Atiprosin

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Atiprosin
Atiprosin structure.png
Systematic (IUPAC) name
(4aR,12bS)-1-ethyl-12-methyl-4-(propan-2-yl)-1,2,3,4,4a,5,6,12b-octahydropyrazino[2',3':3,4]pyrido[1,2-a]indole
Clinical data
Legal status
  • Uncontrolled
Routes of
administration
Oral
Identifiers
CAS Number 89303-63-9 N
ATC code none
PubChem CID: 71770
ChemSpider 64808 YesY
UNII ALS52889WF YesY
ChEMBL CHEMBL2111172 N
Chemical data
Formula C20H29N3
Molecular mass 311.46 g/mol
  • n23c1ccccc1c(c2[C@H]4N(CCN([C@@H]4CC3)C(C)C)CC)C
  • InChI=1S/C20H29N3/c1-5-21-12-13-22(14(2)3)18-10-11-23-17-9-7-6-8-16(17)15(4)19(23)20(18)21/h6-9,14,18,20H,5,10-13H2,1-4H3/t18-,20+/m1/s1 YesY
  • Key:WXNVFYIBELASJW-QUCCMNQESA-N YesY
 NYesY (what is this?)  (verify)

Atiprosin (AY-28,228) is an antihypertensive agent which acts as a selective α1-adrenergic receptor antagonist.[1][2][3][4] It also possesses some antihistamine activity, though it is some 15-fold weaker in this regard than as an alpha blocker.[3] It was never marketed.[1]

See also

References

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