O
1680, 1681, 1682.

HO
OH
OH
OO
OH
HO
O
OO
HO
OH
OH
OH
OH
H
H
OH
485
8848 Glyfoline
8853 Glypentoside C
C18H19NO7 (361.35). Pharm: Antineoplastic (caused tumor cell death
selectively, without showing any cytotoxicity to normal fibroblasts). Source:
Source: JIU BING YE Glycosmis pentaphylla (stem). Ref: 4424.
SHAN XIAO JU Glycosmis citrifolia. Ref: 5042.

O
OH
O
HO
OH
HO
HO
OH
O
8849 Glyoxal
OH
O O O
[107-22-2] C2H2O2 (58.04). Source: SHENG JIANG Zingiber officinale. Ref: 2.

O
OO
OH
OH OH
O
8850 Glypallichalcone
8854 Glyurallin A
4-Hydroxy-2,4'-dimethoxychalcone C17H16O4 (284.31). Yellow columnar
Crystals, mp 140~142C. Source: CI GUO GAN CAO Glycyrrhiza

pallidiflora. Ref: 243.
HO
OH
OH
8855 Glyuranolide
8851 Glypentoside A
3,22-Digydroxy-11-oxo-12-olean-ene-27-methoxy carbonyl-29-oic acid
Methoxyquinol 4-O-[(5-O-trans-p-coumaroyl)--D-apiofuranosyl-(12)--
(29,22) lactone [123914-44-3] C31H44O6 (512.69). White rhomboid crystals,
D-glucopyranoside C27H32O14 (580.55). Amorphous powder, []D25 = 7.5 (c
mp 301~303C, []D14 = +46 (c = 0.087). Source: GAN CAO Glycyrrhiza
= 0.33, MeOH). Source: JIU BING YE Glycosmis pentaphylla (stem). Ref:
4424.
O
O
OH
HO
OO
OH
HO
OH
O O O
H
HO
OH OH
8852 Glypentoside B
8856 Glyyunnanprosapogenin D
4-Demethylantiarol 4-O-[(3-methoxy-4-hydroxy-benzoyl)--D-apiofura-
Oleana-11,13(18)-dien-29-oic acid 3,21-di-O--D-glucuronopyranoside
nosyl-(12)--D-glucopyranoside C27H34O16 (614.56). Amorphous powder,
[139979-69-4] C42H62O16 (822.95). Source: YUN NAN GAN CAO
25
[]D = 60.7 (c = 0.48, MeOH). Source: JIU BING YE Glycosmis
Glycyrrhiza yunnanensis. Ref: 170.
pentaphylla (stem). Ref: 4424.

O
HO
O
OH
OO
OH
HO
HO
OH
O O O
O
HO
OO
OH
OH
OH OH
OH
H
H
HO
O
OH
OH
OH
486
8857 Glyyunnansapogenin A
8861 Glyyunnansapogenin F
3,24-Dihydroxy-16-oxo-olean-12-en-29-oic acid [131137-98-9] C30H46O5
3,24-Dihydroxy-16-oxo-oleana-11,13(18)-dien-30-oic acid [139953-40-5]
(486.70). Colorless crystals. Source: YUN NAN GAN CAO Glycyrrhiza
C30H44O5 (484.68). Source: YUN NAN GAN CAO Glycyrrhiza yunnanensis.
Ref: 170, 1521.

O
O
OH
OH
H
H
HO
HO
H
OH
H
OH
8862 Glyzaglabrin
8858 Glyyunnansapogenin B
Ref: 2, 1521.
3,21,24-Trihydroxy-olean-12-en-30-oic acid [20528-70-5] C30H48O5

(488.71). Colorless crystals, mp 287~289C. Source: YUN NAN GAN CAO
HO
OH
Glycyrrhiza yunnanensis. Ref: 160.
O
O
O
OH
HO
8863 Gmelofuran
[70863-78-4] C15H18O3 (246.31). Crystals, mp 122~123C, []D25 = 900
(CHCl3). Source: CHEN XIANG Aquilaria agallocha, GAO HONG JIN
Hibiscus elatus, TAI WAN FU RONG Hibiscus taiwanensis, YUN NAN SHI
H
HO
ZI Gmelina arborea. Ref: 13, 1521, 2529.
H
OH
O
O
8859 Glyyunnansapogenin B1
C30H48O5 (488.71). White acicular crystals, mp 303~305C. Source: YUN
NAN GAN CAO Glycyrrhiza yunnanensis. Ref: 321.

8864 Gmephiloside
1-O-(8-Epi-loganoyl)--D-glucopyranose C22H34O15 (538.51). White
O
OH
OH
amorphous powder. Source: FEI LV BIN SHI ZI Gmelina philippensis (aerial

parts). Ref: 3954.
HO
HO
OH
OH
O
OH
O
H
OH
OH O
HO
OH
8860 Glyyunnansapogenin B2
OH
C30H50O2 (442.73). White powder, mp 224~228C. Source: YUN NAN GAN
OO
OH
CAO Glycyrrhiza yunnanensis. Ref: 321.

8865 Gnaphaliin
OH
C17H14O6 (314.30). Pharm: Anti-inflammatory[4415]. Source: YI DA LI LA JU

Helichrysum italicum Ref: 4415.
O
OH
O
HO
OH
O
487
8866 Gnemonol A
8870 Gnemonol E
C42H32O10 (696.72). White amorphous powder. Source: XIAN ZHOU MAI
MA TENG Gnetum gnemon (root). Ref: 4200.
Pharm: Antioxidant (super oxide scavenger, IC50 = 72mol/L, control
HO
-Viniferin, IC50 = 20mol/L; lipid peroxide inhibitory activity, IC50 =
OH
H
47mol/L, control -Viniferin, IC50 = 33mol/L). Source: XIAN ZHOU MAI
HO
MA TENG Gnetum gnemon (root: yield = 0.0040%dw). Ref: 4306.
OH
OH
H H
OH
OH
OH
OH
HO
H
OH
OH
H
O
HO
8867 Gnemonol B
HO
OH
8871 Gnemonol F
HO

OH
-Viniferin, IC50 = 20mol/L; lipid peroxide inhibitory activity, IC50 >

OH
100mol/L, control -Viniferin, IC50 = 33mol/L). Source: XIAN ZHOU
OH
MAI MA TENG Gnetum gnemon (root: yield = 0.0005%dw). Ref: 4306.
H
OH
OH
OH
H
H
OH
HO
OH
OH
HO
OH
OH

OH
HO
H
OH
8872 Gnemonol K

H
H
OH O
H
H
MeOH). Pharm: Antioxidant (superoxide anion scavenger, IC50 = 69mol/L;

inhibits lipid peroxidization, IC50 = 19mol/L). Source: XIAN ZHOU MAI
OH
MA TENG Gnetum gnemon. Ref: 2045.
HO
HO
H
OH
OH
8869 Gnemonol D
-Viniferin, IC50 = 20mol/L; lipid peroxide inhibitory activity, IC50 >
100mol/L, control -Viniferin, IC50 = 33mol/L). Source: XIAN ZHOU
MAI MA TENG Gnetum gnemon (root: yield = 0.0023%dw). Ref: 4306.
OH
OH
8873 Gnemonol L
MeOH). Pharm: Antioxidant (superoxide anion scavenger, IC50 = 59mol/L;
inhibits lipid peroxidization, IC50 = 7mol/L). Source: XIAN ZHOU MAI
MA TENG Gnetum gnemon. Ref: 2045.
HO
OH
OH
OH
HO
OH
OH
H
HO
HO
OH
HO
H
OH
OH
OH
H
H
HO
HO
OH
OH
8868 Gnemonol C
HO
OH
HO
OH
OH
H
OH
488
8874 Gnemonol M
8878 Gnetin
C30H26O8 (514.54). Colorless amorphous powder, []D = 28 (c = 0.12,
[56041-27-1] C16H14O3 (254.29). Crystals (CHCl3pet. ether), mp 121~122C.
MeOH). Source: XIAN ZHOU MAI MA TENG Gnetum gnemon. Ref: 2045.
Source: YIN DU MAI MA TENG Gnetum ula. Ref: 1521.
OH
O
O
O
OH
HO
8879 Gnetin C
C28H22O6 (454.48). Yellowish powder (acetone), mp 146~147C. Source: AI
OH
OH
DA HUANG Rheum nanum. Ref: 4807.
OH
HO
HO
O
8875 Gnemonoside E
HO
C40H42O16 (778.77). Brown amorphous powder. Source: MA LAI XI YA MAI
OH
MA TENG Gnetum gnemonoides (stem). Ref: 4200.

OH
OO
HO
8880 Gnetin E
OH
OH
C42H32O9 (680.72). Source: XIAN ZHOU MAI MA TENG Gnetum gnemon
OH
(root), MA LAI XI YA MAI MA TENG Gnetum gnemonoides (stem). Ref:
OH
HO
4200.
HO
OH
OH
OO
HO
OH
OH
OH
O
H
OH
OH
8876 Gnemonoside K
MeOH). Source: XIAN ZHOU MAI MA TENG Gnetum gnemon. Ref: 2045.
OO
OO
OH
OH
2234.
H
OH
OH
OH
OH
8881 Gnetin F
C28H24O6 (456.50). Source: BAI SUI YE Welwitschia mirabilis. Ref: 2233,
OH
HO
OH
OH
HO
H
H
OH
HO
OH
HO
OH
HO
OO
OH
OH
OH
OH
OH
8882 Gnetuhainin A
C28H22O7 (470.48). Source: HAI NAN MAI MA TENG Gnetum hainanense.
8877 Gnetal
C21H16O6 (364.36). White amorphous powder. Source: MA LAI XI YA MAI
Ref: 2233, 2234.
MA TENG Gnetum gnemonoides (stem). Ref: 4200.

OH
HO
HO
OH
OH
OH
HO
H
HO
OH
C60H62O24 (1167.15). Colorless amorphous powder, []D = 36 (c = 0.52,

HO
OH
OH
489
8883 Gnetuhainin C
8888 Gnetuhainin J
Ref: 2233, 2234.
Ref: 2234.
OH
HO
HO
OH
OH
OH
H
HO
HO
OH
OH
OH
8884 Gnetuhainin F
OH
HO
OH
Ref: 2233, 2234.

HO
8889 Gnetuhainin K
HO
Ref: 2234.
OH
OH
OH
HO
OH
8885 Gnetuhainin G
O
25
C30H22O9 (526.50). Greenish amorphous powder, []D = 0 (c = 0.084,
HO
H
MeOH). Source: HAI NAN MAI MA TENG Gnetum hainanense. Ref: 3995.
OH
HO
HO
O
O
OH
HO
OH
8890 Gnetuhainin M
OH
OH
Ref: 2233, 2234.
8886 Gnetuhainin H
25
C30H24O9 (528.52). Yellowish amorphous powder, []D = +16.0 (c = 0.072,
OH
OH
MeOH). Source: HAI NAN MAI MA TENG Gnetum hainanense. Ref: 3995.
OH
HO
O
HO
H
OH
HO
HO
OH
H
OH
HO
OH
OH
OH
8891 Gnetuhainin Q
8887 Gnetuhainin I
Ref: 2234.

Ref: 2234.
OH
HO
O
OH
HO
OH
HO
O
H
OH
OH
OH
OH
O
OH
OH
490
8892 Gnetulin
8896 Gnetumontanin D
C30H26O8 (514.54). Pale brownish amorphous solid. Source: XIAO YE MAI
C31H32O12 (596.59). Yellowish amorphous powder, []D20 = 24.0 (c = 0.075,
MA TENG Gnetum parvifolium [Syn. Gnetum indicum] (bark), YIN DU MAI
MeOH). Source: DA ZI MAI MA TENG Gnetum montanum f. megalocarpum.
MA TENG Gnetum ula. Ref: 2234, 3550.
Ref: 4936.
O
OH
OH
OH
HO
OH
OH
O
OH
OH
OH
OH
8893 Gnetumontanin A
C28H22O8 (486.48). Yellowish amorphous powder, mp 233~234C, []D22 =
+17.0 (c = 0.10, MeOH). Source: DA ZI MAI MA TENG Gnetum montanum
f. megalocarpum. Ref: 4936.
HO
OH
8897 Gnetupendin A
10-(4-Hydroxybenzyl)-isorhapontigenin C22H20O5 (364.40). Pale yellow solid.
Source: CHUI ZI MAI MA TENG Gnetum pendulum. Ref: 5199.
OH
OH
H
O
OO
HO
HO
OH
OH
HO
OH
H
OH
OH
8894 Gnetumontanin B
OH
22
C42H32O11 (712.72). Off-white amorphous powder, mp 209~210C, []D =

16.0 (c = 0.10, MeOH). Pharm: TNF- inhibitor (IC50 = 1.49mol/L)[4936].
8898 Gnetupendin B
Source: DA ZI MAI MA TENG Gnetum montanum f. megalocarpum. Ref:
10-(3,4-Dihydroxybenzyl)-isorhapontigenin C22H20O6 (380.40). Brown solid.
4936.
Pharm: PGE2 production inhibitor (mouse peritoneal macrophages,

LPS-induced, 0.1mol/L, InRt = 24.4%, P<0.05; control Meloxicam, IC50 =
0.0286mol/L; may have cyclo-oxygenase-2 inhibition activity). Source:
OH
HO
CHUI ZI MAI MA TENG Gnetum pendulum. Ref: 5199.
OH
H
HO
HO
O
H
OH
OH
OH
OH
OH
O
HO
H
OH
O
OH
OH
8895 Gnetumontanin C
C25H22O7 (434.45). Yellowish amorphous powder, mp 72~73C, []D20 = 0 (c
= 0.04, MeOH). Source: DA ZI MAI MA TENG Gnetum montanum f.
8899 Gnidicin-20-palmitate
C52H66O11 (867.10). Amorphous powder, []D25 = +41.7 (c = 0.56, CHCl3).
megalocarpum. Ref: 4936.

O
OH
O
O
OO
OH
OH
O
OH
HO
O
O
491
8900 Gnidilatidin
8905 Gomaline
[60195-70-2] C37H44O10 (648.76). Source: YOU RUI XIANG Daphne
oleoides. Ref: 2410.

O
O
O
OO
N
H
OH
O
HO
OH
8906 Gomisin A
OH
Wuweizi alcohol B [58546-54-6] C23H28O7 (416.48). mp 54~56C, []D22 =
8901 Gnidilatidin 20-palmitate
+60.8 (c = 0.58, chloroform); mp 88~89C, []D = +67.9. Pharm:
[60195-68-8] C53H74O11 (887.17). Source: YOU RUI XIANG Daphne
Antineoplastic (screened as potential antitumor promoters, EBV-EA induced
oleoides. Ref: 2410.
by TPA, mol ratio/TPA = 1000, relative percentage of EBV-EA = (7.10.4)%

(positive control value 32pmol, 20ng TPA =100%), viability of Raji cells =
70%)[4644]; antihepatotoxin, reduces excess SGPT (orl 100mg/kg); prevents
toxicosis (mus, due to CCl4 or thioacetamide); promotes biosynthesis of
hepatic glycogen (normal hungry mus); toxin (mus, orl, 250mg/kg, mortality
O
OO
= 2/4; mus, ip, 250mg/kg, mortality = 2/3). Source: NEI NAN WU WEI ZI
Kadsura interior (stem)[4644], REN SHEN Panax ginseng [Syn. Panax
OH
schinseng], WU WEI ZI Schisandra chinensis (dried ripe fruit: mean content
HO
of 11 origins = 0.23%[5508]). Ref: 2, 661, 1582, 4644, 5508.
O
O
8902 Gnoscopine
[6035-40-1] C23H25NO6 (411.46). mp 232C. Source: YA PIAN Papaver
somniferum. Ref: 6.
O
O
OH
O
O
O
N
O
O
8907 Gomisin B
Schizantherin B; Schisantherin B; Wuweizi ester B; Schisanhenrin
[58546-55-7] C28H34O9 (514.58). Prismatic crystals (etherpetroleum ether),
mp 88C, []D23 = 27 (c = 1.0, chloroform); mp 97~99C. Pharm:
Antihepatotoxin (mus, orl, 50mg/(kgd), reduces activity of SGPT); amino

8903 Gobicusin A
C18H20O5 (316.36). Colorless gum, []D21 = +51.6 (c = 5.50, Me2CO). Source:
GE BI TIAN MEN Asparagus gobicus (root). Ref: 4975.
(HbsAg: 100g/mL InRt = 74.1%, 50g/mL InRt = 28.9%, 25g/mL InRt =

3.3%; HbeAg: 100g/mL InRt = 34.1%, 50g/mL InRt = 28.2%, 25g/mL InRt
= 15.7%; DMSO 2.5l/mL, InRt = 0%)[4397]. Source: HUA ZHONG WU WEI
O
OH
HO
HO
transferase inhibitor (mus, hepatitis induced by CCl4)[658]; antihepatitis
ZI Schisandra sphenanthera, WU WEI ZI Schisandra chinensis, YI GENG

WU WEI ZI Schisandra henryi, A LI SHAN WU WEI ZI Schisandra
OH
arisanensis (stem). Ref: 2, 4, 6, 658, 4397.
8904 Gobicusin B
C19H18O4 (310.35). White powder, mp 127~129C (CHCl3), []D21 = 92.0
(c =
0.80, CHCl3). Source: GE BI TIAN MEN Asparagus gobicus (root). Ref: 4975.
OH
O
O
O
HO
O
O
492
8908 Gomisin C
8911 Gomisin F
Wuweizi ester A; Schisantherin A [58546-56-8] C30H32O9 (536.58). mp
[62956-47-2] C28H34O9 (514.58). Source: WU WEI ZI Schisandra chinensis.
116~118C, 122~124C. Pharm: Antineoplastic (screened as potential
Ref: 2.
antitumor promoters, EBV-EA induced by TPA, mol ratio/TPA = 1000,

relative percentage of EBV-EA = (19.70.5)% (positive control value 32pmol,
20ng TPA =100%), viability of Raji cells = 60%)[4644]; antihepatotoxin (mus,
orl, 100mg/(kgd), repairs hepatic injury induced by CCl4 or thioacetamide,
amino transferase inhibitor in rat). Source: HUA ZHONG WU WEI ZI
Schisandra sphenanthera (dried ripe fruit: content scope of 12 origins =
0.03%~2.69%, mean content = 1.27%[5508]), NEI NAN WU WEI ZI Kadsura
O
O
OH
O
O
interior (stem)[4644], WU WEI ZI Schisandra chinensis (dried ripe fruit:
content scope of 6 origins = 0.08%~1.95%, mean content = 0.76%[5508]). Ref:

2, 4, 6, 658, 4644, 5508.
8912 Gomisin G
[62956-48-3] C30H32O9 (536.58). Prisms (Me2CO/Et2O), mp 97~98C, []D25
O
O
= 126 (c = 0.427, CHCl3). Pharm: Antihepatitis (HbsAg: 100g/mL InRt =

76.3%, 50g/mL InRt = 42.4%, 25g/mL InRt = 17.9%; HbeAg:
OH
100g/mL InRt = 22.1%, 50g/mL InRt = 20.0%, 25g/mL InRt = 6.3%;

DMSO 2.5l/mL, InRt = 0%)[4397]; antineoplastic (screened as potential
O
O
antitumor promoters, EBV-EA induced by TPA, mol ratio/TPA = 1000,
relative percentage of EBV-EA = (18.90.6)% (positive control value 32pmol,

20ng TPA =100%), viability of Raji cells = 60%)[4644]. Source: NEI NAN WU
WEI ZI Kadsura interior (stem)[4644], WU WEI ZI Schisandra chinensis, A LI
8909 Gomisin D
SHAN WU WEI ZI Schisandra arisanensis (stem). Ref: 2, 1521, 4397, 4644.

Ref: 2.
O
O
O
O
OH
O
O
O
O
OH
O
O
O
OH
8913 Gomisin H
[66056-20-0] C23H30O7 (418.49). Pharm: Inhibits vasomotion (dog mesenteric
8910 Gomisin E
artery, calcium-induced vasomotion, IC50 = 530mol/L, induced by
[72960-21-5] C28H34O9 (514.58). []D23 = +25.0 (c = 0.40, CHCl3). Pharm:
prostaglandin F2, IC50 = 41mol/L); antihepatotoxin (rat, hepatic cells, GPTs
NFAT transcription inhibitor (IC50 = (4.730.09)mol/L, control Cyclosporin
increase induced by galactosamine, 1.0mg/mL shows weak action). Source:
A, IC50 = (1.200.29)nmol)[5343]. Source: WU WEI ZI Schisandra chinensis.
WU WEI ZI Schisandra chinensis (dried ripe fruit: mean content of 11 origins
Ref: 2, 5343.
= 0.31%[5508]). Ref: 2, 1730, 1731, 5508.
OH
HO
O
OH
493
8914 Gomisin J
8917 (+)-Gomisin K3
[66280-25-9] C22H28O6 (388.46). Pharm: Inhibits vasomotion (dog mesenteric
Schisanhenol; Schizanhenol [69363-14-0] C23H30O6 (402.49). Pharm:
artery, calcium-induced vasomotion, IC50 = 12mol/L, induced by
Antihepatitis (HbsAg: 100g/mL InRt = 76.3%, 50g/mL InRt = 42.4%,
prostaglandin F2, IC50 = 17mol/L); increases coronary flow (anesthetic dog);
25g/mL InRt = 17.9%; HbeAg: 50g/mL InRt = 20.0%, 25g/mL InRt =
antihepatotoxin (rat, hepatic cells, CCl4-induced increase of GPT level,
16.1%; DMSO 2.5l/mL, InRt = 0%)[4397]; antihepatotoxin (mus, orl,
2+
1.0mg/mL); antioxidant (mitochondria of rat hepatic cells, Fe /VC-induced
200mg/kg). Source: A LI SHAN WU WEI ZI Schisandra arisanensis (stem),
lipid peroxidization, IC50 = 5.5mol/L, ADP/NADPH-induced lipid
HONG HUA WU WEI ZI Schisandra rubriflora, HUA ZHONG WU WEI ZI
peroxidization, IC50 = 4.7mol/L); cardioprotective agent (inhibits
Schisandra sphenanthera (dried ripe fruit: content scope of 12 origins =
malondialdehyde (MDA) formed by abnormity of calcium concentration in
0.11%~7.57%, mean content = 1.07%)[5508], WU WEI ZI Schisandra
cardiac muscle cells, 10mol/L); cAMP phosphodiesterase inhibitor (IC50 =
chinensis (dried ripe fruit: content scope of 3 origins = 0.021%~0.41%, mean
136mol/L); antineoplastic (mus, TPA-induced skin tumor); anti-HIV (in
content = 0.14%[5508]). Ref: 2, 2, 658, 4397, 5501, 5508.
vitro); inhibits gastric ulcer (mus, orl, 100mg/kg, gastric ulcer induced by
experimental stress). Source: WU WEI ZI Schisandra chinensis. Ref: 2, 1730,
1731, 1732, 1733, 1734, 1735, 1736.
OH
O
O
O
HO
O
O
8918 ()-Gomisin L1
O
OH

Ref: 2.
O
O
8915 ()-Gomisin K1
O
HO
Ref: 2.
OH
O
O
8919 ()-Gomisin L2
Ref: 2.
O
O
O
O
O
8916 (+)-Gomisin K2
Ref: 2.
O
O
HO
OH
O
8920 ()-Gomisin M1
Ref: 2.
O
O
HO
O
O
O
494
8921 (+)-Gomisin M2
8926 Gomisin T
Gomisin T-ol [119139-66-1] C23H30O7 (418.49). White amorphous powder,

[]D23 = +60 (c = 0.50, chloroform). Pharm: 5-Lipoxygenase inhibitor
(100mol/mL, InRt = 55.6%). Source: WU WEI ZI Schisandra chinensis. Ref:
2, 1023.
O
HO
OH
8922 Gomisin N
[69176-52-9] C23H28O6 (400.48). []D23 = 83.4 (c = 1.07, CHCl3). Pharm:
O
OH
NFAT transcription inhibitor (IC50 = (1.330.05)mol/L, control Cyclosporin

[5343]
A, IC50 = (1.200.29)nmol/L)
. Source: WU WEI ZI Schisandra chinensis.
Ref: 5343.
8927 Gomphrenin I
[17008-59-2] C24H26N2O13 (550.48). Pharm: Purple phytochrome. Source:

QIAN RI HONG Gomphrena globosa. Ref: 15, 658.
O
O
O
HO
OO
HO
OH
OH
8923 Gomisin O
OH
HO
[72960-22-6] C23H28O7 (416.48). Source: HONG HUA WU WEI ZI

Schisandra rubriflora, WU WEI ZI Schisandra chinensis. Ref: 2, 39.
N
H
OH
O
O
8928 Gomphrenin II
[17008-60-5] C24H26N2O13 (550.48). Source: QIAN RI HONG Gomphrena
O
O
globosa. Ref: 15.

OH
HO
8924 Gomisin R
HO
OH
OH
OH
HO
O
N
H
OH
O
OH
O
8929 Gomphrenin III
8925 Gomisin S
[119239-49-5] C23H30O7 (418.49). Colorless rhombic Crystals, mp 172~176C,
C33H32 N2O15 (696.63). Source: QIAN RI HONG Gomphrena globosa.

Ref: 6, 15.
[]D23 = 63 (c = 0.49, chloroform). Pharm: Aldose reductase inhibitor (rat
OH
eye lens, 0.1ng/mL, InRt = 28%). Source: WU WEI ZI Schisandra chinensis.

Ref: 2, 1023.
O
O
OH
HO
O
H
O
OH
OH
O
OH
O
O
OH
OO
OH
N
H
O
OH
495
8930 Gomphrenin V
8934 (6R,7R,8R)-Goniodiol
[16955-52-5] C34H34N2O16 (726.65). Pharm: Purple phytochrome. Source:
C13H14O4 (234.25). Pharm: Cytotoxic (HepG2, IC50 = 9.15g/mL, control
QIAN RI HONG Gomphrena globosa. Ref: 6, 15, 658.

1.20g/mL). Source: TAI WAN GE NA XIANG Goniothalamus amuyon
HO
H
HO
O
OO
OH
OH
OH
H
O
OH
O
N
H
OH
OH
OH
8935 Goniodiol-7-monoacetate
8931 Gomphrenin VI
C15H16 O5 (276.29). Pharm: Cytotoxic (in vitro, NUGC, IC 50 = 4.12g/mL;
[16955-53-6] C34H34N2O16 (726.65). Source: QIAN RI HONG Gomphrena
HONE-1, IC50 = 5.69g/mL; control Actinomycin, NUGC, IC50 =
globosa. Ref: 6, 15.
6.61g/mL; HONE-1, IC50 = 4.53g/mL) [4686]; cytotoxic (HepG2,

inactive; Hep3B, IC50 = 7.85g/mL, control Doxorubicin, IC50 =
0.36g/mL; MDA-MB-231, inactive; MCF7, inactive)[5056]. Source: TAI
HO
HO
OO
WAN GE NA XIANG Goniothalamus amuyon (fresh leaf: yield =
OH
0.028%fw; stem: yield = 0.0016%fw). Ref: 4686, 5056.
OH
OH
O
OH
N
H
O
OH
HO
H
O
O
8932 Goniobutenolide A
1.20g/mL; MCF7, inactive). Source: TAI WAN GE NA XIANG
8936 Goniodiol-8-monoacetate
C15H16O5 (276.29). Pharm: Cytotoxic (in vitro, NUGC, IC50 = 5.02g/mL;
HONE-1, IC50 = 6.09g/mL; control Actinomycin, NUGC, IC50 = 6.61g/mL;
HONE-1, IC50 = 4.53g/mL)[4686]; cytotoxic (HepG2, inactive; Hep3B, IC50 =
4.63g/mL, control Doxorubicin, IC50 = 0.36g/mL; MDA-MB-231, IC50 =
8.05g/mL, Doxorubicin, IC50 = 1.20g/mL; MCF7, inactive)[5056]. Source:
TAI WAN GE NA XIANG Goniothalamus amuyon (fresh leaf: yield =
OH
OH
0.0044%fw). Ref: 4686, 5056.

O
O
O
8933 Goniobutenolide B
OH
H
8937 Gonioffithine
10-Amino-2,4-dimethoxyphenanthrene-1-carboxylic acid lactam
[240122-32-1] C17H13NO4 (295.30). Yellow acicular Crystals, mp 312~314C.
1.20g/mL; MCF7, inactive). Source: TAI WAN GE NA XIANG
Source: DA HUA GE NA XIANG Goniothalamus griffithii. Ref: 848, 5453.

O
OH
O
NH
HO
OH
O
496
8938 Goniofupyrone A
8942 Goniolactone D
C13H14O4 (234.25). Colorless plates, mp 154~156C, []D23 = 25.6 (c =
C28H24O8 (488.5). White needles, mp 158~160C, []D20 = +17.6 (c = 0.42, EtOH).
0.08, MeOH). Pharm: Cytotoxic inactive (HepG2, Hep3B, MDA-MB-231,
Pharm: Cytotoxic inactive (in vitro, A2780, HCT8 and KB). Source: GE NA
MCF7). Source: TAI WAN GE NA XIANG Goniothalamus amuyon (stem
XIANG Goniothalamus cheliensis (root: yield = 0.00021%dw). Ref: 4631.
and leaf). Ref: 5056.

HO
O
HO
HO
C26H24O7 (448.48). White needles, mp 166~168C, []D20 = +83.6 (c = 0.26,

EtOH). Pharm: Cytotoxic (in vitro, showed no significant inhibitory activities
toward A2780, HCT8 and KB). Source: GE NA XIANG Goniothalamus
cheliensis (root: yield = 0.00025%dw). Ref: 4631.
8943 Goniolactone E
C28H24O7 (472.5). White powder, mp 238~240C, []D20 = 0 (c = 0.10, EtOH).
Source: GE NA XIANG Goniothalamus cheliensis (root: yield =
0.00003%dw). Ref: 4631.
OH
O
O
O
O
8939 Goniolactone A
OH
H OH
H O
O
8944 Goniolactone F
OH

EtOH). Pharm: Cytotoxic inactive (in vitro, A2780, HCT8 and KB). Source: GE
NA XIANG Goniothalamus cheliensis (root: yield = 0.00013%dw). Ref: 4631.
8940 Goniolactone B
OH
C28H24O7 (472.5). Amorphous powder, mp 176~178C, []D20 = +33.7 (c =

0.92, EtOH). Pharm: Cytotoxic (in vitro, A2780, IC50 = 7.4mol/L; HCT8,
O
IC50 = 4.43mol/L; KB, IC50 = 7.23mol/L). Source: GE NA XIANG
Goniothalamus cheliensis (root: yield = 0.00029%dw). Ref: 4631.
H O
O
H
O
HO
8945 Goniothalactam
C17H13NO4 (295.30). Source: Goniothalamus sp. Ref: 2447.
HO
OH
O
NH
HO
8941 Goniolactone C
C28H24 O7 (472.5). Colorless oil, []D20 = 53.9 (c = 0.71, EtOH). Source:
8946 cis-Goniothalamicin
GE NA XIANG Goniothalamus cheliensis (root: yield = 0.00005%dw).
[172586-14-0] C35H64O7 (596.90). White amorphous powder (hexane), mp 80C,
Ref: 4631.
[]D25 = 7.2 (c = 0.03, chloroform). Pharm: Cytotoxic (A549, IC50 = 0.13g/mL,

MCF7, IC50 = 1.05g/mL, HT29, IC50 = 0.0053g/mL); cytotoxic (BST, LC50 =
OH
5.2g/mL, PD experiment, InRt = 47%); cytotoxic (in vitro HepG2, EC50 =

0.202g/mL, Hep3B, EC50 = 3.11g/mL; control Doxorubicin, HepG2, EC50 =
HO
O
H O
0.38g/mL, Hep3B, EC50 = 0.36g/mL)[5035]. Source: CI GUO FAN LI ZHI

Annona muricata, SHAN FAN LI ZHI Annona montana (seed). Ref: 1062, 5035.
OH
OH
OH
O
O
OH
OH
497
8947 Goniothalamin
8951 (5S,6S,10S)-Gorgona-1,4(15),11-triene
[17303-67-2] C13H12O2 (200.24). White crystals, mp 85C, [] D25 = +170 (c
(4S,4aS,8aS)-8a-Methyl-5-methylene-4-(1-methylvinyl)-1,2,3,4,4a,5,6,8a-octa
= 1.38, CHCl 3); [] D20 = 183.9 (c = 0.6, MeOH). Pharm: Cytotoxic
hydro-naphthalene C15H22 (202.34). Colorless oil. Source: Saccogyna
(HepG2, IC50 = 0.31g/mL, control Doxorubicin, IC50 = 0.38g/mL; Hep3B,
viticulosa (essential oil). Ref: 3839.
IC50 = 1.07g/mL, control Doxorubicin, IC50 = 0.36g/mL; MDA-MB-231,

IC50 = 1.07g/mL, control Doxorubicin, IC50 = 1.20g/mL; MCF7, IC50 =
4.65g/mL, control Doxorubicin, IC50 = 2.51g/mL)[5056]. Source: DA HUA
H
GE NA XIANG Goniothalamus griffithii, JIN PING GE NA XIANG

Goniothalamus leiocarpus, TAI WAN GE NA XIANG Goniothalamus
amuyon (stem and leaf), TAI WAN GE NA XIANG Goniothalamus amuyon
8952 (+)-(5R,6S,10S)--Gorgonene
(fresh leaf: yield = 0.00061%fw)[4686]. Ref: 420, 4686, 5056, 5453.
(+)-(1S,4aS,8aR)-4a,8-Dimethyl-1-(1-methylvinyl)-1,2,3,4,4a,5,6,8a-octahydr
o-naphthalene C15H24 (204.36). Colorless oil. Source: Saccogyna viticulosa
8948 Goniothalamin epoxide

C13H12O3 (216.24). Pharm: Cytotoxic (in vitro, NUGC, IC50 = 32.1g/mL;
8953 -Gorgonene
HONE-1, IC50 = 36.3g/mL; control Actinomycin, NUGC, IC50 = 6.61g/mL;
(+)-(5S,6S,10S)--Gorgonene C15H24 (204.36). Source: Saccogyna viticulosa
HONE-1, IC50 = 4.53g/mL)[4686]; cytotoxic (HepG2, IC50 = 0.19g/mL,
control Doxorubicin, IC50 = 0.38g/mL; Hep3B, IC50 = 3.29g/mL,

Doxorubicin, IC50 = 0.36g/mL; MDA-MB-231, IC50 = 1.23g/mL,
Doxorubicin, IC50 = 1.20g/mL; MCF7, IC50 = 1.94g/mL, Doxorubicin, IC50
= 2.51g/mL)[5056]. Source: TAI WAN GE NA XIANG Goniothalamus
amuyon (fresh leaf: yield = 0.00035%fw; stem: yield = 0.00047%fw). Ref:

4686, 5056.
8954 ()-(4R,5R,6S,10S)-Gorgon-11-en-4-ol
()-(1R,4aS,8S,9R)-1,4a-Dimethyl-8-(1-methylethenyl)-decahydro-naphthalen
-1-ol C15H26O (222.37). Colorless oil. Source: Saccogyna viticulosa
O
O
HO
8949 (5S,6R,7R,8R)-Goniotriol
C 13 H 14 O 5 (250.25). Source: TAI WAN GE NA XIANG Goniothalamus
amuyon (fresh leaf: yield = 0.0059%fw; stem: yield = 0.00047%fw).
8955 Gorlic acid
Ref: 4686.
C18H30O2 (278.44). Pharm: Antileprotic (inhibits Mycobacterium leprae).

Source: DA FENG ZI Hydnocarpus anthelminticus (seed: content scope =
H OH OH
HO H
0.57%~1.03%). Ref: 5501.

OH
O
O
8950 (5S,6R,7S,8S)-Goniotriol
C13H14O5 (250.25). Source: TAI WAN GE NA XIANG Goniothalamus
amuyon (fresh leaf: yield = 0.00065%fw). Ref: 4686.
8956 Goshuyic acid

Goshuynic acid [39039-37-7] C14H24O2 (224.35). Source: WU ZHU YU
Evodia rutaecarpa. Ref: 6, 1521.
H OH OH
HO H
OH
H
O
H H
498
8957 Goshuyuamide I
8962 Gossypetin-3--D-(2-O--D-glucopyranosylglucopyranoside)-
[126223-62-9] C19H19N3O (305.38). Source: WU ZHU YU Evodia rutaecarpa.
8--D-glucopyranoside
Ref: 2, 347, 877.
C33H40O23 (804.67). Source: MU ZEI Equisetum hiemale. Ref: 2.

OO
HO
OH
N
H
OH
OH
OH OHOHO
OH
HN
8958 GoshuyuamideII
HO
[95274-42-3] C19H17N3O2 (319.37). Source: WU ZHU YU Evodia rutaecarpa.
OO
HO
Ref: 2, 877.
OH
OH
OH
N
H
OH
OH
8963 Gossypetin hexamethyl ether

C21H22O8 (402.40). mp 159~161C, 170~171C. Source: JI CAI Capsella
bursa-pastoris. Ref: 6.
O
8959 Gossypetin
O
O
[489-35-0] C15H10O8 (318.24). mp 311~313C. Pharm: Antibacterial

(Pseudomonas maltophilia and Enterobacter cloacae). Source: BAI HUA
YING SHAN HONG Rhododendron mucronatum, HENG GEN FEI CAI
Sedum kamtschaticum, MAN SHAN HONG Rhododendron dauricum, XIAO

YE PI PA Rhododendron anthopogonoides, YING SHAN HONG
Rhododendron mucronulatum, ZHAO SHAN BAI Rhododendron micranthum.
Ref: 6, 658.
OH
[18799-01-4] C16H12O8 (332.27). Source: DI YANG QUE Lotus corniculatus. Ref: 6.

OH
O
OH
O
OH
HO
8964 Gossypetin-7-methylether
O
OH
OH
O
OH
OH
OH
OH
8965 Gossypin
[652-78-8] C21H20O13 (480.39). mp 230C (dec). Pharm: Analgesic;
8960 Gossypetin-3,5-dimethyl ether

C17H14O8 (346.30). Source: KE SHI FAN YING TAO Eugenia edulis (leaf).
Ref: 3469.
ulcer). Source: HENG GEN FEI CAI Sedum kamtschaticum, MO PAN CAO
Gossypium indicum. Ref: 6, 661.
OH
OH
O
permeability caused by variety of phlogogenic agents); antiulcerative (gastric

Abutilon indicum, PU TAO YE MU JIN Hibiscus vitifolius, YIN DU MIAN
OH
OH
HO
anti-inflammatory (reduces swollen foot and increase of blood capillary
OH
HO
HO
8961 Gossypetin-3,8-dimethyl ether-5-O--glucoside
OO
OH
OH
C23H24O13 (508.44). Source: KE SHI FAN YING TAO Eugenia edulis (leaf).
Ref: 3469.
OH
OH
OH
8966 Gossypitrin
[489-34-9] C21H20O13 (480.39). mp 252C. Source: MU ZEI Equisetum hiemale,
OH
O
HO
MO PAN CAO Abutilon indicum, WEN JING Equisetum arvense. Ref: 2.

OH
OH
O
OH
O
OO
HO
OH
OH
HO
OO
OH
OH
OH
O
OH
OH
OH
OH
499
8967 Gossypol
8969 Graecunin E
[303-45-7] C30H30O8 (518.57). mp 184C, 199C, 214C. Pharm: Antibacterial
C51H82 O22 (1047.21). Source: HU LU BA Trigonella foenum-graecum.
(Staphylococcus aureus, hemolytic streptococcus); antineoplastic (mus, P388,
Ref: 2458.
hysteromyoma, deciduoma caused by luteosterone); anti-fertility agent

O
(inhibits generation and movement of sperma, D-isomer has no activity);

antiviral (-influenza virus PR8 and Japanese encephalitis virus); promotes
regeneration of muscle tissue (ointment); LD50 (mus, orl) = 315mg/kg.
OH
Source: DI TANG HUA Kerria japonica, HAI DAO MIAN Gossypium

barbadense] (root cortex: content = 1.8%
[5508]
), LU DI MIAN Gossypium
OH
MIAN HUA Gossypium herbaceum, MIAN HUA GEN Gossypium

[5508]
herbaceum (root cortex: content = 1.3%
), MIAN ZI YOU Gossypium
herbaceum (seed: mean content of 5 batch samples = 0.13%[5508]). Ref: 4, 5, 6,

658, 5508.
OH
OH
O
OH
O
OH
OH
8970 Graecunin G
C45 H 72 O17 (885.07). Source: HU LU BA Trigonella foenum-graecum.
Ref: 2458.
O
OH
OH
O
OH
HO
O
HO
hirsutum [Syn. Gossypium mexicanum] (root cortex: content = 1.6%)[5508],
OO
OH
O
OH
HO
OH
HO
OH
O
H
OH
OO
O
OH
HO
8968 Gracillin
Gracilline [19083-00-2] C45H72O17 (885.07). Colorless rhombic crystals

(methanol), mp 287~289C (dec); 298~302C; 290~293C, []D20 = 86.2 (c
= 0.12, dimethylformamide). Pharm: Antibacterial (Bacillus dysenteriae, MIC
= 2.5mg/mL; Serratia marcescens, MIC = 2.5mg/mL; Bacillus coli, MIC =
5.0mg/mL; drug-fast Staphylococcus aureus, MIC = 2.5mg/mL; sensitive
Staphylococcus aureus, MIC = 2.5mg/mL); antifungal (Trichophyton
mentagrophytes); cardiotonic; cytotoxic (in vitro, HeLa, IC50 = 12.74g/mL;
control Cisplatin, HeLa, IC50 = 0.75g/mL)[4788]; hemolytic (extremely strong);
antineoplastic (inhibits TPA-induced 32P combines with phospholipid in HeLa
cells, 5g/mL, InRt = 11.5%); cAMP phosphodiesterase inhibitor (in vitro,
IC50 = 61mol/L). Source: BA QIA Smilax china [Syn. Smilax japonica], CI
OH
OH
OH
OH
O
OH
O
OH
8971 Gramine
Donaxine [87-52-5] C11H14N2 (174.25). Acicular or lamellar crystals,
(acetone), mp 138~139C, soluble in ethanol, ether, chloroform, slightly
soluble in cold acetone, insoluble in petroleum ether, water.[5507] Pharm: Insect
antifeedant; toxin (sheep, causes Phalaris blind stagger). Source: HONG HUA
QI Acer rubrum, JI MU Loropetalum chinense, LU ZHU GEN Arundo donax,
MAI YA Hordeum vulgare, YI CAO Phalaris arundinacea, YIN BAI QI Acer
saccharinum, Lupinus sp. Ref: 4, 6, 658, 5507.
JI LI Tribulus terrestris, DUN YE SHU YU Dioscorea zingiberensis, FU

ZHOU SHU YU Dioscorea futschauensis, HAI JIN BI XIE Dioscorea
spongiosa (Rhizome: yield = 0.00041%)[4692], HU BEI HUANG JING
Polygonatum zanlanscianense (rhizome: yield = 0.00045%dw)[4788], SHU
N
N
H
KUI YE SHU YU Dioscorea althaeoides, XIAN XI SHU YU Dioscorea

gracillima, ZHANG LIU TOU Costus speciosus, XIAO HUA DUN YE SHU
8972 Gramine methohydroxide
YU Dioscorea parviflora, Costus sp. Ref: 6, 10, 15, 660, 900, 4692, 4788.
O
N
H
HO
HO
O
OH
OH
OO
O
OH
OH
N
H
H
H
8973 Gramine Nb-oxide

O
OH
O
OH
N
OH OH
N
H
500
8974 Grandiamide A
8979 Grandisin
C38H44N2O9 (672.78). Amorphous powder, []D25 = 108.8 (c = 0.25, CHCl3).
[53250-50-3] C24H32O7 (432.52). Pharm: Inhibits PAF; antitrypanosomal
Source: JU DA MI ZI LAN Aglaia grandis (leaf). Ref: 3947.
(trypomastigote form of Trypanosoma cruzi (Y strain), IC50 = 8.74g/mL)[3450].

Source: DA MU JIANG ZI Litsea grandis, Piper solmsianum. Ref: 658, 3450.
O
HO H N
O
N
H
O
H
O
O
O
8980 cis-Grandmarin
8975 Grandiamide B
C18H24N2O2 (300.40). mp 99~102C (Hexane-EtOH). Source: JU DA MI ZI
LAN Aglaia grandis (leaf). Ref: 3947.

HN
O
H
H
N
H
Source: Citrus tamurana. Ref: 5048.

O
8976 Grandiamide C
C18H24N2O3 (316.40). Amorphous powder, []D20 = 0 (c = 1.13, CHCl3).
Source: JU DA MI ZI LAN Aglaia grandis (leaf). Ref: 3947.

OH
OH
O
HN
N
H
8981 trans-Grandmarin isovalerate
OH

8977 Grandifloroside
racemosa] (leaf, flower and twig: yield = 0.0046%dw). Ref: 4723.
O
HO
Source: Citrus hassaku. Ref: 5048.
O
OH
HO
O
O
O
OH
O
OH
OH
OH
O
OH
8978 Grandifloroside 11-methyl ester

26
8982 Granilin
Source: JI ZI MU Sinoadina Racemosa [Syn. Adina racemosa] (leaf, flower
[40737-97-1] C15H20O4 (264.32). Pharm: Antibacterial. Source: A SHI HAO
and twig: yield = 0.0018%dw). Ref: 4723.
Artemisia ashurbajevii, DA YE TU MU XIANG Inula grandis, DUO SUI

TUN CAO Ambrosia polystachya, TIAN MING JING Carpesium
O
HO
abrotanoides. Ref: 658, 1521.
O
OH
HO
O
O
OH
O
OH
OH
OH
O
HO
501
8983 Grasshopperketone
8987 Gravacridonolchlorine
C13H20O3 (224.30). Source: RI BEN HUANG BAI Phellodendron japonicum
[38494-85-8] C19H18ClNO5 (375.81). mp 233~237C. Source: CHOU CAO
(leaf). Ref: 4502.
Ruta graveolens. Ref: 6.

OH
OH
O Cl
N
OH
HO
OH
8984 Gravacridonechlorine
8988 Gravelliferone
[38494-84-7] C19H18ClNO4 (359.81). mp 254~257C. Source: CHOU CAO
[21316-80-3] C19H22O3 (298.39). mp 116~118C. Source: CHOU CAO Ruta
Ruta graveolens. Ref: 6, 2101.
graveolens. Ref: 6.
OH
N
HO
Cl
8989 Gravelliferone methyl ether

C20H24 O3 (312.41). Pharm: Vasodilator (cerebral, pig, in vitro). Source:
O
OH
SHAN MO LI YUN XIANG Ruta oreojasme, CHOU CAO Ruta

graveolens. Ref: 6, 658.
8985 Gravacridonediol
[37551-75-0] C19H19NO5 (341.37). Yellow amorphous powder, mp
224~227C, []D = 111.1 (c = 0.1, MeOH). Pharm: Antileishmanial
(Leishmania major promastigote, 10mol/L, survival = (54.01.1)%, 1mol/L,
8990 Graveobioside A
survival = (97.22.2)%, control Amphotericin B, 10mol/L, survival =
Luteolin-7-apio-glucoside [63808-23-1] C26H28O15 (580.50). mp 251~252C.
(0.20.04)%, 1mol/L, survival = (71.94.4)%; Leishmania major amastigote,
Source: HAN QIN Apium graveolens. Ref: 6, 1521.
10mol/L, survival = (9.51.0)%, 1mol/L, survival = (58.03.1)%, control

Amphotericin B, 10mol/L, survival = (0.40.02)%, 1mol/L, survival =
OH
(0.50.03)%)[3797]; antifungal inactive (silica gel TLC, Cladosporium

cucumerinum, control Nystatin, MIA = 0.2g)[3797]; algicidal (Oscillatoria
perornata, LCIC = 10mg/L; Selenastrum capricornutum, LCIC >
100mg/L)[5328]. Source: CHOU CAO Ruta graveolens, Thamnosma rhodesica
(root). Ref: 6, 3797, 5328, 1521.
O
O
HO
OH
OH
OH
OH
O
HO
O
OH
OH OH
8991 Graveoline
N
OH OH
[485-61-0] C17H13NO3 (279.30). mp 204~205C. Source: CHOU CAO Ruta

graveolens, WU ZHU YU Evodia rutaecarpa (fruit). Ref: 6, 5031.
8986 Gravacridonediol monomethyl ether
C20H21 NO5 (355.39). mp 219~221C. Source: CHOU CAO Ruta

graveolens. Ref: 6.
O
O
8992 Graveolinine
[4179-37-7] C17H17NO3 (279.30). mp 115~116C. Source: CHOU CAO Ruta
O
O OH
OH
graveolens. Ref: 6.
O
O
O
502
8993 Grayanotoxin I
8998 Grevirobstol A
C22H36O7 (412.53). Source: MU LI LU Leucothoe grayana (in 1971 the
C28H38O4 (438.61). Yellowish oil. Source: YIN HUA Grevillea robusta (leaf).
compound was isolated from the plant)[5505]. Ref: 5505, 5507.
Ref: 3905.
HO
H
HO
O
OH
OH
OH
OH
OH
HO
OH
8994 Grayanotoxin III
8999 Grevirobstol B
C20H34O6 (370.49). Source: MU LI LU Leucothoe grayana (in 1971 the compound
C28H40O4 (440.63). Amorphous powder. Source: YIN HUA Grevillea robusta
was isolated from the plant)[5505], RI BEN MA ZUI MU Pieris japonica (in 1959
the compound was separated from the plant)[5505]. Ref: 5505, 5507.
(leaf). Ref: 3905.

OH
OH
HO
HO
H
HO
OH
OH
OH
OH
9000 Grevirobstol C
C28H36O4 (436.60). Yellowish oil. Source: YIN HUA Grevillea robusta (leaf).
8995 Grayanotoxin II
Ref: 3905.
C20H32O5 (352.48). Source: MU LI LU Leucothoe grayana (the compound

was isolated from the plant in 1971)[5505], NAO YANG HUA Rhododendron
OH
O
HO
molle (flower: yield = 0.00023%dw). Ref: 5505, 4780.

HO
H
HO
OH
OH
OH
OH
9001 Grifficyclocin A
C43H62N8O8 (819.02). []D20 = 132 (c = 0.12, MeOH). Source: DA HUA GE
8996 Grayanotoxin XVIII
NA XIANG Goniothalamus griffithii. Ref: 5453.
C20H32O4 (336.48). White solid. Source: JIN YE ZI Craibiodendron

yunnanese (leaf). Ref: 4575.
H
OH
HO
H
HN
N
H
NH
OH
OH
NH
O
O
N
O
N
8997 Grevillol
9002 Griffinin
5-Tridecyl-1,3-benzenediol [5259-01-8] C19H32O2 (292.47). Acicular crystals
C19H15NO4 (321.34). mp > 250C. Source: DA HUA GE NA XIANG
(benzene), mp 82~83C. Pharm: Dermatitic (causes contact dermatitis);
Goniothalamus griffithii. Ref: 5453.
5-lipoxygenase inhibitor; irritant (to skin). Source: YIN HUA Grevillea
robusta, Grevillea spp. Ref: 658, 2108.
HO
OH
OH
N
503
9003 Griffipavixanthone
9008 Griffonianone B
C36H28O12 (652.62). Pharm: Antioxidant (DPPH scavenger, EC50 =
C22H18O7 (394.38). Yellowish amorphous solid. Source: Millettia griffoniana
0.115g/mL, control BHA, EC50 = 0.136g/mL, Vitamin E, EC50 =
(root cortex). Ref: 5134.
0.138g/mL). Source: DUO ZHI ZHI TENG HUANG Garcinia virgata (stem
cortex). Ref: 3874.
OH
HO
O
HO
O
OH
OH
9009 Griffonianone C
C17H28O6 (448.52). White crystals (MeOH), mp 138~139C. Source: Millettia
OH
HO
griffoniana (root cortex). Ref: 5134.
OH
OH
O
9004 Griffithazanone A
C14H11NO4 (257.25). Source: DA HUA GE NA XIANG Goniothalamus
griffithii. Ref: 2447.
C22H30O2 (326.5). Pharm: Antihistamine (inhibits histamine release, rat
OH
9010 Grifolin
N
H
peritoneal mast cells, compound 48/80-induced). Source: MAN SHAN

HONG Rhododendron dauricum (twig and leaf: yield = 0.0031%) Ref: 4755.
OH
9005 Griffithazanone B
griffithii. Ref: 2447.
OH
9011 Groenlandicin
O
C19H16NO4+ (322.34). Pharm: Cytotoxic (topoisomerase I inhibitor in

vitro)[5369]. Source: Coptis groenlandica. Ref: 1521, 5369.
N
H
OH
9006 Griffithdione
griffithii. Ref: 2447, 5453.
9012 Grosmomoside I
Mogro-3-O--D-glucopyranoside-24-O{[-D-glucopyranosyl (21)]-[-D-
O
O
glucopyranosyl(61)]--D-glucopyranoside} C54H92O24 (1125.32). White
amorphous powder. Source: LUO HAN GUO Siraitia grosvenorii [Syn.
NH
Momordica grosvenorii]. Ref: 4805.

HO
OH
OO
HO
O
OH
OH
OH
HO
9007 Griffonianone A
OO
OH
C28H32O8 (496.56). Yellowish amorphous solid. Source: Millettia griffoniana
OH
(root cortex). Ref: 5134.
HO
H
O
HO
OO
HO
O
OH
OH
O
O
OH
OH
OH
OH
504
9013 Grossamide
9017 GS-2
2-(4-Hydroxy-3-methoxyphenyl)-3-[N-2-(4-hydroxyphenyl)ethyl]carbamoyl-
C20H24N2O5 (372.42). Amorphous. Source: CHANG LV GOU WEN
5-[N-2-(4-hydroxyphenyl)ethyl]carbamoylethenyl-7-methoxybenzodihydrofur
Gelsemium sempervirens (stem and leaf). Ref: 4395.
an C36H36N2O8 (624.70). Yellowish oil. Pharm: Cytotoxic (in vitro, LNCaP,

IC50 = 33mol/L)[4607]; feeding deterrent[4607]. Source: DA MA JIN Hibiscus
H
OH
cannabinus (bark), LANG DANG ZI Hyoscyamus niger (seed: yield =

H N
0.006%dw)[4607]. Ref: 4607, 5233.

O
O
HO
H
N
O
NH
9018 GS-3
OH

O
OH
H
OH
9014 Grossamide K
2-(4-Hydroxy-3-methoxyphenyl)-3-hydroxymethyl-5-[N-2-(4-hydroxyphenyl)
ethyl]carbamoylethenyl-7-methoxybenzodihydrofuran C28H29NO7 (491.55).
H N
H
Yellowish oil. Source: DA MA JIN Hibiscus cannabinus (bark). Ref: 5233.

9019 GSIR-1
C10H15O3 (182.22). Amorphous. Source: CHANG LV GOU WEN Gelsemium
O
HO
sempervirens (stem and leaf). Ref: 4395.
OH
NH
O
H
OH
HO
9020 (+)-Guaiacin
C20H24O4 (328.41). Pharm: Neuroprotective (glutamate-induced neurotoxicity
9015 Grossheimin
Grosheimin C15H18O4 (262.31). mp 200~202C, []D20 = +159.9 (c = 1.14,
chloroform); mp 205C (methanol), []D20 = +137.7 (c = 0.225, methanol).
Pharm: Antineoplastic; cytotoxic (HeLa, ED50 = 2.5g/mL); insect antifeedant.
in primary cultures of cortical cells, 0.1mol/L, protection rate =

(16.71.1)%, MK-801: 1.0mol/L, protection rate = (83.62.0)%, p<0.001,
CNQX: 1.0mol/L, protection rate = (70.51.5)%, p<0.001). Source: HONG
NAN PI Machilus thunbergii. Ref: 4927.
Source: BO LIN JU Chartolepis intermedia, CAI JI Cynara scolymus, NI JIN

ZHAN JU Venidium decurrens. Ref: 661.
H
O
HO
OH
H
OH
9021 Guaiacol
o-Methoxy phenol [90-05-1] C7H8O2 (124.14). mp 32C, bp 205C. Pharm:

9016 GS-1
Antitussive (dispels phlegm). Source: AN YE Eucalyptus globulus, CHAI HU
Bupleurum chinense, DANG GUI Angelica sinensis, HAN QIN Apium
graveolens, SANG YE Morus alba, WU HUA GUO YE Ficus carica, Betula

sp. Ref: 2, 658.
H
OH
H N
O
N
O
OH
O
505
9022 erythro-Guaiacylglycerol
9027 (1'S,2'R)-Guaiacyl glycerol 3'-O--D-glucopyranoside

OH
H
OH
OH
OH
O
OH
HO
HO
OH
OH
OH
9023 D-threo-Guaiacylglycerol 8--D-glucopyranoside
OH
C16H24O10 (376.36). White powder, []D20 = 30.2 (c = 0.26, MeOH). Source:

XIAO YE SHI NAN Photinia parvifolia (stem). Ref: 4553.
OH
9028 threo-Guaiacylglycerol
OH
HO
H
HO
HO
OH
HO
OH
OH
OH
OH
9024 L-threo-Guaiacylglycerol 8--D-glucopyranoside

9029 ()-Guaia-1(10),11-dien-15-al
[133593-95-0] C15H22O (218.34). Source: CHEN XIANG Aquilaria

agallocha. Ref: 13.
OH
O
OH
H
OO
HO
OH
OH
OH
OH
9030 ()-Guaia-1(10),11-dien-15-carboxylic acid

9025 (1'R,2'R)-Guaiacyl glycerol 3'-O--D-glucopyranoside
OH
HO
O
OH
HO
HO
OH
OH
OH
9031 ()-Guaia-1,11-dien-10-ol
9026 (1'R,2'R)-Guaiacyl glycerol 4-O--D-glucopyranoside

C15H24O (220.36). White solid, mp 117~118C, []D = 66.1 (c = 0.40,

CHCl3); mp 118.5C, []D = 79.2 (c = 0.71, CHCl3). Pharm:
Antitrypanosomal (epimastigotes of Trypanosoma cruzi, in vitro, MLC >
200mmol/L)[2551]. Source: GUANG HUO XIANG Pogostemon cablin [Syn.
OH
O
HO
OO
Mentha cablin]. Ref: 2551.

OH
HO
OH
OH
OH
H
OH
506
9032 ()-Guaia-1(10),11-dien-15-ol
9037 Guaia-1(10),2,4,11(13)-tetraen-12,6-olide
C15H24O (220.36). Colorless oil, []D = 8.3 (c = 0.15, EtOH); []D = 11.6
C15H16O2 (228.29). Gum, []D = 34.2 (c = 0.12, CHCl3). Source: YI KUA
(c = 1.0, EtOH). Pharm: Antitrypanosomal (epimastigotes of Trypanosoma
Artemisia myriantha (aerial parts). Ref: 4618.
cruzi, in vitro, MLC > 200mmol/L)[2551]. Source: CHEN XIANG Aquilaria

agallocha, GUANG HUO XIANG Pogostemon cablin [Syn. Mentha cablin].
Ref: 13, 2551.
HO
O
O
9038 Guaiazulene
[489-84-9] C15H18 (198.31). Blue oil, mp 31.5C, bp 165~170C/10mmHg,

176C/17mmHg. Pharm: Anti-inflammatory; 5-reductase inhibitor (IC50 =
9033 (+)-Guaia-10(15),11-dien-1-ol
(100.89.3)mol/L; control Finasteride, IC 50 = (0.380.06)mol/L;
C15H24O (220.36). White solid, mp 64~65C, []D = +67.6 (c = 0.23, CHCl3);
-Linolenic acid, IC50 = (160.324.6)mol/L)[5398]. Source: MU
69.5C, []D = +67.1 (c = 0.73, CHCl3). Pharm: Antitrypanosomal
Matricaria chamomilla [Syn. Matricaria recutita], YU CHUANG MU
(epimastigotes of Trypanosoma cruzi, in vitro, MLC > 200mmol/L). Source:
Guajacum officinale. Ref: 658, 5398.
(3)
JU
GUANG HUO XIANG Pogostemon cablin [Syn. Mentha cablin]. Ref: 2551.
HO
9039 ()-(1S*,5S*,7S*)-Guai-3,9-dien-5,11-oxide
9034 ()-Guaia-1(10),11-dien-15,2-olide
2,2,6,9-Tetramethyl-3,4,6a,7-tetrahydro-2H-3,9a-methanocyclopent[b]oxocin
e C15H22O (218.34). Colorless oil. Source: XIAO E TAI Mylia taylorii
H
9035 1,7,10H-Guaia-4,11-dien-3-one
C15H22O (218.34). Colorless oil, []D24 = +63.1 (c = 0.23, CHCl3). Pharm:
9040 (+)-(1S*,5S*,7S*)-Guai-3,10(14)-dien-5,11-oxide
Cytotoxic (P388, ED50 = 1.19g/mL, control Mithramycin, ED50 = 0.08g/mL;
2,2,9-Trimethyl-6-methylene-3,4,5,6,6a,7-hexahydro-2H-3,9a-methanocyclopent[b
HT29, ED50 > 50g/mL, Mithramycin, ED50 = 0.07g/mL; A549, ED50 >
]oxocine C15H22O (218.34). Colorless oil. Source: XIAO E TAI Mylia taylorii
50g/mL, Mithramycin, ED50 = 0.06g/mL). Source: PI ZHEN XING YAO
HUA Wikstroemia lanceolata (stem and root). Ref: 4947.
H
H
O
9036 (+)-Guaia-1(10),11-dien-9-one
20
C15H22O (218.34). Oil, []D = +27.2 (c = 0.07, CHCl3). Source: CHEN

XIANG Aquilaria agallocha. Ref: 13, 1521.
O
9041 -Guaiene
[3691-12-1] C15H24 (204.36). bp 78~79C/2.5mmHg. Source: CANG ZHU
Atractylodes lancea, GUANG HUO XIANG Pogostemon cablin [Syn. Mentha
cablin], REN SHEN Panax ginseng [Syn. Panax schinseng], SAN QI Panax
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng]. Ref: 2, 660.
507
9042 -Guaiene
9046 Guan-fu base F
[3691-11-0] C15H24 (204.36). bp 118C/8mmHg. Source: CANG ZHU
C26H35NO6 (457.57). Source: HUANG HUA WU TOU Aconitum coreanum
Atractylodes lancea, DANG SHEN Codonopsis pilosula, GUANG HUO
(tuberoid). Ref: 4593.
XIANG Pogostemon cablin [Syn. Mentha cablin], HUA DONG LAN CI
TOU Echinops grijsii, SAN QI Panax pseudo-ginseng var. notoginseng [Syn.
HO
Panax notoginseng]. Ref: 2, 660.
OH
9047 Guan-fu base G

9043 Guaijaverin
O O
Quercetin-3-O-arabinoside; Foeniculin [22255-13-6] C20H18O11 (434.36). mp

256C. Source: DIAO GAN MA Celastrus angulatus, FAN SHI LIU GAN
OH
Polygonum multiflorum, HUI XIANG JING YE Foeniculum vulgare, HU

ZHANG Polygonum cuspidatum. Ref: 2, 6.
Psidium guajava, FAN SHI LIU YE Psidium guajava, HE SHOU WU
OH
OH
HO
9048 Guan-fu base I

OH
OH O O
OH
OH
HO
OH
OH
9044 Guaiol
1(5)-Guaien-11-ol; ()-Guaiol [489-86-1] C15H26O (222.37). mp 91C, bp
288C. Pharm: 5-Reductase inhibitor (IC50 = (81.610.2)mol/L; control
Finasteride, IC50 = (0.380.06)mol/L; -Linolenic acid, IC50 =
9049 Guan-fu base K
(160.324.6)mol/L)[5398]. Source: AN YE Eucalyptus globulus, CANG ZHU
Atractylodes lancea, DU HUO Angelica pubescens f. biserrata [Syn. Angelica
pubescens], HOU PO Magnolia officinalis, NING MENG Citrus limon,

QIANG HUO Notopterygium incisum. Ref: 2, 660, 5398.
O
OH
HO
OH
9050 Guan-fu base P

9045 Guan-fu aminealcohol
11,13-Diacetyl-14-hydroxy-2-isobutyryl hetisine C28H37NO7 (499.61).

Yellowish resin. Source: HUANG HUA WU TOU Aconitum coreanum
O O
OH
O
O
HO
HO
OH
N
O
OH
508
9051 Guanfu base Q
9055 Guangsangon C
13-Dehydro-1-acetyl-2,6-dihydroxyhetisine C22H27NO5 (385.46).
Colorless needles, mp 235~236C. Source: HUANG HUA WU TOU Aconitum
MeOH). Pharm: Antioxidant (100mol/L, InRt of MDA = 96.2%, control
coreanum (stem and leaf). Ref: 4872.
Vitamin E, InRt of MDA = 81.5%; 10mol/L, InRt of MDA = 81.7%, Vitamin

E, InRt of MDA = 33.9%). Source: NAI SANG Morus macroura (stem
O
O
HO
HH
O
cortex). Ref: 5013.
H
H
OH
HO
O
HO
HO
OH
OH
9052 Guan-fu base Z
OH
HO

OH
OH
HO
9056 Guangsangon D
OH

E, InRt of MDA = 33.9%); anti-inflammation (polymorphonuclear leukocytes,
9053 Guangsangon A
C39H38O10 (666.73). Yellow amorphous powder,
[]D29 =
408.5 (c = 0.13, MeOH).
lysosome enzyme release inhibitor, 10mol/L, InRt = 24.3%, p<0.05, control
Pharm: Antioxidant (100mol/L, InRt of MDA = 102.7%, control Vitamin E, InRt
Ginkgolide B, InRt = 58.9%). Source: NAI SANG Morus macroura (stem
of MDA = 81.5%; 10mol/L, InRt of MDA = 84.9%, Vitamin E, InRt of MDA =
cortex). Ref: 5013.
33.9%); anti-inflammation (polymorphonuclear leukocytes, lysosome enzyme

release inhibitor, 10mol/L, InRt = 19.0%, p<0.05, control Ginkgolide B, InRt =
HO
58.9%). Source: NAI SANG Morus macroura (stem cortex). Ref: 5013.
OH
HO
OH
OH
O
OH
OH
O
HO
HO
OH
HO
OH
OH
OH
OH
9057 Guangsangon E
9054 Guangsangon B
C39H36O9 (648.72). Brown amorphous powder, []D29 = +139.7 (c = 0.11,
C34H30O8 (566.61). Brown amorphous powder, []D29 = 394.7 (c = 0.11, MeOH).
Pharm: Antioxidant (100mol/L, InRt of MDA = 95.1%, control Vitamin E, InRt of
MDA = 81.5%; 10mol/L, InRt of MDA = 83.7%, Vitamin E, InRt of MDA =
E, InRt of MDA = 33.9%). Source: NAI SANG Morus macroura (stem
33.9%); anti-inflammation (polymorphonuclear leukocytes, lysosome enzyme
cortex). Ref: 5013.
release inhibitor, 10mol/L, InRt = 57.3%, p<0.001, control Ginkgolide B, InRt =

58.9%). Source: NAI SANG Morus macroura (stem cortex). Ref: 5013.
OH
HO
HO
O
HO
OH
OH
HO
HO
OH
HO
OH
OH
OH
OH
509
9058 Guangsangon F
9061 Guangsangon I
C40H36O10 (676.73). Brown amorphous powder, []D21 = 112.1 (c = 0.13,
MeOH). Source: NAI SANG Morus macroura (stem cortex). Ref: 3891.
MeOH). Pharm: Antioxidant (to determine inhibitory rates of

malondialdehyde (MDA) (H. Lu, et al., Chem Biol Interact, 1991, 78, 77-84.),
OH
10mol/L, InRt = 93.9%, control Vitamin E, InRt = 33.4%);

HO
HO
InRt = 43.8%, control Ginkgolide B, InRt = 58.9%). Source: NAI SANG

Morus macroura (stem cortex). Ref: 3891.
O
HO
OH
O
OH
OH
HO
9059 Guangsangon G
O
OH
HO

MeOH). Source: NAI SANG Morus macroura (stem cortex). Ref: 3891.
OH
HO
HO
OH
O
OH
9062 Guangsangon J
HO
HO
OH

malondialdehyde (MDA), 10mol/L, InRt = 91.1%, control Vitamin E, InRt
O
OH
HO
= 33.4%); anti-inflammatory (to determine release of lysosome enzyme from


OH
O
OH
HO
9060 Guangsangon H
HO

malondialdehyde (MDA) (H. Lu, et al., Chem Biol Interact, 1991, 78, 77-84.),
OH
OH
O
O
HO
OH
10mol/L, InRt = 93.1%, control Vitamin E, InRt = 33.4%);

9063 Guangsangon K
MeOH). Pharm: Antioxidant (microsomal lipid peroxidization induced by

ferrous-cysteine in vitro, determined by the content of malondialdehyde,
10mol/L, InRt = 91.8%, control Vitamin E, InRt = 18.2%). Source: NAI
OH
HO
HO
SANG Morus macroura. Ref: 2570.
OH
HO
OH
O
HO
HO
OH
O
HO
O
OH
OH
OH
OH
O
OH
510
9064 Guangsangon L
9068 4-Guanidino-1-butanol
C5H13N3O (131.18). Source: YI MU CAO Leonurus heterophyllus [Syn.
Leonurus artemisia]. Ref: 6.

OH

H2N
HO
OH
O
HO
9069 -Guanidinobutyric acid
OH
HO
N
H
HN
4-Guanidino-butyric acid [463-00-3] C5H11N3O2 (145.16). mp 276~278C

(dec). Source: WANG GUA ZI Trichosanthes cucumeroides, WEI NAO
OH
OH
Erinaceus europaeus; Hemiechinus dauuricus; Hemiechinus auritus, YI MU

CAO Leonurus heterophyllus [Syn. Leonurus artemisia]. Ref: 6.
9065 Guangsangon M
OH

HO
occurring in DNA and RNA. Source: DONG CHONG XIA CAO Cordyceps
OH
sinensis (dried fungal stroma growing on larva of a caterpillar: content =

O
OH
HN
[73-40-5] C5H5N5O (151.13). mp > 300C. Pharm: Nitrogen-containing base
O
HO
N
H
9070 Guanine (1,7-Dihydro-form)
OH
HO
H2N
0.018%)[5512], QIU YIN Pheretima aspergillum; Allolobophora caliginosa

trapezoides, REN GONG YONG CHONG CAO Cordyceps militaris cv.
(sclerotium and stroma: content = 0.011%)[5512]. Ref: 6, 5512.

O
OH
H
N
HN
9066 Guangsangon N
H2N

9071 Guanosine
10mol/L, InRt = 100%, control Vitamin E, InRt = 18.2%). Source: NAI
9--Ribofuranosylguanine [118-00-3] C10H13N5O5 (283.25). mp 230~235C
(dec). Source: BAN XIA Pinellia ternata (dried tuber: content scope of 4
HO
origins = 0.0038%~0.0220%, mean content = 0.0107%[5508]), DANG GUI
OH
Angelica sinensis (root: content = 0.019%)[5514], DONG CHONG XIA CAO
O
HO
HO
Cordyceps sinensis (dried fungal stroma growing on larva of a caterpillar:
OH
content = 0.135%)[5512], GUAN HUA ROU CONG RONG Cistanche tubulosa

O
OH
(fleshy stem: content = 0.007%)[5514], HUANG QI Astragalus membranaceus

(root: content = 0.032%)[5514], MAI DONG Ophiopogon japonicus (tuberoid:
content = 0.003%)[5514], MAI JIAO Claviceps purpurea, REN GONG YONG

CHONG CAO Cordyceps militaris cv. (sclerotium and stroma: content =
OH
9067 Guanidine
0.274%)[5512], REN SHEN Panax ginseng [Syn. Panax schinseng] (root:

content = 0.035%)[5514]. Ref: 2, 5508, 5512, 5514.
[113-00-8] CH5N3 (59.07). Pharm: Supertoxic agent (orl). Source: GUI GAI
Coprinus atramentarius, QIU YIN Pheretima aspergillum; Allolobophora
caliginosa trapezoides, SHUI NIU JIAO Bubalus bubalis. Ref: 6.
N
H
O
HN
H2N
HO
N
N
N
O
H
OH OH
511
9072 (+)-Guatteboline
9076 Guggulsterone M
C35H34N2O6 (578.67). Amorphous, []D20 = +138 (c = 0.8, CHCl3). Pharm:
C22H30O3 (342.48). Needles (mp 206~208C (MeCN), []D = +93 (c = 0.65,
Antitrypanosomal (inhibits trypomastigote form of Trypanosoma cruzi, strain Y,
MeOH). Source: A MAN SU DAN MO YAO Commiphora wightii. Ref:
IC50 = 57.9g/mL, IC90 = 96.5g/mL)[3976]; antimalarial (Plasmodium
2062.
O
falciparum D6, LC50 = 207.5ng/mL, SI = 29; Plasmodium falciparum W2,

[3976]
LC50 = 72.5ng/mL, SI = 83); cytotoxic (KB, LC50 = 6000ng/mL)
. Source:
O
H
Guatteria boliviana (stem cortex). Ref: 3976.

H
O
O
H
9077 Guiachrysine
C40H44N4O3 (628.82). Orange-colored amorphous powder. Pharm: Supertoxic

agent (LD100 = 4~6mg/kg, death occurs fairly rapidly in 5~10min)[3943];
O
OH
neuromuscular toxicity (neuromuscular transmission inhibitor, IC50 =

12.5mol/L; Venezuelan calabash curare, IC50 = 6.5mol/L)[5202]. Source:
Strychnos guianensis (stem cortex). Ref: 3943, 5202.
9073 Guavacoumaric acid

2,3-Dihydroxy-24-p-z-coumaroyloxyurs-12-en-28-oic acid C39H54O7
(634.86). Colorless needles (CHCl3:MeOH = 1:1), mp 188~190C. Source:

FAN SHI LIU YE Psidium guajava. Ref: 1922.
H
N
OH
OH
H
N
H
HO
OH
HO
H
O
9078 Guiaflavine
O
C40H42N4O2 (610.81). Pharm: Neuromuscular toxicity (neuromuscular
OH
transmission inhibitor, IC50 = 25.5mol/L; Venezuelan calabash curare, IC50 =
9074 Guavanoic acid

20-Acetoxy-2,3-dihydroxyurs-12-en-28-oic acid C32H50O6 (530.75).
6.5mol/L)[5202]. Source: Strychnos guianensis (stem cortex). Ref: 3943, 5202.
Colorless needles (CHCl3:MeOH = 1:1), mp 221~222C. Source: FAN SHI

LIU YE Psidium guajava. Ref: 1922.
H
N
H
HO
OH
HO
H
N
9075 Guggulsterol Y
9079 Guibourtinidol-(46)-catechin
C27H46O4 (434.67). Needles, mp 236~238C (MeCN), []D = 28.8 (c = 0.5,
[27277-74-7] C30H26O10 (546.54). Pharm: Tanning agent. Source: LE SHI JIN
MeOH) Source: A MAN SU DAN MO YAO Commiphora wightii. Ref: 2062.
HE HUAN Acacia luederitzii. Ref: 658.

OH
OH
OH
OH
OH
H
H
HO
HO
HO
HO
OH
OH
OH
512
9080 Guidongnin
9085 Gummosin
Guidongnin A C20H26O6 (362.43). mp 235~237C, []D22 = 160 (c = 1.0,
C24H30O4 (382.50). Source: A WEI Ferula assafoetida (root). Ref: 5243.
C5H5N). Pharm: Cytotoxic (in vitro, K562, IC50 = 0.3g/mL; control

cis-Platin, IC 50 = 0.52g/mL)[4732]. Source: DONG LING CAO Rabdosia
rubescens, LU SHI DONG LING CAO Isodon rubescens var. lushiensis (leaf:
yield = 0.0026%dw)[4732]. Ref: 4067, 4732.
HO
HO
9086 Gurillin G
OH
O
C39H64O13 (740.94). Source: WAN QU TIAN MEN DONG Asparagus
curillus. Ref: 697.
9081 Guidongnin B
Ludongnin B C20H26O5 (346.43). mp 296~299C. Pharm: Cytotoxic inactive
(in vitro, K562, IC50 > 50g/mL; control cis-Platin, IC50 = 0.52g/mL)[4732].
Source: LU SHI DONG LING CAO Isodon rubescens var. lushiensis (leaf:
O
H
yield = 0.00021%dw). Ref: 4067, 4732.
H
O
HO
H
H
OO
OH
HO
OO
OH
OH
OH
9082 Guidongnin C
OH
C20H26O6 (362.43). Pharm: Cytotoxic inactive (in vitro, K562, IC50 >
50g/mL; control cis-Platin, IC50 = 0.52g/mL)[4732]. Source: LU SHI
DONG LING CAO Isodon rubescens var. lushiensis (leaf: yield =
0.00016%dw). Ref: 4732.
HO
C45H74O17 (887.08). Source: WAN QU TIAN MEN DONG Asparagus

curillus. Ref: 697.
9087 Gurillin H
O
O
9083 Guineensine
OH
H
H
OO
C24H33NO3 (383.54). Colorless crystals; crystalline solid. Pharm: Protective

gastric lesions (rat, ethanol-induced, 25mg/kg orl, length = (78.613.0)mm,
HO
control, length = (118.616.2)mm, InRt = 33.7%; indomethacin-induced in

rats, dose, 25mg/kg orl, length = (54.39.8)mm, control, length =
(89.59.8)mm, InRt = 39.3%)[4935]; ACAT inhibitor (dose-dependent manner,
IC50 = 3.12mol/L)[5005]. Source: BI BA Piper longum (fruit), Piper chaba
(fruit). Ref: 4935, 5005.
O
O
OH
OO
OH
OO
HO
OH
OH
OH
OH
9088 -Guriunene
N
H
C15H24 (204.36). bp 114~116C/10mmHg. Source: BAI ZHI Angelica

dahurica [Syn. Angelica porphyrocaulis], GUANG HUO XIANG
Pogostemon cablin [Syn. Mentha cablin], NAN HE SHI Daucus carota, REN
SHEN Panax ginseng [Syn. Panax schinseng], SAN QI Panax
9084 Guisinol
C23H35ClO5 (416.91). Yellowish oil. Source: Emericella unguis. Ref: 1890.
OH
OH
Cl
Kaempferia galanga, SHUI CAI Menyanthes trifoliata. Ref: 2, 660.
O
HO
pseudo-ginseng var. notoginseng [Syn. Panax notoginseng], SHAN NAI
513
9089 Guttiferone A
9093 Guvacoline
C38H50O6 (602.82). Yellow oil, []D20 = +32 (c = 0.04, CHCl3). Pharm:
[495-19-2] C7H11NO2 (141.17). mp 27C, bp 114C/14mmHg. Source: BING
Cytotoxic (hmn ovarian A2780 cell line, IC50 = 6.8g/mL, control
LANG Areca catechu (dried ripe seed: content scope 0.03%0.06%[5508]). Ref:
Actinomycin D, IC50 = 0.003g/mL). Source: Garcinia macrophylla (twig).
2, 5508.
Ref: 5442.
O
O
N
H
OH
O
HO
9094 Gycomoside I
O
O
1,3,12,20(S),26-Pentahydroxy-dammer-24(25)-en-20(S)-O--D-glucopyra
nosyl-(16)--D-gluco-pyranoside [150626-50-9] C42H72O15 (817.03).
OH
Colorless acicular Crystals, mp 196~197C, []D22 = + 18.56 (c= 1.67,

MeOH). Source: BIAN GUO JIAO GU LAN Gynostemma compressum. Ref:
9090 Guttiferone G
266.

CHCl3). Pharm: Cytotoxic (hmn ovarian A2780 cell line, IC50 = 8.0g/mL,
HO
(twig). Ref: 5442.
OO
OO
OH
control Actinomycin D, IC50 = 0.003g/mL). Source: Garcinia macrophylla
OH
OH
OH
OH
OH H
OH
OH
OH
H
HO
OH
O
HO
9095 Gycomoside II
O
O
1,3,12,20(S)-Tetrahydroxy-dammer-24(25)-en-3-O--D-glucopyranosyl-2
0(S)-O--D-glucopyranosyl-(16)--D-glucopyranoside [150626-51-0]
OH

MeOH). Source: BIAN GUO JIAO GU LAN Gynostemma compressum. Ref:
9091 Guttiferone I
266, 1521.
C38H50O6 (602.82). Bright yellow solid, mp 60~62C, []D = 68 (c = 1.2,

HO
CHCl3). Source: GE LI FEI SI TENG HUANG Garcinia griffithii (stem
OO
OO
OH
cortex). Ref: 5311.
OH
OH
OH
OH OH OH
OH
H
O
HO
OH
H
HO
OO
OH
O
OH
OH
OH
9096 Gycomoside III

9092 Guvacine
1,3,12,20(S),26-Pentahydroxy-dammer-24(25)-en-20(S)-O--D-glucopyra
[498-96-4] C6H9NO2 (127.14). mp 285C (dec). Pharm: Inhibits absorption of
noside C36H62O10 (654.89). Yellowish powder, mp 178~180C, []D22 =
GABA and -alanine (cat, myeloid section and cerebral section);
+23.73 (c = 0.59, MeOH). Source: BIAN GUO JIAO GU LAN Gynostemma
Antidyskinetic (inhibits spontaneous movement, mus, 50~100mg/kg, ip).
compressum. Ref: 266.
Source: BING LANG Areca catechu (dried ripe seed: content scope
HO
0.19%0.72%, middle value = 0.46%[5508]). Ref: 6, 658, 5508.
OO
OH
OH
O
OH
N
H
OH
OH
OH
H
HO
OH
H
514
9097 Gycomoside IV
9100 Gymconopin B
1,3,12,20(S),26-Pentahydroxy-dammer-24(25)-en-3-O--D-glucopyranosy
C22H20O4 (348.40). White powder. Pharm: Antiallergic -Hexosaminidase
l-20(S)-O--D-glucopyranosyl-(16)--D-glucopyranoside C48H82O20
(979.18). White powder, mp 207~209C, []D22 = +12.96 (c = 1.08, MeOH).
Source: BIAN GUO JIAO GU LAN Gynostemma compressum. Ref: 266.

HO
OO
OO
OH
OH
OH
OH
OH
OH
OH
OH
OH
H
OH
H
HO
OO
OH
OH
OH
OH
9101 Gymconopin C
OH
C30H26O6 (482.54). White powder. Source: SHOU ZHANG SHEN

9098 Gylongiposide I
C46H76O16 (885.11). White crystalline powder, mp 219.5~220.0C, [] D20 =
1.7 (c = 1, methanol). Source: CHANG GENG JIAO GU LAN
HO
OH
Gynostemma longipes. Ref: 390.
HO
HO
OH
HO
H
O
H
OH
OO
OO
OH

OH
OH
9102 Gymconopin D
OO
OH
fumarate, InRt = (72.50.9)mol/L, p<0.01)[5022]. Source: SHOU ZHANG

SHEN Gymnadenia conopsea (tuber). Ref: 5022.
OH OH
HO
9099 Gymconopin A
HO


9103 Gymnaconitine
[103956-41-8] C34H47NO8 (597.76). White acicular Crystals, mp 110~111C,
OH
[]D17 = +18.2. Source: LU RUI WU TOU Aconitum gymnandrum. Ref: 52.
H
OH
OH
OH
O
O
O
O
OH
515
9104 Gymnasterkoreaside A
9109 Gymnasterkoreayne G
(3R)-8-Decene-4,6-diyne-1,3-diol 1-O--D-glucopyraside C16H22O7 (326.35).
C17H24O3 (276.38). Orange oil, []D20 = +40.0 (c = 0.3, CHCl3). Pharm:
Bright yellow oil, []D20 = 28 (c = 1, MeOH). Source: CHAO XIAN LUO
NFAT transcription factor inhibitor (IC50 = (43.92.2)mol/L, positive
WAN Gymnaster koraiensis (root). Ref: 4196.
control Cyclosporin A, IC50 = (0.310.01)mol/L). Source: CHAO XIAN

LUO WAN Gymnaster koraiensis (leaf). Ref: 4511.
HO
OO
HO
OH
OH
OH
OH
OH
OH
9105 Gymnasterkoreaside B
9110 Gymnemic acid I
(3R)-8-Decene-4,6-diyne-1,3-diol
[122168-40-5] C43H66O14 (807.00). Pharm: Flavorant. Source: CHI GENG
1-O--D-apiofuranosyl-(16)--D-glucopyraside C21H30O11 (458.47). Bright
TENG Gymnema sylvestre. Ref: 658.
20
yellow oil, []D = 78 (c = 1, MeOH). Source: CHAO XIAN LUO WAN

Gymnaster koraiensis (root). Ref: 4196.
O
O
HO
HO
OO
OH OH
OH
OH
OH
H
O
HO
OH
OO
20
C17H22O2 (258.36). []D = +163.0 (c = 0.3, CHCl3). Pharm: NFAT

transcription factor inhibitor (IC50 = (1.440.59)mol/L, control Cyclosporin
A, IC50 = (0.310.01)mol/L). Source: CHAO XIAN LUO WAN Gymnaster
koraiensis (leaf). Ref: 4511.
OH
OH
9106 Gymnasterkoreayne B
OH
OH
OH
9111 Gymnoside VIII

C44H60O24 (972.95). White powder, []D24 = 37.3 (c = 0.39, MeOH). Source:
SHOU ZHANG SHEN Gymnadenia conopsea (tuber: yield = 0.0003%). Ref:
2089.
OH
O
20
C17H24O3 (276.38). []D = +87.9 (c = 0.3, CHCl3). Pharm: NFAT

Cyclosporin A, IC50 = (0.310.01)mol/L)
[4511]
. Source: CHAO XIAN LUO
OO
HO
OH
WAN Gymnaster koraiensis (leaf). Ref: 4511.
OH
transcription factor inhibitor (IC50 = (7.240.42)mol/L, positive control
OH
H
9107 Gymnasterkoreayne E
HO
OH
OH
OH
OH
OH O
9112 Gymnoside IX
OH

Source: SHOU ZHANG SHEN Gymnadenia conopsea (tuber: yield =
OH
0.013%). Ref: 2089.

9108 Gymnasterkoreayne F
C17H22O2 (258.36). []D20 = +134.0 (c = 0.3, CHCl3). Pharm: NFAT
transcription factor inhibitor (IC50 = (10.60.5)mol/L, control Cyclosporin

A, IC50 = (0.310.01)mol/L)[4511]. Source: CHAO XIAN LUO WAN
Gymnaster koraiensis (leaf). Ref: 4511.
OO
HO
OH
OH
OH
HO
O
OH
O
OH
OH
O
O
O
O
OH
OO
HO
OH
OH
OH
516
9113 Gymnoside X
9117 Gynoside B
(20S,24S)-20,24-Epoxy-12,25-dihydroxydammaran-3-yl O--D-glucopy-
Source: SHOU ZHANG SHEN Gymnadenia conopsea (tuber: yield =
ranosyl-(12)--D-glucopyranoside C42H72O14 (801.03). Amorphous powder,
0.0005%). Ref: 2089.
mp 194~196C, []D20 = +0.10 (c = 0.05, MeOH). Source: JIAO GU LAN

Gynostemma pentaphyllum (leaf: yield = 0.00025%dw). Ref: 4757.
O
O
O
OO
HO
OH
OH
HO
OH
O
OH
OH
OH
O
O
OH
O
OH
OH
OH
H
HO
9114 Gynocardin
[14332-17-3] C12H17NO8 (303.27). Pharm: Toxin. Source: MA DAN GUO
HO
HO
HO
HO
HO
Gynocardia odorata. Ref: 658.
O O
OH
9118 Gynoside C
OO
OH
HO
OH
OH
HO
(20S,24R)-20,24-Epoxy-12,25-dihydroxydammaran-3-yl O--D-glucopyranosyl-(12)--D-xylopyranoside C41H70O13 (771.01). Amorphous powder,

mp 194~196C, []D20 = 8.0 (c = 0.1,MeOH). Source: JIAO GU LAN
HO
OH
9115 Gynosaponin TN1

C36H62O9 (638.89). Source: JIAO GU LAN Gynostemma pentaphyllum (leaf:
yield = 0.036%dw). Ref: 4757.
HO
HO
HO
OH
OH OH
H
HO
HO
HO
HO
HO
HO
O O
OH
HO
9119 Gynoside D
(20S,24S)-20,24-Epoxy-12,23,25-trihydroxydammaran-3-yl O--D-gluco9116 Gynoside A
pyranosyl-(12)--D-xylopyranoside C41H70O14 (787.01). Amorphous
(20S,24S)-20,-24-Epoxy-12,25-dihydroxydammaran-3-yl O--D-glucopyra-
powder, mp 195~197C, []D20 = +0.61 (c = 0.1, MeOH). Source: JIAO GU
nosyl-(12)--D-xylopyranoside C41H70O13 (771.01). Colorless plates, mp
LAN Gynostemma pentaphyllum (leaf: yield = 0.00077%dw). Ref: 4757.
203~205C, []D20 = 0.47 (c = 0.9, MeOH). Source: JIAO GU LAN

OH
OH
OH
OH
OH
H
O
HO
HO
HO
HO
HO
O
O
OH
HO
HO
HO
HO
HO
O
OO
OH
517
9120 Gynoside E
9124 Gypenoside I
(12R,20S,24S)-20,24;20,12-Diepoxy-25-hydroxydammaran-3-yl
C60H102O27 (1255.47). Source: JIAO GU LAN Gynostemma pentaphyllum.
O--D-glucopyranosyl-(12)--D-xylopyranoside C41 H68O13 (768.99).
Ref: 2.
Amorphous powder, mp 207~209C, []D20 = +2.0 (c = 0.15, MeOH).

Source: JIAO GU LAN Gynostemma pentaphyllum (leaf: yield =
HO
0.0001%dw). Ref: 4757.
OO
OH
HO
O O
OH
OH
OH
HO
HO
HO
HO
HO
OO
OH OHOH
HO
OO
OH
OH
OH H
OO
OH
OH
OH
OH
OH
OH
9125 Gypenoside II
9121 Gynunol
C11H14O3 (194.23). Colorless oil. Source: TUO YUAN SAN QI CAO Gynura
elliptica. Ref: 763.

Ref: 2.
OH
OH
OO
OO
OH
HO
OH
H
OH
OH
OH OH
OH OO
OO
9122 (+)-Gynunone
TUO YUAN SAN QI CAO Gynura elliptica. Ref: 763.
OH
OH OH OH
HO
OH
H
O
O
HO
OH
OH
9126 Gypenoside V
9123 ()-Gynuraone
Gynosaponin E [80321-60-4] C54H92O22 (1093.32). Source: JIAO GU LAN
Gynostemma pentaphyllum. Ref: 2, 1521.
Platelet aggregation inhibitor (washed rabbit platelets, 100g/mL, 100mol/L

AA-induced, AggRt = 7.2%, control 50mol/L Aspirin, AggRt = 100%;
10g/mL collagen-induced, AggRt = 7.5%, 100mol/L Aspirin, AggRt = 4.9%;
OH
OO
OH
0.1U/mL thrombin-induced, AggRt = 4.0%, 100mol/L Aspirin, AggRt =

1.7%; 2ng/mL PAF-induced, AggRt = 2.9%, 100mol/L Aspirin, AggRt =
OH OH
OH
OH
H
OH
2.1%). Source: SAN QI CAO Gynura segetum [Syn. Gynura japonica]

H
HO
OO
OH
HO
O
HO
OH
HO
OO
OH
OH
OH
518
9127 Gypenoside VI
9131 Gypenoside XI
C54H92O22 (1093.32). Source: JIAO GU LAN Gynostemma pentaphyllum. Ref: 2.
Gynosaponin K [80321-64-8] C48H82O17 (931.18). Source: JIAO GU LAN
HO
OO
OH
OH
OH
H
OO
HO
OH
OH
OH
OH
OO
OH OH
OH
OH OO
OH
OH OH
OH
OH
9132 Gypenoside XII
9128 Gypenoside VII

Gynosaponin G [80321-62-6] C54H92O21 (1077.32). Source: JIAO GU LAN

OH OO
HO
OO
OH
OH
H
OH
OH OH
OH
OO
OH
OH OH
OH
9133 Gypenoside XIII

Gynosaponin M [80325-22-0] C41H70O12 (755.01). Source: JIAO GU LAN
[52705-93-8] C48H82O18 (947.18). Source: JIAO GU LAN Gynostemma
pentaphyllum (aerial parts: yield = 0.0041%dw)[4751]. Ref: 2, 4751.

O
OH
OH
H
OO
9134 Gypenoside XVII

Gynosaponin S C48H82O18 (947.18). Pharm: Hepatoprotective (inhibits
activation of macrophages, inhibits increase in sALT and sAST levels, in vivo,

D-GalN/LPS-induced liver injury in mouse, 100mg/kg ip for sALT, InRt =
OH
95%; 100mg/kg ip for sAST, InRt = 91%; control Hydrocortisone, 20mg/kg
OH
ip for sALT, InRt = 99%; 20mg/kg ip for sAST, InRt = 97%)[4702]. Source:
9130 Gypenoside IX
pentaphyllum, SAN QI HUA LEI Panax pseudo-ginseng var. notoginseng
[Syn. Panax notoginseng] (flower bud: yield = 0.11%dw)[4702]. Ref: 2, 1521,
4702.
JIAO GU LAN Gynostemma pentaphyllum, SAN QI HUA LEI Panax

pseudo-ginseng var. notoginseng [Syn. Panax notoginseng] (flower bud: yield
= 0.18%dw)[4702]. Ref: 2, 1521, 4702.
HO
OH
OH
OHH
OO
OH
OH
OH
OH
H
OH
H
HO
OO
OH
OH
OH
OH
OH
H
HO
OH
OO
OO
OH
OH
OH
OH
OH
OH
H
HO
OH
O
OH
H
OH
OH
OH
OH
HO
OH
OH
H
HO
OO
OO
OH
OH
OH
OH
9129 Gypenoside VIII
OH
OH
OH
HO
OH
H
OO
H
OH
HO
OO
O
OH
OH
OH
OH
OH
OO
OH
OH
HO
OH
OO
OH
H
OH
519
9135 Gypenoside XVIII
9139 Gypenoside XXII
C54H92 O22 (1093.32). Source: JIAO GU LAN Gynostemma pentaphyllum.
Ref: 2.
Ref: 2.
OH
OO
OO
OH
OH
OH OH
OH
OO
OH
OH
H
OO
OO
OO
OH
OO
OH
OH
OH
OH OH
H
HO
OH
OH
OHHO OH
OH
OH
H
OH
OH
HO
OH
9136 Gypenoside XIX

OH O O
OH
OH
9140 Gypenoside XXVI
OH
OH
H
OH
OH OH
OH
OH
Ref: 2.
OO
HO
OH
OO
HO
OH
H
OH O O
OH
OH
OO
HO
OH
O OH
OH
HO
OH
OH
OO
OH
OH
9137 Gypenoside XX
OH
9141 Gypenoside XXIX
Ref: 2, 1521.

Ref: 2.
OO
HO
OH
OH
OO
OH
OH OH
HO
OH
OH
H
OH
H
OH
OH
OO
OO
HO
OH OHOH
HO
OO
OH
OH
OH
OH
OH
OH
OO
OH
9142 Gypenoside XXX
OH
9138 Gypenoside XXI
C41H70O13 (771.01). Source: JIAO GU LAN Gynostemma pentaphyllum. Ref:
Ref: 2.
2, 1521.
HO
OO
OH
OH
OO
OH
OHOH
OH
H
OH
OH
HO OH
OH
H
HO
H
HO
OO
OH
OO
OH
OH
OH
520
9143 Gypenoside XXXIV
9146 Gypenoside XXXVII
Ref: 2.
Ref: 2.
OH OO
OO
H
OH
OH OH O OH
OO
OO
OH
OH
OH
H
OH
OH
OO
OH
OH
HO
OO
OH
OH
O
O
HO
H
HO
OH
O OH
OO
HO
OH
OH
OH
OH
OH
OH
9144 Gypenoside XXXV
9147 Gypenoside XXXVIII
Ref: 2.
Ref: 2.
OO
OO
OH
OH
OH O OH
HO
OH
OH
H
H
HO
H
H
HO
OO
OH
HO
OH
OH
OH
HO
OO
HO
OO
OH
OO
OH
OH
OH
OH
OH
9145 Gypenoside XXXVI
9148 Gypenoside XXXIX
Ref: 2.
Ref: 2.
OH
HO
OH
H
OO
OO
OH
OH
OH OH O OH
HO
H
H
HO
OO
OH
OH
O
O
HO
OH
OO
HO
OH
OH
O
HO
OH
OH
OH
OH
OH
521
9149 Gypenoside XL
9152 Gypenoside XLIII
C 53 H 90 O 22 (1079.30). Source: JIAO GU LAN Gynostemma
Ref: 2.
HO
OH
OH
OO
H
HO
OH
OO
OH
HO
OH
OH
OH OH
OH
OH
H
OH
H
HO
O
O
OO
OH
OH
O
O
HO
OH
OH
OH
OH
OH
9150 Gypenoside XLI

Ref: 2.
9153 Gypenoside XLIV

C 47 H 80 O 18 (933.15). Source: HUI GUO JIAO GU LAN Gynostemma
yixingense, JIAO GU LAN Gynostemma pentaphyllum. Ref: 2, 329.
HO
H
HO
HO
H
HO
OO
OH
OO
OH
OH
HO
OO
OH
OH
OH
O
O
HO
OH
H
OH
OH
OH
OH
OH
OH
OH
OH
9151 Gypenoside XLII

C53H90 O23 (1095.29). Source: HUI GUO JIAO GU LAN Gynostemma
yixingense, JIAO GU LAN Gynostemma pentaphyllum (leaf)
OO
O
OH
H
OH
OH
. Ref: 2,
9154 Gypenoside XLV

Ref: 2.
329, 4757.
HO
[4757]
OH
OH
OH
OH
OH
OH
OH
OH OH
H
OO
HO
OH
O
O
OH
OH
OH
OH
OH
OH
H
OO
HO
OH
OH
HO
O
O
OO
OH
H
522
9155 Gypenoside XLVI
9158 Gypenoside LIII
yield = 0.051%dw)[4757]. Ref: 2, 4757.
HO
OH
OH
H
OH
OHH
OH
OH
OH
OO
OH
O
O
HO
OH
OH
HO
OO
OH
H
HO
OH
OH
OH
9159 Gypenoside LIV
OH
OH

OH
OH
H
9156 Gypenoside LI
HO
Ref: 2.
H
OH
OH
OH
H
O
O
HO
OH
H
OO
OH
OH
OH
9160 Gypenoside LV
OH
O
O
HO
OH
HO
HO
OO
OH
OO
OH
OH
OH
O
O
OH
OH
OH
OH
OH
OH
H
HO
9157 Gypenoside LII
OO
OH

Ref: 2.
OH
OH
9161 Gypenoside LVI

C53H90O22 (1079.30). Source: JIAO GU LAN Gynostemma pentaphyllum
OO
HO
(leaf: yield = 0.00063%dw)[4757]. Ref: 2, 1521, 4757.
OH
HO
OHH
OH
O
OH
OO
OH
H
OH
OO
OH
OH
OO
OH
OH
OH
OH
OH
H
HO
OO
OH
OH
OH OH
OO
OH
HO
O
O
OH
OH
OH
523
9162 Gypenoside LVII
9166 Gypenoside LXII
yield = 0.051%dw)[4757]. Ref: 2, 1521, 4757.

OO
OO
OO
OH
OH
OH
OH
OH
OH
H
OH
OH
HO
OH
H
O
O
HO
OH
OO
OH
OH
H
OH
OH HO OH
H
HO
OO
OH
OH
OH
OO
HO
OH
OH
OH
OH
9163 Gypenoside LVIII
9167 Gypenoside LXIII
OO
OH
OH
OO
OHOH
OH
OH
H
HO
O
O
OH
OH
OO
OO
HO
OH
OH
OH
OH
OH HO OH
OH
HO
OO
OH
OH
H
OH
OO
OO
OH
OH
OH
OH
OH
9168 Gypenoside LXIV

9164 Gypenoside LIX

pentaphyllum. Ref: 2, 1521.
O
O
OO
OH
OH
OO
OH
O
O
OH
OH
OH
H
OH
OH
OH
HO
OH
OH
OH
OH
OH
OH
HO
H
O
O
HO
H
HO
OH
OH
OH
9165 Gypenoside LX
yield = 0.00023%dw)[4757]. Ref: 2, 4757.
OO
OH
OH
OH
OH
H
OH
O
O
OO
OO
OH
OH
9169 Gypenoside LXV
OH
OH
OH
OH
OH
OH HO OH
HO
H
H
HO
HO
OH
H
524
9170 Gypenoside LXVII
9174 Gypenoside LXXII

Ref: 2.
OO
OO
OH
OH
OH
OH
OH HO OH
HO
HO
H
OH
OH
OH OH
OH
OH
OH
OO
OO
OH
9175 Gypenoside LXXIII
OH
9171 Gypenoside LXVIII

Ref: 2.
OH
Ref: 2.
OH
OH
H
OH
OH
OH
HO
OH
OH
OH
OH
HO
H
OO
HO
OH
OH
OH OH
OH
HO
H
O
O
HO
OO
OO
OH
O
O
OO
OH
OH
OH
OH
HO
OH
OH
OH
OH
H
OH
H
O
O
HO
9176 Gypenoside LXXIV
OH
Ref: 2.
OH
OH
HO
9172 Gypenoside LXX

Ref: 2.
OH
OH
OH
OH
OH
H
OH
H
OH
OH HO OH
OH
OO
OO
OH
OH
OO
OO
OH
OH
HO
OH
9177 Gypenoside LXXV

H
O
O
HO
OH
OH
HO
H
HO
O
O
OH
OH
OH
O
O
OO
OH
OH
OH
OH
OH
OH
H
OH
HO
9173 Gypenoside LXXI
C41H70O12 (755.01). Source: JIAO GU LAN Gynostemma pentaphyllum

(aerial parts: yield = 0.0012%dw)[4751]. Ref: 2, 4751.
9178 Gypenoside LXXVI

OO
OH
OH
OH
OO
OO
HO
OH
OH
OH
OH
OH
OH
OH
HO OH
H
HO
H
HO
525
9179 Gypenoside LXXVII
9183 Gypsogenin
[639-14-5] C30H46O4 (470.70). mp 274C. Pharm: Toxin (mammal). Source:
yield = 0.061%dw)[4757]. Ref: 2, 4757.
YIN CHAI HU Stellaria dichotoma var. lanceolata, SHAN YIN CHAI HU

Gypsophila pacifica, MAI XIAN WENG Agrostemma githago. Ref: 6, 658.
OO
OO
OH
OH
OH
OH
OH
OHH
OH
HO
OH
HO
H
H
9180 Gypenoside LXXVIII

Ref: 2.
9184 Gypsoside
[15588-68-8] C80H126O44 (1791.87). mp 215~220C (dec), []D20 = 22.1 2 (c
OO
OH
OH
OH
= 3.07, water). Pharm: Antispasmodic (delays convulsive spasm, mus,
OO
OH
HO
OH
OH
caused by corazol, camphor or coffeine); hypnotic (mus hypnotic synergism

H
with barbital sodium and chloral hydrate); antihypercholesterolemic (atherosis
OH
rbt, reduces the level of cholesterol in serum, cholesterol/cephalin coefficient,

and lipoid content in aorta); anticonvulsant (caused by strychnine). Source:
H
HO
SHAN YIN CHAI HU Gypsophila pacifica. Ref: 661.
9181 Gypenoside LXXIX

Ref: 2.
H
HO
OO
HO
OH
HO OH
OO
OO
OH
HO
HO
OO
OH
OH
OH
HO
H
HO
O
OO
OH
H
D-fucop
HO
O O
O O
O OH OH
OH
OH
OH
OH OH
OH
OH
O
OH
OH
OH
OH
OO
O
OH
OH
OH
OH
9182 Gypentonoside A
[20S]-3,20-Dihydroxy-24-dammaren-12,23-dione-3-O-[-L-rhamnopyranosy
l-(12)-[-L-rhamnopyra-nosyl-(13)]--L-rhamnopyranosyl-(16)]--D-
9185 Gyrophoric acid
glucopyranoside C54H88O21 (1073.29). White powder, mp 272~274C. Source:
[548-89-0] C24H20O10 (468.42). mp 220C (dec). Source: SHI HUA Parmelia
JIAO GU LAN Gynostemma pentaphyllum. Ref: 364.
saxatilis. Ref: 6.
HO
O
H
H
OH
OO
OO
O
OH
OH
OH OH
OO
OH O
OH OH
OH OH
OH
O
HO
OH
OH
OH

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What is the book about?

What is the book about?

What information is provided about each entry?

What information is provided about each entry?

Encyclopedia of Traditional Chinese Medicines

Molecular Structures, Pharmacological Activities,

Jiaju Zhou Guirong Xie Xinjian Yan

Cover design: deblik, Berlin

Encyclopedia of Traditional Chinese Medicines

Volume 5 Isolated Compounds (T-Z)

JJ Zhou, GR Xie and XJ Yan

Normalization of Pharmacological Data. More than 8,000 TCM components in this

In order to standardize abbreviations of cancer cells, such as BT474, CHAGO,

Other six cases are:

Translation of TCM Effects Terms. In the Volume 5 of the encyclopedia, 6,926

Translation of TCM Indications Terms. Based on Wisemans terminological system,

In summary, this encyclopedia provides a collection of more than 23,000 TCM

Jiangsu New Medical College Ed., Chinese Medicine Dictionary, Shanghai

Nigel Wiseman, English-Chinese, Chinese-English Dictionary of Chinese

(Comprehensive data sources of compounds)

Tatsuo Karikome, Wenben Yang translated, Phytochemistry, Science Press,

How to Use the Books

Plant T0001 effects, indications

Sketch Map of Three Important Many to Many Relationships

2. Seven Useful Indexes

with related compound codes. For example, if there is a question as:

Index 3 (Compound Synonym Index) is useful for searching a compound from a

3. Data Survey Example of Compound Entry

22270 Ursolic acid

Pharm: (27 items)

(66912)mol/L, ASA, IC 50 = (66.02.1)mol/L; 1~5mol/L PGH2/TXA2

RONG SHU Ficus microcarpa (aerial root),

Abbreviations and Symbols

I-Transforming Growth Factor-1

2,2'-Azino-Bis-(3-ethylbenzThiazoline 6-Sulphonic acid), radical

Angiotensin Converting Enzyme

macrophage inflammatory protein (MIP-1), monocyte chemotactic

95% Fiducial Limits (=95% Confidence Interval)

protein (MCP-2), and C lymphotactin (ltn) (a chemokine family)

Minimum cytotoxic concentration

IC50 of cytotoxicity (concentration of the 50% cytotoxic effect)

concentration required to double enzyme (induction) activity

Concentration required to double quinone reductase (induction)

medium Convulsive Dose

cyclic guanosine monophosphate

Caffeic Acid Phenethyl Ester

Chinese hamster ovarian

acquired immunodeficiency syndrome

Chemopreventive index (=IC50/CD)

amyotrophic lateral sclerosis

complete inhibiting minimum concentration

avian myeloblastosis virus

6-Cyano-7-nitroquinoxaline-2,3-dione (non-NMDA receptor

dl-2-Amino-5-phosphonovaleric acid (a competitive antagonist of the

central nervous system

aspartate transaminase; aspartate aminotransferase

corticotrophin releasing factor

corticotrophin releasing hormone-1

Butylated HydroxyAnisole; 3-tert-Butyl-4-HydroxyAnisole

Cytochrome P450 2D6